Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(3R,5S)-N-benzyl-1-[(6-methoxypyridin-3-yl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
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 PubChem ID
CID: 134146171
Canonical SMILES
COc1ccc(CN2C[C@@H](C)N([C@@H](C)c3ccccc23)C(=O)NCc2ccccc2)cn1
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Compound Formula C26H30N4O2
Compound Structure
Protein Name
 Protein Info 
Voltage-dependent T-type calcium channel subunit alpha-1G
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Voltage-gated calcium channel
Uniprot ID
O43497
Gene Name
CACNA1G
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 45 nM
   TI
   LI
   LO
   TS