| Compound ID |
Compound Name |
Compound Formula |
|
CP0284641
|
US8957093, 75
Show/Hide
|
C38H32N2O3
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0004968
|
(2R)-2-[[6-[(2,4-dichlorophenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C21H22Cl2N2O4S3
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0521731
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-2-fluorobenzenesulfonamide
Show/Hide
|
C21H12BrCl2FN2O3S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0359362
|
2-[[6-[(2,4-dichlorophenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C21H22Cl2N2O4S3
|
1
|
| 1 |
EC50 = 2.2 nM
|
|
|
|
CP0264243
|
US8957093, 97
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 3 nM
|
|
|
|
CP0474313
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-2-(trifluoromethoxy)benzenesulfonamide
Show/Hide
|
C22H12BrCl2F3N2O4S
|
1
|
| 1 |
EC50 = 4 nM
|
|
|
|
CP0429811
|
4'-((2,3-dimethyl-5-(1-phenylpropylcarbamoyl)-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 13 nM
|
|
|
|
CP0300477
|
US8957093, 106
Show/Hide
|
C33H30N2O3
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0231789
|
US8957093, 113
Show/Hide
|
C33H29FN2O3
|
1
|
| 1 |
EC50 = 47 nM
|
|
|
|
CP0459347
|
2-[[6-[(4-chlorophenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C21H23ClN2O4S3
|
1
|
| 1 |
EC50 = 50 nM
|
|
|
|
CP0109205
|
US8957093, 98
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0368278
|
US8957093, 23
Show/Hide
|
C34H32N2O4
|
1
|
| 1 |
EC50 = 53 nM
|
|
|
|
CP0058863
|
2-[4-[[5-[[(S)-cyclopropyl-(3-propan-2-ylphenyl)methyl]carbamoyl]-2,3-dimethylindol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C38H38N2O3
|
1
|
| 1 |
EC50 = 60 nM
|
|
|
|
CP0250079
|
US8957093, 253
Show/Hide
|
C35H34N2O4
|
1
|
| 1 |
EC50 = 86 nM
|
|
|
|
CP0521730
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-2-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C22H12BrCl2F3N2O3S
|
1
|
| 1 |
EC50 = 94 nM
|
|
|
|
CP0096783
|
2-(3-chloro-4-(3-(3-ethyl-7-propylbenzo[d]isoxazol-6-yloxy)propylthio)phenyl)acetic acid
Show/Hide
|
C23H26ClNO4S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0148936
|
2-[4-[[2,3-dimethyl-5-[[(1S)-2,2,2-trifluoro-1-(3-propan-2-ylphenyl)ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C36H33F3N2O3
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0325068
|
US8957093, 198
Show/Hide
|
C37H38N2O3
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0013457
|
US10322118, Entry 1
Show/Hide
|
C14H8I4O4
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0336862
|
2-[4-[[5-[[(1S)-1-(3-chlorophenyl)ethyl]carbamoyl]-2,3-dimethylindol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C33H29ClN2O3
|
1
|
| 1 |
EC50 = 116 nM
|
|
|
|
CP0487300
|
2-[4-[[2,3-dimethyl-5-[[(1S)-1-(3-propan-2-ylphenyl)pentyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C39H42N2O3
|
1
|
| 1 |
EC50 = 116 nM
|
|
|
|
CP0548493
|
1-[(3-fluorophenyl)methyl]-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
|
C23H17F4N3O2
|
1
|
| 1 |
EC50 = 120 nM
|
|
|
|
CP0127594
|
US8957093, 13
Show/Hide
|
C36H36N2O3
|
1
|
| 1 |
EC50 = 124 nM
|
|
|
|
CP0351547
|
US8957093, 6
Show/Hide
|
C33H29BrN2O3
|
1
|
| 1 |
EC50 = 129 nM
|
|
|
|
CP0548476
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-2,5-difluorobenzenesulfonamide
Show/Hide
|
C21H11BrCl2F2N2O3S
|
1
|
| 1 |
EC50 = 131 nM
|
|
|
|
CP0170588
|
2-[4-[[2,3-dimethyl-5-[(3-propan-2-ylphenyl)methylcarbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C35H34N2O3
|
1
|
| 1 |
EC50 = 133 nM
|
|
|
|
CP0565798
|
2-[4-[[2,3-dimethyl-5-[[(1S)-2-methyl-1-(3-propan-2-ylphenyl)propyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C38H40N2O3
|
1
|
| 1 |
EC50 = 133 nM
|
|
|
|
CP0565931
|
4-bromo-2-chloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H12BrCl3N2O3S
|
1
|
| 1 |
EC50 = 134 nM
|
|
|
|
CP0127601
|
US8957093, 252
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 147 nM
|
|
|
|
CP0324477
|
US8957093, 254
Show/Hide
|
C33H29BrN2O3
|
1
|
| 1 |
EC50 = 147 nM
|
|
|
|
CP0257897
|
2-[4-[[2,3-dimethyl-5-[[(1S)-2-phenyl-1-(3-propan-2-ylphenyl)ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C42H40N2O3
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0355825
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]-2-methylindole-5-carboxamide
Show/Hide
|
C29H26F4N2O3S
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
|
CP0472394
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H13BrCl2N2O3S
|
1
|
| 1 |
EC50 = 151 nM
|
|
|
|
CP0440910
|
(2S)-2-[[6-[(2,4-dichlorophenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C21H22Cl2N2O4S3
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0565932
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-3-fluorobenzenesulfonamide
Show/Hide
|
C21H12BrCl2FN2O3S
|
1
|
| 1 |
EC50 = 169 nM
|
|
|
|
CP0158747
|
2,4-dichloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
|
C21H12Cl4N2O3S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0385101
|
US8957093, 81
Show/Hide
|
C32H34N2O3
|
1
|
| 1 |
EC50 = 179 nM
|
|
|
|
CP0474942
|
2-[4-[[2,3-dimethyl-5-[[(1S)-1-[3-(trifluoromethyl)phenyl]ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C34H29F3N2O3
|
1
|
| 1 |
EC50 = 185 nM
|
|
|
|
CP0058831
|
US8957093, 103
Show/Hide
|
C33H30N2O4
|
1
|
| 1 |
EC50 = 188 nM
|
|
|
|
CP0548464
|
1-[(3-fluorophenyl)methyl]-N-[[4-(methanesulfonamido)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
|
C25H21F4N3O3S
|
1
|
| 1 |
EC50 = 190 nM
|
|
|
|
CP0429812
|
US8957093, 83
Show/Hide
|
C30H26N2O3S
|
1
|
| 1 |
EC50 = 196 nM
|
|
|
|
CP0534068
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-(2-methylpropyl)indole-5-carboxamide
Show/Hide
|
C25H27F3N2O3S
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0542790
|
N-[[4-(cyclopropylsulfonylamino)-2-(trifluoromethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]indole-5-carboxamide
Show/Hide
|
C27H23F4N3O3S
|
1
|
| 1 |
EC50 = 220 nM
|
|
|
|
CP0058864
|
2-[4-[[2,3-dimethyl-5-[[(1S)-3-methyl-1-(3-propan-2-ylphenyl)butyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C39H42N2O3
|
1
|
| 1 |
EC50 = 226 nM
|
|
|
|
CP0440909
|
2-[[6-[(4-phenylphenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C27H28N2O4S3
|
1
|
| 1 |
EC50 = 260 nM
|
|
|
|
CP0429825
|
4'-((5-(benzylcarbamoyl)-2,3-dimethyl-1H-indol-1-yl)methyl)biphenyl-2-carboxylic acid
Show/Hide
|
C32H28N2O3
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0139102
|
2-[3-bromo-4-(4-hydroxy-3,5-diiodophenoxy)-5-iodophenyl]acetic acid
Show/Hide
|
C14H8BrI3O4
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0425602
|
US8957093, 255
Show/Hide
|
C35H34N2O3
|
1
|
| 1 |
EC50 = 334 nM
|
|
|
|
CP0576686
|
1-(cyclopropylmethyl)-N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
|
C25H25F3N2O3S
|
1
|
| 1 |
EC50 = 340 nM
|
|
|
|
CP0231207
|
2-[4-[[2,3-dimethyl-5-[[(1S)-1-(4-methylphenyl)ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C34H32N2O3
|
1
|
| 1 |
EC50 = 344 nM
|
|
|
|
CP0474943
|
2-[4-[[5-[[(1S)-1-(4-tert-butylphenyl)ethyl]carbamoyl]-2,3-dimethylindol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C37H38N2O3
|
1
|
| 1 |
EC50 = 355 nM
|
|
|
|
CP0266195
|
US8957093, 105
Show/Hide
|
C33H30N2O3
|
1
|
| 1 |
EC50 = 363 nM
|
|
|
|
CP0395305
|
2-[4-(4,4''-bis-trifluoromethyl-[1,1';3',1'']terphenyl-5'-ylmethoxy)-phenoxy]-2-methyl-propionic acid
Show/Hide
|
C31H24F6O4
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0024380
|
2-[4-(4-hydroxy-3-iodophenoxy)-3,5-diiodophenyl]acetic acid
Show/Hide
|
C14H9I3O4
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0357725
|
N-[[4-(ethylsulfonylamino)-2-(trifluoromethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]indole-5-carboxamide
Show/Hide
|
C26H23F4N3O3S
|
1
|
| 1 |
EC50 = 370 nM
|
|
|
|
CP0573180
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-ethylindole-5-carboxamide
Show/Hide
|
C23H23F3N2O3S
|
1
|
| 1 |
EC50 = 440 nM
|
|
|
|
CP0544269
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-propan-2-ylindole-5-carboxamide
Show/Hide
|
C24H25F3N2O3S
|
1
|
| 1 |
EC50 = 490 nM
|
|
|
|
CP0456883
|
2-[4-[[5-[[(1S)-1-(3-tert-butylphenyl)ethyl]carbamoyl]-2,3-dimethylindol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C37H38N2O3
|
1
|
| 1 |
EC50 = 499 nM
|
|
|
|
CP0328412
|
US8957093, 72
Show/Hide
|
C33H29N3O5
|
1
|
| 1 |
EC50 = 503 nM
|
|
|
|
CP0127592
|
US8957093, 12
Show/Hide
|
C32H27BrN2O3
|
1
|
| 1 |
EC50 = 516 nM
|
|
|
|
CP0429827
|
US8957093, 1
Show/Hide
|
C33H29BrN2O3
|
1
|
| 1 |
EC50 = 516 nM
|
|
|
|
CP0273832
|
1-benzyl-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
|
C23H18F3N3O2
|
1
|
| 1 |
EC50 = 540 nM
|
|
|
|
CP0073193
|
(2S)-2-ETHOXY-3-{4-[2-(10H-PHENOXAZIN-10-YL)ETHOXY]PHENYL}PROPANOIC ACID
Show/Hide
|
C25H25NO5
|
1
|
| 1 |
EC50 = 570 nM
|
|
|
|
CP0373977
|
2-(4-((4-(4-(N-Isopropyl-N-methyl)benzamide)-5-(4-(trifluoromethoxy)phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C31H29F3N2O7
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0461713
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-3-methylbenzenesulfonamide
Show/Hide
|
C22H15BrCl2N2O3S
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0549554
|
2-methyl-2-[4-[2-[4-phenyldiazenyl-2-(trifluoromethyl)phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
|
C25H23F3N2O4
|
1
|
| 1 |
EC50 = 600 nM
|
|
|
|
CP0573215
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-2-methyl-1-propan-2-ylsulfonylindole-5-carboxamide
Show/Hide
|
C25H27F3N2O5S2
|
1
|
| 1 |
EC50 = 630 nM
|
|
|
|
CP0045084
|
US8957093, 107
Show/Hide
|
C33H30N2O3
|
1
|
| 1 |
EC50 = 632 nM
|
|
|
|
CP0100041
|
US8957093, 112
Show/Hide
|
C33H29FN2O3
|
1
|
| 1 |
EC50 = 638 nM
|
|
|
|
CP0534067
|
1-(3-fluorophenyl)sulfonyl-N-[[4-(methylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
|
C25H20F4N2O5S2
|
1
|
| 1 |
EC50 = 660 nM
|
|
|
|
CP0459344
|
2-[[6-[(4-tert-butylphenyl)sulfonylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C25H32N2O4S3
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0357719
|
1-(cyclohexylmethyl)-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
|
C23H24F3N3O2
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0407205
|
2-[4-[(3,5-diphenylphenyl)methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H24O4
|
1
|
| 1 |
EC50 = 740 nM
|
|
|
|
CP0438503
|
2-[[6-[(4-phenylphenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C28H30N2O2S2
|
1
|
| 1 |
EC50 = 770 nM
|
|
|
|
CP0549559
|
2-methyl-2-[4-[2-[4-phenyldiazenyl-2-(trifluoromethyl)phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
|
C25H23F3N2O4
|
1
|
| 1 |
EC50 = 770 nM
|
|
|
|
CP0000254
|
(Z)-2-(3-(4-(methylthio)benzylidene)-6-fluoro-2-methyl-3H-inden-1-yl)acetic acid
Show/Hide
|
C20H17FO2S
|
1
|
| 1 |
EC50 = 800 nM
|
|
|
|
CP0496449
|
2-[4-[2-(2-chloro-4-phenyldiazenylphenoxy)ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C24H23ClN2O4
|
1
|
| 1 |
EC50 = 820 nM
|
|
|
|
CP0357727
|
N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-[3,3,3-trifluoro-2-(trifluoromethyl)propyl]indole-5-carboxamide
Show/Hide
|
C25H21F9N2O3S
|
1
|
| 1 |
EC50 = 820 nM
|
|
|
|
CP0227236
|
US8957093, 110
Show/Hide
|
C32H27N3O5
|
1
|
| 1 |
EC50 = 822 nM
|
|
|
|
CP0127347
|
US8957093, 119
Show/Hide
|
C32H27N3O5
|
1
|
| 1 |
EC50 = 831 nM
|
|
|
|
CP0534066
|
1-[(3-fluorophenyl)methyl]-N-[[4-methoxy-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
|
C25H20F4N2O2
|
1
|
| 1 |
EC50 = 850 nM
|
|
|
|
CP0235717
|
2-[4-[[2,3-dimethyl-5-[[(1S)-1-(3-propan-2-ylphenyl)ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
|
C36H36N2O3
|
1
|
| 1 |
EC50 = 852 nM
|
|
|
|
CP0549555
|
2-[4-[2-(2-chloro-4-phenyldiazenylphenoxy)ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C24H23ClN2O4
|
1
|
| 1 |
EC50 = 920 nM
|
|
|
|
CP0553524
|
Sulindac analogue, 11
Show/Hide
|
C26H21FO3
|
2
|
| 1 |
EC50 = 930 nM
|
|
|
| 2 |
Kd = 960 nM
|
|
|
|
CP0474315
|
4-bromo-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-3-(trifluoromethyl)benzenesulfonamide
Show/Hide
|
C22H12BrCl2F3N2O3S
|
1
|
| 1 |
EC50 = 957 nM
|
|
|
|
CP0373720
|
2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H24F3N3O7
|
1
|
| 1 |
EC50 = 980 nM
|
|
|
|
CP0479953
|
(2S)-2-(2-benzoylanilino)-3-(4-phenyldiazenylphenyl)propanoic acid
Show/Hide
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C28H23N3O3
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1
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| 1 |
EC50 = 1000 nM
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CP0578041
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1-[(3,4-dichlorophenyl)methyl]-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
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C23H16Cl2F3N3O2
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1
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| 1 |
EC50 = 1000 nM
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CP0577975
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1-benzyl-N-[[4-methoxy-2-(trifluoromethyl)phenyl]methyl]-2-oxo-3H-benzimidazole-5-carboxamide
Show/Hide
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C24H20F3N3O3
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1
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| 1 |
EC50 = 1010 nM
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CP0535047
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-(3-fluorophenyl)sulfonylindole-5-carboxamide
Show/Hide
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C27H22F4N2O5S2
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1
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| 1 |
EC50 = 1020 nM
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CP0384227
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2-(4-((4-(2-Morpholinopyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C28H25F3N4O7
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1
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| 1 |
EC50 = 1030 nM
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CP0528254
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-propan-2-ylsulfonylindole-5-carboxamide
Show/Hide
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C24H25F3N2O5S2
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1
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| 1 |
EC50 = 1050 nM
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CP0535045
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1-[(3-fluorophenyl)methyl]-N-[[4-methoxy-2-(trifluoromethyl)phenyl]methyl]-2-oxo-3H-benzimidazole-5-carboxamide
Show/Hide
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C24H19F4N3O3
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1
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| 1 |
EC50 = 1090 nM
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CP0548463
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1-[(3-fluorophenyl)methyl]-N-[[4-methoxy-2-(trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxamide
Show/Hide
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C24H19F4N3O2
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1
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| 1 |
EC50 = 1120 nM
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CP0109245
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2-[4-[[2,3-dimethyl-5-[[(1S)-1-(4-propan-2-ylphenyl)ethyl]carbamoyl]indol-1-yl]methyl]phenyl]benzoic acid
Show/Hide
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C36H36N2O3
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1
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| 1 |
EC50 = 1141 nM
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CP0549816
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-methylindole-5-carboxamide
Show/Hide
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C22H21F3N2O3S
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1
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| 1 |
EC50 = 1160 nM
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CP0485288
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2-[(3Z)-6-fluoro-2-methyl-3-[(3-phenoxyphenyl)methylidene]inden-1-yl]acetic acid
Show/Hide
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C25H19FO3
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2
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| 1 |
EC50 = 1178 nM
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| 2 |
Kd = 1730 nM
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CP0442513
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2-[4-[(3,5-diphenylphenyl)methoxy]phenoxy]acetic acid
Show/Hide
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C27H22O4
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1
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| 1 |
EC50 = 1200 nM
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CP0373958
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2-(4-((4-(4-(N-Isopropyl-N-methyl)benzamide)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C31H29F3N2O6S
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1
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| 1 |
EC50 = 1200 nM
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CP0496450
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2-methyl-2-[4-[2-(2-methyl-4-phenyldiazenylphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
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C25H26N2O4
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1
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| 1 |
EC50 = 1200 nM
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CP0549556
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2-methyl-2-[4-[2-[2-methyl-4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C26H28N2O4
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1
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| 1 |
EC50 = 1200 nM
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CP0568733
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2-methyl-2-[4-[2-[4-[(4-methylphenyl)diazenyl]-2-(trifluoromethyl)phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C26H25F3N2O4
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1
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| 1 |
EC50 = 1200 nM
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CP0479955
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(2S)-2-(2-benzoylanilino)-3-(4-phenyldiazenylphenyl)propanoic acid
Show/Hide
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C28H23N3O3
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1
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| 1 |
EC50 = 1300 nM
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CP0496448
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2-methyl-2-[4-[2-[4-[(4-methylphenyl)diazenyl]-2-(trifluoromethyl)phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C26H25F3N2O4
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1
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| 1 |
EC50 = 1300 nM
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CP0381222
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2-Ethoxy-3-(4-(5-(4-(trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxyphenyl)propanoic Acid
Show/Hide
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C29H26F3NO5S
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1
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| 1 |
EC50 = 1310 nM
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CP0535046
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1-[(3-fluorophenyl)methyl]-N-[[4-[(2,2,2-trifluoroacetyl)amino]-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C26H18F7N3O2
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1
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| 1 |
EC50 = 1310 nM
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CP0273836
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1-[1-(3-fluorophenyl)ethyl]-N-[[4-(methylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C27H24F4N2O3S
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1
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| 1 |
EC50 = 1340 nM
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CP0170639
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US8957093, 96
Show/Hide
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C32H27N3O5
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1
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| 1 |
EC50 = 1344 nM
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CP0576685
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1-[(3-fluorophenyl)methyl]-N-[[4-(methylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C26H22F4N2O3S
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1
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| 1 |
EC50 = 1350 nM
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CP0551249
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1-(3-fluorobenzoyl)-N-[[4-(methylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C26H20F4N2O4S
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1
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| 1 |
EC50 = 1360 nM
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CP0534065
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1-[(3-fluorophenyl)methyl]-N-[[2-(trifluoromethyl)phenyl]methyl]benzimidazole-5-carboxamide
Show/Hide
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C23H17F4N3O
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1
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| 1 |
EC50 = 1410 nM
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CP0357726
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1-[(3-fluorophenyl)methyl]-N-[[4-(methylsulfanylmethyl)-2-(trifluoromethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C26H22F4N2OS
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1
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| 1 |
EC50 = 1430 nM
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CP0544266
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1H-indole-5-carboxamide
Show/Hide
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C21H19F3N2O3S
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1
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| 1 |
EC50 = 1480 nM
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CP0438505
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2-[[6-[(3-chlorophenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C22H25ClN2O2S2
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1
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| 1 |
EC50 = 1500 nM
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CP0400446
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2-(4-((4-(4-((Piperidin-1-yl)methanone)phenyl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C32H29F3N2O6S
|
1
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| 1 |
EC50 = 1560 nM
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CP0495437
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1-[(3-fluorophenyl)methyl]-N-[[4-methoxy-2-(trifluoromethyl)phenyl]methyl]indazole-5-carboxamide
Show/Hide
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C24H19F4N3O2
|
1
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| 1 |
EC50 = 1590 nM
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CP0479954
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(2S)-2-(2-benzoylanilino)-3-[4-[(4-chlorophenyl)diazenyl]phenyl]propanoic acid
Show/Hide
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C28H22ClN3O3
|
1
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| 1 |
EC50 = 1600 nM
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CP0567292
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1-[(3-fluorophenyl)methyl]-N-[[2-(trifluoromethyl)phenyl]methyl]indazole-5-carboxamide
Show/Hide
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C23H17F4N3O
|
1
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| 1 |
EC50 = 1600 nM
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CP0548496
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N-[[2-fluoro-4-(methylsulfonylmethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]indole-5-carboxamide
Show/Hide
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C25H22F2N2O3S
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1
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| 1 |
EC50 = 1620 nM
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CP0561931
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N-[[4-amino-2-(trifluoromethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]indole-5-carboxamide
Show/Hide
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C24H19F4N3O
|
1
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| 1 |
EC50 = 1680 nM
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CP0459348
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2-[[6-(benzylamino)-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C22H26N2O2S2
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1
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| 1 |
EC50 = 1700 nM
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CP0496444
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2-methyl-2-[4-[2-(2-methyl-4-phenyldiazenylphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
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C25H26N2O4
|
1
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| 1 |
EC50 = 1700 nM
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CP0485340
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2-[(3Z)-3-[(3-chlorophenyl)methylidene]-6-fluoro-2-methylinden-1-yl]acetic acid
Show/Hide
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C19H14ClFO2
|
2
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| 1 |
EC50 = 1740 nM
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| 2 |
Kd = 1220 nM
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CP0438502
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2-[[6-[[4-(trifluoromethyl)phenyl]methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C23H25F3N2O2S2
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1
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| 1 |
EC50 = 1800 nM
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CP0487235
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2-[(3Z)-6-fluoro-3-[(3-fluorophenyl)methylidene]-2-methylinden-1-yl]acetic acid
Show/Hide
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C19H14F2O2
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2
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| 1 |
EC50 = 1840 nM
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| 2 |
Kd = 1800 nM
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CP0357720
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1-[(3,5-difluorophenyl)methyl]-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
|
C23H16F5N3O2
|
1
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| 1 |
EC50 = 1960 nM
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CP0227223
|
US8957093, 19
Show/Hide
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C34H32N2O4
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1
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| 1 |
EC50 = 2076 nM
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CP0496510
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2-methyl-2-[4-[2-[4-[(4-propan-2-ylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C27H30N2O4
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1
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| 1 |
EC50 = 2100 nM
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CP0573179
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N-[[2-chloro-4-(methylsulfonylmethyl)phenyl]methyl]-1-[(3-fluorophenyl)methyl]indole-5-carboxamide
Show/Hide
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C25H22ClFN2O3S
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1
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| 1 |
EC50 = 2140 nM
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CP0561932
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N-[[4-(methylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1H-indole-5-carboxamide
Show/Hide
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C19H17F3N2O3S
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1
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| 1 |
EC50 = 2190 nM
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CP0492310
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5-[(4-phenyldiazenylphenyl)methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C16H13N3O2S
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1
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| 1 |
EC50 = 2200 nM
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CP0547691
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5-[[4-[[4-(trifluoromethyl)phenyl]diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C17H12F3N3O2S
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1
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| 1 |
EC50 = 2200 nM
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CP0391209
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2-(3-(4,5-bis(4-methoxyphenyl)thiazol-2-ylthio)phenyl)propanoic acid
Show/Hide
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C26H23NO4S2
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1
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| 1 |
EC50 = 2300 nM
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CP0572661
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2-methyl-2-[4-[2-[2-methyl-4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
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C26H28N2O4
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1
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| 1 |
EC50 = 2300 nM
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CP0520395
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2-[[6-[(4-chlorophenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C22H25ClN2O2S2
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1
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| 1 |
EC50 = 2400 nM
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CP0373728
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2-(4-((4-(6-Morpholinopyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H26F3N3O7
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1
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| 1 |
EC50 = 2490 nM
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CP0404425
|
US8957093, 94
Show/Hide
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C32H29N3O3
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1
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| 1 |
EC50 = 2532 nM
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CP0373710
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2-(4-(4-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)butoxy)-3-chlorophenyl)acetic Acid
Show/Hide
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C29H28ClNO6S2
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1
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| 1 |
EC50 = 2560 nM
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CP0496446
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2-methyl-2-[4-[2-[4-[(4-propan-2-ylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
Show/Hide
|
C27H30N2O4
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1
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| 1 |
EC50 = 2600 nM
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CP0470919
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2-methyl-2-[4-[2-(4-phenyldiazenylphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
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C24H24N2O4
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1
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| 1 |
EC50 = 2670 nM
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CP0317939
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2-[(3Z)-3-benzylidene-6-fluoro-2-methylinden-1-yl]acetic acid
Show/Hide
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C19H15FO2
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2
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| 1 |
EC50 = 2780 nM
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| 2 |
Kd = 7940 nM
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CP0438504
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2-[[6-[(3,4-dichlorophenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
|
C22H24Cl2N2O2S2
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1
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| 1 |
EC50 = 2800 nM
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CP0448032
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5-[[4-[[4-(2-methylphenyl)phenyl]diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C23H19N3O2S
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1
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| 1 |
EC50 = 2800 nM
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CP0440908
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2-[[6-[(3,5-dichlorophenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C22H24Cl2N2O2S2
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1
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| 1 |
EC50 = 2900 nM
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CP0486825
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5-[[4-[(4-chlorophenyl)diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C16H12ClN3O2S
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1
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| 1 |
EC50 = 2900 nM
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CP0518732
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2-[[6-(naphthalen-2-ylmethylamino)-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C26H28N2O2S2
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1
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| 1 |
EC50 = 3000 nM
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CP0470920
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2-[4-[2-[4-[(4-chlorophenyl)diazenyl]phenoxy]ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C24H23ClN2O4
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1
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| 1 |
EC50 = 3200 nM
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CP0573181
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-(oxetan-3-ylmethyl)indole-5-carboxamide
Show/Hide
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C25H25F3N2O4S
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1
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| 1 |
EC50 = 3200 nM
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CP0548475
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N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)-2,4,6-trimethylbenzenesulfonamide
Show/Hide
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C24H20Cl2N2O3S
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1
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| 1 |
EC50 = 3314 nM
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CP0548462
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1-[(2-chlorophenyl)methyl]-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
|
C23H17ClF3N3O2
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1
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| 1 |
EC50 = 3330 nM
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CP0559357
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1-[(3-fluorophenyl)methyl]-N-[[4-(methylsulfonylmethyl)phenyl]methyl]indole-5-carboxamide
Show/Hide
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C25H23FN2O3S
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1
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| 1 |
EC50 = 3540 nM
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CP0459343
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2-[[6-[(4-tert-butylphenyl)methylamino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C26H34N2O2S2
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1
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| 1 |
EC50 = 3700 nM
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CP0459350
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2-[[6-[(4-tert-butylbenzoyl)amino]-1,3-benzothiazol-2-yl]sulfanyl]hexanoic acid
Show/Hide
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C24H28N2O3S2
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1
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| 1 |
EC50 = 3700 nM
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CP0534064
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2-oxo-N,1-bis[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
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C24H17F6N3O2
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1
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| 1 |
EC50 = 3700 nM
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CP0077898
|
CHEBI:11684
Show/Hide
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C15H12I3NO4
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1
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| 1 |
EC50 = 3800 nM
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CP0261047
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1-[(3-chlorophenyl)methyl]-2-oxo-N-[[2-(trifluoromethyl)phenyl]methyl]-3H-benzimidazole-5-carboxamide
Show/Hide
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C23H17ClF3N3O2
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1
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| 1 |
EC50 = 4100 nM
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CP0252490
|
US8957093, 73
Show/Hide
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C33H29N3O5
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1
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| 1 |
EC50 = 4288 nM
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CP0548477
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N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)naphthalene-2-sulfonamide
Show/Hide
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C25H16Cl2N2O3S
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1
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| 1 |
EC50 = 4289 nM
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CP0438501
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2-[[6-[(4-tert-butylbenzoyl)amino]-1,3-benzothiazol-2-yl]sulfanyl]octanoic acid
Show/Hide
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C26H32N2O3S2
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1
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| 1 |
EC50 = 4300 nM
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CP0551259
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N-[[4-(cyclopropylsulfonylmethyl)-2-(trifluoromethyl)phenyl]methyl]-1-(2-methoxyethyl)indole-5-carboxamide
Show/Hide
|
C24H25F3N2O4S
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1
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| 1 |
EC50 = 4300 nM
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CP0231206
|
US8957093, 297
Show/Hide
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C36H34N2O3
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1
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| 1 |
EC50 = 4391 nM
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CP0549557
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2-[4-[2-[2-chloro-4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H25ClN2O4
|
1
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| 1 |
EC50 = 4500 nM
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CP0430580
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2-(4-(3-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)propoxy)-3-chlorophenyl)acetic Acid
Show/Hide
|
C28H26ClNO6S2
|
1
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| 1 |
EC50 = 4610 nM
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CP0511832
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2-[(3Z)-3-[(3-bromophenyl)methylidene]-6-fluoro-2-methylinden-1-yl]acetic acid
Show/Hide
|
C19H14BrFO2
|
2
|
| 1 |
EC50 = 4610 nM
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| 2 |
Kd = 1710 nM
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CP0496443
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2-[4-[2-[2-chloro-4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
|
C25H25ClN2O4
|
1
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| 1 |
EC50 = 4800 nM
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CP0520397
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2-[(6-benzamido-1,3-benzothiazol-2-yl)sulfanyl]octanoic acid
Show/Hide
|
C22H24N2O3S2
|
1
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| 1 |
EC50 = 4900 nM
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CP0415933
|
2-[(2E)-3,7-dimethylocta-2,6-dienyl]-3-hydroxy-5-pentylcyclohexa-2,5-diene-1,4-dione
Show/Hide
|
C21H30O3
|
1
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| 1 |
EC50 = 4900 nM
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CP0366392
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US8957093, 257
Show/Hide
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C36H36N2O4
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1
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| 1 |
EC50 = 4907 nM
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CP0547692
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(2S)-2-(2-benzoylanilino)-3-[4-[(4-chlorophenyl)diazenyl]phenyl]propanoic acid
Show/Hide
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C28H22ClN3O3
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1
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| 1 |
EC50 = 5000 nM
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CP0545725
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2-[(3E)-6-fluoro-2-methyl-3-[(3-methylphenyl)methylidene]inden-1-yl]acetic acid
Show/Hide
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C20H17FO2
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2
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| 1 |
EC50 = 5250 nM
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| 2 |
Kd = 21570 nM
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CP0077320
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2-[(3Z)-6-fluoro-3-[(3-methoxyphenyl)methylidene]-2-methylinden-1-yl]acetic acid
Show/Hide
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C20H17FO3
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2
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| 1 |
EC50 = 5300 nM
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| 2 |
Kd = 2460 nM
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CP0488451
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2-methyl-2-[4-[(4-phenyldiazenylphenoxy)methyl]phenoxy]propanoic acid
Show/Hide
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C23H22N2O4
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1
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| 1 |
EC50 = 5400 nM
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CP0406483
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(4-{2-[4,5-Bis(4-methoxyphenyl)thiazol-2-ylsulfanyl]ethoxy}-2-methylphenoxy)acetic Acid
Show/Hide
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C28H27NO6S2
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1
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| 1 |
EC50 = 5660 nM
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CP0381070
|
US8957093, 89
Show/Hide
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C29H28N2O3
|
1
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| 1 |
EC50 = 5665 nM
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CP0026502
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(2R)-2-amino-3-[4-(4-hydroxy-3-iodophenoxy)-3,5-diiodophenyl]propanoic acid
Show/Hide
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C15H12I3NO4
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1
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| 1 |
EC50 = 5800 nM
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CP0474314
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2-chloro-N-(3,5-dichloro-4-quinolin-3-yloxyphenyl)benzenesulfonamide
Show/Hide
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C21H13Cl3N2O3S
|
1
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| 1 |
EC50 = 5810 nM
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CP0411105
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2-(4-(2-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)ethoxy)-3-chlorophenyl)acetic Acid
Show/Hide
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C27H24ClNO6S2
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1
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| 1 |
EC50 = 5870 nM
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CP0496442
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2-methyl-2-[4-[2-(4-phenyldiazenylphenoxy)ethyl]phenoxy]propanoic acid
Show/Hide
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C24H24N2O4
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1
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| 1 |
EC50 = 6000 nM
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CP0548322
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2-[(3Z)-6-fluoro-3-[(3-hydroxyphenyl)methylidene]-2-methylinden-1-yl]acetic acid
Show/Hide
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C19H15FO3
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2
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| 1 |
EC50 = 6290 nM
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| 2 |
Kd = 5520 nM
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CP0484980
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5-[(4-phenyldiazenylphenyl)methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C16H13N3O2S
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1
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| 1 |
EC50 = 6300 nM
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CP0402047
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2-(4-(4-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)butoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C30H31NO6S2
|
1
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| 1 |
EC50 = 6360 nM
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CP0551803
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5-[[4-[[4-(2-methylphenyl)phenyl]diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C23H19N3O2S
|
1
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| 1 |
EC50 = 6400 nM
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CP0527505
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2-[(3Z)-6-fluoro-2-methyl-3-[(3-propan-2-ylphenyl)methylidene]inden-1-yl]acetic acid
Show/Hide
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C22H21FO2
|
2
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| 1 |
EC50 = 6410 nM
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|
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| 2 |
Kd = 2470 nM
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CP0479956
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5-[[4-[[4-(trifluoromethyl)phenyl]diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
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C17H12F3N3O2S
|
1
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| 1 |
EC50 = 6500 nM
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CP0569284
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2-methyl-2-[4-[(4-phenyldiazenylphenoxy)methyl]phenoxy]propanoic acid
Show/Hide
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C23H22N2O4
|
1
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| 1 |
EC50 = 6600 nM
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CP0391207
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2-(4-(3-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)propoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H29NO6S2
|
1
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| 1 |
EC50 = 6890 nM
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|
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CP0538427
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5-[[4-[(4-chlorophenyl)diazenyl]phenyl]methyl]-1,3-thiazolidine-2,4-dione
Show/Hide
|
C16H12ClN3O2S
|
1
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| 1 |
EC50 = 7000 nM
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|
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CP0374830
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2-[2-methyl-4-[[3-(4-phenylphenyl)-5-[4-(trifluoromethyl)phenyl]phenyl]methoxy]phenoxy]acetic acid
Show/Hide
|
C35H27F3O4
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0374831
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2-[4-[[3,5-bis[4-(dimethylamino)phenyl]phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C32H34N2O4
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0374832
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2-[4-[[3,4-bis[4-(trifluoromethoxy)phenyl]phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C30H22F6O6
|
1
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| 1 |
EC50 > 10000 nM
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CP0374833
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2-[4-[[3-(4-methoxyphenyl)-5-[4-(trifluoromethyl)phenyl]phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C30H25F3O5
|
1
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| 1 |
EC50 > 10000 nM
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CP0374834
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2-[4-[[2,6-bis(4-methoxyphenyl)pyrimidin-4-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C28H26N2O6
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0374836
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2-[2-methyl-4-[[3-[4-(trifluoromethoxy)phenyl]-5-[4-(trifluoromethyl)phenyl]phenyl]methoxy]phenoxy]acetic acid
Show/Hide
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C30H22F6O5
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0374837
|
2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methoxy]-3-chlorophenyl]acetic acid
Show/Hide
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C29H19ClF6O3
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0377033
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2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C30H22F6O4
|
1
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| 1 |
EC50 > 10000 nM
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CP0378780
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2-[4-[[5,6-bis[4-(trifluoromethyl)phenyl]pyridin-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C29H21F6NO4
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0378782
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2-[4-[[4,6-bis(4-methoxyphenyl)pyrimidin-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H26N2O6
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0378783
|
2-[4-[[3,4-bis(4-methoxyphenyl)phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C30H28O6
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0378784
|
2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methylsulfanyl]-3-chlorophenyl]acetic acid
Show/Hide
|
C29H19ClF6O2S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0395304
|
2-[4-[[2,6-bis[4-(trifluoromethoxy)phenyl]pyrimidin-4-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H20F6N2O6
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0395306
|
2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methoxy]-3-methylphenoxy]acetic acid
Show/Hide
|
C30H22F6O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0407206
|
2-[4-[[2,6-bis[4-(trifluoromethyl)phenyl]pyrimidin-4-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H20F6N2O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0407207
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2-[4-[[4,6-bis[4-(trifluoromethoxy)phenyl]pyrimidin-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H20F6N2O6
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0407209
|
2-[4-[[3,5-bis[4-(trifluoromethoxy)phenyl]phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C30H22F6O6
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0433449
|
2-[4-[[3,5-bis(4-methoxyphenyl)phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C30H28O6
|
1
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| 1 |
EC50 > 10000 nM
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CP0433450
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2-[2-methyl-4-[[3-(4-methylphenyl)-5-[4-(trifluoromethyl)phenyl]phenyl]methoxy]phenoxy]acetic acid
Show/Hide
|
C30H25F3O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0433451
|
2-[4-[[3,5-bis(4-chlorophenyl)phenyl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C28H22Cl2O4
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0446019
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2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methoxy]phenoxy]acetic acid
Show/Hide
|
C29H20F6O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0446020
|
2-[4-[[3,5-bis[4-(trifluoromethyl)phenyl]phenyl]methylsulfanyl]-2-methylphenoxy]acetic acid
Show/Hide
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C30H22F6O3S
|
1
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| 1 |
EC50 > 10000 nM
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CP0449790
|
2-[4-[[4,6-bis[4-(trifluoromethyl)phenyl]pyrimidin-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C28H20F6N2O4
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0453735
|
2-[2-methyl-4-[[3-[3-(trifluoromethyl)phenyl]-5-[4-(trifluoromethyl)phenyl]phenyl]methoxy]phenoxy]acetic acid
Show/Hide
|
C30H22F6O4
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0043946
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2-[2-methyl-4-[[4-(4-propan-2-yloxyphenyl)-5-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]methoxy]phenoxy]acetic acid
Show/Hide
|
C29H26F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0043958
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2-(4-((4-(6-Methoxypyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C26H21F3N2O7
|
1
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| 1 |
EC50 > 10000 nM
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CP0221664
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2-(4-((4-(6-Isopropoxypyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C28H25F3N2O6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0244563
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2-(4-((4-(2-Isopropoxypyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H24F3N3O6S
|
1
|
| 1 |
EC50 > 10000 nM
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CP0244640
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2-[4-[[4-(6-methoxypyridin-3-yl)-5-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C26H21F3N2O6S
|
1
|
| 1 |
EC50 > 10000 nM
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CP0254301
|
2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C31H28F3NO6S
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0287050
|
2-(4-((4-(4-(Cyclopentyloxy)phenyl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C31H28F3NO7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0345351
|
2-(4-((4-(4-Isopropoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H26F3NO7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373747
|
2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C25H20F3N3O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373793
|
2-(5-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-1H-indol-1-yl)acetic Acid
Show/Hide
|
C28H21F3N2O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373795
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-3-chlorophenyl)acetic Acid
Show/Hide
|
C26H19ClF3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373843
|
2-(4-((4-(3-Methoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373952
|
2-(4-((4-(4-(N,N-Dimethyl)benzamide)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H25F3N2O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373953
|
2-(4-((4-(4-(Diethylamino)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H29F3N2O5S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0373954
|
2-(4-((4-(4-(Piperidin-1-yl)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C31H29F3N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373955
|
2-(4-((4-(4-Isobutoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H28F3NO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373956
|
2-(4-((4-(4-(Pyrrolidin-1-yl)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H27F3N2O5S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0373957
|
2-(4-((4-(6-Benzo[d]oxazol-2(3H)-one)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H19F3N2O7S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0373961
|
2-(4-((4-(2,3-Dihydrobenzo[b][1,4]dioxin-6-yl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C28H22F3NO7S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373962
|
2-(4-((4-(4-(Trifluoromethyl)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H19F6NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373964
|
2-(4-((4-(Benzo[d][1,3]dioxol-5-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H20F3NO7S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373970
|
2-(4-((5-(6-Chloropyridin-3-yl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C25H21ClN2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373971
|
2-(4-((4-(4-Methoxyphenyl)-5-(4-propylphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H29NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373973
|
2-(4-((4-(4-Methoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373974
|
2-(4-((4-(4-Methoxyphenyl)-5-(naphthalen-3-yl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H25NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0373975
|
2-(4-((4-(4-Methoxyphenyl)-5-(4-(trifluoromethylthio)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374025
|
2-(4-((4-(2-Methoxypyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C25H20F3N3O7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374026
|
2-(4-((4-(Pyridin-3-yl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C25H19F3N2O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374033
|
2-(1-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)naphthalen-4-yloxy)acetic Acid
Show/Hide
|
C30H22F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374035
|
2-[4-[[4-(4-methoxyphenyl)-5-[4-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]methoxy]-2-propylphenoxy]acetic acid
Show/Hide
|
C29H26F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374036
|
3-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-(trifluoromethyl)phenyl)propanoic Acid
Show/Hide
|
C28H21F6NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374037
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenyl)acetic Acid
Show/Hide
|
C27H22F3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0374038
|
3-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenyl)propanoic Acid
Show/Hide
|
C28H24F3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0375799
|
2-(4-((4-(4-(Piperidin-1-yl)phenyl)-5-(4-(trifluoromethoxy)-phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C32H29F3N2O7
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0381224
|
2-(3-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)phenoxy)acetic Acid
Show/Hide
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C26H20F3NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0381225
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5-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)benzofuran-2-carboxylic Acid
Show/Hide
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C27H18F3NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0382779
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2-(4-((4-(3,4-Dihydro-2H-benzo[b][1,4]dioxepin-8-yl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C29H24F3NO7S
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1
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| 1 |
EC50 > 10000 nM
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CP0382782
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2-(4-((4-(4-Ethoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C28H24F3NO6S
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1
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| 1 |
EC50 > 10000 nM
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CP0382787
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2-(4-((5-(4-methoxyphenyl)-4-phenylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C26H23NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0384129
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2-[4-[[4,5-bis(4-methoxyphenyl)-1,3-thiazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C27H25NO6S
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1
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| 1 |
EC50 > 10000 nM
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CP0384228
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2-(2-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)naphthalen-5-yl)acetic Acid
Show/Hide
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C30H22F3NO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384231
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2-(4-((4-(2-Morpholinopyrimidin-5-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C28H25F3N4O6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384232
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2-(4-((4-(Pyrimidin-5-yl)-5-(4-(trifluoromethoxy)phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C24H18F3N3O6
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1
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| 1 |
EC50 > 10000 nM
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CP0384306
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2-(4-((5-(4-chlorophenyl)-4-methylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C20H18ClNO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384307
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2-(4-((5-(4-chlorophenyl)-4-phenylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C25H20ClNO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384308
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2-(4-((4-(4-chlorophenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C19H16ClNO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384309
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2-(4-((4-(4-methoxyphenyl)-5-phenylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C26H23NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0384310
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2-(4-((5-(4-methoxyphenyl)-4-methylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C21H21NO5S
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1
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| 1 |
EC50 > 10000 nM
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CP0384312
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2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C27H22F3NO6
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1
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| 1 |
EC50 > 10000 nM
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CP0384313
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2-[4-[[4-(4-methoxyphenyl)-5-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
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C27H22F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384314
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2-(4-((5-(4-Chlorophenyl)-4-(4-methoxyphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C26H22ClNO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384315
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2-(4-((4-(4-Methoxyphenyl)-5-styrylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C28H25NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384316
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2-(4-((5-(4-tert-Butylphenyl)-4-(4-methoxyphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C30H31NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384336
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2-(4-((4,5-bis(4-chlorophenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C25H19Cl2NO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384337
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2-(4-((4-(4-methoxyphenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C20H19NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384338
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2-(4-((4-(4-chlorophenyl)-5-phenylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C25H20ClNO4S
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1
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| 1 |
EC50 > 10000 nM
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CP0384342
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2-(2-methyl-4-((4-methyl-5-p-tolylthiazol-2-yl)methoxy)phenoxy)acetic acid
Show/Hide
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C21H21NO4S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384364
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2-(4-((4-(4-Propoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C29H26F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0384368
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2-(4-((4-(4-Biphenyl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C32H24F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0384444
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5-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)-2,3-dihydrobenzofuran-2-carboxylic Acid
Show/Hide
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C27H20F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0390053
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2-(4-((4,5-Bis(4-methoxyphenyl)oxazol-2-yl)methylthio)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H25NO6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0400397
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2-(2-methyl-4-((4-(pyridin-3-yl)-5-p-tolylthiazol-2-yl)methoxy)phenoxy)acetic acid
Show/Hide
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C25H22N2O4S
|
1
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| 1 |
EC50 > 10000 nM
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CP0400404
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2-(4-((4,5-diphenylthiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C25H21NO4S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0400408
|
2-(4-((4-(4-Methoxyphenyl)-5-(quinolin-3-yl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C29H24N2O5S
|
1
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| 1 |
EC50 > 10000 nM
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CP0400419
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2-(4-((5-(4-Chlorophenyl)-4-(4-methoxyphenyl)oxazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C26H22ClNO6
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0400421
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C27H22F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0400436
|
2-[4-[[4-(4-methoxyphenyl)-5-(4-phenylphenyl)-1,3-oxazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C32H27NO6
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0402025
|
2-(4-(3-(4-bromophenyl)-5-(4-(trifluoromethyl)phenyl)pent-2-en-4-ynyloxy)-2-methylphenoxy)acetic acid
Show/Hide
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C27H20BrF3O4
|
1
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| 1 |
EC50 > 10000 nM
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CP0402048
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2-(4-((4,5-Bis(4-methoxyphenyl)thiazol-2-yl)methylthio)-3-chlorophenyl)acetic Acid
Show/Hide
|
C26H22ClNO5S2
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0411101
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2-(4-((4,5-Bis(4-methoxyphenyl)thiazol-2-yl)methylthio)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H25NO5S2
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0411102
|
2-[4-[[4,5-bis(4-methoxyphenyl)-1,3-oxazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C27H25NO7
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0411103
|
2-[4-[[4,5-bis(4-methoxyphenyl)-1,3-thiazol-2-yl]sulfanylmethyl]-2-methylphenoxy]acetic acid
Show/Hide
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C27H25NO5S2
|
1
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| 1 |
EC50 > 10000 nM
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CP0411104
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2-(4-((4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)methyl)-3-chlorophenyl)acetic Acid
Show/Hide
|
C26H22ClNO5S2
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0415384
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2-(4-((4-(Pyridin-3-yl)-5-(4-(trifluoromethoxy)phenyl)oxazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C25H19F3N2O6
|
1
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| 1 |
EC50 > 10000 nM
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CP0415556
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2-(4-((4-(4-Butoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
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C30H28F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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CP0415559
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2-(4-((4-(4-sec-Butoxyphenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H28F3NO6S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0417948
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2-(4-((4-(4-Methoxyphenyl)-5-(quinolin-3-yl)oxazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H24N2O6
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0429900
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2-(2-methyl-4-((5-methyl-4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)methoxy)phenoxy)acetic acid
Show/Hide
|
C21H18F3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0430315
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2-(4-((4,5-bis(4-(trifluoromethyl)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
|
C27H19F6NO4S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0430316
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2-(4-((4-(biphenyl-4-yl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
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C25H21NO4S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0430319
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2-(4-((5-(4-Biphenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C32H27NO5S
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0430321
|
2-(4-((5-(Benzofuran-2-yl)-4-(4-methoxyphenyl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C28H23NO6S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0430323
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2-(4-((4-(4-Methoxyphenyl)-5-(4-propylphenyl)oxazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H29NO6
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0430578
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2-(4-((4,5-Bis(4-methoxyphenyl)thiazol-2-yl)methoxy)-3-chlorophenyl)acetic Acid
Show/Hide
|
C26H22ClNO6S
|
1
|
| 1 |
EC50 > 10000 nM
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|
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CP0433721
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2-(4-((5-(4-Phenyl-3-(trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C33H26F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
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|
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CP0433723
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2-(4-((5-(3-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO5S
|
1
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| 1 |
EC50 > 10000 nM
|
|
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CP0433724
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2-[4-[[4-(4-methoxyphenyl)-5-[3-(trifluoromethyl)phenyl]-1,3-oxazol-2-yl]methoxy]-2-methylphenoxy]acetic acid
Show/Hide
|
C27H22F3NO6
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0433725
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2-(4-((4-(4-Methoxyphenyl)-5-(naphthalen-1-yl)thiazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H25NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0433727
|
2-(4-((5-(3,4-Dichlorophenyl)-4-(4-methoxyphenyl)oxazol-2-yl)-methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C26H21Cl2NO6
|
1
|
| 1 |
EC50 > 10000 nM
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|
|
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CP0433777
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2-(4-((4-(3-Fluoro-4-methoxyphenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H21F4NO6S
|
1
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| 1 |
EC50 > 10000 nM
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|
|
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CP0446570
|
2-[4-[[4,5-bis(4-methoxyphenyl)-1,3-thiazol-2-yl]sulfanyl]-2-methylphenoxy]acetic acid
Show/Hide
|
C26H23NO5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0447369
|
2-(4-((4,5-di(biphenyl-4-yl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic acid
Show/Hide
|
C37H29NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0450405
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-3-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0450406
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methylthio)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO4S2
|
1
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| 1 |
EC50 > 10000 nM
|
|
|
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CP0450407
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)phenoxy)acetic Acid
Show/Hide
|
C26H20F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0452568
|
2-(2-methyl-4-((4-p-tolylthiazol-2-yl)methoxy)phenoxy)acetic acid
Show/Hide
|
C20H19NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0453895
|
2-(4-((4,5-Bis(4-methoxyphenyl)oxazol-2-yl)methylthio)-3-chlorophenyl)acetic acid
Show/Hide
|
C26H22ClNO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0458870
|
2-(4-((4-(Pyrimidin-5-yl)-5-(4-(trifluoromethoxy)phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C24H18F3N3O5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0459077
|
2-(4-((4-(4-Morpholinophenyl)-5-(4-(trifluoromethoxy)phenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C30H27F3N2O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0459078
|
2-(4-((4-(4-(Methylsulfonamide)phenyl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H23F3N2O7S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0469809
|
2-(4-((5-(3-Chloro-4-methoxyphenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H24ClNO6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0471526
|
2-(4-((5-(2-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C27H22F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0473861
|
2-(4-(4,5-Bis(4-methoxyphenyl)thiazol-2-ylthio)-3-chlorophenyl)acetic Acid
Show/Hide
|
C25H20ClNO5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0476150
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methylthio)-3-chlorophenyl)acetic Acid
Show/Hide
|
C26H19ClF3NO3S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0494207
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)phenoxy)-2-methylpropanoic Acid
Show/Hide
|
C28H24F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0496147
|
2-(2-methyl-4-((4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)methoxy)phenoxy)acetic acid
Show/Hide
|
C20H16F3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0497630
|
2-(3-(4-(2-(3,5-dichlorophenoxy)ethylcarbamoyl)-5-phenylisoxazol-3-yl)phenyl)acetic acid
Show/Hide
|
C26H20Cl2N2O5
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0499456
|
2-(2-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)-thiazol-2-yl)methoxy)phenoxy)acetic Acid
Show/Hide
|
C26H20F3NO5S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0499457
|
2-(4-((5-(4-(Trifluoromethyl)phenyl)-4-(4-methoxyphenyl)thiazol-2-yl)methoxy)phenyl)acetic Acid
Show/Hide
|
C26H20F3NO4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0510492
|
2-(4-((4-(6-Morpholinopyridin-3-yl)-5-(4-(trifluoromethoxy)-phenyl)thiazol-2-yl)methoxy)-2-methylphenoxy)acetic Acid
Show/Hide
|
C29H26F3N3O6S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0393671
|
(3R)-3-[5-[[3-(2,6-dimethylphenyl)phenyl]methoxy]thiophen-2-yl]-3-ethoxypropanoic acid
Show/Hide
|
C24H26O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
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CP0408053
|
3-[5-[[3-(2,6-dimethylphenyl)phenyl]methoxy]thiophen-2-yl]propanoic acid
Show/Hide
|
C22H22O3S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0420403
|
(3R)-3-[5-[[3-[2,6-dimethyl-4-(3-methylsulfonylpropoxy)phenyl]phenyl]methoxy]thiophen-2-yl]hex-4-ynoic acid
Show/Hide
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C29H32O6S2
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1
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| 1 |
EC50 > 10000 nM
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CP0157489
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Lmb763
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C27H22ClN3O4
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1
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| 1 |
EC50 > 10000 nM
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CP0496445
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2-[4-[2-[4-[(4-chlorophenyl)diazenyl]phenoxy]ethyl]phenoxy]-2-methylpropanoic acid
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C24H23ClN2O4
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1
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| 1 |
EC50 > 10000 nM
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CP0496511
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2-methyl-2-[4-[2-[4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
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C25H26N2O4
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1
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| 1 |
EC50 > 10000 nM
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CP0571163
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2-methyl-2-[4-[2-[4-[(4-methylphenyl)diazenyl]phenoxy]ethyl]phenoxy]propanoic acid
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C25H26N2O4
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1
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| 1 |
EC50 > 10000 nM
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CP0576735
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3-hydroxy-2-[(1R,6R)-3-methyl-6-prop-1-en-2-ylcyclohex-2-en-1-yl]-5-pentylcyclohexa-2,5-diene-1,4-dione
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C21H28O3
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1
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| 1 |
EC50 = 10500 nM
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CP0534334
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2-[(3Z)-6-fluoro-3-[(4-fluorophenyl)methylidene]-2-methylinden-1-yl]acetic acid
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C19H14F2O2
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2
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| 1 |
EC50 = 11660 nM
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| 2 |
Kd = 6670 nM
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CP0041554
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Thyroxine
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C15H11I4NO4
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1
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| 1 |
EC50 = 12000 nM
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CP0545724
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2-[(3Z)-6-fluoro-2-methyl-3-[(3-methylphenyl)methylidene]inden-1-yl]acetic acid
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C20H17FO2
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2
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| 1 |
EC50 = 12020 nM
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| 2 |
Kd = 4000 nM
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CP0414716
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(2S)-2-amino-3-[3-bromo-4-(4-hydroxy-3,5-diiodophenoxy)-5-iodophenyl]propanoic acid
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C15H11BrI3NO4
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1
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| 1 |
EC50 = 12900 nM
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CP0252290
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4-tert-butyl-N-[[2-chloro-4-(methanesulfonamido)phenyl]methyl]benzamide
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C19H23ClN2O3S
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1
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| 1 |
EC50 = 14700 nM
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CP0562195
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2-methyl-2-(4-methylpent-3-enyl)-7-pentylchromene-5,8-dione
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C21H28O3
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1
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| 1 |
EC50 = 14700 nM
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CP0273107
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2-[(2E)-3,7-dimethylocta-2,6-dienyl]-5-pentylbenzene-1,3-diol
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C21H32O2
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1
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| 1 |
EC50 = 15700 nM
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CP0044444
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(Z)-5-Fluoro-2-methyl-1-((p-(methylsulfinyl)phenyl)methylene)-1H-indene-3-acetic acid
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C20H17FO3S
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2
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| 1 |
EC50 = 22650 nM
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| 2 |
Kd > 100000 nM
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CP0527206
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6,6,9-trimethyl-3-pentylbenzo[c]chromene-1,4-dione
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C21H24O3
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1
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| 1 |
EC50 = 23100 nM
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CP0109180
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2-(6-Isopropenyl-3-methyl-cyclohex-2-enyl)-5-pentyl-benzene-1,3-diol
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C21H30O2
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1
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| 1 |
EC50 > 25000 nM
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CP0260066
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6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol
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C21H26O2
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1
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| 1 |
EC50 > 25000 nM
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CP0260077
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2-Methyl-2-(4-methyl-pent-3-enyl)-7-pentyl-2H-chromen-5-ol(cannabichromene)
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C21H30O2
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1
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| 1 |
EC50 > 25000 nM
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CP0238477
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2-[(3Z)-6-fluoro-2-methyl-3-[(4-propan-2-ylphenyl)methylidene]inden-1-yl]acetic acid
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C22H21FO2
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2
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| 1 |
EC50 > 50000 nM
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| 2 |
Kd > 100000 nM
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CP0485286
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2-[(3Z)-6-fluoro-2-methyl-3-[(4-phenoxyphenyl)methylidene]inden-1-yl]acetic acid
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C25H19FO3
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2
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| 1 |
EC50 > 50000 nM
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| 2 |
Kd > 100000 nM
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CP0487236
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2-[(3Z)-2-methyl-3-[(3-methylphenyl)methylidene]inden-1-yl]acetic acid
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C20H18O2
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2
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| 1 |
EC50 > 50000 nM
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| 2 |
Kd > 100000 nM
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CP0511833
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2-[(3Z)-6-fluoro-2-methyl-3-[(4-phenylmethoxyphenyl)methylidene]inden-1-yl]acetic acid
Show/Hide
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C26H21FO3
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2
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| 1 |
EC50 > 50000 nM
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| 2 |
Kd > 100000 nM
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CP0548323
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2-[(3E)-2-methyl-3-[(3-methylphenyl)methylidene]inden-1-yl]acetic acid
Show/Hide
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C20H18O2
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2
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| 1 |
EC50 > 50000 nM
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| 2 |
Kd > 100000 nM
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CP0057167
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2-[2-methyl-4-[[4-(6-propan-2-yloxypyridin-3-yl)-5-[4-(trifluoromethoxy)phenyl]-1,3-oxazol-2-yl]methoxy]phenoxy]acetic acid
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C28H25F3N2O7
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1
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| 1 |
EC50 = 70000 nM
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CP0576275
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-[[4-(trifluoromethoxy)phenyl]methoxy]phenyl]methylidene]hexanoic acid
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C33H29F6NO6
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1
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| 1 |
IC50 = 1900 nM
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CP0427118
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C32H29F4NO5
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1
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| 1 |
IC50 = 2300 nM
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CP0384330
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-[(1-methylpiperidin-4-yl)methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H35F3N2O5
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1
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| 1 |
IC50 = 2500 nM
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CP0469448
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(2E)-2-[[2-[[4-(difluoromethoxy)phenyl]methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C33H30F5NO6
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1
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| 1 |
IC50 = 2600 nM
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CP0562317
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H27F4NO5
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1
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| 1 |
IC50 = 3200 nM
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CP0403133
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(2E)-2-[[2-[(2-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H27F4NO5
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1
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| 1 |
IC50 = 3500 nM
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CP0403135
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4-methoxy-7-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-1-propylindole-2-carboxylic acid
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C25H23F3N2O5
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1
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| 1 |
IC50 = 3900 nM
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CP0534298
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(2E)-2-[[2-[(3-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H27F4NO5
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1
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| 1 |
IC50 = 3900 nM
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CP0534302
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[(2-methylquinolin-6-yl)methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C30H28FNO4
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1
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| 1 |
IC50 = 4200 nM
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CP0148416
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-[[4-(trifluoromethyl)phenyl]methoxy]phenyl]methylidene]hexanoic acid
Show/Hide
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C33H29F6NO5
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1
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| 1 |
IC50 = 4300 nM
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CP0176364
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H36F3N3O5
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1
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| 1 |
IC50 = 4700 nM
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CP0543510
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-(pyridin-4-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C30H27F3N2O5
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1
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| 1 |
IC50 = 4700 nM
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CP0435145
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-(quinolin-6-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C29H26FNO4
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1
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| 1 |
IC50 = 5000 nM
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CP0534299
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]butanoic acid
Show/Hide
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C30H25F4NO5
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1
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| 1 |
IC50 = 5700 nM
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CP0467901
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[(1-oxidoquinolin-1-ium-6-yl)methoxy]phenyl]methylidene]pentanoic acid
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C29H26FNO5
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1
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| 1 |
IC50 = 6100 nM
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CP0558524
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-[(2-oxo-1H-quinolin-6-yl)methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C29H26FNO5
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1
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| 1 |
IC50 = 6100 nM
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CP0101191
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methyl 2-[4-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]acetate
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C21H21NO5
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1
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| 1 |
IC50 = 6300 nM
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CP0101189
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methyl 2-[4-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]phenyl]acetate
Show/Hide
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C21H21NO5
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1
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| 1 |
IC50 = 6700 nM
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CP0403134
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-phenylmethoxyphenyl]methylidene]pentanoic acid
Show/Hide
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C31H28F3NO5
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1
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| 1 |
IC50 = 7200 nM
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CP0543514
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(2E)-4-cyclopropyl-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-[(1-methylpiperidin-4-yl)methoxy]phenyl]methylidene]butanoic acid
Show/Hide
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C33H37F3N2O5
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1
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| 1 |
IC50 = 7500 nM
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CP0101190
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methyl 3-[[2-(2-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoate
Show/Hide
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C20H19NO5
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1
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| 1 |
IC50 = 7600 nM
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CP0180022
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methyl 4-[[2-(3-methoxyphenyl)-4-methyl-1,3-oxazol-5-yl]methoxy]benzoate
Show/Hide
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C20H19NO5
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1
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| 1 |
IC50 = 7600 nM
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CP0543512
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(E)-2-(cyclopropylmethyl)-3-[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]prop-2-enoic acid
Show/Hide
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C32H27F4NO5
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1
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| 1 |
IC50 = 8400 nM
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CP0576276
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(E)-3-[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]-2-methylprop-2-enoic acid
Show/Hide
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C29H23F4NO5
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1
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| 1 |
IC50 = 9400 nM
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CP0474178
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(2E)-2-[[2-[(4-fluorobenzoyl)amino]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]methylidene]pentanoic acid
Show/Hide
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C31H26F4N2O5
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1
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| 1 |
IC50 = 9500 nM
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CP0554721
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(2E)-2-[[5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]-2-(2-piperazin-1-ylethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C30H34F3N3O5
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1
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| 1 |
IC50 = 9600 nM
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CP0554719
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(E)-3-[2-[(4-fluorophenyl)methoxy]-5-[[4-methoxy-2-(trifluoromethyl)quinolin-6-yl]methoxy]phenyl]prop-2-enoic acid
Show/Hide
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C28H21F4NO5
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1
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| 1 |
IC50 = 11000 nM
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CP0534301
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-(quinolin-2-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C29H26FNO4
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1
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| 1 |
IC50 = 13100 nM
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CP0558525
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(2E)-2-[[2-[(1-methylpiperidin-4-yl)methoxy]-5-(quinolin-6-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C29H34N2O4
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1
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| 1 |
IC50 = 15100 nM
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CP0534300
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-(naphthalen-2-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C30H27FO4
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1
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| 1 |
IC50 = 15800 nM
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CP0427119
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(2E)-2-[[2-[(4-fluorophenyl)methoxy]-5-(quinolin-7-ylmethoxy)phenyl]methylidene]pentanoic acid
Show/Hide
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C29H26FNO4
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1
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| 1 |
IC50 = 23900 nM
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CP0421524
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3,4-dimethoxy-N-[(2-methyl-1H-indol-3-yl)-[4-(trifluoromethoxy)phenyl]methyl]aniline
Show/Hide
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C25H23F3N2O3
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1
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| 1 |
IC50 > 25000 nM
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