| Compound ID |
Compound Name |
Compound Formula |
|
CP0395854
|
(1S,2S,5R,6R)-2-amino-4-oxobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H9NO5
|
1
|
| 1 |
EC50 = 0.16 nM
|
|
|
|
CP0396103
|
(1R,2S,4R,5R,6R)-2-amino-4-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H10FNO4
|
1
|
| 1 |
EC50 = 0.56 nM
|
|
|
|
CP0411409
|
(1R,2S,4S,5R,6R)-2-amino-4-[[5-(difluoromethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C11H12F2N4O4S
|
3
|
| 1 |
EC50 = 0.58 nM
|
|
|
| 2 |
EC50 = 6.3 nM
|
|
|
| 3 |
Ki = 13.4 nM
|
|
|
|
CP0397345
|
(1R,2S,4S,5R,6R)-2-amino-4-[[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C11H11F3N4O4S
|
3
|
| 1 |
EC50 = 0.65 nM
|
|
|
| 2 |
EC50 = 7.8 nM
|
|
|
| 3 |
Ki = 8.55 nM
|
|
|
|
CP0418878
|
(1S,2S,5R,6S)-2-amino-4-methylidenebicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C9H11NO4
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0397780
|
(1R,2S,4R,5R,6R)-2-amino-4-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H13N5O4S
|
3
|
| 1 |
EC50 = 4.5 nM
|
|
|
| 2 |
EC50 = 13 nM
|
|
|
| 3 |
Ki = 67 nM
|
|
|
|
CP0401464
|
(1R,2S,4S,5R,6R)-2-amino-4-(2H-triazol-4-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H12N4O4S
|
3
|
| 1 |
EC50 = 5.2 nM
|
|
|
| 2 |
EC50 = 19 nM
|
|
|
| 3 |
Ki = 111 nM
|
|
|
|
CP0088338
|
(1R,2S,4R,5R,6R)-2-amino-4-(1H-1,2,4-triazol-5-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H12N4O4S
|
7
|
| 1 |
EC50 = 5.6 nM
|
|
|
| 2 |
EC50 = 20.1 nM
|
|
|
| 3 |
EC50 = 21.1 nM
|
|
|
| 4 |
EC50 = 22.1 nM
|
|
|
| 5 |
EC50 = 46.3 nM
|
|
|
| 6 |
EC50 = 48.2 nM
|
|
|
| 7 |
Ki = 144 nM
|
|
|
|
CP0466979
|
1-[2-hydroxy-4-[[3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]-3-(trifluoromethyl)phenyl]ethanone
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|
C22H16F3N5O4
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0397778
|
(1R,2S,4S,5R,6R)-2-amino-4-[(5-amino-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C10H13N5O4S
|
3
|
| 1 |
EC50 = 6.4 nM
|
|
|
| 2 |
EC50 = 20.1 nM
|
|
|
| 3 |
Ki = 27.8 nM
|
|
|
|
CP0076675
|
(1S,2S,5R,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H11NO4
|
4
|
| 1 |
EC50 = 7 nM
|
|
|
| 2 |
EC50 = 34.4 nM
|
|
|
| 3 |
IC50 = 5.6 nM
|
|
|
| 4 |
Ki = 71.7 nM
|
|
|
|
CP0432878
|
(1S,2S,4S,5R,6R)-2-amino-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H11NO5
|
2
|
| 1 |
EC50 = 7.5 nM
|
|
|
| 2 |
Ki = 230 nM
|
|
|
|
CP0445963
|
(1S,2S,4R,5R,6R)-2-amino-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H11NO5
|
2
|
| 1 |
EC50 = 7.6 nM
|
|
|
| 2 |
Ki = 166 nM
|
|
|
|
CP0385922
|
(1S,2S,4R,5R,6S)-2-amino-4-azidobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H10N4O4
|
1
|
| 1 |
EC50 = 8.2 nM
|
|
|
|
CP0397781
|
(1R,2S,4R,5R,6R)-2-amino-4-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C11H14N4O4S
|
3
|
| 1 |
EC50 = 10.4 nM
|
|
|
| 2 |
EC50 = 39.5 nM
|
|
|
| 3 |
Ki = 121 nM
|
|
|
|
CP0397347
|
(1R,2S,4S,5R,6R)-2-amino-4-(1H-1,2,4-triazol-5-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H12N4O4S
|
3
|
| 1 |
EC50 = 11.2 nM
|
|
|
| 2 |
EC50 = 69.1 nM
|
|
|
| 3 |
Ki = 60.4 nM
|
|
|
|
CP0397779
|
(1R,2S,4R,5R,6R)-2-amino-4-[[5-(difluoromethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C11H12F2N4O4S
|
3
|
| 1 |
EC50 = 11.8 nM
|
|
|
| 2 |
EC50 = 53.6 nM
|
|
|
| 3 |
Ki = 95.8 nM
|
|
|
|
CP0404135
|
(1S,2S,4S,5R,6S)-2-amino-4-azidobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H10N4O4
|
1
|
| 1 |
EC50 = 12.2 nM
|
|
|
|
CP0397350
|
(1R,2S,4R,5R,6R)-2-amino-4-(2H-triazol-4-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H12N4O4S
|
3
|
| 1 |
EC50 = 12.4 nM
|
|
|
| 2 |
EC50 = 46.1 nM
|
|
|
| 3 |
Ki = 142 nM
|
|
|
|
CP0397349
|
(1R,2S,4R,5R,6R)-2-amino-4-[[5-(trifluoromethyl)-1H-1,2,4-triazol-3-yl]sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C11H11F3N4O4S
|
3
|
| 1 |
EC50 = 13.9 nM
|
|
|
| 2 |
EC50 = 54.2 nM
|
|
|
| 3 |
Ki = 84.4 nM
|
|
|
|
CP0397346
|
(1R,2S,4R,5R,6R)-2-amino-4-[(5-propan-2-yl-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C13H18N4O4S
|
3
|
| 1 |
EC50 = 16.5 nM
|
|
|
| 2 |
EC50 = 87.8 nM
|
|
|
| 3 |
Ki = 266 nM
|
|
|
|
CP0465014
|
1-[2-hydroxy-4-[[3-[5-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]-3-(trifluoromethyl)phenyl]ethanone
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|
C22H16F3N5O4
|
1
|
| 1 |
EC50 = 17.9 nM
|
|
|
|
CP0390062
|
(1S,2S,4S,5R,6S)-2,4-diaminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H12N2O4
|
1
|
| 1 |
EC50 = 21.2 nM
|
|
|
|
CP0433480
|
(1S,2S,4S,5R,6S)-2-Amino-4-methyl-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C9H13NO4
|
1
|
| 1 |
EC50 = 28.6 nM
|
|
|
|
CP0463827
|
1-[3-chloro-2-hydroxy-4-[[3-[5-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
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|
C21H16ClN5O4
|
1
|
| 1 |
EC50 = 39.3 nM
|
|
|
|
CP0397777
|
(1R,2S,4S,5R,6R)-2-amino-4-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C11H14N4O4S
|
3
|
| 1 |
EC50 = 44.3 nM
|
|
|
| 2 |
EC50 = 146 nM
|
|
|
| 3 |
Ki = 171 nM
|
|
|
|
CP0468464
|
(1S,2S,4R,5R,6S)-2,4-diaminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C8H12N2O4
|
1
|
| 1 |
EC50 = 47.9 nM
|
|
|
|
CP0372597
|
(1S,2S,4R,5R,6S)-2-Amino-4-methyl-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C9H13NO4
|
1
|
| 1 |
EC50 = 63.6 nM
|
|
|
|
CP0397348
|
(1R,2S,4S,5R,6R)-2-amino-4-[(5-propan-2-yl-1H-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C13H18N4O4S
|
3
|
| 1 |
EC50 = 74 nM
|
|
|
| 2 |
EC50 = 242 nM
|
|
|
| 3 |
Ki = 339 nM
|
|
|
|
CP0510685
|
1-[3-chloro-2-hydroxy-4-[[3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C21H16ClN5O4
|
1
|
| 1 |
EC50 = 87.4 nM
|
|
|
|
CP0523668
|
1-[2-hydroxy-3-propyl-4-[[3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
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|
C24H23N5O4
|
1
|
| 1 |
EC50 = 109.6 nM
|
|
|
|
CP0065724
|
1-[2-hydroxy-3-methyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
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|
C22H19N5O4
|
3
|
| 1 |
EC50 = 201 nM
|
|
|
| 2 |
EC50 > 25000 nM
|
|
|
| 3 |
IC50 > 12500 nM
|
|
|
|
CP0464387
|
1-[2-hydroxy-3-propyl-4-[[3-[3-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
EC50 = 227 nM
|
|
|
|
CP0385921
|
(1S,2S,4S,5R,6S)-4-acetamido-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C10H14N2O5
|
1
|
| 1 |
EC50 = 257 nM
|
|
|
|
CP0356641
|
(1S,2S,4S,5R,6S)-2-amino-4-[(3-methoxybenzoyl)amino]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C16H18N2O6
|
1
|
| 1 |
EC50 = 277 nM
|
|
|
|
CP0468331
|
1-[2-hydroxy-3-methyl-4-[[4-[3-(2H-tetrazol-5-yl)phenoxy]phenyl]methoxy]phenyl]ethanone
Show/Hide
|
C23H20N4O4
|
1
|
| 1 |
EC50 = 293.5 nM
|
|
|
|
CP0385269
|
1-[2-hydroxy-3-propyl-4-[[4-[3-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
EC50 = 309.5 nM
|
|
|
|
CP0464437
|
1-[2-hydroxy-3-propyl-4-[[3-[5-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
EC50 = 319 nM
|
|
|
|
CP0463828
|
2-[3-[(4-acetyl-3-hydroxy-2-propylphenoxy)methyl]phenoxy]pyridine-4-carboxylic acid
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|
C24H23NO6
|
1
|
| 1 |
EC50 = 404.5 nM
|
|
|
|
CP0516489
|
1-[2-hydroxy-3-propyl-4-[[4-[4-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
EC50 = 470 nM
|
|
|
|
CP0450311
|
1-[2-hydroxy-3-propyl-4-[[6-[3-(2H-tetrazol-5-yl)phenoxy]pyridin-3-yl]methoxy]phenyl]ethanone
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|
C24H23N5O4
|
1
|
| 1 |
EC50 = 561.5 nM
|
|
|
|
CP0450312
|
1-[2-hydroxy-3-propyl-4-[[4-[5-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C24H23N5O4
|
1
|
| 1 |
EC50 = 682 nM
|
|
|
|
CP0532782
|
1-[3-fluoro-2-hydroxy-4-[[3-[5-(2H-tetrazol-5-yl)pyridin-2-yl]oxyphenyl]methoxy]phenyl]ethanone
Show/Hide
|
C21H16FN5O4
|
1
|
| 1 |
EC50 = 1076 nM
|
|
|
|
CP0385920
|
(1R,2S,4S,5R,6R)-2-amino-4-phenylsulfanylbicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C14H15NO4S
|
5
|
| 1 |
EC50 = 1170 nM
|
|
|
| 2 |
EC50 > 25000 nM
|
|
|
| 3 |
IC50 > 12500 nM
|
|
|
| 4 |
IC50 = 15300 nM
|
|
|
| 5 |
Ki = 1230 nM
|
|
|
|
CP0466980
|
6-[4-[(4-acetyl-3-hydroxy-2-propylphenoxy)methyl]phenoxy]pyridine-3-carboxylic acid
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|
C24H23NO6
|
1
|
| 1 |
EC50 = 1431 nM
|
|
|
|
CP0002355
|
(2S)-2-aminopentanedioic acid
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|
C5H9NO4
|
4
|
| 1 |
EC50 = 1767 nM
|
|
|
| 2 |
EC50 = 1827 nM
|
|
|
| 3 |
EC50 = 2351 nM
|
|
|
| 4 |
EC50 = 2575 nM
|
|
|
|
CP0411408
|
(1R,2S,4R,5R,6R)-2-amino-4-phenylsulfanylbicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C14H15NO4S
|
5
|
| 1 |
EC50 > 12500 nM
|
|
|
| 2 |
IC50 = 7000 nM
|
|
|
| 3 |
IC50 = 7020 nM
|
|
|
| 4 |
IC50 > 12500 nM
|
|
|
| 5 |
Ki = 420 nM
|
|
|
|
CP0067673
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C15H15Cl2NO6
|
3
|
| 1 |
EC50 > 25000 nM
|
|
|
| 2 |
IC50 = 46 nM
|
|
|
| 3 |
Ki = 20.1 nM
|
|
|
|
CP0959561
|
(1R,2R,3R,4S,5R,6R)-2-Amino-3-[(4-fluoro-3-methyl-phenyl)-sulfanylmethyl]-4-(1H-1,2,4-triazol-3-ylsulfanyl)bicyclo[3.1.0]-hexane-2,6-dicarboxylic Acid Hydrochloride
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|
C18H20ClFN4O4S2
|
1
|
| 1 |
IC50 = 6.6 nM
|
|
|
|
CP0517182
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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|
C15H16Cl3NO5S
|
1
|
| 1 |
IC50 = 9.8 nM
|
|
|
|
CP0385286
|
(1R,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-(1H-1,2,4-triazol-5-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C17H16Cl2N4O5S
|
2
|
| 1 |
IC50 = 12.7 nM
|
|
|
| 2 |
Ki = 7.43 nM
|
|
|
|
CP0555781
|
(1S,2R,3R,4S,5R,6R)-2-amino-4-hydroxy-3-(phenylsulfanylmethyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
Show/Hide
|
C15H18ClNO5S
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0322575
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-difluorophenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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|
C15H16ClF2NO5S
|
1
|
| 1 |
IC50 = 16.2 nM
|
|
|
|
CP0386253
|
(1R,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-(1H-imidazol-2-ylsulfanyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C18H17Cl2N3O5S
|
1
|
| 1 |
IC50 = 16.3 nM
|
|
|
|
CP0537744
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(4-fluoro-3-methylphenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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|
C16H19ClFNO5S
|
1
|
| 1 |
IC50 = 17.2 nM
|
|
|
|
CP0386254
|
(1S,2R,3R,4S,5R,6S)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-(methoxycarbonylamino)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C17H18Cl2N2O7
|
1
|
| 1 |
IC50 = 18.8 nM
|
|
|
|
CP0445993
|
(1R,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-[(2-methyl-1,2,4-triazol-3-yl)sulfanyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
|
C18H18Cl2N4O5S
|
1
|
| 1 |
IC50 = 19.9 nM
|
|
|
|
CP0555783
|
(1S,2R,3S,4S,5R,6R)-2-amino-3-[(4-fluorophenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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|
C15H17ClFNO5S
|
1
|
| 1 |
IC50 = 20.2 nM
|
|
|
|
CP0386261
|
(1S,2R,3R,4S,5R,6S)-4-acetamido-2-amino-3-[(3,4-dichlorophenyl)methoxy]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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|
C17H18Cl2N2O6
|
1
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| 1 |
IC50 = 26.1 nM
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CP0517184
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(1S,2R,3R,4S,5R,6S)-4-acetamido-2-amino-3-[(4-fluoro-3-methylphenyl)sulfanylmethyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C18H22ClFN2O5S
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1
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| 1 |
IC50 = 26.2 nM
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CP0377729
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(1S,2S)-2-((S)-1-amino-1-carboxy-2-(9H-xanthen-9-yl)ethyl)cyclopropanecarboxylic acid
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C20H19NO5
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1
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| 1 |
IC50 = 26.7 nM
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CP0555784
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(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dimethylphenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C17H22ClNO5S
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1
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| 1 |
IC50 = 27.6 nM
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CP0475843
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(1S,2R,3R,4S,5R,6S)-2-amino-4-azido-3-[(3,4-dichlorophenyl)methoxy]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H14Cl2N4O5
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1
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| 1 |
IC50 = 34.5 nM
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CP0517180
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(1S,2R,3R,4S,5R,6S)-2,4-diamino-3-[(4-fluoro-3-methylphenyl)sulfanylmethyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C16H20ClFN2O4S
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1
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| 1 |
IC50 = 45.4 nM
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CP0517183
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(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methylsulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C16H18Cl3NO5S
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1
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| 1 |
IC50 = 49.4 nM
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CP0385282
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(1R,2R,3S,4S,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-fluorobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H14Cl2FNO5
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1
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| 1 |
IC50 = 66.9 nM
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CP0517181
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(1S,2R,3S,4S,5R,6R)-2-amino-3-[(3-fluorophenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C15H17ClFNO5S
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1
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| 1 |
IC50 = 76.2 nM
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CP0555782
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(1S,2R,3S,4S,5R,6R)-2-amino-4-hydroxy-3-(phenylsulfanylmethyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C15H18ClNO5S
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1
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| 1 |
IC50 = 114 nM
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CP0386259
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(2,3-dichlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H15Cl2NO6
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1
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| 1 |
IC50 = 149 nM
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CP0385283
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(3,4-dichlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H15Cl2NO6
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2
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| 1 |
IC50 = 169 nM
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| 2 |
Ki = 76 nM
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CP0401048
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(4-chlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H16ClNO6
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1
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| 1 |
IC50 = 210 nM
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CP0386260
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(4-fluoro-3-methylphenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C16H18FNO6
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1
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| 1 |
IC50 = 215 nM
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CP0401049
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(4-chloro-3-fluorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H15ClFNO6
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1
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| 1 |
IC50 = 225 nM
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CP0386257
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(3-chlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H16ClNO6
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1
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| 1 |
IC50 = 280 nM
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CP0432879
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(1S,2R,3S,4R,5R,6R)-2-amino-4-hydroxy-3-phenylmethoxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H17NO6
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1
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| 1 |
IC50 = 306 nM
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CP0543460
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(1S,2S,3S,5R,6S)-2-amino-3-[(3-chloro-4-fluorophenyl)methyl]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
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C15H15ClFNO4
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2
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| 1 |
IC50 = 312 nM
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| 2 |
IC50 = 408 nM
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CP0560067
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(1S,2R,3S,4R,5R,6R)-2-amino-4-hydroxy-3-(phenylsulfanylmethyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C15H18ClNO5S
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1
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| 1 |
IC50 = 335 nM
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CP0386256
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(1S,2R,3S,4R,5R,6R)-2-amino-3-[(2,5-dichlorophenyl)methoxy]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H15Cl2NO6
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1
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| 1 |
IC50 = 387 nM
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CP0386255
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(1S,2R,3R,4S,5R,6S)-2,4-diamino-3-[(3,4-dichlorophenyl)methoxy]bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C15H16Cl2N2O5
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1
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| 1 |
IC50 = 1130 nM
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CP0565872
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(1S,2R,3S,4S,5R,6R)-2-amino-3-[(2-fluorophenyl)sulfanylmethyl]-4-hydroxybicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C15H17ClFNO5S
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1
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| 1 |
IC50 = 1440 nM
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CP0562206
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(1S,2R,3R,4R,5R,6R)-2-amino-4-hydroxy-3-(phenylsulfanylmethyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid;hydrochloride
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C15H18ClNO5S
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1
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| 1 |
IC50 = 2050 nM
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CP0517185
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(1S,2R,3S,4S,5R,6R)-2-amino-4-hydroxy-3-(propan-2-ylsulfanylmethyl)bicyclo[3.1.0]hexane-2,6-dicarboxylic acid
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C12H19NO5S
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1
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| 1 |
IC50 = 2280 nM
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CP0433479
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(1S,2S,4R,5R,6S)-4-acetamido-2-aminobicyclo[3.1.0]hexane-2,6-dicarboxylic acid
Show/Hide
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C10H14N2O5
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1
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| 1 |
IC50 = 4990 nM
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