Brief Information of the Compound and Protein
Compound Name
4-ethenyl-1,5-diphenyl-N-[[2-(2,2,2-trifluoroethoxy)phenyl]methyl]pyrazole-3-carboxamide
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PubChem ID
CID: 145974461
Canonical SMILES
FC(F)(F)COc1ccccc1CNC(=O)c1nn(c(c1C=C)-c1ccccc1)-c1ccccc1
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Compound Formula C27H22F3N3O2
Compound Structure
Protein Name
Voltage-dependent T-type calcium channel subunit alpha-1G
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O43497
Gene Name
CACNA1G
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 71 nM
   TI
   LI
   LO
   TS