Brief Information of the Compound and Protein
Compound Name
 Compound Info 
8-(4-methylphenyl)thiazolo[4'',5'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidine-2,7(1H,8H)-dione
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 PubChem ID
CID: 16659799
SID: 26519849
Canonical SMILES
Cc1ccc(-n2cnc3c(sc4ncc5sc(=O)[nH]c5c43)c2=O)cc1
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Compound Formula C17H10N4O2S2
Compound Structure
Protein Name
 Protein Info 
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q13255
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 446 nM
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