Brief Information of the Compound and Protein
Compound Name
8-(4-chlorophenyl)-1h-pyrazolo[3'',4'':4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-7(8H)-one
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PubChem ID
CID: 16659642
SID: 26519693
Canonical SMILES
Clc1ccc(cc1)-n1cnc2c(sc3ncc4c[nH]nc4c23)c1=O
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Compound Formula C16H8ClN5OS
Compound Structure
Protein Name
Metabotropic glutamate receptor 1
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
Q13255
Gene Name
GRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 37.6 nM
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   LI
   LO
   TS