Brief Information of the Compound and Protein
Compound Name
6-(4-amino-3-methylphenyl)-2,3,8,10-tetrahydro-[1,4]dioxino[2,3-h][2,3]benzodiazepin-9-one
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PubChem ID
CID: 24882540
SID: 50138280
Canonical SMILES
Cc1cc(ccc1N)C1=NNC(=O)Cc2cc3OCCOc3cc12
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Compound Formula C18H17N3O3
Compound Structure
Protein Name
Glutamate receptor 2
Protein Classification
Ion channel
>
Ligand-gated ion channel
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Ionotropic glutamate receptor
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AMPA receptor
Uniprot ID
P42262
Gene Name
GRIA2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 4000 nM
   TI
   LI
   LO
   TS
CL000107 HEK293S Homo sapiens (Human)  1
1
Ki = 9000 nM
   TI
   LI
   LO
   TS