| Compound ID |
Compound Name |
Compound Formula |
|
CP0037565
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(3-fluoro-4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C29H37FN2O6
|
1
|
| 1 |
IC50 = 0.07 nM
|
|
|
|
CP0320198
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(3,4-dimethoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C30H40N2O7
|
1
|
| 1 |
IC50 = 0.11 nM
|
|
|
|
CP0341585
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-p-tolyl-pyrrolidine-3-carboxylic acid
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|
C29H38N2O5
|
1
|
| 1 |
IC50 = 0.12 nM
|
|
|
|
CP0339897
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-ethyl-phenyl)-pyrrolidine-3-carboxylic acid
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|
C30H40N2O5
|
1
|
| 1 |
IC50 = 0.17 nM
|
|
|
|
CP0203851
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(3-fluoro-4-methoxy-phenyl)-1-{2-[(2-methyl-propane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H37FN2O7S
|
1
|
| 1 |
IC50 = 0.21 nM
|
|
|
|
CP0464147
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(butyl-propyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H36N2O6
|
1
|
| 1 |
IC50 = 0.22 nM
|
|
|
|
CP0037579
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H38N2O6
|
2
|
| 1 |
IC50 = 0.31 nM
|
|
|
| 2 |
IC50 = 0.36 nM
|
|
|
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CP0452000
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C29H38N2O6
|
1
|
| 1 |
IC50 = 0.36 nM
|
|
|
|
CP0372974
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-{[bis-(3-methyl-butyl)-carbamoyl]-methyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H42N2O6
|
1
|
| 1 |
IC50 = 0.43 nM
|
|
|
|
CP0185734
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(hexane-1-sulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H42N2O7S
|
1
|
| 1 |
IC50 = 0.43 nM
|
|
|
|
CP0573120
|
4-Benzo[1,3]dioxol-5-yl-1-(1-dibutylcarbamoyl-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C30H40N2O6
|
1
|
| 1 |
IC50 = 0.46 nM
|
|
|
|
CP0359230
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(3-fluoro-4-methoxy-phenyl)-1-{2-[(3-methyl-butane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H39FN2O7S
|
1
|
| 1 |
IC50 = 0.46 nM
|
|
|
|
CP0325088
|
(2R,3R,4S)-4-Benzofuran-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C30H38N2O5
|
1
|
| 1 |
IC50 = 0.48 nM
|
|
|
|
CP0343065
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(4-methoxy-benzenesulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H36N2O8S
|
1
|
| 1 |
IC50 = 0.53 nM
|
|
|
|
CP0511535
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-dipentylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H42N2O6
|
1
|
| 1 |
IC50 = 0.56 nM
|
|
|
|
CP0345828
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H40N2O7S
|
1
|
| 1 |
IC50 = 0.57 nM
|
|
|
|
CP0160959
|
(2R,3R,4S)-1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzofuran-5-yl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H40N2O5
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0275762
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxymethoxy-phenyl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H42N2O8S
|
1
|
| 1 |
IC50 = 0.62 nM
|
|
|
|
CP0162907
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H40N2O8S
|
1
|
| 1 |
IC50 = 0.66 nM
|
|
|
|
CP0204466
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-{2-[(2-methyl-propane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H38N2O7S
|
1
|
| 1 |
IC50 = 0.78 nM
|
|
|
|
CP0341583
|
1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzofuran-5-yl)-2-p-tolyl-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H40N2O4
|
1
|
| 1 |
IC50 = 0.78 nM
|
|
|
|
CP0374664
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(butyl-phenyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H34N2O6
|
1
|
| 1 |
IC50 = 0.81 nM
|
|
|
|
CP0414847
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(butyl-ethyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H34N2O6
|
1
|
| 1 |
IC50 = 0.85 nM
|
|
|
|
CP0038234
|
(2R,3R,4S)-1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H40N2O6
|
1
|
| 1 |
IC50 = 0.85 nM
|
|
|
|
CP0298671
|
1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzofuran-5-yl)-2-(4-ethyl-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H42N2O4
|
1
|
| 1 |
IC50 = 0.92 nM
|
|
|
|
CP0526731
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-propyl-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H42N2O5
|
1
|
| 1 |
IC50 = 1.06 nM
|
|
|
|
CP0371250
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-[2-(ethanesulfonyl-propyl-amino)-ethyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H34N2O7S
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0106389
|
(2R,3R,4S)-1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzofuran-6-yl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H40N2O5
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
|
CP0395394
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-dipropylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H34N2O6
|
1
|
| 1 |
IC50 = 1.23 nM
|
|
|
|
CP0185724
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-ethoxy-3-fluoro-phenyl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H41FN2O7S
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0329298
|
4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(3,4-difluoro-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H34F2N2O5
|
1
|
| 1 |
IC50 = 1.38 nM
|
|
|
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CP0204761
|
(2R,3R,4S)-1-[2-(Benzenesulfonyl-propyl-amino)-ethyl]-4-benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H34N2O7S
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0083845
|
(2R,3R,4S)-1-Dibutylcarbamoylmethyl-4-indan-5-yl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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|
C31H42N2O4
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
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CP0309383
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-{2-[(propane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H36N2O7S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
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CP0539739
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(isobutyl-methyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H32N2O6
|
1
|
| 1 |
IC50 = 1.88 nM
|
|
|
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CP0185039
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[butyl-(propane-1-sulfonyl)-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H38N2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0207344
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(butane-1-sulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H38N2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0275728
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(3-chloro-propane-1-sulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H35ClN2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0186031
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(3,4-dimethoxy-phenyl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H42N2O8S
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
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CP0366717
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(3-fluoro-4-methoxy-phenyl)-1-[2-(phenylmethanesulfonyl-propyl-amino)-ethyl]-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H35FN2O7S
|
1
|
| 1 |
IC50 = 2.7 nM
|
|
|
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CP0298670
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4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-trifluoromethyl-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H35F3N2O5
|
1
|
| 1 |
IC50 = 3.28 nM
|
|
|
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CP0524074
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-{[bis-(2-methoxy-ethyl)-carbamoyl]-methyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H34N2O8
|
1
|
| 1 |
IC50 = 4.45 nM
|
|
|
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CP0460843
|
(2S,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H38N2O6
|
1
|
| 1 |
IC50 = 4.62 nM
|
|
|
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CP0436711
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(butyl-methyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C26H32N2O6
|
1
|
| 1 |
IC50 = 4.71 nM
|
|
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CP0346459
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(heptane-1-sulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H44N2O7S
|
1
|
| 1 |
IC50 = 5.1 nM
|
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CP0112338
|
(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(2-methoxy-ethanesulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H36N2O8S
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
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CP0293880
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1-Dibutylcarbamoylmethyl-4-(2,3-dihydro-benzo[1,4]dioxin-6-yl)-2-(4-ethyl-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H42N2O5
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
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CP0509522
|
5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[(1-oxa-4-aza-spiro[4.5]decane-4-carbonyl)-amino]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
Show/Hide
|
C31H41N5O6
|
1
|
| 1 |
IC50 = 5.7 nM
|
|
|
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CP0507292
|
(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[(methyl-pentyl-carbamoyl)-methyl]-pyrrolidine-3-carboxylic acid
Show/Hide
|
C27H34N2O6
|
1
|
| 1 |
IC50 = 5.78 nM
|
|
|
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CP0502235
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2-[(R)-1-{(S)-2-[(2,3-Dihydro-indole-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
|
C31H35N5O5
|
1
|
| 1 |
IC50 = 5.9 nM
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CP0241603
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(4-chloro-benzenesulfonyl)-propyl-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C30H33ClN2O7S
|
1
|
| 1 |
IC50 = 6.3 nM
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CP0436708
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[(methyl-propyl-carbamoyl)-methyl]-pyrrolidine-3-carboxylic acid
Show/Hide
|
C25H30N2O6
|
1
|
| 1 |
IC50 = 6.63 nM
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CP0429694
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5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-phenyl-ureido)-pentanoylamino]-ethyl}-1H-imidazole-4-carboxylic acid
Show/Hide
|
C29H34N6O4
|
1
|
| 1 |
IC50 = 7.6 nM
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CP0541133
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(hexyl-methyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H36N2O6
|
1
|
| 1 |
IC50 = 7.61 nM
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CP0257534
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[isobutyl-(propane-1-sulfonyl)-amino]-ethyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C28H38N2O7S
|
1
|
| 1 |
IC50 = 8.1 nM
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CP0507021
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(isobutylcarbamoyl-methyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C25H30N2O6
|
1
|
| 1 |
IC50 = 8.2 nM
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CP0330413
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-{2-[propyl-(toluene-4-sulfonyl)-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
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C31H36N2O7S
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1
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| 1 |
IC50 = 8.3 nM
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CP0147983
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-{2-[methyl-(propane-1-sulfonyl)-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
|
C25H32N2O7S
|
1
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| 1 |
IC50 = 10 nM
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CP0194411
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[2-(phenylmethanesulfonyl-propyl-amino)-ethyl]-pyrrolidine-3-carboxylic acid
Show/Hide
|
C31H36N2O7S
|
1
|
| 1 |
IC50 = 10 nM
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CP0137938
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
|
C29H40N6O4
|
1
|
| 1 |
IC50 = 11 nM
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|
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CP0436816
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5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-phenyl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid
Show/Hide
|
C29H33N5O5
|
1
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| 1 |
IC50 = 16 nM
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|
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CP0460818
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(diisobutylcarbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
|
C29H38N2O6
|
1
|
| 1 |
IC50 = 16.2 nM
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|
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CP0486446
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-cyclopentylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C26H30N2O6
|
1
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| 1 |
IC50 = 16.2 nM
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CP0511000
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2-[(R)-1-{(S)-2-[3-(2-Fluoro-phenyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
|
C29H32FN5O5
|
1
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| 1 |
IC50 = 17 nM
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CP0392962
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-propylcarbamoylmethyl-pyrrolidine-3-carboxylic acid
Show/Hide
|
C24H28N2O6
|
1
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| 1 |
IC50 = 17.2 nM
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CP0456639
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(2-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 18 nM
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CP0113234
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-2-(3,4-difluoro-phenyl)-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H36F2N2O6S
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1
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| 1 |
IC50 = 18 nM
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CP0047104
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-[2-(butyl-butyryl-amino)-ethyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C29H38N2O6
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1
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| 1 |
IC50 = 20 nM
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CP0423199
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(cyclohexyl-methyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H34N2O6
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1
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| 1 |
IC50 = 23.8 nM
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CP0527514
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(3-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 26 nM
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CP0460900
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-diethylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H30N2O6
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1
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| 1 |
IC50 = 32.9 nM
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CP0441811
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2-[(R)-1-{(S)-2-[(3,4-Dihydro-2H-quinoline-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C32H37N5O5
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1
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| 1 |
IC50 = 33 nM
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CP0461056
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(2S,3S,4R)-1-Allylcarbamoylmethyl-4-benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H26N2O6
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1
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| 1 |
IC50 = 34.2 nM
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CP0453434
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2-[(R)-1-[(S)-2-(3-Cyclopentyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C28H38N6O4
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1
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| 1 |
IC50 = 37 nM
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CP0544494
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[2-(propane-1-sulfonyl)-ethyl]-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H29NO7S
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1
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| 1 |
IC50 = 37 nM
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CP0573148
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-butylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H30N2O6
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1
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| 1 |
IC50 = 43 nM
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CP0523827
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-ethanesulfinyl-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C23H27NO6S
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1
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| 1 |
IC50 = 44 nM
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CP0164809
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(2R,3R,4S)-4-Benzo[1,3]dioxol-5-yl-1-{2-[(pentane-1-sulfonyl)-propyl-amino]-ethyl}-2-(4-propoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C31H44N2O7S
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1
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| 1 |
IC50 = 48 nM
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CP0505912
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[(methyl-phenyl-carbamoyl)-methyl]-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H28N2O6
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1
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| 1 |
IC50 = 50.2 nM
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CP0431402
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2-[(R)-1-{(S)-2-[(Indole-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C31H33N5O5
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1
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| 1 |
IC50 = 58 nM
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CP0521942
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4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid amide
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C29H39N3O5
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1
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| 1 |
IC50 = 58 nM
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CP0525362
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2-[(R)-1-[(S)-2-(3-Cycloheptyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 60 nM
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CP0507184
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2-[(R)-1-{(S)-2-[3-(3-Fluoro-phenyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C29H32FN5O5
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1
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| 1 |
IC50 = 66 nM
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CP0510382
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5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-pyridin-2-yl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid
Show/Hide
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C28H32N6O5
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1
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| 1 |
IC50 = 74 nM
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CP0515993
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C28H38N6O4
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1
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| 1 |
IC50 = 75 nM
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CP0463640
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-oxo-3-propyl-hexyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H35NO6
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1
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| 1 |
IC50 = 85 nM
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CP0486417
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-[(methyl-prop-2-ynyl-carbamoyl)-methyl]-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H26N2O6
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1
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| 1 |
IC50 = 106 nM
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CP0395395
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-propoxy-ethyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H29NO6
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1
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| 1 |
IC50 = 108 nM
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CP0535408
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2-[(R)-1-{(S)-2-[3-(4-Hydroxy-cyclohexyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C29H40N6O5
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1
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| 1 |
IC50 = 110 nM
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CP0436565
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-{[(2,2-dimethyl-propyl)-methyl-carbamoyl]-methyl}-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C27H34N2O6
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1
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| 1 |
IC50 = 112 nM
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CP0439666
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2-[(R)-1-{(S)-2-[3-(1-Methoxycarbonyl-cyclohexyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C31H41N5O7
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1
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| 1 |
IC50 = 120 nM
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CP0380409
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-dipropylcarbamoyl-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H36N2O6
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1
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| 1 |
IC50 = 121 nM
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CP0509474
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(4-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 141 nM
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CP0514084
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5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-pyridin-3-yl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid
Show/Hide
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C28H32N6O5
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1
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| 1 |
IC50 = 153 nM
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CP0374625
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-oxo-hexyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H29NO6
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1
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| 1 |
IC50 = 163 nM
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CP0343793
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C29H38N2O6
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1
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| 1 |
IC50 = 171 nM
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CP0430571
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(2-methoxy-ethylcarbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H28N2O7
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1
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| 1 |
IC50 = 178 nM
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CP0456640
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(1-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 200 nM
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CP0183366
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C29H39N5O5
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1
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| 1 |
IC50 = 220 nM
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CP0498081
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-butoxy-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H31NO6
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1
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| 1 |
IC50 = 220 nM
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CP0458844
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(1,2,3,4-tetrahydro-naphthalen-1-yl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
Show/Hide
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C33H39N5O5
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1
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| 1 |
IC50 = 230 nM
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CP0532685
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C29H40N6O4
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1
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| 1 |
IC50 = 280 nM
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CP0401670
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2-[(R)-1-[(S)-2-(3-Cyclopentyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C28H37N5O5
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1
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| 1 |
IC50 = 300 nM
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CP0505913
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-oxo-2-piperidin-1-yl-ethyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C26H30N2O6
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1
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| 1 |
IC50 = 350 nM
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CP0534258
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-dibutylcarbamoyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C28H36N2O6
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1
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| 1 |
IC50 = 396 nM
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CP0401238
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2-[(R)-1-[(S)-2-(3-Cycloheptyl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 400 nM
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CP0403648
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-isobutoxy-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H31NO6
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1
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| 1 |
IC50 = 437 nM
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CP0515823
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2-[(R)-1-[(S)-2-(3-Adamantan-2-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C33H43N5O5
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1
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| 1 |
IC50 = 440 nM
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CP0530843
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-ethoxy-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C23H27NO6
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1
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| 1 |
IC50 = 520 nM
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CP0492625
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C28H38N6O4
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1
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| 1 |
IC50 = 570 nM
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CP0492090
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C29H39N5O5
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1
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| 1 |
IC50 = 620 nM
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CP0504178
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(2-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 650 nM
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CP0524575
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C28H37N5O5
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1
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| 1 |
IC50 = 660 nM
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CP0436748
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[2-(2-methoxy-ethoxy)-ethyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H29NO7
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1
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| 1 |
IC50 = 682 nM
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CP0414778
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-butylcarbamoyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H28N2O6
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1
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| 1 |
IC50 = 684 nM
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CP0520337
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-ethyl-1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 730 nM
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CP0541669
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-isopropyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C30H42N6O4
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1
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| 1 |
IC50 = 730 nM
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CP0504794
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-hex-2-ynyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C25H27NO5
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1
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| 1 |
IC50 = 765 nM
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CP0498083
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[(benzyl-methyl-carbamoyl)-methyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C29H30N2O6
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1
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| 1 |
IC50 = 769 nM
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CP0541130
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(4-methoxy-phenylcarbamoyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C27H26N2O7
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1
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| 1 |
IC50 = 781 nM
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CP0374932
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-dibutylamino-ethyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C29H40N2O5
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1
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| 1 |
IC50 = 794 nM
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CP0448581
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-phenoxy-ethyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C27H27NO6
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1
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| 1 |
IC50 = 885 nM
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CP0480519
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2-[(R)-1-[(S)-2-(3-Adamantan-1-yl-ureido)-4-methyl-pentanoylamino]-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C33H43N5O5
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1
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| 1 |
IC50 = 900 nM
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CP0432308
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(2-pyridin-2-yl-ethyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C26H26N2O5
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1
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| 1 |
IC50 = 900 nM
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CP0523322
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(3-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 960 nM
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CP0524563
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2-[(R)-1-[(S)-2-(3,3-Diethyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C26H36N6O4
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1
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| 1 |
IC50 = 1000 nM
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CP0410063
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-(morpholine-4-carbonyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C24H26N2O7
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1
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| 1 |
IC50 = 1080 nM
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CP0373013
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(butane-1-sulfonyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C23H27NO7S
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1
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| 1 |
IC50 = 1240 nM
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CP0448661
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C28H37N5O5
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1
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| 1 |
IC50 = 1430 nM
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CP0501222
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-ethyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C29H40N6O4
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1
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| 1 |
IC50 = 1500 nM
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CP0464993
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-((E)-5-methyl-hex-2-enyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C26H31NO5
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1
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| 1 |
IC50 = 1630 nM
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CP0505645
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2-[(R)-1-{(S)-2-[3-(4-Fluoro-phenyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
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C29H32FN5O5
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1
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| 1 |
IC50 = 1900 nM
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CP0523273
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({2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carbonyl}-amino)-acetic acid
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C30H40N6O6
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1
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| 1 |
IC50 = 1900 nM
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CP0451623
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-ethyl-oxazole-4-carboxylic acid
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C29H39N5O5
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1
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| 1 |
IC50 = 1900 nM
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CP0511477
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-carbamoylmethyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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C21H22N2O6
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1
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| 1 |
IC50 = 2030 nM
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CP0448068
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2-[(R)-1-[(S)-2-(3-Benzyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
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C29H34N6O4
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1
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| 1 |
IC50 = 2100 nM
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CP0414844
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-2-(4-methoxy-phenyl)-1-phenylcarbamoyl-pyrrolidine-3-carboxylic acid
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C26H24N2O6
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1
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| 1 |
IC50 = 2430 nM
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CP0529123
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-isopropyl-oxazole-4-carboxylic acid
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C30H41N5O5
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1
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| 1 |
IC50 = 2500 nM
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CP0480522
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2-[(R)-1-{(S)-2-[3-(4-Hydroxy-cyclohexyl)-ureido]-4-methyl-pentanoylamino}-2-(1-methyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
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C29H39N5O6
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1
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| 1 |
IC50 = 2520 nM
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CP0511375
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5-Methyl-2-((R)-2-(1-methyl-1H-indol-3-yl)-1-{(S)-4-methyl-2-[3-(4-methyl-cyclohexyl)-ureido]-pentanoylamino}-ethyl)-oxazole-4-carboxylic acid
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C30H41N5O5
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1
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| 1 |
IC50 = 2730 nM
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CP0392718
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-hexyl-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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C25H31NO5
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1
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| 1 |
IC50 = 2870 nM
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CP0509502
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Azepane-1-carboxylic acid {(S)-1-[(R)-1-(4-hydroxycarbamoyl-5-methyl-oxazol-2-yl)-2-(1H-indol-3-yl)-ethylcarbamoyl]-3-methyl-butyl}-amide
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C28H38N6O5
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1
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| 1 |
IC50 = 2900 nM
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CP0380899
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2-[(R)-1-[(S)-2-(3,3-Diethyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
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C26H35N5O5
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1
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| 1 |
IC50 = 3000 nM
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CP0535717
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Azepane-1-carboxylic acid {(S)-1-[(R)-2-(1H-indol-3-yl)-1-(5-methyl-4-methylcarbamoyl-oxazol-2-yl)-ethylcarbamoyl]-3-methyl-butyl}-amide
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C29H40N6O4
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1
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| 1 |
IC50 = 3000 nM
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CP0509096
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5-Methyl-2-{(R)-2-(1-methyl-1H-indol-3-yl)-1-[(S)-4-methyl-2-(3-pentafluorophenyl-ureido)-pentanoylamino]-ethyl}-oxazole-4-carboxylic acid
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C29H28F5N5O5
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1
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| 1 |
IC50 = 3550 nM
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CP0448676
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-cyclopropyl-oxazole-4-carboxylic acid
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C30H39N5O5
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1
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| 1 |
IC50 = 3700 nM
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CP0398023
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(4-fluoro-benzyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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C26H24FNO5
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1
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| 1 |
IC50 = 4320 nM
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CP0482729
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-cyclopropyl-1H-imidazole-4-carboxylic acid
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C30H40N6O4
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1
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| 1 |
IC50 = 5200 nM
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CP0539796
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(furan-2-carbonyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
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C24H21NO7
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1
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| 1 |
IC50 = 5220 nM
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CP0498076
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-(2-dibutylamino-acetyl)-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C29H38N2O6
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1
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| 1 |
IC50 = 6810 nM
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CP0510716
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-phenyl-oxazole-4-carboxylic acid
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C33H39N5O5
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1
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| 1 |
IC50 = 7300 nM
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CP0461837
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-propyl-oxazole-4-carboxylic acid
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C30H41N5O5
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1
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| 1 |
IC50 = 7700 nM
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CP0431347
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-propyl-1H-imidazole-4-carboxylic acid
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C30H42N6O4
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1
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| 1 |
IC50 = 7800 nM
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CP0531743
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-benzyl-1H-imidazole-4-carboxylic acid
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C34H42N6O4
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1
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| 1 |
IC50 = 8000 nM
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CP0548982
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2-[(R)-1-[(S)-2-(3-Benzyl-ureido)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
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C29H33N5O5
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1
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| 1 |
IC50 = 8700 nM
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CP0378376
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2-[2-[(1R)-1-[[(2S)-2-(azepane-1-carbonylamino)-4-methylpentanoyl]amino]-2-(1H-indol-3-yl)ethyl]-5-methyl-1,3-oxazol-4-yl]acetic acid
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C29H39N5O5
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1
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| 1 |
IC50 = 9600 nM
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CP0448977
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-isopropyl-thiazole-4-carboxylic acid
Show/Hide
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C30H41N5O4S
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1
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| 1 |
IC50 = 11000 nM
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CP0500928
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2-[(R)-1-[(S)-2-(3-Cyclohexyl-ureido)-4-methyl-pentanoylamino]-2-(1-ethyl-1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 12900 nM
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CP0423865
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid ethyl ester
Show/Hide
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C30H41N5O5
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1
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| 1 |
IC50 = 13800 nM
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CP0374753
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(2S,3S,4R)-4-Benzo[1,3]dioxol-5-yl-1-[2-(4-fluoro-phenoxy)-acetyl]-2-(4-methoxy-phenyl)-pyrrolidine-3-carboxylic acid
Show/Hide
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C27H24FNO7
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1
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| 1 |
IC50 = 14100 nM
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CP0453552
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-benzyl-oxazole-4-carboxylic acid
Show/Hide
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C34H41N5O5
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1
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| 1 |
IC50 = 16000 nM
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CP0520250
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-1-benzyl-5-methyl-1H-imidazole-4-carboxylic acid
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C35H44N6O4
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1
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| 1 |
IC50 = 16200 nM
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CP0502068
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-1,5-dimethyl-1H-imidazole-4-carboxylic acid
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C29H40N6O4
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1
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| 1 |
IC50 = 23300 nM
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CP0517905
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-cyclopropyl-thiazole-4-carboxylic acid
Show/Hide
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C30H39N5O4S
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1
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| 1 |
IC50 = 24000 nM
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CP0529923
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-propyl-thiazole-4-carboxylic acid
Show/Hide
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C30H41N5O4S
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1
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| 1 |
IC50 = 36000 nM
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CP0502361
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-benzyl-thiazole-4-carboxylic acid
Show/Hide
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C34H41N5O4S
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1
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| 1 |
IC50 = 39000 nM
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CP0448075
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-methyl-thiazole-4-carboxylic acid
Show/Hide
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C28H37N5O4S
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1
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| 1 |
IC50 = 41000 nM
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CP0459225
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-ethyl-thiazole-4-carboxylic acid
Show/Hide
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C29H39N5O4S
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1
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| 1 |
IC50 = 41000 nM
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CP0374651
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-phenyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C33H40N6O4
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1
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| 1 |
IC50 = 51000 nM
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CP0458928
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2-[(R)-1-{(S)-2-[(Azepane-1-carbonyl)-amino]-4-methyl-pentanoylamino}-2-(1H-indol-3-yl)-ethyl]-5-phenyl-thiazole-4-carboxylic acid
Show/Hide
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C33H39N5O4S
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1
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| 1 |
IC50 = 51000 nM
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CP0421336
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(R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-methyl-butyl}-5-(1-methyl-1H-indol-3-ylmethyl)-oxazole-4-carbonyl]-amino}-3-pyridin-2-yl-propionic acid
Show/Hide
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C34H42N6O5
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1
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| 1 |
IC50 = 68000 nM
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CP0448975
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(R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-methyl-butyl}-5-(1-methyl-1H-indol-3-ylmethyl)-thiazole-4-carbonyl]-amino}-3-pyridin-2-yl-propionic acid
Show/Hide
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C34H42N6O4S
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1
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| 1 |
IC50 > 90000 nM
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CP0554893
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(R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-methyl-butyl}-5-(1-methyl-1H-indol-3-yl)-thiazole-4-carbonyl]-amino}-3-pyridin-2-yl-propionic acid
Show/Hide
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C33H40N6O4S
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1
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| 1 |
IC50 > 90000 nM
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CP0509228
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2-[(R)-1-[(S)-2-(Azepane-1-sulfonylamino)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid
Show/Hide
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C27H37N5O6S
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1
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| 1 |
IC50 > 100000 nM
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CP0550895
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2-[(R)-1-[(S)-2-(Azepane-1-sulfonylamino)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-1H-imidazole-4-carboxylic acid
Show/Hide
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C27H38N6O5S
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1
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| 1 |
IC50 > 100000 nM
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CP0482728
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(R)-2-{[2-{(S)-1-[(Azepane-1-carbonyl)-amino]-3-methyl-butyl}-5-(1-methyl-1H-indol-3-yl)-oxazole-4-carbonyl]-amino}-3-pyridin-2-yl-propionic acid
Show/Hide
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C33H40N6O5
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1
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| 1 |
IC50 > 100000 nM
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