| Compound ID |
Compound Name |
Compound Formula |
|
CP0192572
|
AVP
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|
C46H65N15O12S2
|
1
|
| 1 |
EC50 = 0.052 nM
|
|
|
|
CP0083253
|
(5H,11H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-yl)-[2-chloro-4-(3-methyl-pyrazol-1-yl)-phenyl]-methanone
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|
C23H19ClN4O
|
3
|
| 1 |
EC50 = 0.74 nM
|
|
|
| 2 |
IC50 = 80 nM
|
|
|
| 3 |
IC50 = 80.3 nM
|
|
|
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CP0464709
|
(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[4-(3-methyl-pyrazol-1-yl)-2-trifluoromethyl-phenyl]-methanone
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|
C24H18F3N5O
|
2
|
| 1 |
EC50 = 1.67 nM
|
|
|
| 2 |
IC50 = 493 nM
|
|
|
|
CP0040044
|
3-chloro-4-(10,11-dihydro-5H-benzo[e]pyrrolo[1,2-a][1,4]diazepin-10-ylcarbonyl)-1-(5-fluoro-2-methylphenylcarboxamido)benzene
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|
C27H21ClFN3O2
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0464708
|
[2-chloro-4-(3-methylpyrazol-1-yl)phenyl]-(5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl)methanone
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|
C23H18ClN5O
|
1
|
| 1 |
IC50 = 91.5 nM
|
|
|
|
CP0424718
|
[2-chloro-4-(1-methylpyrazol-3-yl)phenyl]-(5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl)methanone
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|
C23H18ClN5O
|
1
|
| 1 |
IC50 = 183 nM
|
|
|
|
CP0469331
|
[2-bromo-4-(3-methylpyrazol-1-yl)phenyl]-(5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl)methanone
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|
C23H18BrN5O
|
1
|
| 1 |
IC50 = 296 nM
|
|
|
|
CP0460147
|
[2-chloro-4-(5-methylpyrazol-1-yl)phenyl]-(5,11-dihydropyrido[3,2-c][1,5]benzodiazepin-6-yl)methanone
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|
C23H18ClN5O
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0469332
|
(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[4-(5-methyl-pyrazol-1-yl)-2-trifluoromethyl-phenyl]-methanone
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|
C24H18F3N5O
|
1
|
| 1 |
IC50 = 413 nM
|
|
|
|
CP0453679
|
[2-chloro-4-(3-methylpyrazol-1-yl)phenyl]-(11-methyl-5H-pyrido[3,2-c][1,5]benzodiazepin-6-yl)methanone
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|
C24H20ClN5O
|
1
|
| 1 |
IC50 = 475 nM
|
|
|
|
CP0424719
|
(5,11-dihydro-benzo[b]pyrido[2,3-e][1,4]diazepin-6-yl)-[2-fluoro-4-(3-methyl-pyrazol-1-yl)-phenyl]-methanone
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|
C23H18FN5O
|
1
|
| 1 |
IC50 = 933 nM
|
|
|
|
CP0373176
|
10-[2-chloro-4-(3-methyl-pyrazol-1-yl)-benzoyl]-1,2,5,10-tetrahydro-benzo[e]pyrrolo[1,2-a][1,4]diazepin-3-one
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|
C23H19ClN4O2
|
1
|
| 1 |
IC50 = 1214 nM
|
|
|
