| Compound ID |
Compound Name |
Compound Formula |
|
CP0862257
|
1-(2-(2,4-dichlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15BrCl2N2O3
|
2
|
| 1 |
IC50 = 0.1318 nM
|
|
|
| 2 |
Ki = 0.4898 nM
|
|
|
|
CP0524351
|
5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methoxybenzoic acid
Show/Hide
|
C26H20BrF2NO4
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0528143
|
2-acetamido-5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C27H21BrF2N2O4
|
1
|
| 1 |
IC50 = 0.3981 nM
|
|
|
|
CP0855046
|
1-(2-(2,4-difluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15BrF2N2O3
|
2
|
| 1 |
IC50 = 0.5248 nM
|
|
|
| 2 |
Ki = 2.63 nM
|
|
|
|
CP0536353
|
5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-(difluoromethoxy)benzoic acid
Show/Hide
|
C26H18BrF4NO4
|
1
|
| 1 |
IC50 = 0.631 nM
|
|
|
|
CP0541250
|
3-amino-5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H22BrFN2O3
|
1
|
| 1 |
IC50 = 0.7943 nM
|
|
|
|
CP0496611
|
6-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-1H-indole-4-carboxylic acid
Show/Hide
|
C27H21ClN2O3
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0526682
|
5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H20BrF2NO3
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0526686
|
5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-fluorobenzoic acid
Show/Hide
|
C25H18BrF2NO3
|
1
|
| 1 |
IC50 = 1.259 nM
|
|
|
|
CP0500444
|
3-amino-5-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H23ClN2O3
|
1
|
| 1 |
IC50 = 1.995 nM
|
|
|
|
CP0526685
|
2-fluoro-5-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
Show/Hide
|
C26H19F4NO3
|
1
|
| 1 |
IC50 = 1.995 nM
|
|
|
|
CP0536367
|
5-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-hydroxybenzoic acid
Show/Hide
|
C25H18BrF2NO4
|
1
|
| 1 |
IC50 = 1.995 nM
|
|
|
|
CP0541251
|
5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-(difluoromethoxy)benzoic acid
Show/Hide
|
C26H19BrF3NO4
|
1
|
| 1 |
IC50 = 1.995 nM
|
|
|
|
CP0484547
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H15ClN2O3
|
1
|
| 1 |
IC50 = 1.995 nM
|
|
|
|
CP0497527
|
4-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-N-(pyridin-2-ylmethyl)benzamide
Show/Hide
|
C31H26ClN3O2
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0383444
|
3-[2-[5-bromo-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
Show/Hide
|
C29H20BrF2NO3
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0526683
|
5-[2-[5-chloro-2-[(2,4-difluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H20ClF2NO3
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0526684
|
5-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-chlorobenzoic acid
Show/Hide
|
C25H18BrClFNO3
|
1
|
| 1 |
IC50 = 2.512 nM
|
|
|
|
CP0490478
|
3-amino-5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H23BrN2O3
|
1
|
| 1 |
IC50 = 3.162 nM
|
|
|
|
CP0854908
|
1-(2-(2-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H16BrClN2O3
|
2
|
| 1 |
IC50 = 3.162 nM
|
|
|
| 2 |
Ki = 28.84 nM
|
|
|
|
CP0099081
|
3-(3-(2-(benzyloxy)-5-chlorophenyl)thiophen-2-yl)benzoic acid
Show/Hide
|
C24H17ClO3S
|
2
|
| 1 |
IC50 = 3.548 nM
|
|
|
| 2 |
Ki = 1.259 nM
|
|
|
|
CP0399459
|
3-amino-2-methyl-5-[2-methyl-5-[2-phenylmethoxy-5-(trifluoromethyl)phenyl]pyrrol-1-yl]benzoic acid
Show/Hide
|
C27H23F3N2O3
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0536352
|
3-amino-5-[2-[2-[(4-fluorophenyl)methoxy]-5-(trifluoromethyl)phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C27H22F4N2O3
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0897556
|
sodium 2-(6-bromo-3-isobutyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C16H14BrN2NaO2S
|
2
|
| 1 |
IC50 = 3.981 nM
|
|
|
| 2 |
Ki = 0.1995 nM
|
|
|
|
CP0513342
|
1-[(5-chloro-2-cyclohexyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C20H21ClN2O3
|
1
|
| 1 |
IC50 = 3.981 nM
|
|
|
|
CP0383448
|
5-[2-[5-chloro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
Show/Hide
|
C26H21ClFNO3
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0436388
|
5-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]-2-(difluoromethoxy)benzoic acid
Show/Hide
|
C26H20BrF2NO4
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0464435
|
3-[2-[5-bromo-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
Show/Hide
|
C29H21BrFNO3
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0877334
|
1-(5-chloro-2-isobutoxybenzyl)-N-(4-((dimethylamino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C25H32Cl2N4O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0461851
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-N-cyclopropyl-5-methylpyrazole-3-carboxamide
Show/Hide
|
C23H20ClN3O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0513357
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxamide
Show/Hide
|
C20H16ClN3O2
|
1
|
| 1 |
IC50 = 5.012 nM
|
|
|
|
CP0390763
|
1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H17ClN2O3
|
2
|
| 1 |
IC50 = 5.012 nM
|
|
|
| 2 |
Ki = 0.3981 nM
|
|
|
|
CP0910972
|
sodium 1-(2-(benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylate
Show/Hide
|
C19H16BrN2NaO3
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0949859
|
N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-cyclohexylacetamide
Show/Hide
|
C26H30ClN3O2
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0082063
|
3-(2-(2-(4-fluorobenzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H19BrFNO3
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0526681
|
3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
Show/Hide
|
C29H22ClNO3
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0766472
|
sodium 2-(2-(benzyloxy)-5-chlorobenzyl)thiazole-4-carboxylate
Show/Hide
|
C18H13ClNNaO3S
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0894514
|
sodium 2-(6-chloro-3-(3,3-dimethylbutyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C18H18ClN2NaO2S
|
2
|
| 1 |
IC50 = 6.31 nM
|
|
|
| 2 |
Ki = 3.981 nM
|
|
|
|
CP0926458
|
sodium 2-((6-chloro-3-isobutyl-1H-indol-1-yl)methyl)thiazole-4-carboxylate
Show/Hide
|
C17H16ClN2NaO2S
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0877333
|
1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-(4-(piperidin-1-ylmethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C28H36Cl2N4O2
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0895579
|
1-(2-(benzyloxy)-5-chlorobenzyl)-N-(4-(hydroxymethyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C26H25Cl2N3O3
|
2
|
| 1 |
IC50 = 6.31 nM
|
|
|
| 2 |
Ki = 39.81 nM
|
|
|
|
CP0907732
|
1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-(4-(pyrrolidin-1-ylmethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C27H34Cl2N4O2
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0432377
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
Show/Hide
|
C25H24ClN3O3
|
1
|
| 1 |
IC50 = 6.31 nM
|
|
|
|
CP0109651
|
1-(2-(benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H17BrN2O3
|
2
|
| 1 |
IC50 = 6.457 nM
|
|
|
| 2 |
Ki = 15.14 nM
|
|
|
|
CP0918721
|
1-(2-(4-fluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H16BrFN2O3
|
2
|
| 1 |
IC50 = 7.413 nM
|
|
|
| 2 |
Ki = 11.75 nM
|
|
|
|
CP0109778
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H20ClNO3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0496610
|
2-fluoro-5-[2-[2-[(4-fluorophenyl)methoxy]-5-(trifluoromethyl)phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C26H18F5NO3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0645981
|
sodium 2-(5-chloro-2-isobutoxybenzyl)thiazole-4-carboxylate
Show/Hide
|
C15H15ClNNaO3S
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0895233
|
sodium 2-(6-chloro-3-isobutyl-1H-indol-1-yl)oxazole-4-carboxylate
Show/Hide
|
C16H14ClN2NaO3
|
2
|
| 1 |
IC50 = 7.943 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0110250
|
3-(2-(2-(benzyloxy)-5-bromophenyl)-5-methyl-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C25H20BrNO3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0870432
|
1-(2-(benzyloxy)-5-chlorobenzyl)-N-(4-((dimethylamino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C28H30Cl2N4O2
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0880929
|
1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-(4-((methylamino)methyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C24H30Cl2N4O2
|
2
|
| 1 |
IC50 = 7.943 nM
|
|
|
| 2 |
Ki = 79.43 nM
|
|
|
|
CP0898976
|
1-(5-chloro-2-isobutoxybenzyl)-N-(4-((ethylamino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C25H32Cl2N4O2
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0904395
|
1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-(4-(morpholinomethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C27H34Cl2N4O3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0400868
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-N-(4-hydroxycyclohexyl)-5-methylpyrazole-3-carboxamide
Show/Hide
|
C26H26ClN3O3
|
1
|
| 1 |
IC50 = 7.943 nM
|
|
|
|
CP0849114
|
1-(2-(4-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H16BrClN2O3
|
2
|
| 1 |
IC50 = 8.71 nM
|
|
|
| 2 |
Ki = 8.71 nM
|
|
|
|
CP0927506
|
1-(2-(benzyloxy)-5-bromobenzyl)-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C18H15BrN2O3
|
2
|
| 1 |
IC50 = 9.772 nM
|
|
|
| 2 |
Ki = 54.95 nM
|
|
|
|
CP0862040
|
sodium 1-(1-(2-(benzyloxy)-5-chlorophenyl)ethyl)-5-methyl-1H-pyrazole-3-carboxylate
Show/Hide
|
C20H18ClN2NaO3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0862989
|
1-(2-(benzyloxy)-5-chlorobenzyl)-N-(2,6-difluorophenyl)-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H20ClF2N3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0906216
|
N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-3,3-dimethylbutanamide
Show/Hide
|
C24H28ClN3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0932840
|
sodium 2-(3-isobutyl-6-methyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C17H17N2NaO2S
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0192990
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrrol-1-yl)benzoic acid
Show/Hide
|
C24H18ClNO3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0784948
|
sodium 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylate
Show/Hide
|
C19H16ClN2NaO3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0846020
|
1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(4-(morpholinomethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C30H32Cl2N4O3
|
2
|
| 1 |
IC50 = 10 nM
|
|
|
| 2 |
Ki = 79.43 nM
|
|
|
|
CP0391228
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methyl-N-propan-2-ylpyrazole-3-carboxamide
Show/Hide
|
C23H22ClN3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0400981
|
N-tert-butyl-1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxamide
Show/Hide
|
C24H24ClN3O2
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0427434
|
1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methyl-N-morpholin-4-ylpyrazole-3-carboxamide
Show/Hide
|
C24H23ClN4O3
|
1
|
| 1 |
IC50 = 10 nM
|
|
|
|
CP0926439
|
N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-phenylacetamide
Show/Hide
|
C26H24ClN3O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0942336
|
N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2,6-difluorobenzamide
Show/Hide
|
C25H20ClF2N3O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0509365
|
3-[2-(5-bromo-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
Show/Hide
|
C29H22BrNO3
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0542857
|
2-fluoro-5-[2-[5-fluoro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]benzoic acid
Show/Hide
|
C25H18F3NO3
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0902810
|
sodium 2-(3-isobutyl-6-(trifluoromethyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C17H14F3N2NaO2S
|
2
|
| 1 |
IC50 = 12.59 nM
|
|
|
| 2 |
Ki = 0.0631 nM
|
|
|
|
CP0109669
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)cyclopent-1-enyl)benzoic acid
Show/Hide
|
C25H21ClO3
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0846022
|
1-(2-(benzyloxy)-5-chlorobenzyl)-N-(4-((ethylamino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
|
C28H30Cl2N4O2
|
1
|
| 1 |
IC50 = 12.59 nM
|
|
|
|
CP0882957
|
1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(4-(pyrrolidin-1-ylmethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
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C30H32Cl2N4O2
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1
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| 1 |
IC50 = 12.59 nM
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CP0904394
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(4-(piperidin-1-ylmethyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
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C31H34Cl2N4O2
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1
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| 1 |
IC50 = 12.59 nM
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CP0921780
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(hydroxymethyl)benzamide hydrochloride
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C23H27Cl2N3O3
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1
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| 1 |
IC50 = 12.59 nM
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CP0921781
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(4-((methylamino)methyl)phenyl)-1H-pyrazole-3-carboxamide hydrochloride
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C27H28Cl2N4O2
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2
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| 1 |
IC50 = 12.59 nM
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| 2 |
Ki = 125.89 nM
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CP0853231
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1-(2-(2,6-difluorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
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C19H15BrF2N2O3
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2
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| 1 |
IC50 = 14.79 nM
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| 2 |
Ki = 104.71 nM
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CP0394372
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N-[1-[(5-chloro-2-phenylmethoxyphenyl)methyl]-5-methylpyrazol-3-yl]benzamide
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C25H22ClN3O2
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1
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| 1 |
IC50 = 15.85 nM
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CP0882800
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-methyl-2-(pyridin-2-yl)propanamide
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C27H27ClN4O2
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1
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| 1 |
IC50 = 15.85 nM
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CP0942337
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)cyclopentanecarboxamide
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C24H26ClN3O2
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1
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| 1 |
IC50 = 15.85 nM
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CP0510896
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2-fluoro-5-[2-[2-[(4-fluorophenyl)methoxy]-5-methylphenyl]-5-methylpyrrol-1-yl]benzoic acid
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C26H21F2NO3
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1
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| 1 |
IC50 = 15.85 nM
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CP0526680
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3-amino-5-[2-[2-[(4-fluorophenyl)methoxy]-5-methylphenyl]-5-methylpyrrol-1-yl]-2-methylbenzoic acid
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C27H25FN2O3
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1
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| 1 |
IC50 = 15.85 nM
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CP0858709
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1-(5-chloro-2-isobutoxybenzyl)-N-(4-((bis(2-hydroxyethyl)amino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
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C27H36Cl2N4O4
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2
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| 1 |
IC50 = 15.85 nM
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| 2 |
Ki = 79.43 nM
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CP0855045
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1-(2-(3-bromobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
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C19H16Br2N2O3
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2
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| 1 |
IC50 = 17.78 nM
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| 2 |
Ki = 128.82 nM
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CP0949858
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-(pyridin-2-yl)acetamide
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C25H23ClN4O2
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1
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| 1 |
IC50 = 19.95 nM
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CP0461852
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1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methyl-N-(piperidin-4-ylmethyl)pyrazole-3-carboxamide
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C26H27ClN4O2
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1
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| 1 |
IC50 = 19.95 nM
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CP0240989
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tert-butyl N-[1-[(5-chloro-2-phenylmethoxyphenyl)methyl]-5-methylpyrazol-3-yl]carbamate
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C23H26ClN3O3
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1
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| 1 |
IC50 = 25.12 nM
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CP0524536
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N-benzyl-3-[2-(5-chloro-2-phenylmethoxyphenyl)-5-methylpyrrol-1-yl]benzamide
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C32H27ClN2O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0876687
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2,2-difluoro-2-(pyridin-2-yl)acetamide
Show/Hide
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C25H21ClF2N4O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0902757
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isobutyl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
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C23H26ClN3O3
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1
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| 1 |
IC50 = 25.12 nM
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CP0942335
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)cyclopentanecarboxamide
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C21H28ClN3O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0945585
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)isobutyramide
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C22H24ClN3O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0949861
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
Show/Hide
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C25H23ClN4O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0500445
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3-[2-[5-fluoro-2-[(4-fluorophenyl)methoxy]phenyl]-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
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C29H21F2NO3
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1
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| 1 |
IC50 = 25.12 nM
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CP0659705
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sodium 2-(2-(benzyloxy)-5-chlorophenylamino)thiazole-4-carboxylate
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C17H12ClN2NaO3S
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1
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| 1 |
IC50 = 25.12 nM
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CP0878014
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sodium 5-(6-chloro-3-isobutyl-1H-indol-1-yl)furan-2-carboxylate
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C17H15ClNNaO3
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2
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| 1 |
IC50 = 25.12 nM
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| 2 |
Ki = 1.259 nM
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CP0882950
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1-(5-chloro-2-isobutoxybenzyl)-N-(4-((2-hydroxyethylamino)methyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
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C25H32Cl2N4O3
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2
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| 1 |
IC50 = 25.12 nM
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| 2 |
Ki = 100 nM
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CP0911611
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-2-(hydroxymethyl)benzamide hydrochloride
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C23H27Cl2N3O3
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1
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| 1 |
IC50 = 25.12 nM
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CP0432376
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N-[1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazol-3-yl]-1-(2,2,2-trifluoroethyl)piperidine-4-carboxamide
Show/Hide
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C27H26ClF3N4O2
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1
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| 1 |
IC50 = 25.12 nM
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CP0484546
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1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methyl-N-(3,3,3-trifluoro-2-hydroxypropyl)pyrazole-3-carboxamide
Show/Hide
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C23H19ClF3N3O3
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1
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| 1 |
IC50 = 25.12 nM
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CP0505921
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1-[(5-chloro-2-propyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
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C17H17ClN2O3
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1
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| 1 |
IC50 = 25.12 nM
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CP0098885
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propan-2-yl N-[1-[(5-chloro-2-phenylmethoxyphenyl)methyl]-5-methylpyrazol-3-yl]carbamate
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C22H24ClN3O3
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1
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| 1 |
IC50 = 31.62 nM
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CP0862036
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)cyclohexanecarboxamide
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C22H30ClN3O2
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1
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| 1 |
IC50 = 31.62 nM
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CP0945564
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tert-butyl 1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C20H28ClN3O3
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1
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| 1 |
IC50 = 31.62 nM
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CP0877641
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sodium 2-(6-chloro-3-propyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C15H12ClN2NaO2S
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1
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| 1 |
IC50 = 31.62 nM
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CP0945207
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sodium 2-(6-chloro-3-neopentyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C17H16ClN2NaO2S
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1
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| 1 |
IC50 = 31.62 nM
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CP0911698
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1-(5-chloro-2-isobutoxybenzyl)-N-(4-(hydroxymethyl)phenyl)-5-methyl-1H-pyrazole-3-carboxamide hydrochloride
Show/Hide
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C23H27Cl2N3O3
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1
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| 1 |
IC50 = 31.62 nM
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CP0910935
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1-(2-(4-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C20H16BrF3N2O3
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2
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| 1 |
IC50 = 35.48 nM
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| 2 |
Ki = 97.72 nM
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CP0399186
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1-[(5-chloro-2-phenylmethoxyphenyl)methyl]-5-methyl-N-phenylpyrazole-3-carboxamide
Show/Hide
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C25H22ClN3O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0862037
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2,2-difluoro-2-phenylacetamide
Show/Hide
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C26H22ClF2N3O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0862987
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1-(2-(benzyloxy)-5-chlorobenzyl)-N-benzyl-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C26H24ClN3O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0878556
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-tetrahydrofuran-2-carboxamide
Show/Hide
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C23H24ClN3O3
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1
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| 1 |
IC50 = 39.81 nM
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CP0926440
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-tetrahydrofuran-3-carboxamide
Show/Hide
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C23H24ClN3O3
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1
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| 1 |
IC50 = 39.81 nM
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CP0927594
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-(pyridin-3-yl)acetamide
Show/Hide
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C25H23ClN4O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0878017
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sodium 2-(5-chloro-3-isobutyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C16H14ClN2NaO2S
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1
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| 1 |
IC50 = 39.81 nM
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CP0880657
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sodium 2-(6-chloro-3-isobutyl-2-methyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C17H16ClN2NaO2S
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1
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| 1 |
IC50 = 39.81 nM
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CP0890928
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sodium 6-(5-chloro-2-isobutoxybenzyl)picolinate
Show/Hide
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C17H17ClNNaO3
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1
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| 1 |
IC50 = 39.81 nM
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CP0896436
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sodium 2-(6-fluoro-3-isobutyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C16H14FN2NaO2S
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1
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| 1 |
IC50 = 39.81 nM
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CP0896437
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sodium 2-(6-chloro-3-isopropyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C15H12ClN2NaO2S
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1
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| 1 |
IC50 = 39.81 nM
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CP0858710
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-1,2,3,4-tetrahydroisoquinoline-6-carboxamide hydrochloride
Show/Hide
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C25H30Cl2N4O2
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2
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| 1 |
IC50 = 39.81 nM
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| 2 |
Ki = 125.89 nM
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CP0904377
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(piperidin-1-ylmethyl)benzamide hydrochloride
Show/Hide
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C28H36Cl2N4O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0400867
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N-[1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazol-3-yl]-4-fluoropiperidine-4-carboxamide
Show/Hide
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C25H24ClFN4O2
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1
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| 1 |
IC50 = 39.81 nM
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CP0875534
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-(pyridin-4-yl)acetamide
Show/Hide
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C25H23ClN4O2
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1
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| 1 |
IC50 = 50.12 nM
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CP0877698
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isopropyl 1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C19H26ClN3O3
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1
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| 1 |
IC50 = 50.12 nM
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CP0945011
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1,1,1-trifluoro-2-methylpropan-2-yl 1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C20H25ClF3N3O3
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1
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| 1 |
IC50 = 50.12 nM
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CP0949860
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
Show/Hide
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C25H23ClN4O2
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1
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| 1 |
IC50 = 50.12 nM
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CP0878018
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sodium 5-(6-chloro-3-isobutyl-1H-indol-1-yl)thiophene-2-carboxylate
Show/Hide
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C17H15ClNNaO2S
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1
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| 1 |
IC50 = 50.12 nM
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CP0109664
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2''-benzyloxy-5''-chloro-[1,1';2',1'']terphenyl-3-carboxylic acid
Show/Hide
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C26H19ClO3
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1
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| 1 |
IC50 = 50.12 nM
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CP0846063
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-ethyl-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7-carboxamide hydrochloride
Show/Hide
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C28H36Cl2N4O2
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2
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| 1 |
IC50 = 50.12 nM
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| 2 |
Ki = 50.12 nM
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CP0850252
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(1-(isobutylamino)ethyl)benzamide hydrochloride
Show/Hide
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C28H38Cl2N4O2
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1
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| 1 |
IC50 = 50.12 nM
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CP0858711
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(morpholinomethyl)benzamide hydrochloride
Show/Hide
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C27H34Cl2N4O3
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1
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| 1 |
IC50 = 50.12 nM
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CP0870439
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(pyrrolidin-1-ylmethyl)benzamide hydrochloride
Show/Hide
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C27H34Cl2N4O2
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2
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| 1 |
IC50 = 50.12 nM
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| 2 |
Ki = 158.49 nM
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CP0915505
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(1-(pyrrolidin-1-yl)ethyl)benzamide hydrochloride
Show/Hide
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C28H36Cl2N4O2
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1
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| 1 |
IC50 = 50.12 nM
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CP0475621
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1-[(5-chloro-2-cyclopropyl-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
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C17H15ClN2O3
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1
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| 1 |
IC50 = 50.12 nM
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CP0399209
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1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methyl-N-morpholin-4-ylpyrazole-3-carboxamide
Show/Hide
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C21H25ClN4O3
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1
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| 1 |
IC50 = 50.12 nM
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CP0475626
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2-[1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methylpyrazol-3-yl]-1H-benzimidazole
Show/Hide
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C23H21ClN4O
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1
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| 1 |
IC50 = 50.12 nM
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CP0862038
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-2-methyl-2-phenylpropanamide
Show/Hide
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C28H28ClN3O2
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1
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| 1 |
IC50 = 63.1 nM
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CP0876509
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tetrahydro-2H-pyran-4-yl 1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C21H28ClN3O4
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1
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| 1 |
IC50 = 63.1 nM
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CP0876689
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)-tetrahydro-2H-pyran-4-carboxamide
Show/Hide
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C24H26ClN3O3
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1
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| 1 |
IC50 = 63.1 nM
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CP0921796
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sodium 6-(6-chloro-3-isobutyl-1H-indol-1-yl)picolinate
Show/Hide
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C18H16ClN2NaO2
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2
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| 1 |
IC50 = 63.1 nM
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| 2 |
Ki = 19.95 nM
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CP0387448
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1-[(2-tert-butyl-5-chloro-1-benzofuran-7-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
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C18H19ClN2O3
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1
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| 1 |
IC50 = 63.1 nM
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CP0520301
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N-[1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazol-3-yl]-2-piperidin-4-ylacetamide
Show/Hide
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C26H27ClN4O2
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1
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| 1 |
IC50 = 63.1 nM
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CP0452089
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1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methyl-N-(oxan-4-yl)pyrazole-3-carboxamide
Show/Hide
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C22H26ClN3O3
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1
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| 1 |
IC50 = 63.1 nM
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CP0524890
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1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methyl-N-[4-(methylaminomethyl)phenyl]pyrazole-3-carboxamide
Show/Hide
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C25H27ClN4O2
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1
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| 1 |
IC50 = 63.1 nM
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CP0862035
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pyridin-2-ylmethyl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C25H23ClN4O3
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1
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| 1 |
IC50 = 79.43 nM
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CP0876446
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benzyl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C26H24ClN3O3
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1
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| 1 |
IC50 = 79.43 nM
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CP0876453
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1-(2-(benzyloxy)-5-chlorobenzyl)-N-(4-fluorophenyl)-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C25H21ClFN3O2
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1
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| 1 |
IC50 = 79.43 nM
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CP0876686
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(S)-tetrahydrofuran-3-yl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C23H24ClN3O4
|
1
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| 1 |
IC50 = 79.43 nM
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CP0876690
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
Show/Hide
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C25H23ClN4O2
|
1
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| 1 |
IC50 = 79.43 nM
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CP0882799
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ethyl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C21H22ClN3O3
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1
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| 1 |
IC50 = 79.43 nM
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CP0383445
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3-[2-[2-[(4-fluorophenyl)methoxy]-5-methylphenyl]-5-methylpyrrol-1-yl]naphthalene-1-carboxylic acid
Show/Hide
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C30H24FNO3
|
1
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| 1 |
IC50 = 79.43 nM
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CP0255576
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3-(3-(2-(benzyloxy)-5-chlorophenyl)pyridin-4-yl)benzoic acid
Show/Hide
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C25H18ClNO3
|
1
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| 1 |
IC50 = 79.43 nM
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CP0871053
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3-(4-(2-(benzyloxy)-5-chlorophenyl)-2-oxo-2,5-dihydrofuran-3-yl)benzoic acid
Show/Hide
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C24H17ClO5
|
1
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| 1 |
IC50 = 79.43 nM
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CP0876027
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3-(5-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrazol-1-yl)benzoic acid
Show/Hide
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C23H17ClN2O3
|
1
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| 1 |
IC50 = 79.43 nM
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CP0882951
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-2,3,4,5-tetrahydro-1H-benzo[d]azepine-7-carboxamide hydrochloride
Show/Hide
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C26H32Cl2N4O2
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1
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| 1 |
IC50 = 79.43 nM
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CP0902759
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1-(2-(benzyloxy)-5-chlorobenzyl)-N,5-dimethyl-1H-pyrazole-3-carboxamide
Show/Hide
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C20H20ClN3O2
|
1
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| 1 |
IC50 = 100 nM
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CP0878019
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sodium 2-(6-chloro-3-isobutyl-1H-indol-1-yl)thiazole-5-carboxylate
Show/Hide
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C16H14ClN2NaO2S
|
1
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| 1 |
IC50 = 100 nM
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CP0924849
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sodium 2-(6-chloro-3-isobutyryl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C16H12ClN2NaO3S
|
1
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| 1 |
IC50 = 100 nM
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CP0140992
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3-(3-(2-(benzyloxy)-5-chlorophenyl)pyridin-2-yl)benzoic acid
Show/Hide
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C25H18ClNO3
|
1
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| 1 |
IC50 = 100 nM
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CP0858712
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-((ethylamino)methyl)benzamide hydrochloride
Show/Hide
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C25H32Cl2N4O2
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2
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| 1 |
IC50 = 100 nM
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| 2 |
Ki = 158.49 nM
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CP0870433
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-2-isopropyl-1,2,3,4-tetrahydroisoquinoline-6-carboxamide hydrochloride
Show/Hide
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C28H36Cl2N4O2
|
1
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| 1 |
IC50 = 100 nM
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CP0895580
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-(pyrrolidin-2-yl)benzamide hydrochloride
Show/Hide
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C26H32Cl2N4O2
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2
|
| 1 |
IC50 = 100 nM
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| 2 |
Ki = 100 nM
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CP0915506
|
N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-4-((dimethylamino)methyl)benzamide hydrochloride
Show/Hide
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C25H32Cl2N4O2
|
1
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| 1 |
IC50 = 100 nM
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CP0432375
|
N-[1-[(5-chloro-2-phenyl-1-benzofuran-7-yl)methyl]-5-methylpyrazol-3-yl]piperidine-4-carboxamide
Show/Hide
|
C25H25ClN4O2
|
1
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| 1 |
IC50 = 100 nM
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CP0513343
|
1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methyl-N-piperidin-1-ylpyrazole-3-carboxamide
Show/Hide
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C22H27ClN4O2
|
1
|
| 1 |
IC50 = 100 nM
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CP0932546
|
1-(2-(3-chlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C19H16BrClN2O3
|
2
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| 1 |
IC50 = 114.82 nM
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| 2 |
Ki = 426.58 nM
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CP0899686
|
1-(2-(benzyloxy)-5-bromobenzyl)-4-fluoro-1H-pyrazole-3-carboxylic acid
Show/Hide
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C18H14BrFN2O3
|
2
|
| 1 |
IC50 = 123.03 nM
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| 2 |
Ki = 691.83 nM
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CP0862039
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1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C16H20ClN3O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0862988
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1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-N-(pyridin-2-yl)-1H-pyrazole-3-carboxamide
Show/Hide
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C24H21ClN4O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0876454
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1-(2-(benzyloxy)-5-chlorobenzyl)-N-isopropyl-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C22H24ClN3O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0949862
|
1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
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C19H18ClN3O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0895232
|
sodium 2-(6-chloro-3-ethyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C14H10ClN2NaO2S
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1
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| 1 |
IC50 = 125.89 nM
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CP0109663
|
3-(5-(2-(benzyloxy)-5-chlorophenyl)-1H-imidazol-1-yl)benzoic acid
Show/Hide
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C23H17ClN2O3
|
1
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| 1 |
IC50 = 125.89 nM
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CP0855042
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1-[5-bromo-2-(3-methyl-benzyloxy)-benzyl]-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C20H19BrN2O3
|
2
|
| 1 |
IC50 = 125.89 nM
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| 2 |
Ki = 524.81 nM
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CP0916714
|
N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-(pyrrolidin-1-ylmethyl)benzamide hydrochloride
Show/Hide
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C27H34Cl2N4O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0475624
|
1-[(6-chloro-2-propan-2-ylindolizin-8-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C17H18ClN3O2
|
1
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| 1 |
IC50 = 125.89 nM
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CP0862983
|
N-(1-(2-(benzyloxy)-5-chlorobenzyl)-1H-pyrazol-3-yl)-2-phenylacetamide
Show/Hide
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C25H22ClN3O2
|
1
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| 1 |
IC50 = 158.49 nM
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CP0878525
|
sodium 6-(2-(benzyloxy)-5-chlorobenzyl)picolinate
Show/Hide
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C20H15ClNNaO3
|
1
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| 1 |
IC50 = 158.49 nM
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CP0882906
|
sodium 2-(3-isobutyl-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C16H15N2NaO2S
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2
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| 1 |
IC50 = 158.49 nM
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| 2 |
Ki = 12.59 nM
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CP0941564
|
sodium 2-(3-benzyl-6-chloro-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C19H12ClN2NaO2S
|
2
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| 1 |
IC50 = 158.49 nM
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| 2 |
Ki = 63.1 nM
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CP0942103
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sodium 2-(2-(6-chloro-3-isobutyl-1H-indol-1-yl)thiazol-4-yl)acetate
Show/Hide
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C17H16ClN2NaO2S
|
1
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| 1 |
IC50 = 158.49 nM
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CP0915977
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1-(2-(benzyloxy)-5-bromobenzyl)-5-(thiophen-2-yl)-1H-pyrazole-3-carboxylic acid
Show/Hide
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C22H17BrN2O3S
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2
|
| 1 |
IC50 = 194.98 nM
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| 2 |
Ki = 616.6 nM
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CP0862985
|
methyl 1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-ylcarbamate
Show/Hide
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C20H20ClN3O3
|
1
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| 1 |
IC50 = 199.53 nM
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CP0926441
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1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-(piperidin-1-yl)-1H-pyrazole-3-carboxamide
Show/Hide
|
C21H29ClN4O2
|
1
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| 1 |
IC50 = 199.53 nM
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CP0945586
|
1-(2-(benzyloxy)-5-chlorobenzyl)-N-(3-fluorophenyl)-5-methyl-1H-pyrazole-3-carboxamide
Show/Hide
|
C25H21ClFN3O2
|
1
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| 1 |
IC50 = 199.53 nM
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CP0684691
|
3-(1-(2-(benzyloxy)-5-chlorophenyl)-5-methyl-1H-pyrrol-2-yl)benzoic acid
Show/Hide
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C25H20ClNO3
|
1
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| 1 |
IC50 = 199.53 nM
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CP0862986
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1-(5-chloro-2-isobutoxybenzyl)-5-methyl-N-morpholino-1H-pyrazole-3-carboxamide
Show/Hide
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C20H27ClN4O3
|
1
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| 1 |
IC50 = 251.19 nM
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CP0945563
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-1H-pyrazol-3-yl)benzamide
Show/Hide
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C24H20ClN3O2
|
1
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| 1 |
IC50 = 251.19 nM
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CP0926459
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sodium 2-(6-chloro-3-(2,2,2-trifluoroethyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
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C14H7ClF3N2NaO2S
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1
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| 1 |
IC50 = 251.19 nM
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CP0895581
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-(morpholinomethyl)benzamide hydrochloride
Show/Hide
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C27H34Cl2N4O3
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1
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| 1 |
IC50 = 251.19 nM
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CP0400857
|
1-[(6-chloro-2-propan-2-yl-1-benzofuran-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
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C17H17ClN2O3
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1
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| 1 |
IC50 = 251.19 nM
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CP0862259
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1-(2-(3-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C20H16BrF3N2O3
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2
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| 1 |
IC50 = 309.03 nM
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| 2 |
Ki = 1096.48 nM
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CP0855271
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazol-3-yl)acetamide
Show/Hide
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C20H20ClN3O2
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1
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| 1 |
IC50 = 316.23 nM
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CP0918935
|
3-(4-(2-(benzyloxy)-5-chlorophenyl)pyridin-3-yl)benzoic acid
Show/Hide
|
C25H18ClNO3
|
1
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| 1 |
IC50 = 316.23 nM
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CP0520289
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1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-N-(4-methoxycyclohexyl)-5-methylpyrazole-3-carboxamide
Show/Hide
|
C24H30ClN3O3
|
1
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| 1 |
IC50 = 316.23 nM
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CP0847058
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1-(2-(2,4-dichlorobenzyloxy)-5-fluorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C19H15Cl2FN2O3
|
2
|
| 1 |
IC50 = 354.81 nM
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| 2 |
Ki = 20.42 nM
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CP0862981
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N-(1-(2-(benzyloxy)-5-chlorobenzyl)-1H-pyrazol-3-yl)-2-(pyridin-2-yl)acetamide
Show/Hide
|
C24H21ClN4O2
|
1
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| 1 |
IC50 = 398.11 nM
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CP0862293
|
3-(3-(2-(benzyloxy)-5-chlorophenyl)pyrazin-2-yl)benzoic acid
Show/Hide
|
C24H17ClN2O3
|
1
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| 1 |
IC50 = 398.11 nM
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CP0846752
|
1-(2-(benzyloxy)-5-bromobenzyl)-4-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C19H17BrN2O3
|
2
|
| 1 |
IC50 = 426.58 nM
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| 2 |
Ki = 1348.96 nM
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CP0854935
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1-(2-(benzyloxy)-5-bromobenzyl)-4-bromo-1H-pyrazole-3-carboxylic acid
Show/Hide
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C18H14Br2N2O3
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2
|
| 1 |
IC50 = 457.09 nM
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| 2 |
Ki < 1995.26 nM
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CP0858713
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-((ethylamino)methyl)benzamide hydrochloride
Show/Hide
|
C25H32Cl2N4O2
|
1
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| 1 |
IC50 = 501.19 nM
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CP0877280
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-(piperidin-1-ylmethyl)benzamide hydrochloride
Show/Hide
|
C28H36Cl2N4O2
|
1
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| 1 |
IC50 = 501.19 nM
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CP0475625
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1-[(6-chloro-2-propan-2-ylimidazo[1,2-a]pyridin-8-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H17ClN4O2
|
1
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| 1 |
IC50 = 501.19 nM
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CP0873295
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1-(2-(4-chloro-3-(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
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C20H15BrClF3N2O3
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2
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| 1 |
IC50 = 575.44 nM
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| 2 |
Ki < 1995.26 nM
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CP0922402
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sodium 3-(6-chloro-3-isobutyl-1H-indol-1-yl)benzoate
Show/Hide
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C19H17ClNNaO2
|
1
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| 1 |
IC50 = 630.96 nM
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CP0877298
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N-(1-(5-chloro-2-isobutoxybenzyl)-5-methyl-1H-pyrazol-3-yl)-3-((dimethylamino)methyl)benzamide hydrochloride
Show/Hide
|
C25H32Cl2N4O2
|
1
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| 1 |
IC50 = 630.96 nM
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CP0853230
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1-(2-(benzyloxy)-5-bromobenzyl)-4-(hydroxymethyl)-1H-pyrazole-3-carboxylic acid
Show/Hide
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C19H17BrN2O4
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2
|
| 1 |
IC50 = 676.08 nM
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| 2 |
Ki < 1995.26 nM
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CP0475627
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1-[(5-chloro-2-propan-2-yl-1-benzofuran-7-yl)methyl]-5-methyl-N-piperidin-4-ylpyrazole-3-carboxamide
Show/Hide
|
C22H27ClN4O2
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1
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| 1 |
IC50 = 794.33 nM
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CP0922404
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sodium 2-(6-chloro-3-(dimethylcarbamoyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C15H11ClN3NaO3S
|
1
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| 1 |
IC50 = 1000 nM
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CP0402565
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7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydroxy-5-phenyl-pentyl)-cyclopentyl]-heptanoic acid
Show/Hide
|
C23H36O5
|
1
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| 1 |
IC50 = 1100 nM
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CP0916316
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1-(2-(4-tert-butylbenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C23H25BrN2O3
|
2
|
| 1 |
IC50 = 1230.27 nM
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| 2 |
Ki < 1995.26 nM
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CP0849112
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1-(2-(benzyloxy)-5-bromobenzyl)-4-(trifluoromethyl)-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H14BrF3N2O3
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2
|
| 1 |
IC50 = 2570.4 nM
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| 2 |
Ki < 1995.26 nM
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CP0449088
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7-{(1R,2R,3R,5S)-2-[(R)-5-(2-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid
Show/Hide
|
C23H35FO5
|
1
|
| 1 |
IC50 = 3100 nM
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CP0466595
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7-{(1R,2R,3R,5S)-2-[(R)-5-(4-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid
Show/Hide
|
C23H35FO5
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1
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| 1 |
IC50 = 3450 nM
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CP0927507
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1-(2-(3,5-bis(trifluoromethyl)benzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C21H15BrF6N2O3
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2
|
| 1 |
IC50 = 5248.07 nM
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| 2 |
Ki < 1995.26 nM
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CP0404058
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7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(3-trifluoromethyl-phenyl)-pentyl]-cyclopentyl}-heptanoic acid
Show/Hide
|
C24H35F3O5
|
1
|
| 1 |
IC50 > 10000 nM
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CP0425924
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7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Cyano-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid
Show/Hide
|
C24H35NO5
|
1
|
| 1 |
IC50 > 10000 nM
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CP0428991
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7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Ethyl-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid
Show/Hide
|
C25H40O5
|
1
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| 1 |
IC50 > 10000 nM
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CP0453390
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7-[(1R,2R,3R,5S)-3,5-Dihydroxy-2-((R)-3-hydroxy-5-o-tolyl-pentyl)-cyclopentyl]-heptanoic acid
Show/Hide
|
C24H38O5
|
1
|
| 1 |
IC50 = 10000 nM
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CP0453409
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7-{(1R,2R,3R,5S)-2-[(R)-5-(3-Fluoro-phenyl)-3-hydroxy-pentyl]-3,5-dihydroxy-cyclopentyl}-heptanoic acid
Show/Hide
|
C23H35FO5
|
1
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| 1 |
IC50 = 10000 nM
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CP0457103
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7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(4-methoxy-phenyl)-pentyl]-cyclopentyl}-heptanoic acid
Show/Hide
|
C24H38O6
|
1
|
| 1 |
IC50 > 10000 nM
|
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CP0456706
|
7-{(1R,2R,3R,5S)-3,5-Dihydroxy-2-[(R)-3-hydroxy-5-(3-methoxy-phenyl)-pentyl]-cyclopentyl}-heptanoic acid
Show/Hide
|
C24H38O6
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0042409
|
2-[2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C28H26N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0042410
|
2-[8-chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H19ClN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0045673
|
2-[2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H16ClFN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055416
|
2-[2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H20N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055418
|
2-[6-chloro-2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H15Cl2FN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055420
|
2-[2-(3-chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H17ClN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055873
|
2-[8-fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C23H20FN3O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055874
|
2-[8-fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C18H15FN2O3S
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0055877
|
2-[2-benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C21H17F3N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0070143
|
2-(2-benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C20H18N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0083568
|
2-[8-fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C26H23FN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0086399
|
2-[6-chloro-2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C28H25ClN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0086409
|
2-[8-fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H21FN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0087804
|
ACT-129968
Show/Hide
|
C24H19FN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0130562
|
2-[8-methyl-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H22N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0156867
|
2-[2-(cyclohexanecarbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H24N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0156868
|
2-[6-chloro-8-fluoro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H18ClFN2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0199029
|
2-(2-benzoyl-8-propan-2-yl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0199053
|
2-(2-benzoyl-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C21H20N2O4
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0261961
|
2-[2-(naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H19F3N2O3
|
1
|
| 1 |
IC50 > 25000 nM
|
|
|
|
CP0876913
|
sodium 2-(6-chloro-3-isobutyl-1H-indol-1-yl)acetate
Show/Hide
|
C14H15ClNNaO2
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0876914
|
sodium 2-(6-chloro-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C12H6ClN2NaO2S
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0877640
|
sodium 2-(6-chloro-3-((dimethylamino)methyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C15H13ClN3NaO2S
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0895231
|
sodium 2-(6-chloro-3-isobutyl-1H-indol-1-yl)benzoate
Show/Hide
|
C19H17ClNNaO2
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0895238
|
sodium 6-(2-(benzyloxy)phenylamino)picolinate
Show/Hide
|
C19H15N2NaO3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0910973
|
sodium 2-(6-chloro-3-(2-(dimethylamino)ethyl)-1H-indol-1-yl)thiazole-4-carboxylate
Show/Hide
|
C16H15ClN3NaO2S
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0889347
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)pyridin-3-yl)benzoic acid
Show/Hide
|
C25H18ClNO3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0889348
|
3-(4-(2-(benzyloxy)-5-chlorophenyl)-5-oxo-2,5-dihydrofuran-3-yl)benzoic acid
Show/Hide
|
C24H17ClO5
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0889349
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)-1H-imidazol-1-yl)benzoic acid
Show/Hide
|
C23H17ClN2O3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0889350
|
3-(2-(2-(benzyloxy)-5-chlorophenyl)-2H-1,2,4-triazol-3-yl)benzoic acid
Show/Hide
|
C22H16ClN3O3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0889351
|
3-(5-(2-(benzyloxy)-5-chlorophenyl)-1H-1,2,4-triazol-1-yl)benzoic acid
Show/Hide
|
C22H16ClN3O3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0894450
|
3-(1-(2-(benzyloxy)-5-chlorophenyl)-1H-pyrazol-5-yl)benzoic acid
Show/Hide
|
C23H17ClN2O3
|
1
|
| 1 |
IC50 < 1000 nM
|
|
|
|
CP0492339
|
1-[(6-chloro-2-propan-2-ylpyrazolo[1,5-a]pyridin-4-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H17ClN4O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0427457
|
1-[(7-chloro-2-propan-2-ylimidazo[1,2-a]pyridin-5-yl)methyl]-5-methylpyrazole-3-carboxylic acid
Show/Hide
|
C16H17ClN4O2
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0849115
|
1-(2-(2,4-dichlorobenzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15Cl3N2O3
|
2
|
| 1 |
IC50 < 1995.26 nM
|
|
|
| 2 |
Ki = 0.5495 nM
|
|
|
|
CP0918353
|
1-(2-(2,4-difluorobenzyloxy)-5-chlorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15ClF2N2O3
|
2
|
| 1 |
IC50 < 1995.26 nM
|
|
|
| 2 |
Ki = 1.122 nM
|
|
|
|
CP0932565
|
1-(2-(2,4-difluorobenzyloxy)-5-fluorobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15F3N2O3
|
2
|
| 1 |
IC50 < 1995.26 nM
|
|
|
| 2 |
Ki = 7.943 nM
|
|
|
|
CP0941379
|
1-(2-(2,4-dichlorobenzyloxy)benzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H16Cl2N2O3
|
2
|
| 1 |
IC50 < 1995.26 nM
|
|
|
| 2 |
Ki = 8.318 nM
|
|
|
|
CP0915925
|
N-[2-(4-hydroxy-3-methylsulfamoyl-phenyl)-ethyl]-2-[(toluene-4-sulfonyl)-o-tolyl-amino]-acetamide
Show/Hide
|
C25H29N3O6S2
|
1
|
| 1 |
Ki = 3.715 nM
|
|
|
|
CP0035659
|
N-[(4-chlorophenyl)methyl]-2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)acetamide
Show/Hide
|
C24H25ClN2O3S
|
1
|
| 1 |
Ki = 11.48 nM
|
|
|
|
CP0918667
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2,3-dimethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C27H32N2O5S
|
1
|
| 1 |
Ki = 12.88 nM
|
|
|
|
CP0897850
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C27H32N2O5S
|
1
|
| 1 |
Ki = 13.49 nM
|
|
|
|
CP0915924
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-(trifluoromethyl)phenylsulfonamido)acetamide
Show/Hide
|
C27H29F3N2O5S
|
1
|
| 1 |
Ki = 19.05 nM
|
|
|
|
CP0913678
|
N-(4-bromobenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C24H25BrN2O3S
|
1
|
| 1 |
Ki = 22.91 nM
|
|
|
|
CP0897833
|
N-(3,4-dimethoxyphenethyl)-2-(4-bromo-N-(2-ethylphenyl)phenylsulfonamido)acetamide
Show/Hide
|
C26H29BrN2O5S
|
1
|
| 1 |
Ki = 28.84 nM
|
|
|
|
CP0897848
|
N-(3,4-dimethoxyphenethyl)-2-(4-methyl-N-(3-(trifluoromethyl)phenyl)phenylsulfonamido)acetamide
Show/Hide
|
C26H27F3N2O5S
|
1
|
| 1 |
Ki = 30.9 nM
|
|
|
|
CP0897847
|
N-(3,4-dimethoxyphenethyl)-2-(4-cyano-N-(2-ethylphenyl)phenylsulfonamido)acetamide
Show/Hide
|
C27H29N3O5S
|
1
|
| 1 |
Ki = 31.62 nM
|
|
|
|
CP0920873
|
N-(3,4-dimethoxyphenethyl)-2-(N-(3-bromophenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H27BrN2O5S
|
1
|
| 1 |
Ki = 34.67 nM
|
|
|
|
CP0484317
|
2-(2-ethyl-N-(4-methylphenyl)sulfonylanilino)-N-[(4-methoxyphenyl)methyl]acetamide
Show/Hide
|
C25H28N2O4S
|
1
|
| 1 |
Ki = 35.48 nM
|
|
|
|
CP0844859
|
N-(3,4-dimethoxyphenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C26H30N2O5S
|
1
|
| 1 |
Ki = 38.9 nM
|
|
|
|
CP0873268
|
N-(3,4-dimethoxyphenethyl)-2-(N-(3-chlorophenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H27ClN2O5S
|
1
|
| 1 |
Ki = 61.66 nM
|
|
|
|
CP0895711
|
N-(3,4-dimethoxyphenethyl)-2-(4-methyl-N-m-tolylphenylsulfonamido)acetamide
Show/Hide
|
C26H30N2O5S
|
1
|
| 1 |
Ki = 61.66 nM
|
|
|
|
CP0844857
|
N-(2-fluoro-3,4-dimethoxyphenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C26H29FN2O5S
|
1
|
| 1 |
Ki = 66.07 nM
|
|
|
|
CP0962766
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-(trifluoromethoxy)phenylsulfonamido)acetamide
Show/Hide
|
C27H29F3N2O6S
|
1
|
| 1 |
Ki = 69.18 nM
|
|
|
|
CP0945784
|
1-(2-(2-methoxybenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C20H19BrN2O4
|
1
|
| 1 |
Ki = 69.18 nM
|
|
|
|
CP0915906
|
N-(4-chlorobenzyl)-2-(N-(1-ethyl-1H-pyrazol-5-yl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C21H23ClN4O3S
|
1
|
| 1 |
Ki = 72.44 nM
|
|
|
|
CP0869852
|
N-(4-(methylsulfonamido)phenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C25H29N3O5S2
|
1
|
| 1 |
Ki = 89.13 nM
|
|
|
|
CP0897846
|
N-(2-fluorobenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C24H25FN2O3S
|
1
|
| 1 |
Ki = 134.9 nM
|
|
|
|
CP0882726
|
N-(3-methoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H28N2O4S
|
1
|
| 1 |
Ki = 138.04 nM
|
|
|
|
CP0844855
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-2-methylphenylsulfonamido)acetamide
Show/Hide
|
C27H32N2O5S
|
1
|
| 1 |
Ki = 165.96 nM
|
|
|
|
CP0873261
|
N-(4-methoxyphenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C25H28N2O4S
|
1
|
| 1 |
Ki = 169.82 nM
|
|
|
|
CP0922539
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-4-methoxyphenylsulfonamido)acetamide
Show/Hide
|
C27H32N2O6S
|
1
|
| 1 |
Ki = 169.82 nM
|
|
|
|
CP0935548
|
N-(3-hydroxyphenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C24H26N2O4S
|
1
|
| 1 |
Ki = 204.17 nM
|
|
|
|
CP0913677
|
N-(4-(trifluoromethyl)benzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H25F3N2O3S
|
1
|
| 1 |
Ki = 208.93 nM
|
|
|
|
CP0897849
|
N-benzyl-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C24H26N2O3S
|
1
|
| 1 |
Ki = 223.87 nM
|
|
|
|
CP0895710
|
N-(3,4-dimethoxyphenethyl)-2-(3-cyano-N-(2-ethylphenyl)phenylsulfonamido)acetamide
Show/Hide
|
C27H29N3O5S
|
1
|
| 1 |
Ki = 239.88 nM
|
|
|
|
CP0915923
|
N-(3,4-dimethoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C26H30N2O5S
|
1
|
| 1 |
Ki = 281.84 nM
|
|
|
|
CP0942003
|
1-(2-(3-nitrobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H16BrN3O5
|
1
|
| 1 |
Ki = 338.84 nM
|
|
|
|
CP0926452
|
N-(3-(trifluoromethoxy)benzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H25F3N2O4S
|
1
|
| 1 |
Ki = 426.58 nM
|
|
|
|
CP0844860
|
N-(4-chlorobenzyl)-2-(4-methyl-N-(1-methyl-1H-pyrazol-5-yl)phenylsulfonamido)acetamide
Show/Hide
|
C20H21ClN4O3S
|
1
|
| 1 |
Ki = 588.84 nM
|
|
|
|
CP0913667
|
N-(3,4-dimethoxyphenethyl)-2-(4-methyl-N-phenylphenylsulfonamido)acetamide
Show/Hide
|
C25H28N2O5S
|
1
|
| 1 |
Ki = 588.84 nM
|
|
|
|
CP0652436
|
N-(4-chlorophenethyl)-2-(4-methyl-N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C24H25ClN2O3S
|
1
|
| 1 |
Ki = 660.69 nM
|
|
|
|
CP0844852
|
N-(4-chlorobenzyl)-2-(4-methyl-N-(2-methylpyridin-3-yl)phenylsulfonamido)acetamide
Show/Hide
|
C22H22ClN3O3S
|
1
|
| 1 |
Ki = 676.08 nM
|
|
|
|
CP0844853
|
N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-3-(trifluoromethoxy)phenylsulfonamido)acetamide
Show/Hide
|
C27H29F3N2O6S
|
1
|
| 1 |
Ki = 707.95 nM
|
|
|
|
CP0939751
|
N-(3,4-dimethoxyphenethyl)-2-(N-o-tolylphenylsulfonamido)acetamide
Show/Hide
|
C25H28N2O5S
|
1
|
| 1 |
Ki = 741.31 nM
|
|
|
|
CP0940083
|
1-(2-(benzyloxy)-5-bromobenzyl)-5-butyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C22H23BrN2O3
|
1
|
| 1 |
Ki = 977.24 nM
|
|
|
|
CP0939749
|
N-(2-methoxybenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H28N2O4S
|
1
|
| 1 |
Ki = 1071.52 nM
|
|
|
|
CP0945783
|
1-(2-(3,5-dichlorobenzyloxy)-5-bromobenzyl)-5-methyl-1H-pyrazole-3-carboxylic acid
Show/Hide
|
C19H15BrCl2N2O3
|
1
|
| 1 |
Ki = 1122.02 nM
|
|
|
|
CP0962767
|
N-(3,4-dimethoxyphenethyl)-2-(N-(4-chlorophenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C25H27ClN2O5S
|
1
|
| 1 |
Ki = 1288.25 nM
|
|
|
|
CP0941207
|
2-(4-methyl-N-o-tolylphenylsulfonamido)-N-phenethylacetamide
Show/Hide
|
C24H26N2O3S
|
1
|
| 1 |
Ki = 1348.96 nM
|
|
|
|
CP0939750
|
N-(3-chlorobenzyl)-2-(N-(2-ethylphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
|
C24H25ClN2O3S
|
1
|
| 1 |
Ki = 1412.54 nM
|
|
|
|
CP0876565
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N-(3,4-dimethoxyphenethyl)-2-(N-(2-ethylphenyl)-3-methylphenylsulfonamido)acetamide
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C27H32N2O5S
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1
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| 1 |
Ki = 1659.59 nM
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CP0913679
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N-(3,4-dimethoxyphenethyl)-2-(2-chloro-N-(2-ethylphenyl)phenylsulfonamido)acetamide
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C26H29ClN2O5S
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1
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| 1 |
Ki = 1995.26 nM
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CP0897317
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N-(3,4-dimethoxyphenethyl)-2-(4-methyl-N-p-tolylphenylsulfonamido)acetamide
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C26H30N2O5S
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1
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| 1 |
Ki < 1122.02 nM
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CP0895712
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N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-3-yl)phenylsulfonamido)acetamide
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C22H22ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0902805
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N-(4-chlorobenzyl)-2-(4-methyl-N-(6-methylpyridin-2-yl)phenylsulfonamido)acetamide
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C22H22ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0915907
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N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
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C21H20ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0918668
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N-(4-chlorobenzyl)-2-(4-methyl-N-(pyridin-3-yl)phenylsulfonamido)acetamide
Show/Hide
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C21H20ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0918673
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N-(4-chlorobenzyl)-2-(4-methyl-N-(5-methylpyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
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C22H22ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0942223
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N-(4-chlorobenzyl)-2-(4-methyl-N-(3-methylpyridin-2-yl)phenylsulfonamido)acetamide
Show/Hide
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C22H22ClN3O3S
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1
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| 1 |
Ki < 1445.44 nM
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CP0922540
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N-(3,4-dimethoxyphenethyl)-2-(N-(4-fluorophenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C25H27FN2O5S
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1
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| 1 |
Ki < 1584.89 nM
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CP0939752
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N-(3,4-dimethoxyphenethyl)-2-(N-(4-methoxyphenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C26H30N2O6S
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1
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| 1 |
Ki < 1584.89 nM
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CP0846753
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1-(2-(benzyloxy)-5-bromobenzyl)-1H-imidazole-5-carboxylic acid
Show/Hide
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C18H15BrN2O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0899687
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1-(2-(benzyloxy)-5-bromobenzyl)-1H-imidazole-4-carboxylic acid
Show/Hide
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C18H15BrN2O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0916309
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1-(2-(benzyloxy)-5-bromobenzyl)-4-chloro-1H-pyrazole-3-carboxylic acid
Show/Hide
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C18H14BrClN2O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0916312
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1-(2-(benzyloxy)-5-bromobenzyl)-1H-pyrazole-4-carboxylic acid
Show/Hide
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C18H15BrN2O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0932545
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1-(2-(benzyloxy)-5-bromobenzyl)-1H-1,2,3-triazole-4-carboxylic acid
Show/Hide
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C17H14BrN3O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0941939
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1-(2-(benzyloxy)-5-bromobenzyl)-5-acetamido-1H-pyrazole-3-carboxylic acid
Show/Hide
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C20H18BrN3O4
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1
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| 1 |
Ki < 1995.26 nM
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CP0957120
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1-(2-(benzyloxy)-5-bromobenzyl)-1H-pyrazole-5-carboxylic acid
Show/Hide
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C18H15BrN2O3
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1
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| 1 |
Ki < 1995.26 nM
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CP0873267
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N-(3,4-dimethoxyphenethyl)-2-(2-cyano-N-(2-ethylphenyl)phenylsulfonamido)acetamide
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C27H29N3O5S
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1
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| 1 |
Ki < 3162.28 nM
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CP0924835
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N-(3,4-dimethoxyphenethyl)-2-(N-(4-bromophenyl)-4-methylphenylsulfonamido)acetamide
Show/Hide
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C25H27BrN2O5S
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1
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| 1 |
Ki < 3801.89 nM
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