General Information of the Compound
Compound ID
CP0036041
Compound Name
4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide
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Synonyms
301836-41-9
4-(4-(1,3-Benzodioxole-5-yl)-5-(2-pyridyl)-1H-imidazole-2-yl)benzamide
4-(4-(benzo[d][1,3]dioxol-5-yl)-5-(pyridin-2-yl)-1H-imidazol-2-yl)benzamide
4-(4-Benzo[1,3]dioxol-5-yl-5-pyridin-2-yl-1H-imidazol-2-yl)-benzamide
4-[4-(1,3-BENZODIOXOL-5-YL)-5-(2-PYRIDINYL)-1H-IMIDAZOL-2-YL]BENZAMIDE
4-[4-(3,4-Methylenedioxyphenyl)-5-(2-pyridyl)-1H-imidazol-2-yl]benzamide
C22H16N4O3
CHEMBL440084
E1557V1V0N
SB 431542
SB 431542 hydrate
SB-431542
SB431542
UNII-E1557V1V0N
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Structure
Formula
C22H16N4O3
Molecular Weight
384.395
Canonical SMILES
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
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InChI
InChI=1S/C22H16N4O3/c23-21(27)13-4-6-14(7-5-13)22-25-19(20(26-22)16-3-1-2-10-24-16)15-8-9-17-18(11-15)29-12-28-17/h1-11H,12H2,(H2,23,27)(H,25,26)
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InChIKey
FHYUGAJXYORMHI-UHFFFAOYSA-N
Physicochemical Property
logP
3.6333
Rotatable Bonds
4
Heavy Atom Count
29
Polar Areas
103.12
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
5
Complexity
29

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 4521392
SID: 87231679
ChEMBL ID
CHEMBL440084
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01221, TGF-beta receptor type-1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000150 HaCaT Homo sapiens (Human)  1
1
EC50 = 172 nM
   TI
   LI
   LO
   TS
CL000063 Hep-G2 Homo sapiens (Human)  1
1
IC50 = 250 nM
   TI
   LI
   LO
   TS
CL000775 CHO/IR Cricetulus griseus (Chinese hamster)  1
1
IC50 = 350 nM
   TI
   LI
   LO
   TS
CL000013 Sf9 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 1542 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 66 nM
2 IC50 = 70 nM
3 IC50 = 94 nM
4 IC50 = 125 nM
5 Kd = 170 nM
6 Ki = 17 nM
Protein ID: PT01867, TGF-beta receptor type-2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000025 HEK-293T Homo sapiens (Human)  1
1
IC50 = 66 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Kd > 10000 nM
Clinical Information about the Compound
Drug 1 ( SB-431542 )
Drug Name SB-431542
Indication
Pulmonary fibrosis
Preclinical
Target(s)
TGF-beta receptor type I (TGFBR1)
Inhibitor