| Compound ID |
Compound Name |
Compound Formula |
|
CP0520044
|
2-[4-(3,3-difluorocyclobutyl)phenyl]-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C22H19F4N3O
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0412184
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(3,3-difluoropyrrolidin-1-yl)pyridin-3-yl]acetamide
Show/Hide
|
C21H19F4N5O
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0412187
|
N-[1-[(4-chlorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C20H21ClN4O
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0541307
|
N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-ethyl-4-(2,2,2-trifluoroethoxy)phenyl]acetamide
Show/Hide
|
C22H20F3N5O2
|
1
|
| 1 |
IC50 = 1.1 nM
|
|
|
|
CP0143412
|
2-(4-propan-2-ylphenyl)-N-[(1R)-1-[5-(2,2,2-trifluoroethoxy)pyridin-2-yl]ethyl]acetamide
Show/Hide
|
C20H23F3N2O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0408590
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1,3,3-trimethyl-2-oxoindol-5-yl)acetamide
Show/Hide
|
C23H22F2N4O2
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0412180
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(4-propan-2-ylphenyl)acetamide
Show/Hide
|
C21H21F2N3O
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0471804
|
2-[4-(3,3-difluorocyclobutyl)oxyphenyl]-N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C22H19F4N3O2
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0477388
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C20H20F2N4O
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
|
CP0389186
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-6-yl)acetamide
Show/Hide
|
C20H16F2N4O
|
1
|
| 1 |
IC50 = 1.9 nM
|
|
|
|
CP0255833
|
N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(2,2,2-trifluoroethoxy)phenyl]acetamide
Show/Hide
|
C21H18F3N5O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0396378
|
2-[4-(dimethylamino)phenyl]-N-[1-[[4-(trifluoromethoxy)phenyl]methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C21H21F3N4O2
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0366788
|
N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(trifluoromethoxy)phenyl]acetamide
Show/Hide
|
C20H16F3N5O2
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0404249
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1H-indol-5-yl)acetamide
Show/Hide
|
C20H16F2N4O
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0412191
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(3-methyloxetan-3-yl)phenyl]acetamide
Show/Hide
|
C22H21F2N3O2
|
1
|
| 1 |
IC50 = 2.4 nM
|
|
|
|
CP0412194
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-[(3S)-3-fluoropyrrolidin-1-yl]pyridin-3-yl]acetamide
Show/Hide
|
C21H20F3N5O
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0227177
|
N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]-2-[3-methyl-4-(3,3,3-trifluoropropoxy)phenyl]acetamide
Show/Hide
|
C22H20F3N5O2
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0412178
|
2-(4-tert-butylphenyl)-N-[1-[(5-cyanopyridin-2-yl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C22H23N5O
|
1
|
| 1 |
IC50 = 2.8 nM
|
|
|
|
CP0412200
|
N-[1-[(4-cyano-3-fluorophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C21H20FN5O
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
|
CP0396376
|
N-[1-[(3,5-difluoro-4-methoxyphenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C21H22F2N4O2
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
|
CP0392102
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(2,2-dimethyl-1,3-dioxolan-4-yl)phenyl]acetamide
Show/Hide
|
C23H23F2N3O3
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0446098
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(3-methyl-2-oxo-1,3-benzoxazol-6-yl)acetamide
Show/Hide
|
C20H16F2N4O3
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0481948
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylindazol-5-yl)acetamide
Show/Hide
|
C20H17F2N5O
|
1
|
| 1 |
IC50 = 3.4 nM
|
|
|
|
CP0404251
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-[(3-methyloxetan-3-yl)methoxy]phenyl]acetamide
Show/Hide
|
C23H23F2N3O3
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0408536
|
N-[2-(3,4-Difluoro-benzyl)-2H-[1,2,3]triazol-4-yl]-2-(1-methyl-1H-indazol-5-yl)-acetamide
Show/Hide
|
C19H16F2N6O
|
1
|
| 1 |
IC50 = 3.5 nM
|
|
|
|
CP0382629
|
(3R,5S)-1-[(2-fluorophenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0452703
|
(3R,5S)-3,5-dimethyl-N-pyridin-3-yl-1-[[5-(trifluoromethyl)furan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C23H23F3N4O2
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0008581
|
1-[4-[(2,4-dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C32H30Cl2N2O
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 33 nM
|
|
|
|
CP0412179
|
2-[4-(dimethylamino)phenyl]-N-[1-[(4-fluorophenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C20H21FN4O
|
1
|
| 1 |
IC50 = 4.2 nM
|
|
|
|
CP0481954
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(3-fluorooxetan-3-yl)phenyl]acetamide
Show/Hide
|
C21H18F3N3O2
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0471802
|
N-[4-[(3,4-difluorophenyl)methyl]-1,3-thiazol-2-yl]-2-(4-propan-2-ylphenyl)acetamide
Show/Hide
|
C21H20F2N2OS
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0396377
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[4-(oxetan-3-yloxy)phenyl]acetamide
Show/Hide
|
C21H19F2N3O3
|
1
|
| 1 |
IC50 = 4.6 nM
|
|
|
|
CP0382618
|
(3R,5S)-N-benzyl-1-[(2,3-difluorophenyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H27F2N3O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0471801
|
2-(4-tert-butylphenyl)-N-[1-[(3,4-difluorophenyl)methyl]-1,2,4-triazol-3-yl]acetamide
Show/Hide
|
C21H22F2N4O
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0481950
|
N-(1-benzylpyrazol-3-yl)-2-(4-propan-2-ylphenyl)acetamide
Show/Hide
|
C21H23N3O
|
1
|
| 1 |
IC50 = 5.1 nM
|
|
|
|
CP0424410
|
(3R,5S)-1-benzyl-8-fluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0481946
|
2-[4-(dimethylamino)phenyl]-N-[1-[(4-fluorophenyl)methyl]pyrazol-3-yl]propanamide
Show/Hide
|
C21H23FN4O
|
1
|
| 1 |
IC50 = 6.2 nM
|
|
|
|
CP0085643
|
Act-709478
Show/Hide
|
C22H18F3N5O
|
1
|
| 1 |
IC50 = 6.4 nM
|
|
|
|
CP0408544
|
1-[(3,4-difluorophenyl)methyl]-N-[[6-(3,3-difluoropyrrolidin-1-yl)pyridin-3-yl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C21H19F4N5O
|
1
|
| 1 |
IC50 = 6.5 nM
|
|
|
|
CP0412186
|
N-[1-[[4-(difluoromethoxy)phenyl]methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C21H22F2N4O2
|
1
|
| 1 |
IC50 = 6.8 nM
|
|
|
|
CP0377009
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-[[5-(trifluoromethyl)furan-2-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H26F3N3O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0446022
|
(3R,5S)-N,1-dibenzyl-8-fluoro-3,5-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0477385
|
2-[4-(dimethylamino)phenyl]-N-[1-[(4-methylphenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C21H24N4O
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0412468
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(1-methylpyrrolo[2,3-b]pyridin-5-yl)acetamide
Show/Hide
|
C20H17F2N5O
|
1
|
| 1 |
IC50 = 7.1 nM
|
|
|
|
CP0396285
|
(3R,5S)-1-[(3-fluorophenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0477602
|
(3R,5S)-1-benzyl-N-[(4-methoxyphenyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C27H31N3O2
|
1
|
| 1 |
IC50 = 8 nM
|
|
|
|
CP0446099
|
2-[4-(dimethylamino)phenyl]-N-[1-[(3-methylphenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C21H24N4O
|
1
|
| 1 |
IC50 = 8.1 nM
|
|
|
|
CP0174617
|
methyl 5-[3-(1H-benzimidazol-2-yl)propyl-methylamino]-2-(4-bromophenyl)-2-propan-2-ylpentanoate
Show/Hide
|
C26H34BrN3O2
|
1
|
| 1 |
IC50 = 8.17 nM
|
|
|
|
CP0477386
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(2,2,2-trifluoroethoxy)pyridin-3-yl]acetamide
Show/Hide
|
C19H15F5N4O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0396345
|
N-[1-[(4-cyanophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C21H21N5O
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0481945
|
N-(1-benzylpyrazol-3-yl)-2-(4-methoxy-3-methylphenyl)acetamide
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0382620
|
(3R,5S)-1-benzyl-6,8-difluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H24F2N4O
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0412195
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-[6-(dimethylamino)pyridin-3-yl]acetamide
Show/Hide
|
C19H19F2N5O
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0455946
|
(3R,5S)-N-[(4-methoxyphenyl)methyl]-3,5-dimethyl-1-[[5-(trifluoromethyl)furan-2-yl]methyl]-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27F3N4O3
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0519622
|
(3R,5S)-1-[(3,4-difluorophenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H24F2N4O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0551482
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-[[2-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25F3N4OS
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0429720
|
N-(1-benzylpyrazol-3-yl)-2-[4-(trifluoromethoxy)phenyl]acetamide
Show/Hide
|
C19H16F3N3O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0396344
|
N-(1-benzylpyrazol-3-yl)-2-[4-(dimethylamino)phenyl]acetamide
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0494493
|
2-(4-propan-2-ylphenyl)-N-[1-[2-(2,2,2-trifluoroethoxy)ethyl]pyrazol-3-yl]acetamide
Show/Hide
|
C18H22F3N3O2
|
1
|
| 1 |
IC50 = 14 nM
|
|
|
|
CP0377011
|
(3R,5S)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H28N4O
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0908753
|
2-(6-Cyclopropyl-pyridin-3-yl)-N-[1-(3,4-difluoro-benzyl)-1H-pyrazol-3-yl]-acetamide
Show/Hide
|
C20H18F2N4O
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0377005
|
(3R,5S)-N,1-dibenzyl-8-chloro-3,5-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27ClN4O
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0865116
|
4-(3,4-Difluorobenzyl)-N-(4-(dimethylamino)benzyl)thiazole-2-carboxamide
Show/Hide
|
C20H19F2N3OS
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0865123
|
N-(4-Cyano-1-(3,4-difluorobenzyl)-1H-pyrazol-3-yl)-2-(1-methyl-1H-indazol-5-yl)acetamide
Show/Hide
|
C21H16F2N6O
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0396291
|
(3R,5S)-N,1-dibenzyl-3,5,8-trimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C26H30N4O
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0412188
|
N-[(6-pyrrolidin-1-ylpyridin-3-yl)methyl]-2-[[4-(trifluoromethoxy)phenyl]methyl]-1,3-oxazole-4-carboxamide
Show/Hide
|
C22H21F3N4O3
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0444018
|
(3R,5S)-1-benzyl-6-fluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0396362
|
4-bromo-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H19BrF3N3O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0568717
|
N-[1-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]ethyl]-2-(4-propan-2-ylphenyl)acetamide
Show/Hide
|
C23H25F2N3O
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0382631
|
(3R,5S)-1-(cyclopentylmethyl)-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C23H30N4O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0444013
|
(3R,5S)-3,5-dimethyl-1-(3-methylbutyl)-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C22H30N4O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0865213
|
2-(4-Dimethylamino-phenyl)-N-[1-(4-methoxy-benzyl)-1H-pyrazol-3-yl]-acetamide
Show/Hide
|
C21H24N4O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0446069
|
[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-(oxan-4-yl)methanone
Show/Hide
|
C24H30N2O2
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0412189
|
1-[(3,4-difluorophenyl)methyl]-N-[(4-propan-2-ylphenyl)methyl]pyrazole-3-carboxamide
Show/Hide
|
C21H21F2N3O
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0382630
|
(3R,5S)-1-[(4-fluorophenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0396286
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-[[6-(trifluoromethyl)pyridin-2-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H27F3N4O
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0377008
|
[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-morpholin-4-ylmethanone
Show/Hide
|
C23H29N3O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0452701
|
(3R,5S)-1-benzyl-3,5-dimethyl-N-(oxetan-3-yl)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0455950
|
(3R,5S)-1-[dideuterio(phenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H26N4O
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0408586
|
4-bromo-1-(2-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H18BrF4N3O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0059960
|
N,3-bis(4-fluorophenyl)-5-pyridin-4-yl-3,4-dihydropyrazole-2-carboxamide
Show/Hide
|
C21H16F2N4O
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0396289
|
1-[(3R,5S)-3,5-dimethyl-1-(3-methylbutyl)-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C24H33N3O
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
|
CP0444161
|
1-[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C26H29N3O
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0518118
|
4-bromo-1,5-diphenyl-N-[(2-pyrazol-1-ylphenyl)methyl]pyrazole-3-carboxamide
Show/Hide
|
C26H20BrN5O
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0396287
|
(3R,5S)-3,5-dimethyl-N-pyridin-3-yl-1-[[2-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C22H22F3N5OS
|
1
|
| 1 |
IC50 = 33 nM
|
|
|
|
CP0519621
|
1-[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-2-(1,3-thiazol-5-yl)ethanone
Show/Hide
|
C23H25N3OS
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0482176
|
2-[(3,4-difluorophenyl)methyl]-N-[(1-methylindazol-5-yl)methyl]triazole-4-carboxamide
Show/Hide
|
C19H16F2N6O
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0444064
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-[2-[(2-methylpropan-2-yl)oxy]ethyl]-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H35N3O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0008576
|
1-[4-[(2,4-dimethylphenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C34H36N2O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0412466
|
N-(1-benzylpyrazol-3-yl)-2-(4-methylphenyl)acetamide
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0486052
|
N-(1-benzylpyrazol-3-yl)-2-(4-ethoxyphenyl)acetamide
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0498397
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(2-fluorophenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C25H32F2N2O
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0532988
|
1-[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-2-morpholin-4-ylethanone
Show/Hide
|
C24H31N3O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0410031
|
N-[[1-[2-(tert-butylamino)-2-oxoethyl]piperidin-4-yl]methyl]-3-chloro-5-fluorobenzamide
Show/Hide
|
C19H27ClFN3O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0532987
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-[[5-(trifluoromethyl)furan-2-yl]methyl]-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C24H25F3N4O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0382624
|
(3R,5S)-N-benzyl-1-[(2,3-difluorophenyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H26F2N4O
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0444157
|
1-[(3R,5S)-3,5-dimethyl-1-[[2-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C24H25F3N4OS
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0452712
|
(3R,5S)-1-benzyl-6-fluoro-3,5-dimethyl-N-(oxetan-3-yl)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C22H26FN3O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0378573
|
N-benzyl-2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide
Show/Hide
|
C37H43N5O
|
3
|
| 1 |
IC50 = 41 nM
|
|
|
| 2 |
IC50 = 41.3 nM
|
|
|
| 3 |
IC50 = 260 nM
|
|
|
|
CP0486051
|
N-(1-benzylpyrazol-3-yl)-2-(4-chlorophenyl)acetamide
Show/Hide
|
C18H16ClN3O
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0455947
|
(3R,5S)-1-benzyl-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H26N4O
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0482178
|
N-(1-benzylpyrazol-3-yl)-2-(3-chlorophenyl)acetamide
Show/Hide
|
C18H16ClN3O
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0396294
|
(3R,5S)-N-benzyl-1-[(6-methoxypyridin-3-yl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H30N4O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0510168
|
1-[(3R,5S)-6-fluoro-3,5-dimethyl-1-(3-methylbutyl)-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C24H32FN3O
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0476828
|
4-bromo-1,5-diphenyl-N-[[3-(2,2,2-trifluoroethoxy)pyridin-2-yl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C24H18BrF3N4O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0404250
|
N-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-2-(3-methylbenzimidazol-5-yl)acetamide
Show/Hide
|
C20H17F2N5O
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0521801
|
2-[(3,4-difluorophenyl)methyl]-N-[[4-(dimethylamino)phenyl]methyl]-1,3-thiazole-4-carboxamide
Show/Hide
|
C20H19F2N3OS
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0396364
|
4-(2-hydroxyethyl)-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C27H24F3N3O3
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0408322
|
1-[(3R,5S)-1-benzyl-6-fluoro-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C26H28FN3O
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0452705
|
(3R,5S)-N-benzyl-1-[(2-fluorophenyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
IC50 = 47 nM
|
|
|
|
CP0389185
|
4-(difluoromethyl)-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C26H20F5N3O2
|
1
|
| 1 |
IC50 = 49 nM
|
|
|
|
CP0213567
|
4-[2-(ethylamino)ethyl]-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C29H29F3N4O2
|
1
|
| 1 |
IC50 = 52 nM
|
|
|
|
CP0382579
|
(3R,5S)-N-benzyl-1-[(2-fluoropyridin-3-yl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0412183
|
1-[(3,4-difluorophenyl)methyl]-N-[[4-(3-fluorooxetan-3-yl)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C21H18F3N3O2
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0400923
|
methyl 2-(4-bromophenyl)-5-[3-(5,6-dimethyl-1H-benzimidazol-2-yl)propyl-methylamino]-2-propan-2-ylpentanoate
Show/Hide
|
C28H38BrN3O2
|
1
|
| 1 |
IC50 = 53.02 nM
|
|
|
|
CP0471781
|
3-chloro-2-methyl-N-[[2-(2-methylpropoxy)phenyl]methyl]-5-(trifluoromethyl)-4,5,6,7-tetrahydroisoindole-1-carboxamide
Show/Hide
|
C22H26ClF3N2O2
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0865121
|
N-(1-Benzyl-1H-pyrazol-3-yl)-2-m-tolyl-acetamide
Show/Hide
|
C19H19N3O
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0008577
|
1-[4-[(3-chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C32H31ClN2O
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0408589
|
4-(hydroxymethyl)-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C26H22F3N3O3
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0412463
|
N-[[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]methyl]-2-(4-propan-2-ylphenyl)acetamide
Show/Hide
|
C22H23F2N3O
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0435082
|
methyl 5-[3-(1H-benzimidazol-2-yl)propyl-methylamino]-2-(4-bromophenyl)-5-oxo-2-propan-2-ylpentanoate
Show/Hide
|
C26H32BrN3O3
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0396292
|
(3R,5S)-N,1-dibenzyl-3,5-dimethyl-8-(trifluoromethyl)-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C26H27F3N4O
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0482015
|
4-bromo-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C24H18BrF3N4O2
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0389187
|
1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H20F3N3O2
|
1
|
| 1 |
IC50 = 59 nM
|
|
|
|
CP0486049
|
4-[[2-[(4-fluorophenyl)methyl]-4H-imidazo[4,5-c]pyrazol-5-yl]methyl]-N,N-dimethylaniline
Show/Hide
|
C20H20FN5
|
1
|
| 1 |
IC50 = 60 nM
|
|
|
|
CP0009666
|
1-[4-[(2,3-dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C32H30Cl2N2O
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0377006
|
(3R,5S)-N,1-dibenzyl-7-fluoro-3,5-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
IC50 = 65 nM
|
|
|
|
CP0444045
|
(3R,5S)-1-benzyl-7-fluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0389209
|
1-[(3,4-difluorophenyl)methyl]-N-(1H-indol-5-ylmethyl)pyrazole-3-carboxamide
Show/Hide
|
C20H16F2N4O
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0463423
|
4-ethenyl-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C27H22F3N3O2
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0377007
|
(3R,5S)-N-[(4-methoxyphenyl)methyl]-3,5-dimethyl-1-(3-methylbutyl)-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C24H34N4O2
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0444069
|
(3R,5S)-N,1-dibenzyl-7-chloro-3,5-dimethyl-3,5-dihydro-2H-pyrido[2,3-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27ClN4O
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0444065
|
(3R,5S)-1-benzyl-N-[(4-methoxyphenyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C26H30N4O2
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0009367
|
1-[4-[(4-chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C32H31ClN2O
|
1
|
| 1 |
IC50 = 81 nM
|
|
|
|
CP0531063
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(4-fluorophenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C25H32F2N2O
|
1
|
| 1 |
IC50 = 82 nM
|
|
|
|
CP0520052
|
5-chloro-4-ethyl-1,3-dimethyl-N-[[2-(2-methylpropoxy)phenyl]methyl]pyrrole-2-carboxamide
Show/Hide
|
C20H27ClN2O2
|
1
|
| 1 |
IC50 = 82 nM
|
|
|
|
CP0502930
|
1-benzyl-N-[2-ethyl-2-(4-fluorophenyl)butyl]piperidine-4-carboxamide
Show/Hide
|
C25H33FN2O
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
|
CP0471736
|
3-chloro-N-[(2-ethoxyphenyl)methyl]-2,5,5-trimethyl-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C21H27ClN2O2
|
1
|
| 1 |
IC50 = 87 nM
|
|
|
|
CP0450864
|
4-bromo-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]-1-(2,2,2-trifluoroethyl)pyrazole-3-carboxamide
Show/Hide
|
C21H16BrF6N3O2
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0536149
|
4-bromo-1-(4-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H18BrF4N3O2
|
1
|
| 1 |
IC50 = 88 nM
|
|
|
|
CP0468566
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-(2-phenylethyl)piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O
|
1
|
| 1 |
IC50 = 89 nM
|
|
|
|
CP0499302
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(2-fluorophenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C26H34F2N2O
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0531064
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(3-methoxyphenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O2
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0433089
|
methyl 2-(4-bromophenyl)-5-[4-(2-methoxyphenyl)piperazin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C26H35BrN2O3
|
2
|
| 1 |
IC50 = 95 nM
|
|
|
| 2 |
IC50 = 95040 nM
|
|
|
|
CP0475586
|
(5S,6S)-3-chloro-2,5,6-trimethyl-N-[[2-(2-methylpropoxy)phenyl]methyl]-4,5,6,7-tetrahydroisoindole-1-carboxamide
Show/Hide
|
C23H31ClN2O2
|
1
|
| 1 |
IC50 = 98 nM
|
|
|
|
CP0433657
|
3-(4-chlorobenzyl)-N-(3-(2-ethylpiperidin-1-yl)propyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C26H31ClN4O2S
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0494609
|
ethyl 5-[3-(5,6-dimethyl-1H-benzimidazol-2-yl)propyl-methylamino]-2-phenyl-2-propan-2-ylpentanoate
Show/Hide
|
C29H41N3O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0322289
|
(2R)-1-[4-[(3,4-dichlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
|
C20H23Cl2FN2O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0429388
|
4-bromo-5-cyclopropyl-1-(2-fluorophenyl)-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C22H18BrF4N3O2
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0382615
|
(3R)-N,1-dibenzyl-3-methyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H27N3O
|
1
|
| 1 |
IC50 = 102 nM
|
|
|
|
CP0424412
|
(3R,5S)-1-benzyl-6-fluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C23H24FN5O
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0396296
|
(3R,5S)-3,5-dimethyl-1-[2-[(2-methylpropan-2-yl)oxy]ethyl]-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C23H32N4O2
|
1
|
| 1 |
IC50 = 108 nM
|
|
|
|
CP0397786
|
N-[[4-[(4-fluorophenyl)sulfonylamino]phenyl]methyl]-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide
Show/Hide
|
C34H34FN5O3S
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
IC50 = 200 nM
|
|
|
|
CP0408588
|
4-bromo-5-ethyl-1-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C21H19BrF3N3O2
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0542970
|
1-[(3R,5S)-6-fluoro-3,5-dimethyl-1-[[2-(trifluoromethyl)-1,3-thiazol-5-yl]methyl]-3,5-dihydro-2H-1,4-benzodiazepin-4-yl]-3-pyridin-3-ylpropan-1-one
Show/Hide
|
C24H24F4N4OS
|
1
|
| 1 |
IC50 = 115 nM
|
|
|
|
CP0499301
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(2-methoxyphenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O2
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0536135
|
3-chloro-2,5,5-trimethyl-N-[[2-(pyrazol-1-ylmethyl)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C23H27ClN4O
|
1
|
| 1 |
IC50 = 120 nM
|
|
|
|
CP0373366
|
2-(2-(5-aminopentylamino)-3-(biphenyl-4-yl)-3,4-dihydroquinazolin-4-yl)-N-benzylacetamide
Show/Hide
|
C34H37N5O
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
IC50 = 130.02 nM
|
|
|
|
CP0499080
|
1-benzyl-N-[2-(4-fluorophenyl)-2-methylpropyl]piperidine-4-carboxamide
Show/Hide
|
C23H29FN2O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0504504
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(3-fluorophenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C26H34F2N2O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0531062
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(3-fluorophenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C25H32F2N2O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0482016
|
N-[(2-fluorophenyl)methyl]-1,5-diphenylpyrazole-3-carboxamide
Show/Hide
|
C23H18FN3O
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0373363
|
2-(3-(5-aminopentyl)-2-(biphenyl-4-ylamino)-3,4-dihydroquinazolin-4-yl)-N-benzylacetamide
Show/Hide
|
C34H37N5O
|
2
|
| 1 |
IC50 = 139.96 nM
|
|
|
| 2 |
IC50 = 140 nM
|
|
|
|
CP0512771
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(3-methoxyphenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C27H37FN2O2
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0444047
|
(3R,5S)-N,1-dibenzyl-6-fluoro-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27FN4O
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0475589
|
3-bromo-N-[[2-(ethoxymethyl)phenyl]methyl]-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophene-1-carboxamide
Show/Hide
|
C21H26BrNO2S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0002873
|
1-[4-[(2-chlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
|
C32H31ClN2O
|
1
|
| 1 |
IC50 = 141 nM
|
|
|
|
CP0421177
|
tert-butyl N-[5-[[4-[2-(benzylamino)-2-oxoethyl]-3-(4-phenylphenyl)-1,4-dihydroquinazolin-2-ylidene]amino]pentyl]carbamate
Show/Hide
|
C39H45N5O3
|
2
|
| 1 |
IC50 = 159.96 nM
|
|
|
| 2 |
IC50 = 160 nM
|
|
|
|
CP0482012
|
4-(difluoromethyl)-1-(4-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C26H19F6N3O2
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0373851
|
2-(3-Phenyl-2-piperidin-1-yl-3,4-dihydro-quinazolin-4-yl)-N-[4-(toluene-4-sulfonylamino)-benzyl]-acetamide
Show/Hide
|
C35H37N5O3S
|
3
|
| 1 |
IC50 = 169.82 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
| 3 |
IC50 = 250 nM
|
|
|
|
CP0421176
|
tert-butyl N-[5-[4-[2-(benzylamino)-2-oxoethyl]-2-(4-phenylanilino)-4H-quinazolin-3-yl]pentyl]carbamate
Show/Hide
|
C39H45N5O3
|
2
|
| 1 |
IC50 = 169.82 nM
|
|
|
| 2 |
IC50 = 170 nM
|
|
|
|
CP0505875
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(2-methoxyphenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C27H37FN2O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0475587
|
3-chloro-2-methyl-N-[[2-(2-methylpropoxy)phenyl]methyl]-5,6-dihydro-4H-cyclopenta[c]pyrrole-1-carboxamide
Show/Hide
|
C20H25ClN2O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0482179
|
N-(1-benzylpyrazol-3-yl)-2-(4-methoxyphenyl)acetamide
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0396153
|
(3R,5S)-1-benzyl-9-fluoro-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C24H25FN4O
|
1
|
| 1 |
IC50 = 178 nM
|
|
|
|
CP0503162
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(4-fluorophenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C26H34F2N2O
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0396309
|
3-chloro-N-[[2-(ethoxymethyl)phenyl]methyl]-2,5,5-trimethyl-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C22H29ClN2O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0470836
|
3-chloro-2,5,5-trimethyl-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C20H23ClF3N3O2
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0481947
|
3-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-5-[(4-propan-2-ylphenyl)methyl]-1H-1,2,4-triazole
Show/Hide
|
C22H21F2N5
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0475697
|
(3R,5S)-1-benzyl-3,5-dimethyl-N-pyridin-3-yl-8-(2,2,2-trifluoroethoxy)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H27F3N4O2
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0382580
|
(3R,5S)-1-benzyl-6-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O2
|
1
|
| 1 |
IC50 = 188 nM
|
|
|
|
CP0514526
|
methyl 5-[3-(1H-benzimidazol-2-yl)propyl-methylamino]-2-(4-methoxyphenyl)-2-propan-2-ylpentanoate
Show/Hide
|
C27H37N3O3
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0470878
|
1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-yl)-4-(cyclohexylmethylamino)butan-1-one
Show/Hide
|
C28H38ClN3O
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0450863
|
4-(difluoromethyl)-1-(2-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C26H19F6N3O2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0444160
|
(5S)-N,1-dibenzyl-5-methyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H27N3O
|
1
|
| 1 |
IC50 = 193 nM
|
|
|
|
CP0395729
|
1-[(3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepin-4-yl]-3-(4-fluorophenyl)propan-1-one
Show/Hide
|
C26H28FN3O
|
1
|
| 1 |
IC50 = 196 nM
|
|
|
|
CP0013607
|
2-methoxyacetic acid [(1S,2S)-2-[2-[3-(1H-benzimidazol-2-yl)propyl-methyl-amino]ethyl]-6-fluoro-1-isopropyl-tetralin-2-yl] ester;hydrate;hydrochloride
Show/Hide
|
C29H38FN3O3
|
6
|
| 1 |
IC50 = 200 nM
|
|
|
| 2 |
IC50 = 560 nM
|
|
|
| 3 |
IC50 = 830 nM
|
|
|
| 4 |
IC50 = 840 nM
|
|
|
| 5 |
IC50 = 860 nM
|
|
|
| 6 |
IC50 = 1340 nM
|
|
|
|
CP0504503
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[(4-methoxyphenyl)methyl]piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0463422
|
4-[2-(cyclopropylamino)ethyl]-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C30H29F3N4O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0482011
|
N-benzyl-1,5-diphenylpyrazole-3-carboxamide
Show/Hide
|
C23H19N3O
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0085972
|
3-chloro-2,5,5-trimethyl-N-[[2-(propan-2-yloxymethyl)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C23H31ClN2O2
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0450850
|
3-bromo-N-[(2-ethoxyphenyl)methyl]-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophene-1-carboxamide
Show/Hide
|
C20H24BrNO2S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0396283
|
(2R,5S)-N,1-dibenzyl-2,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H29N3O
|
1
|
| 1 |
IC50 = 211 nM
|
|
|
|
CP0512770
|
1-benzyl-N-[[1-(4-fluorophenyl)cyclopentyl]methyl]piperidine-4-carboxamide
Show/Hide
|
C25H31FN2O
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0452704
|
(3R,5S)-N,1-dibenzyl-7-chloro-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H27ClN4O
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0450861
|
4-bromo-1-(3-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H18BrF4N3O2
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0396298
|
(3R,5S)-1-benzyl-3,5,8-trimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O
|
1
|
| 1 |
IC50 = 227 nM
|
|
|
|
CP0378571
|
methyl 2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetate
Show/Hide
|
C31H38N4O2
|
2
|
| 1 |
IC50 = 230 nM
|
|
|
| 2 |
IC50 = 230.14 nM
|
|
|
|
CP0345360
|
(2S)-1-[4-[(3,4-dichlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
|
C20H23Cl2FN2O2
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0475592
|
(2R,4S)-N-[[4-(ethoxymethyl)phenyl]methyl]-3,3,9-trimethyl-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
|
C22H27NO2S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0528908
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-(3-phenylpropyl)piperidine-4-carboxamide
Show/Hide
|
C27H37FN2O
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0396363
|
4-[2-(diethylamino)ethyl]-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C31H33F3N4O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0450852
|
5-chloro-3-ethyl-1,4-dimethyl-N-[[2-(2-methylpropoxy)phenyl]methyl]pyrrole-2-carboxamide
Show/Hide
|
C20H27ClN2O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0475590
|
3-chloro-2,5,5-trimethyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C21H24ClF3N2O2
|
1
|
| 1 |
IC50 = 240 nM
|
|
|
|
CP0400920
|
ethyl 5-[3-(1H-benzimidazol-2-yl)propyl-methylamino]-2-phenyl-2-propan-2-ylpentanoate
Show/Hide
|
C27H37N3O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0431125
|
methyl 2-(4-bromophenyl)-5-[3-(6-methoxy-1H-benzimidazol-2-yl)propyl-methylamino]-2-propan-2-ylpentanoate
Show/Hide
|
C27H36BrN3O3
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0528909
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-(4-phenylbutyl)piperidine-4-carboxamide
Show/Hide
|
C28H39FN2O
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0396361
|
1-benzyl-4-(difluoromethyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C27H22F5N3O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0429392
|
4-(difluoromethyl)-1-methyl-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C21H18F5N3O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0429377
|
3-chloro-2,5,5-trimethyl-N-[[3-(2,2,2-trifluoroethoxy)pyridin-2-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C20H23ClF3N3O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0412202
|
2-[4-(dimethylamino)phenyl]-N-[1-[(2-methylphenyl)methyl]pyrazol-3-yl]acetamide
Show/Hide
|
C21H24N4O
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0396297
|
(3R,5S)-N-benzyl-3,5-dimethyl-1-phenyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H27N3O
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0090639
|
N-benzyl-2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide
Show/Hide
|
C39H45N5O
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
IC50 = 260.02 nM
|
|
|
|
CP0503532
|
ethyl 5-[4-[(4-fluorophenyl)methyl]piperazin-1-yl]-2-phenyl-2-propan-2-ylpentanoate
Show/Hide
|
C27H37FN2O2
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0508263
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-(2-phenoxyethyl)piperidine-4-carboxamide
Show/Hide
|
C26H35FN2O2
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0670565
|
N-benzyl-2-(3-(biphenyl-4-yl)-2-((5-(dimethylamino)pentyl)(methyl)amino)-3,4-dihydroquinazolin-4-yl)acetamide dihydrochloride
Show/Hide
|
C37H45Cl2N5O
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0870883
|
(+/-)-N-Benzyl-3,5-dimethyl-1-(phenylmethyl-d2)-1,2,3,5-tetrahydro-4H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H28N4O
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0475588
|
3-bromo-N-[[2-(methoxymethyl)phenyl]methyl]-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophene-1-carboxamide
Show/Hide
|
C20H24BrNO2S
|
1
|
| 1 |
IC50 = 260 nM
|
|
|
|
CP0396293
|
(3S,5R)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H29N3O
|
1
|
| 1 |
IC50 = 262 nM
|
|
|
|
CP0396284
|
(3S,5S)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C26H29N3O
|
1
|
| 1 |
IC50 = 279 nM
|
|
|
|
CP0373492
|
4-(4-(4-chlorobenzyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C21H24Cl3N3O
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0547181
|
methyl 2-(4-bromophenyl)-2-propan-2-yl-5-[4-[[3-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]pentanoate
Show/Hide
|
C27H34BrF3N2O2
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0398604
|
4-(4-Isopropylbenzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C31H38ClN3O
|
1
|
| 1 |
IC50 = 280 nM
|
|
|
|
CP0408587
|
4-bromo-1-methyl-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
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C20H17BrF3N3O2
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1
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| 1 |
IC50 = 280 nM
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CP0446025
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(3R,5S)-1-benzyl-8-bromo-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C24H25BrN4O
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1
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| 1 |
IC50 = 286 nM
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CP0382616
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(2S,5S)-N,1-dibenzyl-2,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C26H29N3O
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1
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| 1 |
IC50 = 293 nM
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CP0485975
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methyl 2-[3-(5-aminopentyl)-2-(4-phenylanilino)-4H-quinazolin-4-yl]acetate
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C28H32N4O2
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2
|
| 1 |
IC50 = 299.92 nM
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| 2 |
IC50 = 300 nM
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CP0382627
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(3R,5S)-N,1-dibenzyl-3,5-dimethyl-2-oxo-3,5-dihydro-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C26H27N3O2
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1
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| 1 |
IC50 = 304 nM
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CP0382626
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N,1-dibenzyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C24H25N3O
|
1
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| 1 |
IC50 = 305 nM
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CP0196973
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2-[2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide
Show/Hide
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C38H44N6O2
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1
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| 1 |
IC50 = 310 nM
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CP0538997
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N-benzyl-2-[2-[4-(dimethylamino)butyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide
Show/Hide
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C36H41N5O
|
1
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| 1 |
IC50 = 310 nM
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CP0482595
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3-chloro-2,6,6-trimethyl-N-[[2-(2-methylpropoxy)phenyl]methyl]-5,7-dihydro-4H-isoindole-1-carboxamide
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C23H31ClN2O2
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1
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| 1 |
IC50 = 310 nM
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CP0443299
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methyl 2-(4-bromophenyl)-2-propan-2-yl-5-[4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-1-yl]pentanoate
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C29H41BrN2O5
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1
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| 1 |
IC50 = 320 nM
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CP0396895
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1-[(3,4-dimethoxyphenyl)methyl]-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]piperidine-4-carboxamide
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C28H37FN2O3
|
1
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| 1 |
IC50 = 320 nM
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CP0538996
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2-[2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-fluorophenyl)methyl]acetamide
Show/Hide
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C37H41FN6O
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1
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| 1 |
IC50 = 320 nM
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CP0429373
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3-cyano-2,5,5-trimethyl-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
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C21H23F3N4O2
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1
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| 1 |
IC50 = 320 nM
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CP0486197
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(2R,4S)-3,3,9-trimethyl-N-[[2-(trifluoromethyl)phenyl]methyl]-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
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C20H20F3NOS
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1
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| 1 |
IC50 = 320 nM
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CP0536131
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(2R,4S)-3,3,9-trimethyl-N-[[3-(trifluoromethoxy)phenyl]methyl]-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
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C20H20F3NO2S
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1
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| 1 |
IC50 = 330 nM
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CP0429394
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1-benzyl-4-bromo-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
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C26H21BrF3N3O2
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1
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| 1 |
IC50 = 335 nM
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CP0372203
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methyl 2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetate
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C33H40N4O2
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2
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| 1 |
IC50 = 339.63 nM
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| 2 |
IC50 = 340 nM
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CP0431127
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ethyl 5-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-2-phenyl-2-propan-2-ylpentanoate
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C28H40N2O3
|
1
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| 1 |
IC50 = 340 nM
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CP0390395
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2-(2-(dimethylamino)-3-phenyl-3,4-dihydroquinazolin-4-yl)-N-(4-nitrobenzyl)acetamide
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C25H25N5O3
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2
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| 1 |
IC50 = 349.95 nM
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| 2 |
IC50 = 350 nM
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CP0389183
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tert-butyl 3-chloro-2-methyl-1-[[2-(2-methylpropoxy)phenyl]methylcarbamoyl]-4,6-dihydropyrrolo[3,4-c]pyrrole-5-carboxylate
Show/Hide
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C24H32ClN3O4
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1
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| 1 |
IC50 = 350 nM
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CP0507628
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1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-yl)-4-(isobutylamino)butan-1-one
Show/Hide
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C25H34ClN3O
|
1
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| 1 |
IC50 = 360 nM
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CP0477601
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(3R,5S)-1-benzyl-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
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C23H25N5O
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1
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| 1 |
IC50 = 360 nM
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CP0463421
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4-(difluoromethyl)-1-(3-fluorophenyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
Show/Hide
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C26H19F6N3O2
|
1
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| 1 |
IC50 = 360 nM
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CP0420024
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methyl 2-[3-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentyl]-2-(4-phenylanilino)-4H-quinazolin-4-yl]acetate
Show/Hide
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C33H40N4O4
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2
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| 1 |
IC50 = 369.83 nM
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| 2 |
IC50 = 370 nM
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CP0464415
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4-(4-(4-chlorobenzyl)piperazin-1-yl)-N-(4-chlorophenyl)butanamide
Show/Hide
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C21H25Cl2N3O
|
1
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| 1 |
IC50 = 370 nM
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CP0396896
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1-benzyl-N-[2-(4-fluorophenyl)-2-propylpentyl]piperidine-4-carboxamide
Show/Hide
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C27H37FN2O
|
1
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| 1 |
IC50 = 370 nM
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CP0382622
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(3R,5S)-1-benzyl-8-fluoro-7-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H27FN4O2
|
1
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| 1 |
IC50 = 370 nM
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CP0894010
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1-[4-(9H-Fluoren-9-yl)-piperazin-1-yl]-3,3-diphenyl-propan-1-one
Show/Hide
|
C32H30N2O
|
1
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| 1 |
IC50 = 371 nM
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CP0497857
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N-[(4-aminophenyl)methyl]-2-[2-(dimethylamino)-3-phenyl-4H-quinazolin-4-yl]acetamide
Show/Hide
|
C25H27N5O
|
1
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| 1 |
IC50 = 380 nM
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CP0534565
|
2,5,5-trimethyl-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]-3-(trifluoromethyl)-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C21H23F6N3O2
|
1
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| 1 |
IC50 = 380 nM
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CP0400919
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2-(4-Bromo-phenyl)-2-isopropyl-5-[4-(3-methyl-benzyl)-piperazin-1-yl]-pentanoic acid methyl ester
Show/Hide
|
C27H37BrN2O2
|
1
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| 1 |
IC50 = 390 nM
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CP0457424
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1-benzyl-N-[[1-(4-fluorophenyl)cyclobutyl]methyl]piperidine-4-carboxamide
Show/Hide
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C24H29FN2O
|
1
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| 1 |
IC50 = 390 nM
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CP0457359
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2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide
Show/Hide
|
C38H45N5O2
|
1
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| 1 |
IC50 = 390 nM
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CP0382581
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(3R,5S)-1-benzyl-7-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O2
|
1
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| 1 |
IC50 = 390 nM
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CP0934290
|
1-(4-Benzhydryl-piperazin-1-yl)-2-(9H-fluoren-9-yl)-ethanone
Show/Hide
|
C32H30N2O
|
1
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| 1 |
IC50 = 404 nM
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CP0389184
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4-(difluoromethyl)-5-phenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]-1-(2,2,2-trifluoroethyl)pyrazole-3-carboxamide
Show/Hide
|
C22H17F8N3O2
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1
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| 1 |
IC50 = 410 nM
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CP0398605
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1-(4-((4-Chlorophenyl)(phenyl)methyl)piperazin-1-yl)-4-(ethylamino)butan-1-one
Show/Hide
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C23H30ClN3O
|
1
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| 1 |
IC50 = 420 nM
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CP0382617
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benzyl (3R,5S)-1-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxylate
Show/Hide
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C26H28N2O2
|
1
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| 1 |
IC50 = 420 nM
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CP0504392
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2-[2-(dimethylamino)-3-phenyl-4H-quinazolin-4-yl]-N-[[4-[(4-fluorophenyl)sulfonylamino]phenyl]methyl]acetamide
Show/Hide
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C31H30FN5O3S
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1
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| 1 |
IC50 = 429.54 nM
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CP0446027
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(3R,5S)-1-[dideuterio(phenyl)methyl]-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C23H25N5O
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1
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| 1 |
IC50 = 441 nM
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CP0376226
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(3S,5S)-N-benzyl-5-[(4-chlorophenyl)methyl]-6-oxomorpholine-3-carboxamide
Show/Hide
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C19H19ClN2O3
|
1
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| 1 |
IC50 = 450 nM
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CP0446070
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(3R,5S)-N,1-dibenzyl-N,3,5-trimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C27H31N3O
|
1
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| 1 |
IC50 = 457 nM
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CP0433018
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2-[2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-methylphenyl)methyl]acetamide
Show/Hide
|
C38H44N6O
|
1
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| 1 |
IC50 = 460 nM
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CP0429371
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3-bromo-N-[[4-(methoxymethyl)phenyl]methyl]-5,5-dimethyl-6,7-dihydro-4H-2-benzothiophene-1-carboxamide
Show/Hide
|
C20H24BrNO2S
|
1
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| 1 |
IC50 = 460 nM
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CP0471731
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3-chloro-2,5,5-trimethyl-N-[[2-(3,3,3-trifluoropropoxy)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C22H26ClF3N2O2
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1
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| 1 |
IC50 = 460 nM
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CP0455948
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(3R,5S)-N-benzyl-3,5-dimethyl-1-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O
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1
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| 1 |
IC50 = 476 nM
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CP0494610
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methyl 2-(4-bromophenyl)-5-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C27H37BrN2O3
|
1
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| 1 |
IC50 = 480 nM
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CP0144570
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(2S)-1-[4-(3-methoxyphenyl)piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
|
C21H25F3N2O3
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1
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| 1 |
IC50 = 480 nM
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CP0471738
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3-chloro-2,5,5-trimethyl-N-[[2-(1,2,4-triazol-1-ylmethyl)phenyl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C22H26ClN5O
|
1
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| 1 |
IC50 = 480 nM
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CP0471814
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N-(1-benzylpyrazol-3-yl)-2-(2-methylphenyl)acetamide
Show/Hide
|
C19H19N3O
|
1
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| 1 |
IC50 = 490 nM
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CP0549582
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1-benzyl-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]piperidine-4-carboxamide
Show/Hide
|
C26H33FN2O
|
1
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| 1 |
IC50 = 510 nM
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CP0470835
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3-chloro-2,5,5-trimethyl-N-[[5-methyl-4-(pyrazol-1-ylmethyl)-1,2-oxazol-3-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C21H26ClN5O2
|
1
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| 1 |
IC50 = 510 nM
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CP0461373
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N-[[4-[bis(methylsulfonyl)amino]phenyl]methyl]-2-[2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide;hydrochloride
Show/Hide
|
C39H48ClN7O5S2
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1
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| 1 |
IC50 = 520 nM
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CP0450851
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3-bromo-5,5-dimethyl-N-[(2-propan-2-yloxyphenyl)methyl]-6,7-dihydro-4H-2-benzothiophene-1-carboxamide
Show/Hide
|
C21H26BrNO2S
|
1
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| 1 |
IC50 = 530 nM
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CP0471735
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(2R,4S)-3,3,9-trimethyl-N-[[3-(trifluoromethyl)phenyl]methyl]-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
|
C20H20F3NOS
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1
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| 1 |
IC50 = 540 nM
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CP0408655
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N-benzyl-2-[2-[6-(dimethylamino)hexyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetamide
Show/Hide
|
C38H45N5O
|
1
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| 1 |
IC50 = 550 nM
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CP0372201
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methyl 2-[2-(5-aminopentylimino)-3-(4-phenylphenyl)-1,4-dihydroquinazolin-4-yl]acetate
Show/Hide
|
C28H32N4O2
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2
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| 1 |
IC50 = 559.76 nM
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| 2 |
IC50 = 560 nM
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CP0504395
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tert-butyl N-[5-[[4-[2-(benzylamino)-2-oxoethyl]-3-phenyl-1,4-dihydroquinazolin-2-ylidene]amino]pentyl]carbamate
Show/Hide
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C33H41N5O3
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2
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| 1 |
IC50 = 570 nM
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| 2 |
IC50 = 570.16 nM
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CP0519761
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(3R,5S)-1-benzyl-3,5-dimethyl-4-(1-methylimidazol-4-yl)sulfonyl-3,5-dihydro-2H-1,4-benzodiazepine
Show/Hide
|
C22H26N4O2S
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1
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| 1 |
IC50 = 576 nM
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CP0396288
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(3R,5S)-1-benzyl-8-cyano-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H25N5O
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1
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| 1 |
IC50 = 582 nM
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CP0382582
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(3R,5S)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,2-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C25H28N4O
|
1
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| 1 |
IC50 = 597 nM
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CP0398606
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4-(4-Nitrobenzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C28H31ClN4O3
|
1
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| 1 |
IC50 = 600 nM
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CP0469337
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2-[2-[3-(dimethylcarbamoylamino)propyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-fluorophenyl)methyl]acetamide;hydrochloride
Show/Hide
|
C36H40ClFN6O2
|
1
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| 1 |
IC50 = 600 nM
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CP0486214
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(2R,4S)-N-[(2-chlorophenyl)methyl]-3,3,9-trimethyl-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
|
C19H20ClNOS
|
1
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| 1 |
IC50 = 600 nM
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CP0446023
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(3R,5S)-N-benzyl-3,5-dimethyl-1-(pyridin-2-ylmethyl)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O
|
1
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| 1 |
IC50 = 605 nM
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CP0444163
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(3R,5S)-3,5-dimethyl-1-(3-methylbutyl)-N-pyridin-3-yl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
Show/Hide
|
C21H29N5O
|
1
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| 1 |
IC50 = 613 nM
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CP0408320
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(3R,5S)-1-benzyl-8-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C25H28N4O2
|
1
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| 1 |
IC50 = 627 nM
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CP0461401
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2-(2-(dimethylamino)-3-phenyl-3,4-dihydroquinazolin-4-yl)-N-(4-(4-methylphenylsulfonamido)benzyl)acetamide
Show/Hide
|
C32H33N5O3S
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2
|
| 1 |
IC50 = 629.51 nM
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|
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| 2 |
IC50 = 630 nM
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CP0439136
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N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]-3-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]propan-1-amine
Show/Hide
|
C27H33F3N4O
|
1
|
| 1 |
IC50 = 650 nM
|
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CP0458312
|
methyl 2-(4-bromophenyl)-5-[4-(2-methoxyphenyl)piperazin-1-yl]-5-oxo-2-propan-2-ylpentanoate
Show/Hide
|
C26H33BrN2O4
|
1
|
| 1 |
IC50 = 654 nM
|
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CP0382628
|
(3R)-1-benzyl-3-methyl-4-(2-phenylethyl)-2,3-dihydro-1,4-benzodiazepin-5-one
Show/Hide
|
C25H26N2O
|
1
|
| 1 |
IC50 = 676 nM
|
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CP0421175
|
methyl 2-[2-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentylimino]-3-(4-phenylphenyl)-1,4-dihydroquinazolin-4-yl]acetate
Show/Hide
|
C33H40N4O4
|
2
|
| 1 |
IC50 = 679.2 nM
|
|
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| 2 |
IC50 = 680 nM
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CP0445464
|
2-[2-[6-(dimethylamino)hexyl-methylamino]-3-naphthalen-2-yl-4H-quinazolin-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide;hydrochloride
Show/Hide
|
C37H46ClN5O2
|
1
|
| 1 |
IC50 = 730 nM
|
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CP0400921
|
methyl 2-(4-bromophenyl)-5-[4-[(2-fluorophenyl)methyl]piperazin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
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C26H34BrFN2O2
|
1
|
| 1 |
IC50 = 740 nM
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CP0000413
|
1-[4-[bis(4-methoxyphenyl)methyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
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C34H36N2O3
|
1
|
| 1 |
IC50 = 745 nM
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CP0510802
|
4-(4-(3,4-dichlorobenzyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
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C21H23Cl4N3O
|
1
|
| 1 |
IC50 = 750 nM
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CP0531061
|
1-benzyl-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]-N-methylpiperidine-4-carboxamide
Show/Hide
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C27H35FN2O
|
1
|
| 1 |
IC50 = 750 nM
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CP0396295
|
(3R,5S)-N-benzyl-1-ethyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C21H27N3O
|
1
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| 1 |
IC50 = 754 nM
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CP0144569
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(2S)-1-[4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
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C21H23ClF4N2O2
|
1
|
| 1 |
IC50 = 760 nM
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CP0471732
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2,5,5-trimethyl-N-[[2-(2,2,2-trifluoroethoxy)pyridin-3-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C20H24F3N3O2
|
1
|
| 1 |
IC50 = 760 nM
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CP0472469
|
N-[2-ethyl-2-(4-fluorophenyl)butyl]-1-[2-(4-methoxyphenyl)ethyl]piperidine-4-carboxamide
Show/Hide
|
C27H37FN2O2
|
1
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| 1 |
IC50 = 770 nM
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CP0311384
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methyl 2-[[4-[3-(4-bromophenyl)-3-(4-fluorophenyl)propanoyl]piperazin-1-yl]methyl]-1,3-oxazole-4-carboxylate
Show/Hide
|
C25H25BrFN3O4
|
1
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| 1 |
IC50 = 860 nM
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CP0549584
|
N-(1-benzylpiperidin-4-yl)-2-[1-(4-fluorophenyl)cyclohexyl]acetamide
Show/Hide
|
C26H33FN2O
|
1
|
| 1 |
IC50 = 860 nM
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CP0510407
|
2-(3-ethyl-2-piperidin-1-yl-4H-quinazolin-4-yl)-N-[(4-nitrophenyl)methyl]acetamide
Show/Hide
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C24H29N5O3
|
1
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| 1 |
IC50 = 868.96 nM
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CP0408539
|
(2R,4S)-3,3,9-trimethyl-N-[(2-methylphenyl)methyl]-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
|
C20H23NOS
|
1
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| 1 |
IC50 = 870 nM
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CP0475698
|
(3R,5S)-3,5-dimethyl-1-(oxan-2-ylmethyl)-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
|
C23H30N4O2
|
1
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| 1 |
IC50 = 875 nM
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CP0494611
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methyl 5-[3-(6-methoxy-1H-benzimidazol-2-yl)propyl-methylamino]-2-(4-methoxyphenyl)-2-propan-2-ylpentanoate
Show/Hide
|
C28H39N3O4
|
1
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| 1 |
IC50 = 880 nM
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CP0373186
|
N-benzyl-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide
Show/Hide
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C28H30N4O
|
2
|
| 1 |
IC50 = 900 nM
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| 2 |
IC50 = 1160 nM
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CP0475591
|
3-chloro-2,5,5-trimethyl-N-[[3-(2,2,2-trifluoroethoxy)pyridin-4-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C20H23ClF3N3O2
|
1
|
| 1 |
IC50 = 910 nM
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CP0483098
|
N-(1-benzylpyrazol-3-yl)-1-(4-methoxyphenyl)cyclopropane-1-carboxamide
Show/Hide
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C21H21N3O2
|
1
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| 1 |
IC50 = 920 nM
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CP0906036
|
2-(4-chlorobenzyl)-N-(3-(2-methylpiperidin-1-yl)propyl)-1,3-dioxoisoindoline-5-carboxamide hydrochloride
Show/Hide
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C25H29Cl2N3O3
|
1
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| 1 |
IC50 = 930 nM
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CP0373356
|
2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazolin-4-yl)-N-(4-(4-methylphenylsulfonamido)benzyl)acetamide
Show/Hide
|
C31H37N5O3S
|
2
|
| 1 |
IC50 = 959.4 nM
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| 2 |
IC50 = 960 nM
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CP0943785
|
2-(4-chlorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
Show/Hide
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C23H25Cl2N3O3
|
1
|
| 1 |
IC50 = 960 nM
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CP0517063
|
methyl 2-(4-bromophenyl)-5-[4-[(3-fluorophenyl)methyl]piperazin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C26H34BrFN2O2
|
1
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| 1 |
IC50 = 980 nM
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CP0376203
|
(3S,5S)-N-benzyl-6-oxo-5-propan-2-ylmorpholine-3-carboxamide
Show/Hide
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C15H20N2O3
|
1
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| 1 |
IC50 = 990 nM
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CP0450867
|
(2R,4S)-3,3,9-trimethyl-N-[(4-methylphenyl)methyl]-8-thiatricyclo[4.3.0.02,4]nona-1(9),6-diene-7-carboxamide
Show/Hide
|
C20H23NOS
|
1
|
| 1 |
IC50 = 1000 nM
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CP0344603
|
(2S)-2-(2,4-dihydroxyphenyl)-5,7-dihydroxy-8-[(2R)-5-methyl-2-(prop-1-en-2-yl)hex-4-en-1-yl]-2,3-dihydro-4H-chromen-4-one
Show/Hide
|
C25H28O6
|
1
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| 1 |
IC50 = 1000 nM
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CP0450628
|
(2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-8-(3-methylbut-2-en-1-yl)-3,4-dihydro-2H-1-benzopyran-4-one
Show/Hide
|
C20H20O5
|
1
|
| 1 |
IC50 = 1000 nM
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CP0538721
|
2-(4-hydroxyphenyl)-6-(3-methylbut-2-enyl)-5,7-bis(oxidanyl)-2,3-dihydrochromen-4-one
Show/Hide
|
C20H20O5
|
1
|
| 1 |
IC50 = 1000 nM
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CP0390360
|
2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)-N-thiophen-2-ylsulfonylacetamide
Show/Hide
|
C25H26N4O3S2
|
1
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| 1 |
IC50 = 1009.25 nM
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CP0464413
|
4-(4-(3-chlorophenyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C20H22Cl3N3O
|
1
|
| 1 |
IC50 = 1010 nM
|
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CP0490485
|
5-(4-(3,4-dichlorobenzyl)piperazin-1-yl)-N-(2-chlorophenyl)pentanamide
Show/Hide
|
C22H26Cl3N3O
|
1
|
| 1 |
IC50 = 1010 nM
|
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CP0376234
|
(3S,5S)-N,5-dibenzyl-6-oxomorpholine-3-carboxamide
Show/Hide
|
C19H20N2O3
|
1
|
| 1 |
IC50 = 1010 nM
|
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CP0531908
|
N-[[3-[2-(trifluoromethyl)phenyl]-1,2-oxazol-5-yl]methyl]-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine
Show/Hide
|
C24H24F6N4O
|
1
|
| 1 |
IC50 = 1020 nM
|
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CP0373598
|
4-(2,6-Dichlorobenzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C28H30Cl3N3O
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
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CP0373357
|
2-(3-ethyl-2-(piperidin-1-yl)-3,4-dihydroquinazolin-4-yl)-N-(4-(4-fluorophenylsulfonamido)benzyl)acetamide
Show/Hide
|
C30H34FN5O3S
|
2
|
| 1 |
IC50 = 1039.92 nM
|
|
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| 2 |
IC50 = 1040 nM
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CP0469338
|
N-benzyl-2-[3-(4-cyclohexylphenyl)-2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-4H-quinazolin-4-yl]acetamide;hydrochloride
Show/Hide
|
C37H49ClN6O
|
1
|
| 1 |
IC50 = 1040 nM
|
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CP0127762
|
(2S)-1-(4-chlorophenoxy)-3-[4-[(4-chlorophenyl)methyl]piperazin-1-yl]propan-2-ol
Show/Hide
|
C20H24Cl2N2O2
|
1
|
| 1 |
IC50 = 1080 nM
|
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CP0099020
|
3-(4-chlorobenzyl)-N-(3-(4-methylpiperidin-1-yl)propyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C25H29ClN4O2S
|
1
|
| 1 |
IC50 = 1100 nM
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CP0431126
|
methyl 2-(4-bromophenyl)-5-[4-[(4-fluorophenyl)methyl]piperazin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C26H34BrFN2O2
|
1
|
| 1 |
IC50 = 1110 nM
|
|
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CP0485245
|
2-[2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[[4-[(4-methylphenyl)sulfonylamino]phenyl]methyl]acetamide
Show/Hide
|
C28H33N5O3S
|
1
|
| 1 |
IC50 = 1119.44 nM
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CP0467237
|
(3S,5S)-N-benzyl-5-[(4-nitrophenyl)methyl]-6-oxomorpholine-3-carboxamide
Show/Hide
|
C19H19N3O5
|
1
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| 1 |
IC50 = 1130 nM
|
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CP0519502
|
(5S,7R)-N,9-dibenzyl-5,7-dimethyl-7,8-dihydro-5H-pyridazino[3,4-e][1,4]diazepine-6-carboxamide
Show/Hide
|
C24H27N5O
|
1
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| 1 |
IC50 = 1139 nM
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CP0486053
|
N-(1-benzylpyrazol-3-yl)-2-phenylacetamide
Show/Hide
|
C18H17N3O
|
1
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| 1 |
IC50 = 1140 nM
|
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CP0389181
|
3,5-dichloro-4-cyclopropyl-1-methyl-N-[[2-(2-methylpropoxy)phenyl]methyl]pyrrole-2-carboxamide
Show/Hide
|
C20H24Cl2N2O2
|
1
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| 1 |
IC50 = 1150 nM
|
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CP0464384
|
3-(4-chlorobenzyl)-4-oxo-N-(3-(pyrrolidin-1-yl)propyl)-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C23H25ClN4O2S
|
1
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| 1 |
IC50 = 1160 nM
|
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CP0487830
|
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]propan-1-amine
Show/Hide
|
C27H36N4O
|
1
|
| 1 |
IC50 = 1190 nM
|
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CP0373364
|
tert-butyl N-[5-[2-anilino-4-[2-(benzylamino)-2-oxoethyl]-4H-quinazolin-3-yl]pentyl]carbamate
Show/Hide
|
C33H41N5O3
|
1
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| 1 |
IC50 = 1199.5 nM
|
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CP0505874
|
1-(1-benzylpiperidin-4-yl)-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]methanamine
Show/Hide
|
C26H35FN2
|
1
|
| 1 |
IC50 = 1200 nM
|
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CP0549583
|
1-benzyl-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]piperidine-3-carboxamide
Show/Hide
|
C26H33FN2O
|
1
|
| 1 |
IC50 = 1200 nM
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CP0456439
|
(3S,5S)-N-benzyl-5-butan-2-yl-6-oxomorpholine-3-carboxamide
Show/Hide
|
C16H22N2O3
|
1
|
| 1 |
IC50 = 1220 nM
|
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CP0096004
|
2-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-N-(4-(trifluoromethyl)phenyl)acetamide
Show/Hide
|
C22H24F3N5O
|
1
|
| 1 |
IC50 = 1230 nM
|
|
|
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CP0368241
|
(2R)-1-[4-[(3,4-dichlorophenyl)methyl]piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
|
C21H23Cl2F3N2O2
|
1
|
| 1 |
IC50 = 1270 nM
|
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CP0055685
|
3-(4-fluorophenyl)-1-(4-((6-methylbenzo[d]oxazol-2-yl)methyl)piperazin-1-yl)-3-phenylpropan-1-one
Show/Hide
|
C28H28FN3O2
|
1
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| 1 |
IC50 = 1290 nM
|
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CP0487800
|
N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]-2-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine
Show/Hide
|
C26H31F3N4O
|
1
|
| 1 |
IC50 = 1300 nM
|
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CP0400141
|
3-(4-(4-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C26H33ClN4O
|
1
|
| 1 |
IC50 = 1310 nM
|
|
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CP0467239
|
(3R,5S)-5-[(4-chlorophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]morpholine-3-carboxamide
Show/Hide
|
C20H21ClN2O3
|
1
|
| 1 |
IC50 = 1330 nM
|
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CP0458666
|
5-[3-(1H-benzimidazol-2-yl)propyl-methylamino]-2-(4-bromophenyl)-2-propan-2-ylpentanoic acid
Show/Hide
|
C25H32BrN3O2
|
1
|
| 1 |
IC50 = 1360 nM
|
|
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CP0441800
|
(3S,5S)-5-[(4-hydroxyphenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]morpholine-3-carboxamide
Show/Hide
|
C20H22N2O4
|
1
|
| 1 |
IC50 = 1390 nM
|
|
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CP0389208
|
2-[4-(dimethylamino)phenyl]-N-(1-phenylpyrazol-3-yl)acetamide
Show/Hide
|
C19H20N4O
|
1
|
| 1 |
IC50 = 1400 nM
|
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CP0511052
|
3-(4-chlorobenzyl)-N-(3-(azepan-1-yl)propyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C25H29ClN4O2S
|
1
|
| 1 |
IC50 = 1410 nM
|
|
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CP0284837
|
(2S)-1-[4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl]-3-(4-chlorophenoxy)propan-2-ol
Show/Hide
|
C20H23Cl2FN2O2
|
1
|
| 1 |
IC50 = 1420 nM
|
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CP0489476
|
2-(4-(3-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H31ClN4O
|
1
|
| 1 |
IC50 = 1450 nM
|
|
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CP0372256
|
2-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-N-(2-chlorophenyl)acetamide
Show/Hide
|
C21H24ClN5O
|
1
|
| 1 |
IC50 = 1470 nM
|
|
|
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CP0373493
|
4-(4-(3-chlorobenzyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C21H24Cl3N3O
|
1
|
| 1 |
IC50 = 1480 nM
|
|
|
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CP0441795
|
(3R,5S)-5-[(4-fluorophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]morpholine-3-carboxamide
Show/Hide
|
C20H21FN2O3
|
1
|
| 1 |
IC50 = 1480 nM
|
|
|
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CP0897230
|
2-(2-chlorobenzyl)-N-(3-(2-methylpiperidin-1-yl)propyl)-1,3-dioxoisoindoline-5-carboxamide hydrochloride
Show/Hide
|
C25H29Cl2N3O3
|
1
|
| 1 |
IC50 = 1520 nM
|
|
|
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CP0505345
|
2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-(trifluoromethyl)phenyl)isoxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H29F3N4O
|
1
|
| 1 |
IC50 = 1530 nM
|
|
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CP0493048
|
4-(2-Ethylbutylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C27H38ClN3O
|
1
|
| 1 |
IC50 = 1540 nM
|
|
|
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CP0322288
|
(2S)-1-[4-[(4-chlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
|
C20H24ClFN2O2
|
1
|
| 1 |
IC50 = 1560 nM
|
|
|
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CP0453053
|
(3S,5S)-5-[(4-chlorophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]morpholine-3-carboxamide
Show/Hide
|
C20H21ClN2O3
|
1
|
| 1 |
IC50 = 1610 nM
|
|
|
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CP0904316
|
2-(4-chlorobenzyl)-1,3-dioxo-N-(3-(pyrrolidin-1-yl)propyl)isoindoline-5-carboxamide hydrochloride
Show/Hide
|
C23H25Cl2N3O3
|
1
|
| 1 |
IC50 = 1620 nM
|
|
|
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CP0373490
|
4-(4-(benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C22H25Cl2N3O3
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
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CP0411904
|
4-(Benzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)-butan-1-one
Show/Hide
|
C28H32ClN3O
|
1
|
| 1 |
IC50 = 1670 nM
|
|
|
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CP0487801
|
2-(4-(2,3-dimethylphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C27H36N4O
|
1
|
| 1 |
IC50 = 1710 nM
|
|
|
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CP0332364
|
methyl 2-[[4-[3-(4-fluorophenyl)-3-[4-(trifluoromethyl)phenyl]propanoyl]piperazin-1-yl]methyl]-1,3-oxazole-4-carboxylate
Show/Hide
|
C26H25F4N3O4
|
1
|
| 1 |
IC50 = 1730 nM
|
|
|
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CP0452341
|
3-(4-(3-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C26H33ClN4O
|
1
|
| 1 |
IC50 = 1750 nM
|
|
|
|
CP0504250
|
3-(4-(2,3-dimethylphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C28H38N4O
|
1
|
| 1 |
IC50 = 1780 nM
|
|
|
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CP0144571
|
(2R)-1-[4-(2-methoxyphenyl)piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
|
C21H25F3N2O3
|
1
|
| 1 |
IC50 = 1790 nM
|
|
|
|
CP0405418
|
4-(4-(3-chlorobenzyl)piperazin-1-yl)-N-(4-chlorophenyl)butanamide
Show/Hide
|
C21H25Cl2N3O
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0920185
|
2-(3-chlorobenzyl)-N-(3-(2-methylpiperidin-1-yl)propyl)-1,3-dioxoisoindoline-5-carboxamide hydrochloride
Show/Hide
|
C25H29Cl2N3O3
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0373489
|
5-(4-(4-chlorobenzyl)piperazin-1-yl)-1-(4-(2-fluorophenyl)piperazin-1-yl)pentan-1-one
Show/Hide
|
C26H34ClFN4O
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0445463
|
benzyl 2-[2-[4-[2-(dimethylamino)ethyl]piperazin-1-yl]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]acetate
Show/Hide
|
C37H41N5O2
|
1
|
| 1 |
IC50 = 1810 nM
|
|
|
|
CP0918657
|
2-(3-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid [3-(2-methyl-piperidin-1-yl)-propyl]-amide hydrochloride
Show/Hide
|
C26H32ClN3O3
|
1
|
| 1 |
IC50 = 1840 nM
|
|
|
|
CP0510408
|
methyl 2-[2-(5-aminopentylimino)-3-phenyl-1,4-dihydroquinazolin-4-yl]acetate
Show/Hide
|
C22H28N4O2
|
1
|
| 1 |
IC50 = 1840.77 nM
|
|
|
|
CP0467248
|
(3S,5S)-N-benzyl-5-(2-methylsulfanylethyl)-6-oxomorpholine-3-carboxamide
Show/Hide
|
C15H20N2O3S
|
1
|
| 1 |
IC50 = 1860 nM
|
|
|
|
CP0433685
|
N-(2-chlorophenyl)-5-[4-(3-chlorophenyl)piperazin-1-yl]pentanamide
Show/Hide
|
C21H25Cl2N3O
|
1
|
| 1 |
IC50 = 1910 nM
|
|
|
|
CP0886006
|
2-(3-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid (2-piperidin-1-yl-ethyl)-amide hydrochloride
Show/Hide
|
C24H28ClN3O3
|
1
|
| 1 |
IC50 = 1930 nM
|
|
|
|
CP0400135
|
N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine
Show/Hide
|
C26H31F3N4O
|
1
|
| 1 |
IC50 = 1940 nM
|
|
|
|
CP0512493
|
1-(1-benzylpiperidin-4-yl)-3-[1-(4-fluorophenyl)cyclohexyl]propan-1-one
Show/Hide
|
C27H34FNO
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0429851
|
methyl 2-[2-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentylimino]-3-phenyl-1,4-dihydroquinazolin-4-yl]acetate
Show/Hide
|
C27H36N4O4
|
1
|
| 1 |
IC50 = 2018.37 nM
|
|
|
|
CP0560308
|
2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((3-(2-methoxyphenyl)isoxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H32N4O2
|
1
|
| 1 |
IC50 = 2020 nM
|
|
|
|
CP0920184
|
2-(4-fluorobenzyl)-N-(3-(2-methylpiperidin-1-yl)propyl)-1,3-dioxoisoindoline-5-carboxamide hydrochloride
Show/Hide
|
C25H29ClFN3O3
|
1
|
| 1 |
IC50 = 2030 nM
|
|
|
|
CP0511051
|
N-[[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl]-2-[4-[3-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine
Show/Hide
|
C24H27F3N4O2
|
1
|
| 1 |
IC50 = 2040 nM
|
|
|
|
CP0467247
|
(3S,5S)-N-benzyl-5-[(4-methoxyphenyl)methyl]-6-oxomorpholine-3-carboxamide
Show/Hide
|
C20H22N2O4
|
1
|
| 1 |
IC50 = 2040 nM
|
|
|
|
CP0933152
|
2-(2-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid [3-(2-methyl-piperidin-1-yl)-propyl]-amide hydrochloride
Show/Hide
|
C26H32ClN3O3
|
1
|
| 1 |
IC50 = 2070 nM
|
|
|
|
CP0484902
|
3-(4-chlorobenzyl)-4-oxo-N-(3-(piperidin-1-yl)propyl)-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C24H27ClN4O2S
|
1
|
| 1 |
IC50 = 2080 nM
|
|
|
|
CP0477532
|
2-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-N-(2,6-diethylphenyl)acetamide
Show/Hide
|
C25H33N5O
|
1
|
| 1 |
IC50 = 2080 nM
|
|
|
|
CP0489479
|
N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]-2-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]ethanamine
Show/Hide
|
C26H31F3N4O
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0427132
|
(2R)-1-[4-[(3-chlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
|
C20H24ClFN2O2
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0429387
|
(2S,4R)-N-[(2-methoxyphenyl)methyl]-3,3,9-trimethyl-8,9-diazatricyclo[4.3.0.02,4]nona-1(6),7-diene-7-carboxamide
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
IC50 = 2100 nM
|
|
|
|
CP0441794
|
(3S,5S)-5-[(4-nitrophenyl)methyl]-6-oxo-N-[(1S)-1-phenylethyl]morpholine-3-carboxamide
Show/Hide
|
C20H21N3O5
|
1
|
| 1 |
IC50 = 2130 nM
|
|
|
|
CP0542728
|
2-[2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[(4-nitrophenyl)methyl]acetamide
Show/Hide
|
C21H25N5O3
|
1
|
| 1 |
IC50 = 2167.7 nM
|
|
|
|
CP0464575
|
(3S,5S)-5-benzyl-N-cyclohexyl-6-oxomorpholine-3-carboxamide
Show/Hide
|
C18H24N2O3
|
1
|
| 1 |
IC50 = 2180 nM
|
|
|
|
CP0531060
|
1-benzyl-N-[[4-(4-fluorophenyl)oxan-4-yl]methyl]piperidine-4-carboxamide
Show/Hide
|
C25H31FN2O2
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0452339
|
2-(4-(3,4-dimethylphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C27H36N4O
|
1
|
| 1 |
IC50 = 2220 nM
|
|
|
|
CP0489477
|
2-(4-(2,4-dimethylphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C27H36N4O
|
1
|
| 1 |
IC50 = 2220 nM
|
|
|
|
CP0504394
|
methyl 2-[2-anilino-3-[5-[(2-methylpropan-2-yl)oxycarbonylamino]pentyl]-4H-quinazolin-4-yl]acetate
Show/Hide
|
C27H36N4O4
|
1
|
| 1 |
IC50 = 2269.86 nM
|
|
|
|
CP0406217
|
4-(4-(Dimethylamino)benzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C30H37ClN4O
|
1
|
| 1 |
IC50 = 2320 nM
|
|
|
|
CP0401627
|
2-(7-amino-3-phenyl-2-(piperidin-1-yl)-3,4-dihydroquinazolin-4-yl)-N-(4-nitrobenzyl)acetamide
Show/Hide
|
C28H29N5O3
|
2
|
| 1 |
IC50 = 2338.84 nM
|
|
|
| 2 |
IC50 = 2500 nM
|
|
|
|
CP0455786
|
3-chloro-N-[[3-[(3S)-3-fluoropyrrolidin-1-yl]pyridin-2-yl]methyl]-2,5,5-trimethyl-6,7-dihydro-4H-isoindole-1-carboxamide
Show/Hide
|
C22H28ClFN4O
|
1
|
| 1 |
IC50 = 2360 nM
|
|
|
|
CP0411274
|
2-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-N-(3,4-dimethylphenyl)acetamide
Show/Hide
|
C23H29N5O
|
1
|
| 1 |
IC50 = 2390 nM
|
|
|
|
CP0427580
|
4-(4-(2-chloro-6-fluorobenzyl)piperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C21H23Cl3FN3O
|
1
|
| 1 |
IC50 = 2400 nM
|
|
|
|
CP0464412
|
5-(4-(3-chlorobenzyl)piperazin-1-yl)-1-(4-(2-fluorophenyl)piperazin-1-yl)pentan-1-one
Show/Hide
|
C26H34ClFN4O
|
1
|
| 1 |
IC50 = 2440 nM
|
|
|
|
CP0370654
|
3-(4-methoxyphenyl)-1-(4-((6-methylbenzo[d]oxazol-2-yl)methyl)piperazin-1-yl)-3-phenylpropan-1-one
Show/Hide
|
C29H31N3O3
|
1
|
| 1 |
IC50 = 2480 nM
|
|
|
|
CP0433659
|
3-(4-chlorobenzyl)-N-(3-(4-ethylpiperazin-1-yl)propyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C25H30ClN5O2S
|
1
|
| 1 |
IC50 = 2530 nM
|
|
|
|
CP0417564
|
(2S)-1-[4-[(3-chlorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
|
C20H24ClFN2O2
|
1
|
| 1 |
IC50 = 2580 nM
|
|
|
|
CP0433687
|
N-(4-chlorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]butanamide
Show/Hide
|
C21H26ClN3O2
|
1
|
| 1 |
IC50 = 2610 nM
|
|
|
|
CP0405419
|
N-(4-chlorophenyl)-4-[4-(4-chlorophenyl)piperazin-1-yl]butanamide
Show/Hide
|
C20H23Cl2N3O
|
1
|
| 1 |
IC50 = 2640 nM
|
|
|
|
CP0432629
|
methyl 2-(4-bromophenyl)-5-[4-(2-methoxyphenyl)piperidin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C27H36BrNO3
|
1
|
| 1 |
IC50 = 2650 nM
|
|
|
|
CP0373494
|
4-(4-(benzo[d][1,3]dioxol-5-ylmethyl)piperazin-1-yl)-N-(4-chlorophenyl)butanamide
Show/Hide
|
C22H26ClN3O3
|
1
|
| 1 |
IC50 = 2730 nM
|
|
|
|
CP0391004
|
(3S,5S)-N-benzyl-5-[(4-fluorophenyl)methyl]-6-oxomorpholine-3-carboxamide
Show/Hide
|
C19H19FN2O3
|
1
|
| 1 |
IC50 = 2750 nM
|
|
|
|
CP0373497
|
N-(4-chlorophenyl)-4-[4-(3-methoxyphenyl)piperazin-1-yl]butanamide
Show/Hide
|
C21H26ClN3O2
|
1
|
| 1 |
IC50 = 2780 nM
|
|
|
|
CP0400140
|
3-(4-(2-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C26H33ClN4O
|
1
|
| 1 |
IC50 = 2800 nM
|
|
|
|
CP0400129
|
2-(4-(4-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H31ClN4O
|
1
|
| 1 |
IC50 = 2820 nM
|
|
|
|
CP0427693
|
5-(4-(3,4-dichlorobenzyl)piperazin-1-yl)-1-(4-phenylpiperazin-1-yl)pentan-1-one
Show/Hide
|
C26H34Cl2N4O
|
1
|
| 1 |
IC50 = 2910 nM
|
|
|
|
CP0531059
|
1-benzyl-N-[[1-(4-fluorophenyl)cyclohexyl]methyl]piperidine-2-carboxamide
Show/Hide
|
C26H33FN2O
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0487832
|
3-(4-(3,4-dimethylphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C28H38N4O
|
1
|
| 1 |
IC50 = 3020 nM
|
|
|
|
CP0501983
|
3-(4-(3-fluorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C26H33FN4O
|
1
|
| 1 |
IC50 = 3030 nM
|
|
|
|
CP0429831
|
2-[2-(5-aminopentylimino)-3-phenyl-1,4-dihydroquinazolin-4-yl]-N-benzylacetamide
Show/Hide
|
C28H33N5O
|
1
|
| 1 |
IC50 = 3126.08 nM
|
|
|
|
CP0427695
|
4-(4-benzylpiperazin-1-yl)-N-(2,4-dichlorophenyl)butanamide
Show/Hide
|
C21H25Cl2N3O
|
1
|
| 1 |
IC50 = 3140 nM
|
|
|
|
CP0325332
|
1-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-2-(2-(trifluoromethyl)phenylamino)ethanone
Show/Hide
|
C22H24F3N5O
|
1
|
| 1 |
IC50 = 3170 nM
|
|
|
|
CP0487829
|
3-(4-(4-fluorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
|
C26H33FN4O
|
1
|
| 1 |
IC50 = 3210 nM
|
|
|
|
CP0525389
|
methyl 2-(4-bromophenyl)-5-[4-(2-methoxyphenyl)-3,6-dihydro-2H-pyridin-1-yl]-2-propan-2-ylpentanoate
Show/Hide
|
C27H34BrNO3
|
1
|
| 1 |
IC50 = 3240 nM
|
|
|
|
CP0458665
|
2-(4-bromophenyl)-5-[4-(2-methoxyphenyl)piperazin-1-yl]-2-propan-2-ylpentanoic acid
Show/Hide
|
C25H33BrN2O3
|
1
|
| 1 |
IC50 = 3260 nM
|
|
|
|
CP0427697
|
4-(4-(2-chloro-6-fluorobenzyl)piperazin-1-yl)-N-(4-chlorophenyl)butanamide
Show/Hide
|
C21H24Cl2FN3O
|
1
|
| 1 |
IC50 = 3270 nM
|
|
|
|
CP0433686
|
N-(2,4-dichlorophenyl)-4-[4-(2-methoxyphenyl)piperazin-1-yl]butanamide
Show/Hide
|
C21H25Cl2N3O2
|
1
|
| 1 |
IC50 = 3340 nM
|
|
|
|
CP0400127
|
2-(4-(3-fluorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H31FN4O
|
1
|
| 1 |
IC50 = 3350 nM
|
|
|
|
CP0427574
|
5-(4-(4-chlorobenzyl)piperazin-1-yl)-1-(4-phenylpiperazin-1-yl)pentan-1-one
Show/Hide
|
C26H35ClN4O
|
1
|
| 1 |
IC50 = 3400 nM
|
|
|
|
CP0465239
|
N-(4-chlorophenyl)-4-[4-(4-fluorophenyl)piperazin-1-yl]butanamide
Show/Hide
|
C20H23ClFN3O
|
1
|
| 1 |
IC50 = 3490 nM
|
|
|
|
CP0373495
|
4-(4-benzylpiperazin-1-yl)-N-(4-chlorophenyl)butanamide
Show/Hide
|
C21H26ClN3O
|
1
|
| 1 |
IC50 = 3520 nM
|
|
|
|
CP0939740
|
2-(4-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid [3-(2-methyl-piperidin-1-yl)-propyl]-amide hydrochloride
Show/Hide
|
C26H32ClN3O3
|
1
|
| 1 |
IC50 = 3530 nM
|
|
|
|
CP0439449
|
N-(4-chlorophenyl)-4-[4-(2-fluorophenyl)piperazin-1-yl]butanamide
Show/Hide
|
C20H23ClFN3O
|
1
|
| 1 |
IC50 = 3630 nM
|
|
|
|
CP0471734
|
4-chloro-5-methyl-N-[[2-(2-methylpropoxy)phenyl]methyl]-2,3-dihydro-1H-pyrrolo[3,4-c]pyrrole-6-carboxamide
Show/Hide
|
C19H24ClN3O2
|
1
|
| 1 |
IC50 = 3700 nM
|
|
|
|
CP0501630
|
4-amino-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
|
C21H26ClN3O
|
1
|
| 1 |
IC50 = 3710 nM
|
|
|
|
CP0373499
|
N-(2,4-dichlorophenyl)-4-[4-(3-methoxyphenyl)piperazin-1-yl]butanamide
Show/Hide
|
C21H25Cl2N3O2
|
1
|
| 1 |
IC50 = 3810 nM
|
|
|
|
CP0401802
|
1-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-2-(2,6-diethylphenylamino)ethanone
Show/Hide
|
C25H33N5O
|
1
|
| 1 |
IC50 = 4000 nM
|
|
|
|
CP0918650
|
2-(3-chlorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
Show/Hide
|
C23H25Cl2N3O3
|
1
|
| 1 |
IC50 = 4090 nM
|
|
|
|
CP0477656
|
2-[2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[[4-[(4-fluorophenyl)sulfonylamino]phenyl]methyl]acetamide
Show/Hide
|
C27H30FN5O3S
|
1
|
| 1 |
IC50 = 4102.04 nM
|
|
|
|
CP0373259
|
N-benzyl-2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-phenyl-4H-quinazolin-4-yl]acetamide
Show/Hide
|
C33H41N5O
|
2
|
| 1 |
IC50 = 4197.59 nM
|
|
|
| 2 |
IC50 = 4200 nM
|
|
|
|
CP0427575
|
N-(2,4-dichlorophenyl)-4-(4-phenylpiperazin-1-yl)butanamide
Show/Hide
|
C20H23Cl2N3O
|
1
|
| 1 |
IC50 = 4210 nM
|
|
|
|
CP0566000
|
(2S)-1-[4-[(4-chlorophenyl)methyl]piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
|
C21H24ClF3N2O2
|
1
|
| 1 |
IC50 = 4230 nM
|
|
|
|
CP0439137
|
2-[4-(2-methylphenyl)piperazin-1-yl]-N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]ethanamine
Show/Hide
|
C26H34N4O
|
1
|
| 1 |
IC50 = 4300 nM
|
|
|
|
CP0501962
|
2-(4-(2-chlorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
Show/Hide
|
C25H31ClN4O
|
1
|
| 1 |
IC50 = 4370 nM
|
|
|
|
CP0373498
|
N-(4-chlorophenyl)-4-(4-phenylpiperazin-1-yl)butanamide
Show/Hide
|
C20H24ClN3O
|
1
|
| 1 |
IC50 = 4470 nM
|
|
|
|
CP0485427
|
2-[3-(5-aminopentyl)-2-anilino-4H-quinazolin-4-yl]-N-benzylacetamide
Show/Hide
|
C28H33N5O
|
1
|
| 1 |
IC50 = 4539.42 nM
|
|
|
|
CP0381851
|
N-benzyl-2-(3-ethyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide
Show/Hide
|
C24H30N4O
|
1
|
| 1 |
IC50 = 4581.42 nM
|
|
|
|
CP0467094
|
3-(4-chlorobenzyl)-N-(3-(benzyl(methyl)amino)propyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
|
C27H27ClN4O2S
|
1
|
| 1 |
IC50 = 4690 nM
|
|
|
|
CP0900128
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2-(4-methoxybenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
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C24H28ClN3O4
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1
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| 1 |
IC50 = 5250 nM
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CP0412197
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2-[4-(dimethylamino)phenyl]-N-[1-[[4-(2-oxopyrrolidin-1-yl)phenyl]methyl]pyrazol-3-yl]acetamide
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C24H27N5O2
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1
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| 1 |
IC50 = 5700 nM
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CP0936779
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2-(4-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid (2-piperidin-1-yl-ethyl)-amide hydrochloride
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C24H28ClN3O3
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1
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| 1 |
IC50 = 5820 nM
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CP0939738
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2-(2-chlorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
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C23H25Cl2N3O3
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1
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| 1 |
IC50 = 5820 nM
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CP0372202
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methyl 2-[2-[methyl(5-pyrrolidin-1-ylpentyl)amino]-3-phenyl-4H-quinazolin-4-yl]acetate
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C27H36N4O2
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2
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| 1 |
IC50 = 5834.45 nM
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| 2 |
IC50 = 5840 nM
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CP0500873
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N-(4-chlorophenyl)-4-[4-(2-chlorophenyl)piperazin-1-yl]butanamide
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C20H23Cl2N3O
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1
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| 1 |
IC50 = 6010 nM
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CP0382619
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(3R,5S)-1-benzoyl-N-benzyl-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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C26H27N3O2
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1
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| 1 |
IC50 = 6070 nM
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CP0382577
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(3R,5S)-1-benzyl-3,5-dimethyl-4-(oxan-4-ylmethyl)-3,5-dihydro-2H-1,4-benzodiazepine
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C24H32N2O
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1
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| 1 |
IC50 = 6110 nM
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CP0382635
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(3R,5S)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[4,3-e][1,4]diazepine-4-carboxamide
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C25H28N4O
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1
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| 1 |
IC50 = 6280 nM
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CP0501961
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2-(4-(4-fluorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
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C25H31FN4O
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1
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| 1 |
IC50 = 7080 nM
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CP0487831
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N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]-3-[4-[4-(trifluoromethyl)phenyl]piperazin-1-yl]propan-1-amine
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C27H33F3N4O
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1
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| 1 |
IC50 = 7250 nM
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CP0501985
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2-(4-benzhydrylpiperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
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C32H38N4O
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1
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| 1 |
IC50 = 7470 nM
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CP0933148
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2-(2-methyl-benzyl)-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid (2-piperidin-1-yl-ethyl)-amide hydrochloride
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C24H28ClN3O3
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1
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| 1 |
IC50 = 8280 nM
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CP0933151
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2-(3-fluorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
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C23H25ClFN3O3
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1
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| 1 |
IC50 = 8520 nM
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CP0489480
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3-[4-(2-methylphenyl)piperazin-1-yl]-N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]propan-1-amine
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C27H36N4O
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1
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| 1 |
IC50 = 8750 nM
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CP0412116
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methyl 2-[[4-[3-(4-chlorophenyl)-3-(4-fluorophenyl)propanoyl]piperazin-1-yl]methyl]-1,3-oxazole-4-carboxylate
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C25H25ClFN3O4
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1
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| 1 |
IC50 = 8800 nM
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CP0939739
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2-(4-fluorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
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C23H25ClFN3O3
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1
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| 1 |
IC50 = 8880 nM
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CP0458863
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methyl 2-[3-(5-aminopentyl)-2-anilino-4H-quinazolin-4-yl]acetate
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C22H28N4O2
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1
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| 1 |
IC50 = 9162.2 nM
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CP0489478
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2-(4-(4-methoxyphenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)ethanamine
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C26H34N4O2
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1
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| 1 |
IC50 = 9200 nM
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CP0377010
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(3R,5S)-N-benzyl-3,5-dimethyl-1,2,3,5-tetrahydro-1,4-benzodiazepine-4-carboxamide
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C19H23N3O
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1
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| 1 |
IC50 > 10000 nM
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CP0444048
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(3S,5R)-N,1-dibenzyl-3,5-dimethyl-3,5-dihydro-2H-pyrido[3,4-e][1,4]diazepine-4-carboxamide
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C25H28N4O
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1
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| 1 |
IC50 > 10000 nM
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CP0446026
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(3R,5S)-1-benzyl-3,5-dimethyl-8-methylsulfonyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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C25H28N4O3S
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1
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| 1 |
IC50 > 10000 nM
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CP0452711
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(3R,5S)-1-(benzenesulfonyl)-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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C23H24N4O3S
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1
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| 1 |
IC50 > 10000 nM
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CP0471733
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3-cyano-2,5,5-trimethyl-N-[[3-(2,2,2-trifluoroethoxy)pyridin-2-yl]methyl]-6,7-dihydro-4H-isoindole-1-carboxamide
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C21H23F3N4O2
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1
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| 1 |
IC50 > 10000 nM
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CP0412185
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N-[1-[(4-acetamidophenyl)methyl]pyrazol-3-yl]-2-[4-(dimethylamino)phenyl]acetamide
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C22H25N5O2
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1
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| 1 |
IC50 > 10000 nM
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CP0412204
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N-(1-benzylpyrazol-3-yl)benzamide
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C17H15N3O
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1
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| 1 |
IC50 > 10000 nM
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CP0483095
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3-[1-[(3,4-difluorophenyl)methyl]pyrazol-3-yl]-5-(4-propan-2-ylphenyl)-1,2,4-oxadiazole
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C21H18F2N4O
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1
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| 1 |
IC50 > 10000 nM
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CP0416434
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2-(4-phenylpiperazin-1-yl)-N-[(4-phenyl-2-propyl-1,3-oxazol-5-yl)methyl]ethanamine
Show/Hide
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C25H32N4O
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1
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| 1 |
IC50 = 10250 nM
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CP0477655
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(2,3-Diphenyl-3,4-dihydro-quinazolin-4-yl)-acetic acid methyl ester
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C23H20N2O2
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2
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| 1 |
IC50 = 10690.55 nM
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| 2 |
IC50 = 10700 nM
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CP0467096
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3-(4-chlorobenzyl)-N-(2-(butyl(methyl)amino)ethyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
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C23H27ClN4O2S
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1
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| 1 |
IC50 = 11370 nM
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CP0490902
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(2S)-1-[4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
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C20H23ClF2N2O2
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1
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| 1 |
IC50 = 11380 nM
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CP0259273
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3-(4-chlorobenzyl)-7-(1-methylpiperazine-4-carbonyl)-2-thioxo-2,3-dihydroquinazolin-4(1H)-one
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C21H21ClN4O2S
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1
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| 1 |
IC50 = 11390 nM
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CP0385832
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(2R)-1-(4-fluorophenoxy)-3-[4-(3-methoxyphenyl)piperazin-1-yl]propan-2-ol
Show/Hide
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C20H25FN2O3
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1
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| 1 |
IC50 = 12000 nM
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CP0500391
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(2R)-1-[4-[(2-chloro-6-fluorophenyl)methyl]piperazin-1-yl]-3-(4-fluorophenoxy)propan-2-ol
Show/Hide
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C20H23ClF2N2O2
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1
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| 1 |
IC50 = 12330 nM
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CP0417726
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2-(4-((1H-benzo[d]imidazol-2-yl)methyl)-1,4-diazepan-1-yl)-N-(2-methoxyphenyl)acetamide
Show/Hide
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C22H27N5O2
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1
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| 1 |
IC50 = 12600 nM
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CP0429830
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2-[7-amino-2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]-N-[(4-aminophenyl)methyl]acetamide
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C21H28N6O
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1
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| 1 |
IC50 = 12705.74 nM
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CP0394045
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N-[(4-aminophenyl)methyl]-2-(3-phenyl-2-piperidin-1-yl-4H-quinazolin-4-yl)acetamide
Show/Hide
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C28H31N5O
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2
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| 1 |
IC50 = 13031.67 nM
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| 2 |
IC50 = 14400 nM
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CP0918649
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2-(3-methoxybenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
Show/Hide
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C24H28ClN3O4
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1
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| 1 |
IC50 = 14120 nM
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CP0900129
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2-(2-fluorobenzyl)-1,3-dioxo-N-(2-(piperidin-1-yl)ethyl)isoindoline-5-carboxamide hydrochloride
Show/Hide
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C23H25ClFN3O3
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1
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| 1 |
IC50 = 14860 nM
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CP0417563
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(2S)-1-[4-(4-fluorophenyl)piperazin-1-yl]-3-[4-(trifluoromethyl)phenoxy]propan-2-ol
Show/Hide
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C20H22F4N2O2
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1
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| 1 |
IC50 = 15500 nM
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CP0406216
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4-(4-Methoxybenzylamino)-1-(4-((4-chlorophenyl)(phenyl)methyl)piperazin-1-yl)butan-1-one
Show/Hide
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C29H34ClN3O2
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1
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| 1 |
IC50 = 16100 nM
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CP0452340
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3-(4-(2-fluorophenyl)piperazin-1-yl)-N-((4-phenyl-2-propyloxazol-5-yl)methyl)propan-1-amine
Show/Hide
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C26H33FN4O
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1
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| 1 |
IC50 = 16130 nM
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CP0412115
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methyl 2-[[4-[3-phenyl-3-[4-(trifluoromethyl)phenyl]propanoyl]piperazin-1-yl]methyl]-1,3-oxazole-4-carboxylate
Show/Hide
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C26H26F3N3O4
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1
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| 1 |
IC50 = 17050 nM
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CP0437414
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methyl 2-[[4-[3-(4-bromophenyl)-3-phenylpropanoyl]piperazin-1-yl]methyl]-1,3-oxazole-4-carboxylate
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C25H26BrN3O4
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1
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| 1 |
IC50 = 21150 nM
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CP0393638
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N-benzyl-2-(2-morpholin-4-yl-3-phenyl-4H-quinazolin-4-yl)acetamide
Show/Hide
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C27H28N4O2
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2
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| 1 |
IC50 = 21577.44 nM
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| 2 |
IC50 = 21600 nM
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CP0918651
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2-benzyl-1,3-dioxo-2,3-dihydro-1H-isoindole-5-carboxylic acid (2-piperidin-1-yl-ethyl)-amide hydrochloride
Show/Hide
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C23H26ClN3O3
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1
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| 1 |
IC50 = 22780 nM
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CP0431941
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N-benzyl-2-[2-(dimethylamino)-3-ethyl-4H-quinazolin-4-yl]acetamide
Show/Hide
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C21H26N4O
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1
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| 1 |
IC50 = 24154.61 nM
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CP0409559
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(3-Phenyl-2-piperidin-1-yl-3,4-dihydro-quinazolin-4-yl)-acetic acid methyl ester
Show/Hide
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C22H25N3O2
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2
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| 1 |
IC50 = 27669.42 nM
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| 2 |
IC50 = 27700 nM
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CP0461115
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N-benzyl-2-[2-(4-methylpiperazin-1-yl)-3-phenyl-4H-quinazolin-4-yl]acetamide
Show/Hide
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C28H31N5O
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2
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| 1 |
IC50 = 35800 nM
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| 2 |
IC50 = 35809.64 nM
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CP0446777
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3-(4-chlorobenzyl)-N-(2-(dimethylamino)ethyl)-4-oxo-2-thioxo-1,2,3,4-tetrahydroquinazoline-7-carboxamide
Show/Hide
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C20H21ClN4O2S
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1
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| 1 |
IC50 = 53500 nM
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CP0001395
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1-[4-[(3,5-dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
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C32H30Cl2N2O
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1
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| 1 |
IC50 > 1000 nM
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CP0005547
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1-[4-[(3,4-dichlorophenyl)-phenylmethyl]piperazin-1-yl]-3,3-diphenylpropan-1-one
Show/Hide
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C32H30Cl2N2O
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1
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| 1 |
IC50 > 1000 nM
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CP0863073
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1-{4-[(2,6-Dichloro-phenyl)-phenyl-methyl]-piperazin-1-yl}-3,3-diphenyl-propan-1-one hydrochloride
Show/Hide
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C32H31Cl3N2O
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1
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| 1 |
IC50 < 1000 nM
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CP0382621
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(3R,5S)-1-benzyl-9-methoxy-3,5-dimethyl-N-pyridin-3-yl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C25H28N4O2
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1
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| 1 |
IC50 > 5300 nM
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CP0382578
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(3R,5S)-N-benzyl-3,5-dimethyl-1-(pyridin-4-ylmethyl)-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Show/Hide
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C25H28N4O
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1
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| 1 |
IC50 > 7260 nM
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CP0534094
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(7R,9S)-N,5-dibenzyl-7,9-dimethyl-7,9-dihydro-6H-pyrimido[5,4-e][1,4]diazepine-8-carboxamide
Show/Hide
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C24H27N5O
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1
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| 1 |
IC50 > 8500 nM
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CP0424411
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(4S,6R)-N,8-dibenzyl-1,4,6-trimethyl-6,7-dihydro-4H-pyrazolo[3,4-e][1,4]diazepine-5-carboxamide
Show/Hide
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C24H29N5O
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1
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| 1 |
IC50 > 9400 nM
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