Brief Information of the Compound and Protein
Compound Name
2-[2-[5-(dimethylamino)pentyl-methylamino]-3-(4-phenylphenyl)-4H-quinazolin-4-yl]-N-[(4-methoxyphenyl)methyl]acetamide
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PubChem ID
CID: 72725613
Canonical SMILES
COc1ccc(CNC(=O)CC2N(C(=Nc3ccccc23)N(C)CCCCCN(C)C)c2ccc(cc2)-c2ccccc2)cc1
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Compound Formula C38H45N5O2
Compound Structure
Protein Name
Voltage-dependent T-type calcium channel subunit alpha-1G
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O43497
Gene Name
CACNA1G
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 390 nM
   TI
   LI
   LO
   TS