Brief Information of the Compound and Protein
Compound Name
 Compound Info 
8-bromo-3-(4-chloro-phenyl)-9-methylamino-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one
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 PubChem ID
CID: 44435349
Canonical SMILES
CNc1c(Br)cnc2sc3c(ncn(-c4ccc(Cl)cc4)c3=O)c12
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Compound Formula C16H10BrClN4OS
Compound Structure
Protein Name
 Protein Info 
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q13255
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 5.9 nM
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