| Compound ID |
Compound Name |
Compound Formula |
|
CP0071769
|
2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)benzimidazol-4-ol
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|
C19H21F2N7O3
|
2
|
| 1 |
IC50 = 1.3 nM
|
|
|
| 2 |
IC50 = 2.9 nM
|
|
|
|
CP0152367
|
N-[2-chloro-5-(4-pyridin-4-ylquinolin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C25H16ClFN4O2S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0072230
|
2-[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-2-[(5-fluoro-6-methoxypyridin-3-yl)amino]imidazo[1,2-a]pyridin-6-yl]propan-2-ol
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|
C20H21FN8O2
|
1
|
| 1 |
IC50 = 4.5 nM
|
|
|
|
CP0071675
|
2-(difluoromethyl)-3-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-7-methoxybenzimidazol-5-amine
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|
C20H24F2N8O3
|
2
|
| 1 |
IC50 = 4.8 nM
|
|
|
| 2 |
IC50 = 8.8 nM
|
|
|
|
CP0199338
|
N-[6-[6-chloro-5-[(4-fluorophenyl)sulfonylamino]pyridin-3-yl]-1,3-benzothiazol-2-yl]acetamide
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|
C20H14ClFN4O3S2
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
|
CP0210324
|
N-[2-chloro-5-(4-pyridin-3-ylquinolin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C25H16ClFN4O2S
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0252844
|
N-[2-chloro-5-(4-morpholin-4-ylquinolin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C24H20ClFN4O3S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0298054
|
N-[2-chloro-5-[3-(4-propan-2-ylpiperazin-1-yl)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C26H26ClFN6O2S
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0090562
|
N-[2-chloro-5-[4-[4-(pyridin-4-ylmethyl)piperazin-1-yl]quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C30H26ClFN6O2S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0491652
|
N-[2-chloro-5-[3-(2-piperidin-1-ylethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C26H26ClFN6O2S
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0649593
|
N-(3-(4-amino-6-methyl-1,3,5-triazin-2-yl)imidazo[1,2-a]pyridin-2-yl)quinolin-7-amine
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|
C20H16N8
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0090561
|
N-[2-chloro-5-(3-morpholin-4-ylquinoxalin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C23H19ClFN5O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0688569
|
4-(3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-2-(5-fluoro-6-methoxypyridin-3-ylamino)imidazo[1,2-a]pyridin-6-yl)-N,N-dimethylpiperazine-1-carboxamide
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|
C24H28FN11O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0491653
|
N-(2-chloro-5-quinazolin-6-ylpyridin-3-yl)-4-fluorobenzenesulfonamide
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|
C19H12ClFN4O2S
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0399013
|
N-[2-chloro-5-(3-pyridin-4-ylquinoxalin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C24H15ClFN5O2S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0750883
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(5-fluoro-6-methoxypyridin-3-yl)-6-(4-(2-methoxyethyl)piperazin-1-yl)imidazo[1,2-a]pyridin-2-amine
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|
C24H29FN10O2
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0452381
|
4-[4-[2-(difluoromethyl)-4-methoxybenzimidazol-1-yl]-6-morpholin-4-yl-1,3,5-triazin-2-yl]morpholine
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|
C20H23F2N7O3
|
2
|
| 1 |
IC50 = 28 nM
|
|
|
| 2 |
IC50 = 55 nM
|
|
|
|
CP0399012
|
N-[2-chloro-5-[4-(4-propan-2-ylpiperazin-1-yl)quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C27H27ClFN5O2S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0007933
|
2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-1H-benzimidazole
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|
C19H21F2N7O2
|
2
|
| 1 |
IC50 = 32 nM
|
|
|
| 2 |
IC50 = 111 nM
|
|
|
|
CP0252600
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(1H-indazol-4-yl)imidazo[1,2-a]pyridin-2-amine
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|
C18H15N9
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0717560
|
4-(3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-2-(6-methoxypyridin-3-ylamino)imidazo[1,2-a]pyridin-6-yl)-N,N-dimethylpiperazine-1-carboxamide
Show/Hide
|
C24H29N11O2
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0177940
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(6-methoxypyridin-3-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C17H16N8O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0750882
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(5-fluoro-6-methoxypyridin-3-yl)-6-(piperazin-1-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C21H23FN10O
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0252843
|
N-[2-chloro-5-[3-(2-morpholin-4-ylethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C25H24ClFN6O3S
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0295372
|
N-[5-(2-amino-1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C18H12ClFN4O2S2
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0431312
|
N-[2-chloro-5-[3-(dimethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C21H17ClFN5O2S
|
1
|
| 1 |
IC50 = 44 nM
|
|
|
|
CP0711390
|
2-(3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-2-(6-methoxypyridin-3-ylamino)imidazo[1,2-a]pyridin-6-yl)propan-2-ol
Show/Hide
|
C20H22N8O2
|
1
|
| 1 |
IC50 = 45 nM
|
|
|
|
CP0427666
|
N-[2-chloro-5-[3-(4-methoxypiperidin-1-yl)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C25H23ClFN5O3S
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0431313
|
N-[2-chloro-5-[3-(2-methoxyethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C22H19ClFN5O3S
|
1
|
| 1 |
IC50 = 54 nM
|
|
|
|
CP0533259
|
N-[2-chloro-5-[3-[2-methoxyethyl(methyl)amino]quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C23H21ClFN5O3S
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0391659
|
N-[2-chloro-5-[4-[4-(dimethylamino)phenyl]quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C28H22ClFN4O2S
|
1
|
| 1 |
IC50 = 61 nM
|
|
|
|
CP0731810
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(6-methoxypyridin-3-yl)-6-(piperazin-1-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C21H24N10O
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0252602
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(5-fluoro-6-methoxypyridin-3-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C17H15FN8O
|
1
|
| 1 |
IC50 = 86 nM
|
|
|
|
CP0475656
|
N-[2-chloro-5-(4-phenylquinolin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C26H17ClFN3O2S
|
1
|
| 1 |
IC50 = 127 nM
|
|
|
|
CP0461919
|
N-[2-chloro-5-(3-piperidin-1-ylquinoxalin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C24H21ClFN5O2S
|
1
|
| 1 |
IC50 = 128 nM
|
|
|
|
CP0431310
|
N-[5-[4-(4-benzylpiperazin-1-yl)quinolin-6-yl]-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
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|
C31H27ClFN5O2S
|
1
|
| 1 |
IC50 = 136 nM
|
|
|
|
CP0390761
|
N-[2-chloro-5-[4-(4-hydroxypiperidin-1-yl)quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C25H22ClFN4O3S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0476557
|
N-[2-chloro-5-[3-(4,4-difluoropiperidin-1-yl)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C24H19ClF3N5O2S
|
1
|
| 1 |
IC50 = 189 nM
|
|
|
|
CP0387479
|
N-[2-chloro-5-[4-(dimethylamino)quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C22H18ClFN4O2S
|
1
|
| 1 |
IC50 = 223 nM
|
|
|
|
CP0173323
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(6-ethoxypyridin-3-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C18H18N8O
|
1
|
| 1 |
IC50 = 229 nM
|
|
|
|
CP0495442
|
N-[2-chloro-5-[3-(2-phenylethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C27H21ClFN5O2S
|
1
|
| 1 |
IC50 = 241 nM
|
|
|
|
CP0461823
|
N-[5-[3-(3-azabicyclo[3.2.2]nonan-3-yl)quinoxalin-6-yl]-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C27H25ClFN5O2S
|
1
|
| 1 |
IC50 = 247 nM
|
|
|
|
CP0505973
|
N-[5-[3-[benzyl(methyl)amino]quinoxalin-6-yl]-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C27H21ClFN5O2S
|
1
|
| 1 |
IC50 = 258 nM
|
|
|
|
CP0399396
|
N-[2-chloro-5-[3-(cyclohexylmethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C26H25ClFN5O2S
|
1
|
| 1 |
IC50 = 281 nM
|
|
|
|
CP0765233
|
3-(4-amino-6-methyl-1,3,5-triazin-2-yl)-N-(5-fluoro-6-methoxypyridin-3-yl)-6-(4-isopropylpiperazin-1-yl)imidazo[1,2-a]pyridin-2-amine
Show/Hide
|
C24H29FN10O
|
1
|
| 1 |
IC50 = 294 nM
|
|
|
|
CP0387452
|
N-(2-chloro-5-quinolin-6-ylpyridin-3-yl)-4-fluorobenzenesulfonamide
Show/Hide
|
C20H13ClFN3O2S
|
1
|
| 1 |
IC50 = 377 nM
|
|
|
|
CP0071674
|
2-(difluoromethyl)-1-(4,6-dimorpholin-4-yl-1,3,5-triazin-2-yl)-5-methoxybenzimidazol-4-ol
Show/Hide
|
C20H23F2N7O4
|
2
|
| 1 |
IC50 = 378 nM
|
|
|
| 2 |
IC50 = 583 nM
|
|
|
|
CP0075331
|
4-[4-[4-(difluoromethoxy)-2-(difluoromethyl)benzimidazol-1-yl]-6-morpholin-4-yl-1,3,5-triazin-2-yl]morpholine
Show/Hide
|
C20H21F4N7O3
|
2
|
| 1 |
IC50 = 418 nM
|
|
|
| 2 |
IC50 = 427 nM
|
|
|
|
CP0461818
|
N-[2-chloro-5-(4-piperidin-1-ylquinolin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C25H22ClFN4O2S
|
1
|
| 1 |
IC50 = 498 nM
|
|
|
|
CP0191632
|
N-[5-(1,3-benzothiazol-6-yl)-2-chloropyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C18H11ClFN3O2S2
|
1
|
| 1 |
IC50 = 769 nM
|
|
|
|
CP0476558
|
N-[2-chloro-5-(1,5-naphthyridin-2-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C19H12ClFN4O2S
|
1
|
| 1 |
IC50 = 784 nM
|
|
|
|
CP0505974
|
N-[2-chloro-5-[4-(2-methoxyethylamino)quinolin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C23H20ClFN4O3S
|
1
|
| 1 |
IC50 = 1020 nM
|
|
|
|
CP0431311
|
N-(2-chloro-5-quinoxalin-6-ylpyridin-3-yl)-4-fluorobenzenesulfonamide
Show/Hide
|
C19H12ClFN4O2S
|
1
|
| 1 |
IC50 = 1450 nM
|
|
|
|
CP0461822
|
N-(2-chloro-5-cinnolin-6-ylpyridin-3-yl)-4-fluorobenzenesulfonamide
Show/Hide
|
C19H12ClFN4O2S
|
1
|
| 1 |
IC50 = 1920 nM
|
|
|
|
CP0431314
|
N-[2-chloro-5-[3-(piperidin-3-ylmethylamino)quinoxalin-6-yl]pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C25H24ClFN6O2S
|
1
|
| 1 |
IC50 = 2710 nM
|
|
|
|
CP0387453
|
N-(2-chloro-5-isoquinolin-6-ylpyridin-3-yl)-4-fluorobenzenesulfonamide
Show/Hide
|
C20H13ClFN3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0387454
|
N-[2-chloro-5-(1,7-naphthyridin-6-yl)pyridin-3-yl]-4-fluorobenzenesulfonamide
Show/Hide
|
C19H12ClFN4O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0041963
|
N-[3-(4-amino-6-methyl-1,3,5-triazin-2-yl)imidazo[1,2-a]pyridin-2-yl]quinolin-6-amine
Show/Hide
|
C20H16N8
|
1
|
| 1 |
IC50 > 780 nM
|
|
|
