4-cyano-5-ethyl-1-methyl-3-(2'-methylsulfanyl-biphenyl-4-yl)-1H-pyrrole-2-carboxylic acid

4-cyano-3-(2'-ethoxy-biphenyl-4-yl)-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

3-(2'-chloro-biphenyl-4-yl)-4-cyano-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

3-(4-tert-butylphenyl)-4-cyano-5-ethylthiophene-2-carboxylic acid

4-cyano-3-(2'-cyano-biphenyl-4-yl)-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

3-(4-tert-butylphenyl)-4-cyano-5-(trifluoromethyl)thiophene-2-carboxylic acid

3-(4-tert-butylphenyl)-4-cyano-5-(methylthio)thiophene-2-carboxylic acid

3-biphenyl-4-yl-4-cyano-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-3-(2'-fluoro-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

3-(4'-chloro-biphenyl-4-yl)-4-cyano-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

N-[2-[4-(4-cyanophenyl)cyclohexyl]propyl]propane-2-sulfonamide

3-biphenyl-4-yl-4-cyano-1-methyl-5-methylsulfanyl-1H-pyrrole-2-carboxylic acid

3-(4-tert-butylphenyl)-4-cyano-5-(dimethylamino)thiophene-2-carboxylic acid

3-(3'-chloro-biphenyl-4-yl)-4-cyano-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-1-methyl-3-(2'-methyl-biphenyl-4-yl)-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-3-(2'-methoxy-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

3-biphenyl-4-yl-4-cyano-1,5-dimethyl-1H-pyrrole-2-carboxylic acid

3-(4-tert-butylphenyl)-4-cyano-5-(methylsulfonyl)thiophene-2-carboxylic acid

4-cyano-5-ethyl-3-(4'-fluoro-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-3-(4'-cyano-biphenyl-4-yl)-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-3-(4'-methoxy-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-3-(3'-methoxy-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

4-cyano-3-(3'-cyano-biphenyl-4-yl)-5-ethyl-1-methyl-1H-pyrrole-2-carboxylic acid

(R)-3,5-difluoro-N-(4-(1-(1-methylethylsulfonamido)propan-2-yl)phenyl)benzamide

N-{5-[3-(1,1-dioxido-2-isothiazolidinyl)phenyl]-2,3-dihydro-1H-inden-2-yl}-2-propanesulfonamide

4-cyano-5-ethyl-1-methyl-3-(4'-methyl-biphenyl-4-yl)-1H-pyrrole-2-carboxylic acid

4-cyano-5-ethyl-3-(3'-fluoro-biphenyl-4-yl)-1-methyl-1H-pyrrole-2-carboxylic acid

(+/-) Propane-2-sulfonic acid [2-(4'-cyano-biphenyl-4-yl)-propyl]-amide

3-(4-tert-butylphenyl)-4-cyano-1-methyl-5-(methylthio)-1H-pyrrole-2-carboxylic acid

N-(5-{4-[(Methylsulfonyl)amino]phenyl}-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide

4-cyano-5-ethyl-1-methyl-3-(3'-methyl-biphenyl-4-yl)-1H-pyrrole-2-carboxylic acid

1-({4-[3-(Trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]-phenyl}methyl)-2-pyrrolidinone

1-({2-Fluoro-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1Hindazol-1-yl]phenyl}methyl)-2-pyrrolidinone

3-(4-tert-butylphenyl)-4-cyano-5-(pyrrolidin-1-yl)thiophene-2-carboxylic acid

N-(5-{3-[Methyl(methylsulfonyl)amino]phenyl}-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide

1-{3-Fluoro-4-[2-oxo-2-(1-pyrrolidinyl)ethyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)acetamide

N-[(2S)-5-(5-fluoropyridin-2-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-[(2S)-5-(6-methylpyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N,N-dimethyl-2-[4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]phenyl]acetamide

N-methyl-N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)acetamide

3-Bicyclo[2.2.1]hept-5-en-2-yl-6-chloro-1,1-dioxo-1,2,3,4-tetrahydro-1lambda*6*-benzo[1,2,4]thiadiazine-7-sulfonic acid amide

N-[(2S)-5-(6-fluoropyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-(5-{3-[(ethylsulfonyl)amino]phenyl}-2,3-dihydro-1H-inden-2-yl)-2-propanesulfonamide

N-[[4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]phenyl]methyl]propanamide

N-[5-(5-methylpyridin-2-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-[5-(6-methyl-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide

1-{4-[2-OXO-2-(1-PYRROLIDINYL)ETHYL]PHENYL}-3-( TRIFLUOROMETHYL)-4,5,6,7-TETRAHYDRO-1H-INDAZOLE

1-{4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}-2-propanone

N-[5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide

1-({4-[3-(Trifluoromethyl)-4,7-dihydropyrano[3,4-c]pyrazol-1(5H)-yl]phenyl}methyl)-2-pyrrolidinone

N-{5-[3-(2-oxopropyl)phenyl]-2,3-dihydro-1H-inden-2-yl}-2-propanesulfonamide

N-[5-(5-fluoro-2-pyridinyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide

N-[5-(5-chloropyridin-2-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

3-(2-x-2,3-dihydro-1H-inden-5-yl)-N,N-dimethylbenzenesulfonamide

N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)methanesulfonamide

1-({4-[3-(Trifluoromethyl)-6,7-dihydropyrano[4,3-c]pyrazol-1(4H)-yl]phenyl}methyl)-2-pyrrolidinone

1-[4-(1-Pyrrolidinylcarbonyl)phenyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

1-{4-[(1,1-Dioxido-2-isothiazolidinyl)methyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)cyclopropanesulfonamide

N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)-2-propanesulfonamide

N-(5-{3-[(2-Oxo-1-pyrrolidinyl)methyl]phenyl}-2,3-dihydro-1Hinden-2-yl)-2-propanesulfonamide

N-(5-pyridin-3-yl-2,3-dihydro-1H-inden-2-yl)propane-2-sulfonamide

N-[5-(2-fluoropyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-butyl-N-methyl-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]benzamide

N-[5-(3-methylpyridin-2-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-[5-(4-methylpyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-[3-(2-{[(1-methylethyl)sulfonyl]amino}-2,3-dihydro-1H-inden-5-yl)phenyl]acetamide

1-({2,6-Difluoro-4-[3-(trifluoromethyl)-6,7-dihydropyrano[4,3-c]pyrazol-1(4H)-yl]phenyl}methyl)-2-pyrrolidinone

1-[4-(1-Pyrrolidinylcarbonyl)phenyl]-3-(trifluoromethyl)-1,4,6,7-tetrahydropyrano[4,3-c]pyrazole

N,N-dimethyl-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]benzenesulfonamide

1-{4-[1,1-difluoro-2-oxo-2-(1-pyrrolidinyl)ethyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

N-Methyl-N-({4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}methyl)methanesulfonamide

1-[4-(4-Morpholinylcarbonyl)phenyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

N,N-dimethyl-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]benzamide

1-{4-[1-methyl-2-oxo-2-(1-pyrrolidinyl)ethyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

N-[(2R)-5-(6-fluoropyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-[5-(2,6-dimethylpyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

1-{4-[3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazol-1-yl]phenyl}ethanone

1-{4-[1-(1-pyrrolidinylcarbonyl)cyclopropyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1Hindazole

1-(4-(methylsulfonyl)phenyl)-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

1-{4-[1-fluoro-2-oxo-2-(1-pyrrolidinyl)ethyl]phenyl}-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1Hindazole

1-({4-[6-Methyl-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-1-yl]phenyl}methyl)-2-pyrrolidinone

N-methyl-N-(2-phenylethyl)-4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]benzamide

N-[5-(3-acetylphenyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide

N-[5-(3-Cyanophenyl)-2,3-dihydro-1H-inden-2-yl]-2-propanesulfonamide

2-Methyl-N-[3-(2-{[(1-methylethyl)sulfonyl]amino}-2,3-dihydro-1H-inden-5-10yl)phenyl]propanamide

N-[5-(5-cyanopyridin-3-yl)-2,3-dihydro-1H-inden-2-yl]propane-2-sulfonamide

N-cyclopentyl-2-[4-[3-(trifluoromethyl)-4,5,6,7-tetrahydroindazol-1-yl]phenyl]acetamide

1-[4-(1-Pyrrolidinylcarbonyl)phenyl]-3-(trifluoromethyl)-1,4,5,7-tetrahydropyrano[3,4-c]pyrazole

1-[4-(1-piperidinylcarbonyl)phenyl]-3-(trifluoromethyl)-4,5,6,7-tetrahydro-1H-indazole

3-(4-tert-butylphenyl)-4-cyanothiophene-2-carboxylic acid

ethyl 3-(4-tert-butylphenyl)-4-cyano-5-methylsulfanylthiophene-2-carboxylate

3-biphenyl-4-yl-5-bromo-4-cyano-1-methyl-1H-pyrrole-2-carboxylic acid

3-biphenyl-4-yl-4-cyano-5-isopropylsulfanyl-1-methyl-1H-pyrrole-2-carboxylic acid

3-biphenyl-4-yl-4-cyano-1-methyl-1H-pyrrole-2-carboxylic acid

2,3-Dihydroxy-6-nitro-benzo[f]quinoxaline-7-sulfonic acid amide

2-(3-(3-bromophenyl)ureido)-4-chlorobenzoic acid

4-Chloro-2-(3-naphthalen-2-yl-ureido)-benzoic acid

(S)-2-Amino-3-(6-chloro-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid

(S)-2-Amino-3-(6-bromo-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid

(S)-2-Amino-3-(5-fluoro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-propionic acid

(S)-2-Amino-3-(5-chloro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-propionic acid

(S)-2-Amino-3-(5-bromo-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-propionic acid

(S)-2-Amino-3-(6-iodo-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid

(2S)-2-amino-3-(3-hydroxy-5-methyl-1,2-oxazol-4-yl)propanoic acid

(S)-2-Amino-3-(5-nitro-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-propionic acid

(S)-2-Amino-3-(5-iodo-2,4-dioxo-3,4-dihydro-2H-pyrimidin-1-yl)-propionic acid

(S)-2-Amino-3-(6-methyl-3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid

(S)-2-Amino-3-(3,5-dioxo-4,5-dihydro-3H-[1,2,4]triazin-2-yl)-propionic acid

(2S)-2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid

(2S)-2-aminopentanedioic acid

6-(4-aminophenyl)-8-(3-bromo-4,5-dihydro-1,2-oxazol-5-yl)-3,10-dihydro-2H-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one

(S)-2-Amino-4-cyclopentylidene-pentanedioic acid

(2S,4E)-2-amino-4-(2-methylpropylidene)pentanedioic acid

4-(8-Methyl-9H-1,3-dioxa-6,7-diaza-cyclohepta[f]inden-5-yl)-phenylamine

6-(4-amino-3-methylphenyl)-2,3,8,10-tetrahydro-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one

6-(4-amino-3,5-dimethylphenyl)-8-[(3-bromo-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3,10-dihydro-2H-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one

LY 457691

LY 458545

(2S,4R)-2-amino-4-[(E)-3-(4-chlorophenyl)prop-2-enyl]pentanedioic acid

(2S,4R)-2-amino-4-[(E)-3-(2-methoxyphenyl)prop-2-enyl]pentanedioic acid

(2S,4R)-2-Amino-4-((E)-3-naphthalen-2-yl-allyl)-pentanedioic acid

(2S-(2alpha,3beta,4beta))-2-carboxy-4-(1-methylethenyl)-3-pyrrolidineacetic acid

6-(4-amino-phenyl)-2,3,8,10-tetrahydro-1,4-dioxa-7,8-diaza-cyclohepta[b]naphthalen-9-one

(2S,4Z)-2-amino-4-(2-methylpropylidene)pentanedioic acid

6-(4-amino-3-methylphenyl)-8-[(3-bromo-4,5-dihydro-1,2-oxazol-5-yl)methyl]-3,10-dihydro-2H-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one

6-(4-amino-3,5-dimethylphenyl)-2,3,8,10-tetrahydro-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one

LY 525327

(3S,4aS,6S,8aR)-6-[2-(1H-Tetrazol-5-yl)-phenoxy]-decahydro-isoquinoline-3-carboxylic acid isobutyl ester

(3S,4aR,6S,8aR)-6-(4-Carboxy-benzyl)-decahydro-isoquinoline-3-carboxylic acid