| Compound ID |
Compound Name |
Compound Formula |
|
CP0129571
|
2-[4-(4-chlorophenyl)piperazin-1-yl)methyl]imidazo[1,2-a]pyridine
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|
C18H19ClN4
|
1
|
| 1 |
EC50 = 2.6 nM
|
|
|
|
CP0384374
|
2-(3',4',-5',6'-tetrahydro-2'H-[2,4'-bipyridine]-1'-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C19H23N3O
|
4
|
| 1 |
EC50 = 2.7 nM
|
|
|
| 2 |
EC50 = 473 nM
|
|
|
| 3 |
IC50 = 68.4 nM
|
|
|
| 4 |
IC50 = 191 nM
|
|
|
|
CP0384667
|
N-(3-methylphenyl)-2-(4-pyrimidin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C17H21N5O
|
4
|
| 1 |
EC50 = 3.4 nM
|
|
|
| 2 |
EC50 = 278 nM
|
|
|
| 3 |
IC50 = 197 nM
|
|
|
| 4 |
IC50 = 463 nM
|
|
|
|
CP0384672
|
N-(3-methylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C18H22N4O
|
4
|
| 1 |
EC50 = 3.6 nM
|
|
|
| 2 |
EC50 = 394 nM
|
|
|
| 3 |
IC50 = 82.7 nM
|
|
|
| 4 |
IC50 = 313 nM
|
|
|
|
CP0058895
|
2-[4-(2-methoxyphenyl)piperazin-1-ylmethyl]imidazo[1,2-a]pyridine
Show/Hide
|
C19H22N4O
|
1
|
| 1 |
EC50 = 4.5 nM
|
|
|
|
CP0384369
|
2-(4-phenylpiperidin-1-yl)-N-(m-tolyl)acetamide
Show/Hide
|
C20H24N2O
|
4
|
| 1 |
EC50 = 15.4 nM
|
|
|
| 2 |
EC50 = 242 nM
|
|
|
| 3 |
IC50 = 2 nM
|
|
|
| 4 |
IC50 = 135 nM
|
|
|
|
CP0384370
|
N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C19H24N4O
|
4
|
| 1 |
EC50 = 28.7 nM
|
|
|
| 2 |
EC50 = 133 nM
|
|
|
| 3 |
IC50 = 370 nM
|
|
|
| 4 |
IC50 = 1311 nM
|
|
|
|
CP0006107
|
CAS_85760-74-3
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|
C13H21N3
|
1
|
| 1 |
EC50 = 49 nM
|
|
|
|
CP0041783
|
1,1-diethyl-3-[(8alpha)-6-methyl-9,10-didehydroergolin-8-yl]urea
Show/Hide
|
C20H26N4O
|
1
|
| 1 |
EC50 = 88.5 nM
|
|
|
|
CP0384375
|
N-(3-methylphenyl)-2-(4-naphthalen-1-ylpiperazin-1-yl)acetamide
Show/Hide
|
C23H25N3O
|
4
|
| 1 |
EC50 = 108.5 nM
|
|
|
| 2 |
EC50 = 9212 nM
|
|
|
| 3 |
IC50 = 2521 nM
|
|
|
| 4 |
IC50 = 4252 nM
|
|
|
|
CP0384679
|
N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperidin-1-yl)propanamide
Show/Hide
|
C20H25N3O
|
3
|
| 1 |
EC50 = 349 nM
|
|
|
| 2 |
IC50 = 3805 nM
|
|
|
| 3 |
IC50 = 6343 nM
|
|
|
|
CP0001212
|
1-(2-methoxyphenyl)-4-[3-[(4-methyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]propyl]piperazine
Show/Hide
|
C23H29N5OS
|
1
|
| 1 |
EC50 = 359.1 nM
|
|
|
|
CP0384677
|
N-(3-ethylphenyl)-2-(4-pyridin-2-ylpiperidin-1-yl)acetamide
Show/Hide
|
C20H25N3O
|
3
|
| 1 |
EC50 = 539 nM
|
|
|
| 2 |
IC50 = 1908 nM
|
|
|
| 3 |
IC50 = 2622 nM
|
|
|
|
CP0384371
|
N-(3-methylphenyl)-3-(4-pyrimidin-2-ylpiperazin-1-yl)propanamide
Show/Hide
|
C18H23N5O
|
3
|
| 1 |
EC50 = 568 nM
|
|
|
| 2 |
IC50 = 430 nM
|
|
|
| 3 |
IC50 = 2120 nM
|
|
|
|
CP0384372
|
N-(3-methylphenyl)-3-(4-pyridin-2-ylpiperazin-1-yl)propanamide
Show/Hide
|
C19H24N4O
|
3
|
| 1 |
EC50 = 612 nM
|
|
|
| 2 |
IC50 = 1086 nM
|
|
|
| 3 |
IC50 = 1629 nM
|
|
|
|
CP0384381
|
N-pyridin-3-yl-2-(4-pyridin-2-ylpiperazin-1-yl)acetamide
Show/Hide
|
C16H19N5O
|
4
|
| 1 |
EC50 = 1075 nM
|
|
|
| 2 |
EC50 = 2657 nM
|
|
|
| 3 |
IC50 = 25780 nM
|
|
|
| 4 |
IC50 = 86493 nM
|
|
|
|
CP0040671
|
8-[4-(4-fluorophenyl)-4-keto-butyl]-1-phenyl-1,3,8-triazaspiro[4.5]decan-4-one
Show/Hide
|
C23H26FN3O2
|
2
|
| 1 |
IC50 = 0.5 nM
|
|
|
| 2 |
Ki = 0.2 nM
|
|
|
|
CP0443508
|
(2S)-4-[(6-chloro-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H21ClN2O2
|
2
|
| 1 |
IC50 = 8 nM
|
|
|
| 2 |
Ki = 2.2 nM
|
|
|
|
CP0401192
|
(2S)-2-[(6-chloropyridin-2-yl)oxymethyl]-4-[(6-fluoro-1H-indol-3-yl)methyl]morpholine
Show/Hide
|
C19H19ClFN3O2
|
2
|
| 1 |
IC50 = 11.9 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0443493
|
(2S)-4-[(6-fluoro-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H21FN2O2
|
2
|
| 1 |
IC50 = 18.9 nM
|
|
|
| 2 |
Ki = 5.2 nM
|
|
|
|
CP0376286
|
(2S)-4-[(6-methoxy-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C21H24N2O3
|
2
|
| 1 |
IC50 = 19.5 nM
|
|
|
| 2 |
Ki = 5.4 nM
|
|
|
|
CP0376284
|
(2S)-4-[(3,4-dimethylphenyl)methyl]-2-(phenylsulfanylmethyl)morpholine
Show/Hide
|
C20H25NOS
|
2
|
| 1 |
IC50 = 27 nM
|
|
|
| 2 |
Ki = 7.4 nM
|
|
|
|
CP0452595
|
(2S)-4-[(4-chlorophenyl)methyl]-2-(phenylsulfanylmethyl)morpholine
Show/Hide
|
C18H20ClNOS
|
2
|
| 1 |
IC50 = 34 nM
|
|
|
| 2 |
Ki = 9.4 nM
|
|
|
|
CP0376281
|
(2S)-4-[(4-chloro-3-methoxyphenyl)methyl]-2-[(3-fluorophenoxy)methyl]morpholine
Show/Hide
|
C19H21ClFNO3
|
2
|
| 1 |
IC50 = 37 nM
|
|
|
| 2 |
Ki = 10.1 nM
|
|
|
|
CP0472286
|
(2S)-4-[(4-chlorophenyl)methyl]-2-[(4-fluorophenoxy)methyl]morpholine
Show/Hide
|
C18H19ClFNO2
|
2
|
| 1 |
IC50 = 38 nM
|
|
|
| 2 |
Ki = 10.4 nM
|
|
|
|
CP0509053
|
(2S)-4-[(3-chloro-4-methoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H22ClNO3
|
2
|
| 1 |
IC50 = 38 nM
|
|
|
| 2 |
Ki = 10.4 nM
|
|
|
|
CP0376289
|
(2S)-4-[(3-chloro-4-methoxyphenyl)methyl]-2-[(3-fluorophenoxy)methyl]morpholine
Show/Hide
|
C19H21ClFNO3
|
2
|
| 1 |
IC50 = 39 nM
|
|
|
| 2 |
Ki = 10.8 nM
|
|
|
|
CP0509058
|
(2S)-4-[(4-chloro-3-methoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H22ClNO3
|
2
|
| 1 |
IC50 = 42 nM
|
|
|
| 2 |
Ki = 11.6 nM
|
|
|
|
CP0563745
|
(2S)-4-[(4-fluoro-3-methoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H22FNO3
|
2
|
| 1 |
IC50 = 42 nM
|
|
|
| 2 |
Ki = 11.6 nM
|
|
|
|
CP0376285
|
(2S)-4-[(3,4-dimethylphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H25NO2
|
2
|
| 1 |
IC50 = 45 nM
|
|
|
| 2 |
Ki = 12.3 nM
|
|
|
|
CP0376288
|
(2S)-2-[(4-fluorophenoxy)methyl]-4-[(4-methoxyphenyl)methyl]morpholine
Show/Hide
|
C19H22FNO3
|
2
|
| 1 |
IC50 = 47 nM
|
|
|
| 2 |
Ki = 13.1 nM
|
|
|
|
CP0443492
|
(2S)-4-[(3-fluoro-4-methoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H22FNO3
|
2
|
| 1 |
IC50 = 56 nM
|
|
|
| 2 |
Ki = 14.3 nM
|
|
|
|
CP0376274
|
(2S)-4-[(4-methylsulfanylphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H23NO2S
|
2
|
| 1 |
IC50 = 58 nM
|
|
|
| 2 |
Ki = 16.1 nM
|
|
|
|
CP0459659
|
(2S)-4-(1H-indol-5-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H22N2O2
|
2
|
| 1 |
IC50 = 58 nM
|
|
|
| 2 |
Ki = 15.9 nM
|
|
|
|
CP0559235
|
(2S)-4-[[3-fluoro-4-(trifluoromethyl)phenyl]methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H19F4NO2
|
2
|
| 1 |
IC50 = 58 nM
|
|
|
| 2 |
Ki = 16.2 nM
|
|
|
|
CP0509054
|
(2S)-4-[(3-chloro-4-fluorophenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C18H19ClFNO2
|
2
|
| 1 |
IC50 = 62 nM
|
|
|
| 2 |
Ki = 170 nM
|
|
|
|
CP0443505
|
(2S)-4-(naphthalen-2-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C22H23NO2
|
2
|
| 1 |
IC50 = 64 nM
|
|
|
| 2 |
Ki = 17.8 nM
|
|
|
|
CP0443507
|
(2S)-4-(2H-indazol-3-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H21N3O2
|
2
|
| 1 |
IC50 = 65 nM
|
|
|
| 2 |
Ki = 18.1 nM
|
|
|
|
CP0376277
|
(2S)-4-[(4-chloro-3-fluorophenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C18H19ClFNO2
|
2
|
| 1 |
IC50 = 69 nM
|
|
|
| 2 |
Ki = 19.1 nM
|
|
|
|
CP0472291
|
(2S)-4-[(6-fluoro-1H-indol-3-yl)methyl]-2-[(6-fluoropyridin-2-yl)oxymethyl]morpholine
Show/Hide
|
C19H19F2N3O2
|
2
|
| 1 |
IC50 = 76 nM
|
|
|
| 2 |
Ki = 21 nM
|
|
|
|
CP0459657
|
(2S)-2-[(3-fluorophenoxy)methyl]-4-[(4-methoxyphenyl)methyl]morpholine
Show/Hide
|
C19H22FNO3
|
2
|
| 1 |
IC50 = 92 nM
|
|
|
| 2 |
Ki = 26 nM
|
|
|
|
CP0376276
|
(2S)-4-[(3,4-dichlorophenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C18H19Cl2NO2
|
2
|
| 1 |
IC50 = 97 nM
|
|
|
| 2 |
Ki = 27 nM
|
|
|
|
CP0339664
|
CHEBI:64217
Show/Hide
|
C21H26ClN3O2
|
1
|
| 1 |
IC50 = 98.2 nM
|
|
|
|
CP0443506
|
(2S)-4-[(4-chlorophenyl)methyl]-2-[(6-chloropyridin-2-yl)oxymethyl]morpholine
Show/Hide
|
C17H18Cl2N2O2
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
Ki = 29 nM
|
|
|
|
CP0509056
|
3-[[(2S)-4-[(4-chloro-3-methoxyphenyl)methyl]morpholin-2-yl]methoxy]benzonitrile
Show/Hide
|
C20H21ClN2O3
|
2
|
| 1 |
IC50 = 100 nM
|
|
|
| 2 |
Ki = 28 nM
|
|
|
|
CP0376272
|
(2S)-4-[(4-chlorophenyl)methyl]-2-(pyridin-3-yloxymethyl)morpholine
Show/Hide
|
C17H19ClN2O2
|
2
|
| 1 |
IC50 = 103 nM
|
|
|
| 2 |
Ki = 47 nM
|
|
|
|
CP0376282
|
(2S)-4-[(4-chlorophenyl)methyl]-2-[(3-methoxyphenoxy)methyl]morpholine
Show/Hide
|
C19H22ClNO3
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
Ki = 36 nM
|
|
|
|
CP0459656
|
3-[[(2S)-4-[(3-chloro-4-methoxyphenyl)methyl]morpholin-2-yl]methoxy]benzonitrile
Show/Hide
|
C20H21ClN2O3
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
Ki = 36 nM
|
|
|
|
CP0459658
|
(2S)-4-(imidazo[1,5-a]pyridin-1-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H21N3O2
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
Ki = 35 nM
|
|
|
|
CP0509059
|
(2S)-4-[(5-chloro-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H21ClN2O2
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
Ki = 37 nM
|
|
|
|
CP0563717
|
(2S)-4-(1H-indol-7-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H22N2O2
|
2
|
| 1 |
IC50 = 130 nM
|
|
|
| 2 |
Ki = 37 nM
|
|
|
|
CP0509051
|
(2S)-4-[(3,4-dimethoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 = 150 nM
|
|
|
| 2 |
Ki = 43 nM
|
|
|
|
CP0509055
|
(2S)-4-[(4-chlorophenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C18H20ClNO2
|
2
|
| 1 |
IC50 = 150 nM
|
|
|
| 2 |
Ki = 42 nM
|
|
|
|
CP0572540
|
(2S)-4-[(4-chlorophenyl)methyl]-2-[(4-methoxyphenoxy)methyl]morpholine
Show/Hide
|
C19H22ClNO3
|
2
|
| 1 |
IC50 = 150 nM
|
|
|
| 2 |
Ki = 42 nM
|
|
|
|
CP0559234
|
(2S)-4-[(4-methoxyphenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H23NO3
|
2
|
| 1 |
IC50 = 160 nM
|
|
|
| 2 |
Ki = 44 nM
|
|
|
|
CP0472285
|
(2S)-4-[(1-methylindazol-5-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H23N3O2
|
2
|
| 1 |
IC50 = 170 nM
|
|
|
| 2 |
Ki = 47 nM
|
|
|
|
CP0509052
|
(2S)-2-(phenoxymethyl)-4-[[4-(trifluoromethoxy)phenyl]methyl]morpholine
Show/Hide
|
C19H20F3NO3
|
2
|
| 1 |
IC50 = 180 nM
|
|
|
| 2 |
Ki = 51 nM
|
|
|
|
CP0563723
|
(2S)-4-[(4-methoxyphenyl)methyl]-2-(pyridin-3-yloxymethyl)morpholine
Show/Hide
|
C18H22N2O3
|
2
|
| 1 |
IC50 = 210 nM
|
|
|
| 2 |
Ki = 59 nM
|
|
|
|
CP0509050
|
(2S)-4-[(2,2-difluoro-1,3-benzodioxol-5-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H19F2NO4
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
Ki = 72 nM
|
|
|
|
CP0509057
|
(2S)-4-[(3-chloro-4-methoxyphenyl)methyl]-2-[(6-fluoropyridin-2-yl)oxymethyl]morpholine
Show/Hide
|
C18H20ClFN2O3
|
2
|
| 1 |
IC50 = 260 nM
|
|
|
| 2 |
Ki = 73 nM
|
|
|
|
CP0566401
|
(2S)-4-[[4-fluoro-3-(trifluoromethyl)phenyl]methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H19F4NO2
|
2
|
| 1 |
IC50 = 320 nM
|
|
|
| 2 |
Ki = 89 nM
|
|
|
|
CP0559236
|
(2S)-2-[(4-methoxyphenoxy)methyl]-4-[(4-methoxyphenyl)methyl]morpholine
Show/Hide
|
C20H25NO4
|
2
|
| 1 |
IC50 = 380 nM
|
|
|
| 2 |
Ki = 110 nM
|
|
|
|
CP0384376
|
N-(3-methylphenyl)-2-[4-(5-methylpyridin-2-yl)piperidin-1-yl]acetamide
Show/Hide
|
C20H25N3O
|
2
|
| 1 |
IC50 = 394 nM
|
|
|
| 2 |
IC50 = 453 nM
|
|
|
|
CP0376283
|
(2S)-4-[(4-chlorophenyl)methyl]-2-[(6-fluoropyridin-2-yl)oxymethyl]morpholine
Show/Hide
|
C17H18ClFN2O2
|
2
|
| 1 |
IC50 = 460 nM
|
|
|
| 2 |
Ki = 130 nM
|
|
|
|
CP0563722
|
(2S)-4-[(5-methoxy-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C21H24N2O3
|
2
|
| 1 |
IC50 = 460 nM
|
|
|
| 2 |
Ki = 130 nM
|
|
|
|
CP0472288
|
(2S)-4-[(3,4-difluorophenyl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C18H19F2NO2
|
2
|
| 1 |
IC50 = 530 nM
|
|
|
| 2 |
Ki = 150 nM
|
|
|
|
CP0448072
|
(2S)-4-(imidazo[1,2-a]pyridin-2-ylmethyl)-2-(phenoxymethyl)morpholine
Show/Hide
|
C19H21N3O2
|
2
|
| 1 |
IC50 = 590 nM
|
|
|
| 2 |
Ki = 160 nM
|
|
|
|
CP0376279
|
(2S)-2-(phenoxymethyl)-4-(quinolin-2-ylmethyl)morpholine
Show/Hide
|
C21H22N2O2
|
2
|
| 1 |
IC50 = 1110 nM
|
|
|
| 2 |
Ki = 310 nM
|
|
|
|
CP0376280
|
(2S)-4-[(4-chlorophenyl)methyl]-2-(pyridin-2-yloxymethyl)morpholine
Show/Hide
|
C17H19ClN2O2
|
2
|
| 1 |
IC50 = 2630 nM
|
|
|
| 2 |
Ki = 730 nM
|
|
|
|
CP0384675
|
N-(3-methylphenyl)-2-[4-(4-methylphenyl)piperidin-1-yl]acetamide
Show/Hide
|
C21H26N2O
|
2
|
| 1 |
IC50 = 3064 nM
|
|
|
| 2 |
IC50 = 7352 nM
|
|
|
|
CP0376273
|
(2S)-4-[(4-fluoro-1H-indol-3-yl)methyl]-2-(phenoxymethyl)morpholine
Show/Hide
|
C20H21FN2O2
|
2
|
| 1 |
IC50 = 3830 nM
|
|
|
| 2 |
Ki = 1060 nM
|
|
|
|
CP0416633
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-methylphenyl)acetamide
Show/Hide
|
C18H21ClN4O
|
2
|
| 1 |
IC50 = 4701 nM
|
|
|
| 2 |
IC50 = 7777 nM
|
|
|
|
CP0384367
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-(3-ethylphenyl)acetamide
Show/Hide
|
C19H23ClN4O
|
2
|
| 1 |
IC50 = 7059 nM
|
|
|
| 2 |
IC50 = 10449 nM
|
|
|
|
CP0494751
|
9-Oxo-1-propyl-2,3,4a,9,10,10a-hexahydro-1H-4-oxa-9lambda*4*-thia-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0418912
|
7-N,7-N-dipropyl-7,8-dihydro-6H-cyclopenta[g][1,3]benzothiazole-2,7-diamine
Show/Hide
|
C16H23N3S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0377202
|
N-methyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C22H25N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0377208
|
N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C21H23N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0398637
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-1-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0416325
|
N-ethyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C23H27N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0416326
|
N-(cyclopropylmethyl)-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417851
|
N-benzyl-N-[3-(4-methylpiperazin-1-yl)phenyl]naphthalene-2-sulfonamide
Show/Hide
|
C28H29N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0417858
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylbenzenesulfonamide
Show/Hide
|
C20H27N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0487098
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propylnaphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0421988
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyridin-3-ylacetamide
Show/Hide
|
C16H18ClN5O
|
2
|
| 1 |
IC50 = 23450 nM
|
|
|
| 2 |
IC50 = 40000 nM
|
|
|
|
CP0384366
|
2-[4-(4-chlorophenyl)piperidin-1-yl]-N-(3-methylphenyl)acetamide
Show/Hide
|
C20H23ClN2O
|
2
|
| 1 |
IC50 = 42357 nM
|
|
|
| 2 |
IC50 = 70157 nM
|
|
|
|
CP0137322
|
1H-indol-2-yl-[4-[2-(4-methoxyphenoxy)ethyl]piperazin-1-yl]methanone
Show/Hide
|
C22H25N3O3
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0384383
|
2-(4-pyridin-2-ylpiperazin-1-yl)-N-pyrimidin-5-ylacetamide
Show/Hide
|
C15H18N6O
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0384678
|
2-[4-(5-chloropyridin-2-yl)piperazin-1-yl]-N-pyrimidin-5-ylacetamide
Show/Hide
|
C15H17ClN6O
|
1
|
| 1 |
IC50 > 100000 nM
|
|
|
|
CP0398640
|
N-[3-(4-methylpiperazin-1-yl)phenyl]-N-propan-2-ylnaphthalene-2-sulfonamide
Show/Hide
|
C24H29N3O2S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0380100
|
2-(3-(3-fluorophenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl)-N,N-dimethylethanamine
Show/Hide
|
C17H18FN3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0405688
|
2-[3-(3-chlorophenyl)sulfonylpyrrolo[2,3-b]pyridin-1-yl]-N,N-dimethylethanamine
Show/Hide
|
C17H18ClN3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0419036
|
N,N-dimethyl-2-(3-naphthalen-1-ylsulfonylpyrrolo[2,3-b]pyridin-1-yl)ethanamine
Show/Hide
|
C21H21N3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0424416
|
2-[3-(Phenylsulfonyl)-1H-pyrrolo[2,3-b]pyridin-1-yl]ethylamine
Show/Hide
|
C15H15N3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0439248
|
2-{3-[(3-Chlorophenyl)sulfonyl]-1H-pyrrolo[2,3-b]pyridin-1-yl}ethylamine
Show/Hide
|
C15H14ClN3O2S
|
1
|
| 1 |
IC50 > 5000 nM
|
|
|
|
CP0393312
|
3-Benzyl-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H19NO3
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0409290
|
(R)-1-Phenoxy-3-(4-phenoxy-piperidin-1-yl)-propan-2-ol
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0008601
|
4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1-(4-fluoro-phenyl)-butan-1-one;propionate(HCl)
Show/Hide
|
C21H23ClFNO2
|
1
|
| 1 |
Ki = 2.2 nM
|
|
|
|
CP0429011
|
3-(4-Chloro-benzyl)-8-hydroxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C19H16ClNO3
|
1
|
| 1 |
Ki = 2.4 nM
|
|
|
|
CP0422922
|
8-Methoxy-3-(4-methyl-benzyl)-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
Ki = 2.6 nM
|
|
|
|
CP0405628
|
3-Benzyl-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H19NO2
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0375013
|
1-Phenoxy-3-(4-phenoxy-piperidin-1-yl)-propan-2-ol
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 3.6 nM
|
|
|
|
CP0448817
|
3-(4-Fluoro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18FNO3
|
1
|
| 1 |
Ki = 4.3 nM
|
|
|
|
CP0502203
|
7-(4-Phenyl-3,6-dihydro-2H-pyridin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H19NO2
|
1
|
| 1 |
Ki = 4.4 nM
|
|
|
|
CP0269449
|
4-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C18H19Cl2N3O
|
1
|
| 1 |
Ki = 5.3 nM
|
|
|
|
CP0269450
|
4-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C19H19ClN4O
|
1
|
| 1 |
Ki = 5.5 nM
|
|
|
|
CP0040248
|
7-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-one
Show/Hide
|
C18H18N2O2
|
1
|
| 1 |
Ki = 5.8 nM
|
|
|
|
CP0178951
|
N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]-4-methylbenzamide
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
Ki = 6.5 nM
|
|
|
|
CP0076889
|
N-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]-3-methylbenzamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
Ki = 6.7 nM
|
|
|
|
CP0402061
|
7-[4-(3-Chloro-4-methyl-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C21H21ClN2O2
|
1
|
| 1 |
Ki = 6.9 nM
|
|
|
|
CP0424524
|
8-Methoxy-3-(4-nitro-benzyl)-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18N2O5
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0439261
|
3-(4-Fluoro-benzyl)-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18FNO2
|
1
|
| 1 |
Ki = 7.5 nM
|
|
|
|
CP0215268
|
N-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]-4-methylbenzamide
Show/Hide
|
C20H25N3O2
|
1
|
| 1 |
Ki = 7.7 nM
|
|
|
|
CP0432916
|
8-Methoxy-3-phenethyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H21NO3
|
1
|
| 1 |
Ki = 7.9 nM
|
|
|
|
CP0375155
|
8-Methoxy-3-(4-trifluoromethyl-benzyl)-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H18F3NO3
|
1
|
| 1 |
Ki = 8.2 nM
|
|
|
|
CP0406449
|
3-(4-Chloro-benzyl)-8,9-dimethoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H20ClNO4
|
1
|
| 1 |
Ki = 8.5 nM
|
|
|
|
CP0159532
|
N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]-3-methylbenzamide
Show/Hide
|
C20H22N4O
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0409709
|
3-(4-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18ClNO3
|
1
|
| 1 |
Ki = 8.7 nM
|
|
|
|
CP0441413
|
7-[(2-p-Tolylamino-ethylamino)-methyl]-chromen-2-one
Show/Hide
|
C19H20N2O2
|
1
|
| 1 |
Ki = 10 nM
|
|
|
|
CP0393326
|
3-(4-Chloro-benzyl)-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18ClNO2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0428725
|
6-(4-p-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0420854
|
(S)-1-Phenoxy-3-(4-phenoxy-piperidin-1-yl)-propan-2-ol
Show/Hide
|
C20H25NO3
|
1
|
| 1 |
Ki = 11.6 nM
|
|
|
|
CP0269448
|
N-[[4-(2-chlorophenyl)piperazin-1-yl]methyl]-4-methylbenzamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0110881
|
4-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C19H22ClN3O2
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0378770
|
7-{[2-(4-Chloro-phenylamino)-ethylamino]-methyl}-chromen-2-one
Show/Hide
|
C18H17ClN2O2
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0460169
|
7-[4-(3,4-Dimethyl-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C22H24N2O2
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0178952
|
3-Chloro-N-[4-(2-methoxy-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C19H22ClN3O2
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0025667
|
2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl-2,3-dihydro-indol-1-yl)-ethanone
Show/Hide
|
C18H19ClN4
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0415028
|
3-Benzyl-7,8-dimethoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H21NO4
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0437764
|
7-(4-o-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0455466
|
7-{[2-(3-Chloro-4-methyl-phenylamino)-ethylamino]-methyl}-chromen-2-one
Show/Hide
|
C19H19ClN2O2
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0449041
|
3-(3-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18ClNO3
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0496150
|
7-(4-p-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0412072
|
(-)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO2S
|
1
|
| 1 |
Ki = 17.6 nM
|
|
|
|
CP0467603
|
1-(Naphthalen-1-yloxy)-3-(4-phenoxy-piperidin-1-yl)-propan-2-ol
Show/Hide
|
C24H27NO3
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0487048
|
1-(4-Benzyl-piperidin-1-yl)-3-(4-chloro-phenoxy)-propan-2-ol
Show/Hide
|
C21H26ClNO2
|
1
|
| 1 |
Ki = 18 nM
|
|
|
|
CP0402815
|
7-(4-Phenyl-piperidin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H21NO2
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0372930
|
7-{[2-(3,4-Dimethyl-phenylamino)-ethylamino]-methyl}-chromen-2-one
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0442595
|
7-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C19H25NOS
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0311650
|
N-[[4-(2-methoxyphenyl)piperazin-1-yl]methyl]benzamide
Show/Hide
|
C19H23N3O2
|
1
|
| 1 |
Ki = 22 nM
|
|
|
|
CP0404069
|
((R)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-(2-thiophen-2-yl-ethyl)-amine
Show/Hide
|
C20H27NOS
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0055058
|
3-(4-(3,6-dihydro-4-phenyl-1(2H)-pyridinyl)butyl)-1H-indol-5-ol
Show/Hide
|
C23H26N2O
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0457060
|
1-(4-Benzyl-piperidin-1-yl)-3-(naphthalen-1-yloxy)-propan-2-ol
Show/Hide
|
C25H29NO2
|
1
|
| 1 |
Ki = 26 nM
|
|
|
|
CP0141757
|
N-[[4-(2-cyanophenyl)piperazin-1-yl]methyl]benzamide
Show/Hide
|
C19H20N4O
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0178940
|
N-[[4-(2-chlorophenyl)piperazin-1-yl]methyl]-3-methylbenzamide
Show/Hide
|
C19H22ClN3O
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0527494
|
7-(4-Phenyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
Ki = 27 nM
|
|
|
|
CP0461830
|
6-(4-Phenyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C20H20N2O2
|
1
|
| 1 |
Ki = 30 nM
|
|
|
|
CP0514194
|
7-[(3-Phenylamino-propylamino)-methyl]-chromen-2-one
Show/Hide
|
C19H20N2O2
|
1
|
| 1 |
Ki = 31 nM
|
|
|
|
CP0439589
|
7-(Methyl-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0110876
|
N-[[4-(2-chlorophenyl)piperazin-1-yl]methyl]benzamide
Show/Hide
|
C18H20ClN3O
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0403331
|
1-(Naphthalen-1-yloxy)-3-(4-phenylsulfanyl-piperidin-1-yl)-propan-2-ol
Show/Hide
|
C24H27NO2S
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0456581
|
1-[4-(4-Fluoro-benzyl)-piperidin-1-yl]-3-(naphthalen-1-yloxy)-propan-2-ol
Show/Hide
|
C25H28FNO2
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0461319
|
7-(4-m-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 32 nM
|
|
|
|
CP0040962
|
3-Chloro-N-[4-(2-cyano-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C19H19ClN4O
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0405629
|
3-(2-Chloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H18ClNO3
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0457280
|
1-(4-Benzyl-piperidin-1-yl)-3-phenoxy-propan-2-ol
Show/Hide
|
C21H27NO2
|
1
|
| 1 |
Ki = 34 nM
|
|
|
|
CP0374678
|
3-Chloro-N-[4-(2-chloro-phenyl)-piperazin-1-ylmethyl]-benzamide
Show/Hide
|
C18H19Cl2N3O
|
1
|
| 1 |
Ki = 41 nM
|
|
|
|
CP0380911
|
7-[(2-Phenoxy-ethylamino)-methyl]-chromen-2-one
Show/Hide
|
C18H17NO3
|
1
|
| 1 |
Ki = 43 nM
|
|
|
|
CP0401205
|
(trans)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO2S
|
1
|
| 1 |
Ki = 44.4 nM
|
|
|
|
CP0375057
|
4-Benzyl-1-[2-methoxy-3-(naphthalen-1-yloxy)-propyl]-piperidine
Show/Hide
|
C26H31NO2
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0496793
|
1-[4-(4-Chloro-benzyl)-piperidin-1-yl]-3-(naphthalen-1-yloxy)-propan-2-ol
Show/Hide
|
C25H28ClNO2
|
1
|
| 1 |
Ki = 45 nM
|
|
|
|
CP0413983
|
(2R,3R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C16H25NO
|
1
|
| 1 |
Ki = 47 nM
|
|
|
|
CP0409085
|
((1S,2R)-5-Methoxy-1-methyl-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine
Show/Hide
|
C18H29NO
|
1
|
| 1 |
Ki = 48 nM
|
|
|
|
CP0449628
|
4-Benzyl-1-[3-(naphthalen-1-yloxy)-propyl]-piperidine
Show/Hide
|
C25H29NO
|
1
|
| 1 |
Ki = 50 nM
|
|
|
|
CP0441504
|
1-[4-(4-Methyl-benzyl)-piperidin-1-yl]-3-(naphthalen-1-yloxy)-propan-2-ol
Show/Hide
|
C26H31NO2
|
1
|
| 1 |
Ki = 52 nM
|
|
|
|
CP0374327
|
(R)6-(Phenethyl-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C21H27NO
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0494825
|
7-(Phenethyl-propyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C21H27NO
|
1
|
| 1 |
Ki = 54 nM
|
|
|
|
CP0343133
|
(S)-6-[Propyl-(2-thiophen-2-yl-ethyl)-amino]-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C19H25NOS
|
1
|
| 1 |
Ki = 55 nM
|
|
|
|
CP0449627
|
1-(4-Benzyl-piperidin-1-yl)-3-(4-nitro-phenoxy)-propan-2-ol
Show/Hide
|
C21H26N2O4
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0425902
|
7-[4-(4-Fluoro-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C20H19FN2O2
|
1
|
| 1 |
Ki = 59 nM
|
|
|
|
CP0419228
|
3-(3,4-Dichloro-benzyl)-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H17Cl2NO3
|
1
|
| 1 |
Ki = 61 nM
|
|
|
|
CP0416309
|
6-(4-o-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 63 nM
|
|
|
|
CP0448444
|
6-[Propyl-(2-thiophen-3-yl-ethyl)-amino]-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C19H25NOS
|
1
|
| 1 |
Ki = 72 nM
|
|
|
|
CP0494343
|
4-Benzyl-1-[2-methyl-3-(naphthalen-1-yloxy)-propyl]-piperidine
Show/Hide
|
C26H31NO
|
1
|
| 1 |
Ki = 72 nM
|
|
|
|
CP0424527
|
8-Methoxy-3-pyridin-4-ylmethyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C19H18N2O3
|
1
|
| 1 |
Ki = 74 nM
|
|
|
|
CP0437431
|
1-[4-(4-Methoxy-benzyl)-piperidin-1-yl]-3-(naphthalen-1-yloxy)-propan-2-ol
Show/Hide
|
C26H31NO3
|
1
|
| 1 |
Ki = 74 nM
|
|
|
|
CP0455465
|
6-(4-m-Tolyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 74 nM
|
|
|
|
CP0502225
|
7-[4-(4-Methoxy-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C21H22N2O3
|
1
|
| 1 |
Ki = 75 nM
|
|
|
|
CP0437030
|
6-Propylamino-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C13H19NO
|
1
|
| 1 |
Ki = 76 nM
|
|
|
|
CP0393313
|
8-Methoxy-3-(4-methoxy-benzyl)-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C21H21NO4
|
1
|
| 1 |
Ki = 84 nM
|
|
|
|
CP0449096
|
7-[4-(4-Chloro-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C20H19ClN2O2
|
1
|
| 1 |
Ki = 93 nM
|
|
|
|
CP0044536
|
(2R)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C16H25NO
|
1
|
| 1 |
Ki = 110 nM
|
|
|
|
CP0338014
|
AJ 76
Show/Hide
|
C15H23NO
|
1
|
| 1 |
Ki = 117 nM
|
|
|
|
CP0420797
|
[(5S,6R)-6-(dipropylamino)-5-methyl-5,6,7,8-tetrahydronaphthalen-1-yl] trifluoromethanesulfonate
Show/Hide
|
C18H26F3NO3S
|
1
|
| 1 |
Ki = 121 nM
|
|
|
|
CP0457281
|
1-(4-Benzyl-piperidin-1-yl)-3-(4-methoxy-phenoxy)-propan-2-ol
Show/Hide
|
C22H29NO3
|
1
|
| 1 |
Ki = 123 nM
|
|
|
|
CP0405312
|
((S)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-(2-thiophen-2-yl-ethyl)-amine
Show/Hide
|
C20H27NOS
|
1
|
| 1 |
Ki = 134 nM
|
|
|
|
CP0127400
|
(-)-Pramipexole
Show/Hide
|
C10H17N3S
|
1
|
| 1 |
Ki = 138 nM
|
|
|
|
CP0420798
|
3-Benzyl-10-hydroxy-8-methyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H19NO3
|
1
|
| 1 |
Ki = 145 nM
|
|
|
|
CP0053493
|
(+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4,9-dioxa-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO3
|
1
|
| 1 |
Ki = 169 nM
|
|
|
|
CP0401215
|
(R)-6-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C16H25NO
|
1
|
| 1 |
Ki = 182 nM
|
|
|
|
CP0405425
|
(cis)1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO2S
|
1
|
| 1 |
Ki = 193 nM
|
|
|
|
CP0462767
|
7-[4-(4-tert-Butyl-phenyl)-piperazin-1-ylmethyl]-chromen-2-one
Show/Hide
|
C24H28N2O2
|
1
|
| 1 |
Ki = 227 nM
|
|
|
|
CP0077378
|
4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-phenylamine
Show/Hide
|
C21H22N2
|
1
|
| 1 |
Ki = 228 nM
|
|
|
|
CP0406988
|
7-Propylamino-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C13H19NO
|
1
|
| 1 |
Ki = 269 nM
|
|
|
|
CP0413018
|
6-N,6-N-dipropyl-6,7-dihydro-5H-cyclopenta[f][1,3]benzothiazole-2,6-diamine
Show/Hide
|
C16H23N3S
|
1
|
| 1 |
Ki = 272 nM
|
|
|
|
CP0211927
|
5-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridin-2-ylamine
Show/Hide
|
C20H21N3
|
1
|
| 1 |
Ki = 278 nM
|
|
|
|
CP0497505
|
6-[(2-Phenylamino-ethylamino)-methyl]-chromen-2-one
Show/Hide
|
C18H18N2O2
|
1
|
| 1 |
Ki = 311 nM
|
|
|
|
CP0409110
|
(5-Cyclopentyloxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-(2-thiophen-2-yl-ethyl)-amine
Show/Hide
|
C24H33NOS
|
1
|
| 1 |
Ki = 324 nM
|
|
|
|
CP0447814
|
((S)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine
Show/Hide
|
C17H27NO
|
1
|
| 1 |
Ki = 335 nM
|
|
|
|
CP0073517
|
6-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridin-3-ylamine
Show/Hide
|
C20H21N3
|
1
|
| 1 |
Ki = 371 nM
|
|
|
|
CP0498455
|
7-{[Ethyl-(2-phenylamino-ethyl)-amino]-methyl}-chromen-2-one
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 410 nM
|
|
|
|
CP0493877
|
3-Benzoyl-8-methoxy-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C20H17NO4
|
1
|
| 1 |
Ki = 420 nM
|
|
|
|
CP0375804
|
(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki = 485 nM
|
|
|
|
CP0275169
|
4-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridine
Show/Hide
|
C20H20N2
|
1
|
| 1 |
Ki = 570 nM
|
|
|
|
CP0442593
|
(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-methyl-amine
Show/Hide
|
C12H17NO
|
1
|
| 1 |
Ki = 603 nM
|
|
|
|
CP0494145
|
[(5S,6R)-5-methyl-6-(propylamino)-5,6,7,8-tetrahydronaphthalen-1-yl] trifluoromethanesulfonate
Show/Hide
|
C15H20F3NO3S
|
1
|
| 1 |
Ki = 621 nM
|
|
|
|
CP0221754
|
(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine
Show/Hide
|
C17H27NO
|
1
|
| 1 |
Ki = 634 nM
|
|
|
|
CP0216424
|
3-[4-(4-Phenyl-3,6-dihydro-2H-pyridin-1-yl)-but-1-ynyl]-pyridine
Show/Hide
|
C20H20N2
|
1
|
| 1 |
Ki = 681 nM
|
|
|
|
CP0428555
|
7-Dimethylamino-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C12H17NO
|
1
|
| 1 |
Ki = 729 nM
|
|
|
|
CP0456715
|
(5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dimethyl-amine
Show/Hide
|
C13H19NO
|
1
|
| 1 |
Ki = 734 nM
|
|
|
|
CP0447817
|
N,N-diethyl-5-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C15H23NO
|
1
|
| 1 |
Ki = 964 nM
|
|
|
|
CP0405626
|
7-(Ethyl-methyl-amino)-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C13H19NO
|
1
|
| 1 |
Ki = 1033 nM
|
|
|
|
CP0419743
|
((R)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dipropyl-amine
Show/Hide
|
C17H27NO
|
1
|
| 1 |
Ki = 1504 nM
|
|
|
|
CP0483810
|
N-ethyl-5-methoxy-1,2,3,4-tetrahydronaphthalen-2-amine
Show/Hide
|
C13H19NO
|
1
|
| 1 |
Ki = 1519 nM
|
|
|
|
CP0424568
|
(5S,6R)-5-Methyl-6-propylamino-5,6,7,8-tetrahydro-naphthalene-1-carboxylic acid methyl ester
Show/Hide
|
C16H23NO2
|
1
|
| 1 |
Ki = 1593 nM
|
|
|
|
CP0460846
|
7-{[2-(Ethyl-phenyl-amino)-ethylamino]-methyl}-chromen-2-one
Show/Hide
|
C20H22N2O2
|
1
|
| 1 |
Ki = 2664 nM
|
|
|
|
CP0537469
|
7-(4-Benzyl-piperazin-1-ylmethyl)-chromen-2-one
Show/Hide
|
C21H22N2O2
|
1
|
| 1 |
Ki = 2700 nM
|
|
|
|
CP0391260
|
(4aS,10bR)-4-propyl-3,4a,5,10b-tetrahydro-1H-chromeno[3,4-d][1,3]oxazin-9-ol
Show/Hide
|
C14H19NO3
|
1
|
| 1 |
Ki = 7000 nM
|
|
|
|
CP0275794
|
5-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine
Show/Hide
|
C11H15NO
|
1
|
| 1 |
Ki > 33333 nM
|
|
|
|
CP0402749
|
(+)-3-(1-Propyl-piperidin-3-yl)-benzonitrile
Show/Hide
|
C15H20N2
|
1
|
| 1 |
Ki > 933 nM
|
|
|
|
CP0448607
|
(-)-Trifluoro-methanesulfonic acid 3-(1-propyl-piperidin-3-yl)-phenyl ester
Show/Hide
|
C15H20F3NO3S
|
1
|
| 1 |
Ki > 933 nM
|
|
|
|
CP0470701
|
(+)-Trifluoro-methanesulfonic acid 3-(1-propyl-piperidin-3-yl)-phenyl ester
Show/Hide
|
C15H20F3NO3S
|
1
|
| 1 |
Ki > 933 nM
|
|
|
|
CP0430802
|
8-Methoxy-3-phenyl-1,2,3,4-tetrahydro-chromeno[3,4-c]pyridin-5-one
Show/Hide
|
C19H17NO3
|
1
|
| 1 |
Ki > 3300 nM
|
|
|
|
CP0442149
|
3-Benzyl-7-methoxy-1,2,3,4-tetrahydro-9-oxa-3-aza-phenanthren-10-one
Show/Hide
|
C20H19NO3
|
1
|
| 1 |
Ki > 3300 nM
|
|
|
|
CP0508599
|
(+)-1-Propyl-2,3,10,10a-tetrahydro-1H,4aH-4-oxa-9-thia-1-aza-phenanthren-6-ol
Show/Hide
|
C14H19NO2S
|
1
|
| 1 |
Ki > 3300 nM
|
|
|
|
CP0431710
|
6-N-propyl-6,7-dihydro-5H-cyclopenta[f][1,3]benzothiazole-2,6-diamine
Show/Hide
|
C13H17N3S
|
1
|
| 1 |
Ki > 3330 nM
|
|
|
|
CP0162288
|
7-Amino-5,6,7,8-tetrahydro-naphthalen-2-ol
Show/Hide
|
C10H13NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0297070
|
7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine
Show/Hide
|
C11H15NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0348498
|
6-Amino-5,6,7,8-tetrahydro-naphthalen-1-ol
Show/Hide
|
C10H13NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0401217
|
((R)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0405129
|
Butyl-(5-methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-amine
Show/Hide
|
C15H23NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0405625
|
((S)-7-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-propyl-amine
Show/Hide
|
C14H21NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0448509
|
(7S)-7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-2-ol
Show/Hide
|
C16H25NO
|
1
|
| 1 |
Ki > 3333 nM
|
|
|
|
CP0777252
|
2-Iodo-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C20H22IN3O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
|
CP0853639
|
2-Chloro-N-(3-(R)-1-pyrrolidin-2-ylmethyl-1H-indol-5-yl)-benzenesulfonamide
Show/Hide
|
C19H20ClN3O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
|
CP0860616
|
3-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
|
CP0873359
|
2-Chloro-N-[3-((R)-1-methyl-pyrrolidin-2-ylmethyl)-1H-indol-5-yl]-benzenesulfonamide
Show/Hide
|
C20H22ClN3O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
|
CP0376224
|
1-(2-Fluoro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H17FN2O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
|
CP0409239
|
1-(2-Chloro-benzenesulfonyl)-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole
Show/Hide
|
C19H17ClN2O2S
|
1
|
| 1 |
Ki > 5000 nM
|
|
|
