| Compound ID |
Compound Name |
Compound Formula |
|
CP0565199
|
4-[[(1S,2S)-2-[(3R)-3-aminopiperidin-1-yl]-4,6-dichloro-2,3-dihydro-1H-inden-1-yl]oxy]-2,3-dichlorobenzenesulfonamide
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|
C20H21Cl4N3O3S
|
1
|
| 1 |
IC50 = 0.2 nM
|
|
|
|
CP0446579
|
1-[(1S,2S)-4,6-dichloro-1-(2-chloro-4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-1,4-diazepane
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|
C21H23Cl3N2O3S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0419623
|
2-[[(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperidin-3-yl]amino]ethanol
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|
C23H28Cl2N2O4S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0470843
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperidin-3-amine
Show/Hide
|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 4 nM
|
|
|
|
CP0470842
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-1,4-diazepane
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|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 6 nM
|
|
|
|
CP0525409
|
2-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-2,7-diazaspiro[4.4]nonane
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|
C23H26Cl2N2O3S
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0446582
|
1-[(1S,2S)-4,6-dichloro-1-[4-(3,5-dimethyl-1,2,4-triazol-4-yl)phenoxy]-2,3-dihydro-1H-inden-2-yl]-4-methyl-1,4-diazepane
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|
C25H29Cl2N5O
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0395693
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-3-methylpiperazine
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|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0530958
|
N'-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-N,N,N'-trimethylethane-1,2-diamine
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|
C21H26Cl2N2O3S
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0667979
|
N-carbamimidoyl-3-(2-((E)-3-(diaminomethyleneamino)-2-methyl-3-oxoprop-1-enyl)-4-methylphenyl)-2-methylacrylamide
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|
C17H22N6O2
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0525410
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
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|
C20H22Cl2N2O3S
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0455982
|
1-[(1S,2S)-4,6-dichloro-1-[4-(3,5-dimethyl-1,2,4-triazol-4-yl)phenoxy]-2,3-dihydro-1H-inden-2-yl]-1,4-diazepane
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|
C24H27Cl2N5O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0566697
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-imidazol-1-ylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperidin-3-amine
Show/Hide
|
C23H24Cl2N4O
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0555868
|
(3aR,6aS)-5-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-2,3,3a,4,6,6a-hexahydro-1H-pyrrolo[3,4-c]pyrrole
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|
C22H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0510180
|
2-[4-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-1,4-diazepan-1-yl]ethanol
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|
C23H28Cl2N2O4S
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0565198
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-[4-(1,2,4-triazol-1-yl)phenoxy]-2,3-dihydro-1H-inden-2-yl]piperidin-3-amine
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|
C22H23Cl2N5O
|
1
|
| 1 |
IC50 = 30 nM
|
|
|
|
CP0555870
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-[4-(3,5-dimethyl-1,2,4-triazol-4-yl)-2-fluorophenoxy]-2,3-dihydro-1H-inden-2-yl]pyrrolidin-3-ol
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|
C23H23Cl2FN4O2
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0573923
|
1-[(1S,2S)-6,7-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-1,4-diazepane
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|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0419626
|
N'-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-N,N,N'-trimethylpropane-1,3-diamine
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|
C22H28Cl2N2O3S
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0555867
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-N-(2-fluoroethyl)piperidin-3-amine
Show/Hide
|
C23H27Cl2FN2O3S
|
1
|
| 1 |
IC50 = 56 nM
|
|
|
|
CP0555866
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-4-(2-methoxyethyl)-1,4-diazepane
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|
C24H30Cl2N2O4S
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0419628
|
4-[3-chloro-4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-3,5-dimethyl-1,2,4-triazole
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|
C23H25ClN4O
|
1
|
| 1 |
IC50 = 78 nM
|
|
|
|
CP0463890
|
(3R)-1-[(1S,2S)-6-chloro-1-[2-chloro-4-(3,5-dimethyl-1,2,4-triazol-4-yl)phenoxy]-2,3-dihydro-1H-inden-2-yl]pyrrolidin-3-ol
Show/Hide
|
C23H24Cl2N4O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0419627
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-4-methyl-1,4-diazepane
Show/Hide
|
C22H26Cl2N2O3S
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0514472
|
4-[3-chloro-4-[[(1S,2S)-6-chloro-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-3,5-dimethyl-1,2,4-triazole
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|
C23H24Cl2N4O
|
1
|
| 1 |
IC50 = 94 nM
|
|
|
|
CP0566871
|
3,5-dimethyl-4-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]-3-(trifluoromethyl)phenyl]-1,2,4-triazole
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|
C24H25F3N4O
|
1
|
| 1 |
IC50 = 118 nM
|
|
|
|
CP0446578
|
1-[(1S,2S)-4-chloro-6-fluoro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
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|
C20H22ClFN2O3S
|
1
|
| 1 |
IC50 = 123 nM
|
|
|
|
CP0458114
|
2,3-dichloro-4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]benzenesulfonamide
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|
C19H20Cl2N2O3S
|
1
|
| 1 |
IC50 = 123 nM
|
|
|
|
CP0419625
|
1-[(1S,2S)-5,7-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
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|
C20H22Cl2N2O3S
|
1
|
| 1 |
IC50 = 135 nM
|
|
|
|
CP0510182
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-3-fluoropyrrolidine
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|
C20H20Cl2FNO3S
|
1
|
| 1 |
IC50 = 166 nM
|
|
|
|
CP0573925
|
1-[(1S,2S)-6-chloro-4-fluoro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
Show/Hide
|
C20H22ClFN2O3S
|
1
|
| 1 |
IC50 = 168 nM
|
|
|
|
CP0514541
|
4-[2,3-dimethyl-4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-3,5-dimethyl-1,2,4-triazole
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|
C25H30N4O
|
1
|
| 1 |
IC50 = 170 nM
|
|
|
|
CP0470846
|
1-methyl-3-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]imidazol-2-one
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|
C23H25N3O2
|
1
|
| 1 |
IC50 = 197 nM
|
|
|
|
CP0572626
|
(3aS,6aR)-5-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-2-methyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole
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|
C23H26Cl2N2O3S
|
1
|
| 1 |
IC50 = 241 nM
|
|
|
|
CP0536432
|
3-cyclopropyl-5-methyl-4-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,2,4-triazole
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|
C25H28N4O
|
1
|
| 1 |
IC50 = 272 nM
|
|
|
|
CP0514474
|
3-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1H-imidazol-2-one
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|
C22H23N3O2
|
1
|
| 1 |
IC50 = 281 nM
|
|
|
|
CP0530960
|
[3-[[(1S,2S)-2-[(3R)-3-aminopiperidin-1-yl]-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]urea
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|
C21H26N4O2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0566699
|
3,5-dimethyl-4-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,2,4-triazole
Show/Hide
|
C23H26N4O
|
1
|
| 1 |
IC50 = 345 nM
|
|
|
|
CP0470845
|
(3S)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]pyrrolidin-3-ol
Show/Hide
|
C20H21Cl2NO4S
|
1
|
| 1 |
IC50 = 384 nM
|
|
|
|
CP0455986
|
3,5-dimethyl-4-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,2-oxazole
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|
C24H26N2O2
|
1
|
| 1 |
IC50 = 411 nM
|
|
|
|
CP0419631
|
N-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]acetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 438 nM
|
|
|
|
CP0463891
|
N-[3-[[(1S,2S)-2-[(3R)-3-aminopiperidin-1-yl]-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]acetamide
Show/Hide
|
C22H27N3O2
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
|
CP0555872
|
2,3-dichloro-N-methyl-4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]benzenesulfonamide
Show/Hide
|
C20H22Cl2N2O3S
|
1
|
| 1 |
IC50 = 475 nM
|
|
|
|
CP0419630
|
4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]benzenesulfonamide
Show/Hide
|
C19H22N2O3S
|
1
|
| 1 |
IC50 = 500 nM
|
|
|
|
CP0395695
|
1-[(1S,2S)-6-chloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
Show/Hide
|
C20H23ClN2O3S
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0455984
|
1-[(1S,2S)-1-(2,3-dichloro-4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]pyrrolidine
Show/Hide
|
C20H21Cl2NO3S
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
|
CP0446585
|
1-[(1S,2S)-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]pyrrolidine
Show/Hide
|
C20H23NO3S
|
1
|
| 1 |
IC50 = 572 nM
|
|
|
|
CP0573926
|
(3R)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]pyrrolidin-3-ol
Show/Hide
|
C20H21Cl2NO4S
|
1
|
| 1 |
IC50 = 588 nM
|
|
|
|
CP0514545
|
3-methyl-4-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,2,4-triazole
Show/Hide
|
C22H24N4O
|
1
|
| 1 |
IC50 = 640 nM
|
|
|
|
CP0419633
|
4-[[(1S,2S)-2-[(3R)-3-aminopiperidin-1-yl]-2,3-dihydro-1H-inden-1-yl]oxy]-2,3-dichlorobenzenesulfonamide
Show/Hide
|
C20H23Cl2N3O3S
|
1
|
| 1 |
IC50 = 650 nM
|
|
|
|
CP0565200
|
1-[(1S,2S)-6-chloro-4-fluoro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]pyrrolidine
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|
C20H21ClFNO3S
|
1
|
| 1 |
IC50 = 737 nM
|
|
|
|
CP0510181
|
(3S)-1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-3-fluoropyrrolidine
Show/Hide
|
C20H20Cl2FNO3S
|
1
|
| 1 |
IC50 = 883 nM
|
|
|
|
CP0514473
|
3-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,3-oxazolidin-2-one
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|
C22H24N2O3
|
1
|
| 1 |
IC50 = 955 nM
|
|
|
|
CP0731184
|
N-carbamimidoyl-3-(3-((E)-3-(diaminomethyleneamino)-2-methyl-3-oxoprop-1-enyl)phenyl)-2-methylacrylamide
Show/Hide
|
C16H20N6O2
|
1
|
| 1 |
IC50 = 1320 nM
|
|
|
|
CP0514543
|
2-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,2-thiazolidine 1,1-dioxide
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|
C22H26N2O3S
|
1
|
| 1 |
IC50 = 1530 nM
|
|
|
|
CP0446580
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]azetidin-3-ol
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|
C19H19Cl2NO4S
|
1
|
| 1 |
IC50 = 1640 nM
|
|
|
|
CP0446583
|
2-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]-1,3-thiazole
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|
C22H22N2OS
|
1
|
| 1 |
IC50 = 1710 nM
|
|
|
|
CP0514542
|
N,N-diethyl-4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]benzamide
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|
C24H30N2O2
|
1
|
| 1 |
IC50 = 2070 nM
|
|
|
|
CP0573908
|
5-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]-3H-2-benzofuran-1-one
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|
C21H21NO3
|
1
|
| 1 |
IC50 = 2440 nM
|
|
|
|
CP0514546
|
N-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]acetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 2770 nM
|
|
|
|
CP0530959
|
1-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]pyrrolidine-2,5-dione
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
IC50 = 2960 nM
|
|
|
|
CP0573924
|
1-[(1S,2S)-6-fluoro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
Show/Hide
|
C20H23FN2O3S
|
1
|
| 1 |
IC50 = 3490 nM
|
|
|
|
CP0419629
|
1-[3-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]phenyl]pyrrolidin-2-one
Show/Hide
|
C23H26N2O2
|
1
|
| 1 |
IC50 = 3520 nM
|
|
|
|
CP0566698
|
1-[(1S,2S)-4,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-4-methylpiperazine
Show/Hide
|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 4040 nM
|
|
|
|
CP0470847
|
4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]benzonitrile
Show/Hide
|
C20H20N2O
|
1
|
| 1 |
IC50 = 4500 nM
|
|
|
|
CP0446584
|
N-[4-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]pyridin-2-yl]acetamide
Show/Hide
|
C20H23N3O2
|
1
|
| 1 |
IC50 = 4530 nM
|
|
|
|
CP0419624
|
1-[(1S,2S)-5,6-dichloro-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]-1,4-diazepane
Show/Hide
|
C21H24Cl2N2O3S
|
1
|
| 1 |
IC50 = 6055 nM
|
|
|
|
CP0555869
|
1-[(1S,2S)-1-(4-methylsulfonylphenoxy)-2,3-dihydro-1H-inden-2-yl]piperazine
Show/Hide
|
C20H24N2O3S
|
1
|
| 1 |
IC50 = 6680 nM
|
|
|
|
CP0514544
|
8-[[(1S,2S)-2-pyrrolidin-1-yl-2,3-dihydro-1H-inden-1-yl]oxy]quinoline
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C22H22N2O
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1
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| 1 |
IC50 = 9520 nM
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CP0864469
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N''-[(3S)-3-(5-fluoro-2-methylphenyl)-3,4-dihydronaphthalen-1(2H)-ylidene]carbonohydrazonic diamide
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C18H19FN4
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1
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| 1 |
IC50 = 11000 nM
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CP0864470
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N''-[(3R)-3-(5-fluoro-2-methylphenyl)-3,4-dihydronaphthalen-1(2H)-ylidene]carbonohydrazonic diamide
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C18H19FN4
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1
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| 1 |
IC50 > 30000 nM
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