| Compound ID |
Compound Name |
Compound Formula |
|
CP0785593
|
(Z)-3-[Phenyl-(4-piperidin-1-ylmethyl-phenylamino)-methylene]-2-oxo-2,3-dihydro-1H-indole-6-carboxylic Acid Ethylamide
Show/Hide
|
C30H32N4O2
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0647120
|
(Z)-3-((4-(N-(2-(dimethylamino)ethyl)acetamido)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C31H35N5O3
|
1
|
| 1 |
EC50 = 102 nM
|
|
|
|
CP0641932
|
(Z)-2-oxo-3-[Phenyl-(4-piperidin-1-ylmethyl-phenylamino)-methylene]-2,3-dihydro-1H-indole-6-carboxylic Acid Ethylmethylamide
Show/Hide
|
C31H34N4O2
|
1
|
| 1 |
EC50 = 105 nM
|
|
|
|
CP0643814
|
(Z)-3-((4-(N-(2-(dimethylamino)ethyl)methylsulfonamido)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C29H33N5O4S
|
1
|
| 1 |
EC50 = 108 nM
|
|
|
|
CP0774796
|
(Z)-3-((4-(2-(dimethylamino)ethyl)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C28H30N4O2
|
1
|
| 1 |
EC50 = 135 nM
|
|
|
|
CP0643877
|
(Z)-N-ethyl-3-((4-((ethylamino)methyl)phenylamino)(phenyl)methylene)-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C28H30N4O2
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0036041
|
4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide
Show/Hide
|
C22H16N4O3
|
1
|
| 1 |
EC50 = 172 nM
|
|
|
|
CP0639868
|
(Z)-3-((4-((dimethylamino)methyl)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C27H28N4O2
|
1
|
| 1 |
EC50 = 185 nM
|
|
|
|
CP0643897
|
(Z)-N,N-dimethyl-2-oxo-3-(phenyl(4-(piperidin-1-ylmethyl)phenylamino)methylene)indoline-5-carboxamide
Show/Hide
|
C30H32N4O2
|
1
|
| 1 |
EC50 = 198 nM
|
|
|
|
CP0785594
|
(Z)-3-((4-(N-(2-(dimethylamino)ethyl)methylsulfonamido)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C30H35N5O4S
|
1
|
| 1 |
EC50 = 209 nM
|
|
|
|
CP0647119
|
(Z)-N,N-dimethyl-2-oxo-3-(phenyl(4-(piperidin-1-ylmethyl)phenylamino)methylene)indoline-6-carboxamide
Show/Hide
|
C30H32N4O2
|
1
|
| 1 |
EC50 = 246 nM
|
|
|
|
CP0778726
|
(Z)-3-((4-(2-(dimethylamino)ethyl)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C29H32N4O2
|
1
|
| 1 |
EC50 = 259 nM
|
|
|
|
CP0729847
|
(Z)-N-ethyl-2-oxo-3-((4-(piperidin-1-ylmethyl)phenylamino)methylene)indoline-6-carboxamide
Show/Hide
|
C24H28N4O2
|
1
|
| 1 |
EC50 = 376 nM
|
|
|
|
CP0647121
|
(Z)-3-((4-(2-(dimethylamino)-N-methylacetamido)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C30H33N5O3
|
1
|
| 1 |
EC50 = 382 nM
|
|
|
|
CP0667581
|
(Z)-3-((4-(N-(3-(dimethylamino)propyl)acetamido)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C32H37N5O3
|
1
|
| 1 |
EC50 = 411 nM
|
|
|
|
CP0774795
|
(Z)-3-((4-(2-(diethylamino)ethylcarbamoyl)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C31H35N5O3
|
1
|
| 1 |
EC50 = 505 nM
|
|
|
|
CP0784804
|
(Z)-3-((4-(2-(diethylamino)ethylcarbamoyl)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C32H37N5O3
|
1
|
| 1 |
EC50 = 542 nM
|
|
|
|
CP0834341
|
(Z)-3-((4-(N-(3-(dimethylamino)propyl)acetamido)phenylamino)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C25H31N5O3
|
1
|
| 1 |
EC50 = 597 nM
|
|
|
|
CP0690546
|
(Z)-3-(phenyl(4-(piperidin-1-ylmethyl)phenylamino)methylene)-6-(pyrrolidine-2-carbonyl)indolin-2-one
Show/Hide
|
C32H34N4O2
|
1
|
| 1 |
EC50 = 696 nM
|
|
|
|
CP0828600
|
(Z)-2-oxo-3-[Phenyl-(4-piperidin-1-ylmethyl-phenylamino)-methylene]-2,3-dihydro-1H-indole-6-carboxylic Acid Isopropylamide
Show/Hide
|
C31H34N4O2
|
1
|
| 1 |
EC50 = 708 nM
|
|
|
|
CP0759858
|
(Z)-N-ethyl-N-methyl-3-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenylamino)(phenyl)methylene)-2-oxoindoline-6-carboxamide
Show/Hide
|
C33H38N6O3
|
1
|
| 1 |
EC50 = 833 nM
|
|
|
|
CP0834506
|
(Z)-N-butyl-2-oxo-3-(phenyl(4-(piperidin-1-ylmethyl)phenylamino)methylene)indoline-6-carboxamide
Show/Hide
|
C32H36N4O2
|
1
|
| 1 |
EC50 = 1065 nM
|
|
|
|
CP0667580
|
(Z)-3-((4-(N-(2-(dimethylamino)ethyl)acetamido)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C30H33N5O3
|
1
|
| 1 |
EC50 = 1066 nM
|
|
|
|
CP0784803
|
(Z)-3-((4-(N-(3-(dimethylamino)propyl)acetamido)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C31H35N5O3
|
1
|
| 1 |
EC50 = 1249 nM
|
|
|
|
CP0826693
|
(Z)-N-ethyl-3-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenylamino)(phenyl)methylene)-2-oxoindoline-6-carboxamide
Show/Hide
|
C32H36N6O3
|
1
|
| 1 |
EC50 = 1370 nM
|
|
|
|
CP0778728
|
(Z)-N-ethyl-3-((4-(N-methyl-2-(4-methylpiperazin-1-yl)acetamido)phenylamino)methylene)-2-oxoindoline-6-carboxamide
Show/Hide
|
C26H32N6O3
|
1
|
| 1 |
EC50 = 2175 nM
|
|
|
|
CP0834372
|
(Z)-3-((4-(2-(dimethylamino)-N-methylacetamido)phenylamino)(phenyl)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C29H31N5O3
|
1
|
| 1 |
EC50 = 3383 nM
|
|
|
|
CP0834502
|
(Z)-3-((4-(2-(dimethylamino)-N-methylacetamido)phenylamino)methylene)-N-ethyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C23H27N5O3
|
1
|
| 1 |
EC50 = 4355 nM
|
|
|
|
CP0667582
|
(Z)-N-ethyl-N-methyl-3-((4-(N-methylmethylsulfonamido)phenylamino)(phenyl)methylene)-2-oxoindoline-6-carboxamide
Show/Hide
|
C27H28N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0818490
|
(Z)-3-((cyclohexylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C25H29N3O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0832208
|
(Z)-N-ethyl-N-methyl-3-((1-methylpiperidin-4-ylamino)(phenyl)methylene)-2-oxoindoline-6-carboxamide
Show/Hide
|
C25H30N4O2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0674919
|
(Z)-2-oxo-3-[Phenyl-(4-piperidin-1-ylmethyl-phenylamino)-methylene]-2,3-dihydro-1H-indole-6-carboxylic Acid Amide
Show/Hide
|
C28H28N4O2
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0784802
|
(Z)-N-(2-hydroxyethyl)-2-oxo-3-(phenyl(4-(piperidin-1-ylmethyl)phenylamino)methylene)indoline-6-carboxamide
Show/Hide
|
C30H32N4O3
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
|
CP0834501
|
(Z)-3-((4-(N-(2-(dimethylamino)-2-oxoethyl)methylsulfonamido)phenylamino)(phenyl)methylene)-N-ethyl-N-methyl-2-oxoindoline-6-carboxamide
Show/Hide
|
C30H33N5O5S
|
1
|
| 1 |
EC50 > 3000 nM
|
|
|
|
CP0055625
|
2-fluoro-N-[[5-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)-1H-imidazol-2-yl]methyl]aniline
Show/Hide
|
C22H18FN7
|
1
|
| 1 |
IC50 = 16.5 nM
|
|
|
|
CP0173805
|
3-((5-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)-1H-imidazol-2-yl)methyl)benzamide
Show/Hide
|
C25H20N6O
|
1
|
| 1 |
IC50 = 19.6 nM
|
|
|
|
CP0015550
|
2-(4-(benzo[d][1,3]dioxol-5-yl)-2-tert-butyl-1H-imidazol-5-yl)-6-methylpyridine
Show/Hide
|
C20H21N3O2
|
1
|
| 1 |
IC50 = 43.8 nM
|
|
|
|
CP0010529
|
GALUNISERTIB
Show/Hide
|
C22H19N5O
|
1
|
| 1 |
IC50 > 100 nM
|
|
|
