Bioactivity Information

Brief Information of the Compound and Protein

Compound Name

Compound Info

2-[(R)-1-[(S)-2-(Azepane-1-sulfonylamino)-4-methyl-pentanoylamino]-2-(1H-indol-3-yl)-ethyl]-5-methyl-oxazole-4-carboxylic acid

Show/Hide

PubChem ID

CID: 10721589

SID: 15756754

Canonical SMILES	CC(C)C[C@H](NS(=O)(=O)N1CCCCCC1)C(=O)N[C@H](Cc1c[nH]c2ccccc12)c1nc(C(O)=O)c(C)o1 Show/Hide
Compound Formula	C27H37N5O6S

Compound Structure

Protein Name

Protein Info

Endothelin-1 receptor

Protein Classification

Membrane receptor

Family A G protein-coupled receptor

Peptide receptor (family A GPCR)

Short peptide receptor (family A GPCR)

Endothelin receptor

Uniprot ID

P26684

Gene Name

EDNRA

Table of Molecular Bioactivities Related to the Compound and Protein

Cell-based Assay