Compound ID |
Compound Name |
Compound Formula |
CP0915507
|
(S)-N-(2-(3-chlorophenyl)pyridin-3-yl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C27H24ClN5O3
|
2
|
1 |
IC50 = 4 nM
|
|
|
2 |
IC50 = 15 nM
|
|
|
CP0656832
|
SID90341472
Show/Hide
|
C23H27N5
|
2
|
1 |
IC50 = 4.74 nM
|
|
|
2 |
IC50 = 25 nM
|
|
|
CP0472109
|
N-[[1-(2-methoxyphenyl)indazol-5-yl]methyl]-2-propylpentanamide
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|
C23H29N3O2
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0479045
|
1-((1-(4-fluorophenyl)-5-methyl-1H-pyrazol-4-yl)methyl)-4-(3-methoxyphenyl)piperazine
Show/Hide
|
C22H25FN4O
|
2
|
1 |
IC50 = 5 nM
|
|
|
2 |
IC50 = 64.7 nM
|
|
|
CP0409410
|
3,4,5-trimethoxy-N-[N'-[4-methyl-3-[(4-phenylbenzoyl)amino]phenyl]carbamimidoyl]benzamide
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|
C31H30N4O5
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0068085
|
2-chloro-N-(4-chloro-3-(pyridin-2-yl)phenyl)-4-(methylsulfonyl)benzamide
Show/Hide
|
C19H14Cl2N2O3S
|
2
|
1 |
IC50 = 5.1 nM
|
|
|
2 |
IC50 = 7 nM
|
|
|
CP0873343
|
(S)-N-(1-(3-fluorophenyl)-1H-pyrazol-5-yl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C25H23FN6O3
|
2
|
1 |
IC50 = 7 nM
|
|
|
2 |
IC50 = 9 nM
|
|
|
CP0125962
|
4-((3-(2-fluoro-6-methoxyphenoxy)azetidin-1-yl)methyl)-5-methyl-1-phenyl-1H-pyrazole
Show/Hide
|
C21H22FN3O2
|
2
|
1 |
IC50 = 8.27 nM
|
|
|
2 |
IC50 = 124 nM
|
|
|
CP0416678
|
1-((5-chloro-3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-(4-fluorophenyl)piperazine
Show/Hide
|
C21H22ClFN4
|
2
|
1 |
IC50 = 10 nM
|
|
|
2 |
IC50 = 1860 nM
|
|
|
CP0887656
|
(S)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)-N-(2-phenylpyridin-3-yl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C27H25N5O3
|
1
|
1 |
IC50 = 12 nM
|
|
|
CP0282016
|
(8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclopropyl]-N-(2-phenylpyrazol-3-yl)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxamide
Show/Hide
|
C26H26N6O3
|
2
|
1 |
IC50 = 13 nM
|
|
|
2 |
IC50 = 22 nM
|
|
|
CP0851877
|
(S)-1,3-dioxo-N-(1-phenyl-1H-pyrazol-5-yl)-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C25H24N6O3
|
2
|
1 |
IC50 = 15 nM
|
|
|
2 |
IC50 = 18 nM
|
|
|
CP0917328
|
(S)-N-(2-(3-cyanophenyl)pyridin-3-yl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C28H24N6O3
|
2
|
1 |
IC50 = 16 nM
|
|
|
2 |
IC50 = 22 nM
|
|
|
CP0873347
|
(S)-N-(1-(3-chlorophenyl)-1H-pyrazol-5-yl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C25H23ClN6O3
|
2
|
1 |
IC50 = 18 nM
|
|
|
2 |
IC50 = 32 nM
|
|
|
CP0966119
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(morpholino)methanone
Show/Hide
|
C26H25ClN4O2S
|
1
|
1 |
IC50 = 18 nM
|
|
|
CP0501233
|
(8aS)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclopropyl]-N-(2-phenylphenyl)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxamide
Show/Hide
|
C29H28N4O3
|
2
|
1 |
IC50 = 19 nM
|
|
|
2 |
IC50 = 60 nM
|
|
|
CP0375517
|
1-((1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl)methyl)-4-(3-methoxyphenyl)piperazine
Show/Hide
|
C23H27FN4O
|
2
|
1 |
IC50 = 20 nM
|
|
|
2 |
IC50 = 823 nM
|
|
|
CP0655728
|
(S)-N-(biphenyl-2-yl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C28H26N4O3
|
2
|
1 |
IC50 = 21 nM
|
|
|
2 |
IC50 = 70 nM
|
|
|
CP0910633
|
(S)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)-N-(2-(thiophen-3-yl)pyridin-3-yl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C25H23N5O3S
|
2
|
1 |
IC50 = 21 nM
|
|
|
2 |
IC50 = 42 nM
|
|
|
CP0416561
|
3,4,5-trimethoxy-N-[[4-methyl-3-[(4-phenylbenzoyl)amino]phenyl]carbamoyl]benzamide
Show/Hide
|
C31H29N3O6
|
1
|
1 |
IC50 = 24 nM
|
|
|
CP0462652
|
N-[[1-(4-methoxyphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C23H29N3O2
|
1
|
1 |
IC50 = 40 nM
|
|
|
CP0043416
|
4-((3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl)methyl)-1-(2-fluorophenyl)-5-methyl-1H-pyrazole
Show/Hide
|
C23H26FN3O2
|
2
|
1 |
IC50 = 40.8 nM
|
|
|
2 |
IC50 = 216 nM
|
|
|
CP0851875
|
(S)-N-(2,6-dichloro-4-(methylsulfonyl)phenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C23H22Cl2N4O5S
|
2
|
1 |
IC50 = 42 nM
|
|
|
2 |
IC50 = 68 nM
|
|
|
CP0967786
|
5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-N-(pyridin-3-yl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine-2-carboxamide
Show/Hide
|
C27H22ClN5OS
|
1
|
1 |
IC50 = 56 nM
|
|
|
CP0416550
|
3,4,5-trimethoxy-N-[[4-methyl-3-[(4-phenylbenzoyl)amino]phenyl]carbamothioyl]benzamide
Show/Hide
|
C31H29N3O5S
|
1
|
1 |
IC50 = 63 nM
|
|
|
CP0136263
|
(3S,3'R,3'aS,6'S,6aS,6bS,7'aR,9R,11aS,11bR)-3',6',10,11b-tetramethylspiro[2,3,4,6,6a,6b,7,8,11,11a-decahydro-1H-benzo[a]fluorene-9,2'-3a,4,5,6,7,7a-hexahydro-3H-furo[3,2-b]pyridine]-3-ol
Show/Hide
|
C27H41NO2
|
1
|
1 |
IC50 = 64 nM
|
|
|
CP0496199
|
N-[[1-(3-methylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C23H29N3O
|
1
|
1 |
IC50 = 70 nM
|
|
|
CP0921973
|
(S)-N-(2,6-dichloro-4-(dimethylcarbamoyl)phenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C25H25Cl2N5O4
|
2
|
1 |
IC50 = 77 nM
|
|
|
2 |
IC50 = 120 nM
|
|
|
CP0051889
|
1-((5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-phenylpiperazine
Show/Hide
|
C21H24N4
|
2
|
1 |
IC50 = 78.4 nM
|
|
|
2 |
IC50 = 96 nM
|
|
|
CP0967785
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-(pyrimidin-2-yl)piperazin-1-yl)methanone
Show/Hide
|
C30H28ClN7OS
|
1
|
1 |
IC50 = 92 nM
|
|
|
CP0462651
|
N-[[1-(3-methoxyphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C23H29N3O2
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0884849
|
(S)-N-(2,6-dichloro-4-cyanophenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C23H19Cl2N5O3
|
2
|
1 |
IC50 = 100 nM
|
|
|
2 |
IC50 = 450 nM
|
|
|
CP0453815
|
1-(4-methoxyphenyl)-4-((5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)piperazine
Show/Hide
|
C22H26N4O
|
2
|
1 |
IC50 = 105 nM
|
|
|
2 |
IC50 = 126 nM
|
|
|
CP0416536
|
N-[(3-benzamidophenyl)carbamoyl]-3,4,5-trimethoxybenzamide
Show/Hide
|
C24H23N3O6
|
1
|
1 |
IC50 = 107 nM
|
|
|
CP0471969
|
N-[[1-(2,3-dimethylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C24H31N3O
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0429379
|
N-[[1-(6-methoxypyridin-3-yl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H28N4O2
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0472092
|
N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H26FN3O
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0968344
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-methylpiperazin-1-yl)methanone
Show/Hide
|
C27H28ClN5OS
|
1
|
1 |
IC50 = 135 nM
|
|
|
CP0505044
|
2-propyl-N-[[1-(5,6,7,8-tetrahydronaphthalen-1-yl)indazol-5-yl]methyl]pentanamide
Show/Hide
|
C26H33N3O
|
1
|
1 |
IC50 = 150 nM
|
|
|
CP0851874
|
(S)-N-(2,6-dichloro-4-fluorophenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C22H19Cl2FN4O3
|
2
|
1 |
IC50 = 180 nM
|
|
|
2 |
IC50 = 520 nM
|
|
|
CP0897580
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-hydroxypiperazin-1-yl)methanone
Show/Hide
|
C27H27ClN4O2S
|
1
|
1 |
IC50 = 192 nM
|
|
|
CP0427252
|
N-[[1-(2-methylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C23H29N3O
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0521125
|
N-[(1-phenylindazol-5-yl)methyl]-2-propylpentanamide
Show/Hide
|
C22H27N3O
|
1
|
1 |
IC50 = 200 nM
|
|
|
CP0952084
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-(3,4-dichlorophenyl)piperazin-1-yl)methanone
Show/Hide
|
C32H28Cl3N5OS
|
1
|
1 |
IC50 = 213 nM
|
|
|
CP0968345
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-(methylsulfonyl)piperazin-1-yl)methanone
Show/Hide
|
C27H28ClN5O3S2
|
1
|
1 |
IC50 = 217 nM
|
|
|
CP0884850
|
(S)-N-(2,3-dichlorophenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C22H20Cl2N4O3
|
2
|
1 |
IC50 = 230 nM
|
|
|
2 |
IC50 = 690 nM
|
|
|
CP0894339
|
(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-(pyrimidin-2-yl)piperazin-1-yl)methanone
Show/Hide
|
C30H29N7OS
|
1
|
1 |
IC50 = 237 nM
|
|
|
CP0858770
|
5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-N-(pyridin-3-yl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine-2-carboxamide
Show/Hide
|
C27H23N5OS
|
1
|
1 |
IC50 = 261 nM
|
|
|
CP0891470
|
(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(morpholino)methanone
Show/Hide
|
C26H26N4O2S
|
1
|
1 |
IC50 = 294 nM
|
|
|
CP0390282
|
N-[(3-benzamidophenyl)carbamothioyl]-3,4,5-trimethoxybenzamide
Show/Hide
|
C24H23N3O5S
|
1
|
1 |
IC50 = 300 nM
|
|
|
CP0508050
|
3-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-1,1-dipropylurea
Show/Hide
|
C21H25FN4O
|
1
|
1 |
IC50 = 310 nM
|
|
|
CP0858771
|
(5-(4-chloro-3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(pyrrolidin-1-yl)methanone
Show/Hide
|
C26H25ClN4OS
|
1
|
1 |
IC50 = 315 nM
|
|
|
CP0952083
|
(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-methylpiperazin-1-yl)methanone
Show/Hide
|
C27H29N5OS
|
1
|
1 |
IC50 = 326 nM
|
|
|
CP0416679
|
1-((5-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-(3-(trifluoromethyl)phenyl)piperazine
Show/Hide
|
C22H23F3N4
|
2
|
1 |
IC50 = 328 nM
|
|
|
2 |
IC50 = 333 nM
|
|
|
CP0505995
|
N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2,2-dimethylpentanamide
Show/Hide
|
C21H24FN3O
|
1
|
1 |
IC50 = 330 nM
|
|
|
CP0462654
|
N-[[1-(2-methoxypyridin-3-yl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H28N4O2
|
1
|
1 |
IC50 = 340 nM
|
|
|
CP0963828
|
N,N-diethyl-5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridine-2-carboxamide
Show/Hide
|
C26H26N4OS
|
1
|
1 |
IC50 = 352 nM
|
|
|
CP0504283
|
N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2-methylpentanamide
Show/Hide
|
C20H22FN3O
|
1
|
1 |
IC50 = 360 nM
|
|
|
CP0967784
|
(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)(4-(methylsulfonyl)piperazin-1-yl)methanone
Show/Hide
|
C27H29N5O3S2
|
1
|
1 |
IC50 = 373 nM
|
|
|
CP0966118
|
(4-hydroxypiperidin-1-yl)(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)methanone
Show/Hide
|
C27H28N4O2S
|
1
|
1 |
IC50 = 431 nM
|
|
|
CP0968342
|
(4-(3,4-dichlorophenyl)piperazin-1-yl)(5-(3-(1-methyl-1H-benzo[d]imidazol-2-yl)phenyl)-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-2-yl)methanone
Show/Hide
|
C32H29Cl2N5OS
|
1
|
1 |
IC50 = 456 nM
|
|
|
CP0917084
|
(R)-N-(2,3-dichlorophenyl)-1,3-dioxo-2-((1S,2R)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C22H20Cl2N4O3
|
1
|
1 |
IC50 = 650 nM
|
|
|
CP0917327
|
(S)-N-(2,3-dichlorophenyl)-1,3-dioxo-2-((1R,2S)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
Show/Hide
|
C22H20Cl2N4O3
|
1
|
1 |
IC50 = 670 nM
|
|
|
CP0514395
|
N-[[1-(3-fluorophenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H26FN3O
|
1
|
1 |
IC50 = 680 nM
|
|
|
CP0514448
|
2-ethyl-N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]butanamide
Show/Hide
|
C20H22FN3O
|
1
|
1 |
IC50 = 720 nM
|
|
|
CP0514371
|
N-[[1-(4-methylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C23H29N3O
|
1
|
1 |
IC50 = 900 nM
|
|
|
CP0514663
|
N-[[1-(2-fluorophenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H26FN3O
|
1
|
1 |
IC50 = 900 nM
|
|
|
CP0508051
|
N-[[1-(2,6-dimethylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C24H31N3O
|
1
|
1 |
IC50 = 950 nM
|
|
|
CP0472093
|
N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]pentanamide
Show/Hide
|
C19H20FN3O
|
1
|
1 |
IC50 = 1200 nM
|
|
|
CP0504285
|
N-[[1-(4-chlorophenyl)indazol-5-yl]methyl]-2-propylpentanamide
Show/Hide
|
C22H26ClN3O
|
1
|
1 |
IC50 = 1200 nM
|
|
|
CP0388253
|
(8aR)-8a-methyl-1,3-dioxo-2-[(1S,2R)-2-phenylcyclopropyl]-N-(2-phenylphenyl)-6,8-dihydro-5H-imidazo[1,5-a]pyrazine-7-carboxamide
Show/Hide
|
C29H28N4O3
|
2
|
1 |
IC50 = 1200 nM
|
|
|
2 |
IC50 = 1600 nM
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CP0505034
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1-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-1-methyl-3,3-dipropylurea
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C22H27FN4O
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1
|
1 |
IC50 = 1300 nM
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|
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CP0462653
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N-[[1-(4-acetylphenyl)indazol-5-yl]methyl]-2-propylpentanamide
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C24H29N3O2
|
1
|
1 |
IC50 = 1400 nM
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|
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CP0473611
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1-((1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl)methyl)-4-(4-methoxyphenyl)piperazine
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C23H27FN4O
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2
|
1 |
IC50 = 1690 nM
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|
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2 |
IC50 = 2000 nM
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CP0851876
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(R)-N-(2,3-dichlorophenyl)-1,3-dioxo-2-((1R,2S)-2-phenylcyclopropyl)hexahydroimidazo[1,5-a]pyrazine-7(1H)-carboxamide
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C22H20Cl2N4O3
|
1
|
1 |
IC50 = 1700 nM
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|
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CP0402634
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tert-butyl 4-[5-[(2-propylpentanoylamino)methyl]indazol-1-yl]benzoate
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C27H35N3O3
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1
|
1 |
IC50 = 1800 nM
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|
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CP0514664
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2-propyl-N-[(1-pyridin-3-ylindazol-5-yl)methyl]pentanamide
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C21H26N4O
|
1
|
1 |
IC50 = 1830 nM
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|
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CP0416673
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1-((3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)methyl)-4-(2-methoxyphenyl)piperazine
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C23H28N4O
|
2
|
1 |
IC50 = 1870 nM
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|
|
2 |
IC50 > 5000 nM
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|
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CP0402633
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N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-N-methyl-2-propylpentanamide
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C23H28FN3O
|
1
|
1 |
IC50 = 3000 nM
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|
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CP0455258
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2-propyl-N-[(1-pyridin-4-ylindazol-5-yl)methyl]pentanamide
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|
C21H26N4O
|
1
|
1 |
IC50 = 4500 nM
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|
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CP0402635
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2-propyl-N-[(1-pyrimidin-2-ylindazol-5-yl)methyl]pentanamide
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C20H25N5O
|
1
|
1 |
IC50 = 6300 nM
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|
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CP0427346
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N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2-phenylacetamide
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C22H18FN3O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0431076
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N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]cyclohexanecarboxamide
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C21H22FN3O
|
1
|
1 |
IC50 = 10000 nM
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|
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CP0455257
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2-propyl-N-[(1-pyridin-2-ylindazol-5-yl)methyl]pentanamide
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C21H26N4O
|
1
|
1 |
IC50 > 10000 nM
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|
|
CP0496436
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N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2-methylpropanamide
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|
C18H18FN3O
|
1
|
1 |
IC50 = 10000 nM
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|
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CP0499036
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N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]-2,2-dimethylpropanamide
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C19H20FN3O
|
1
|
1 |
IC50 = 10000 nM
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|
|
CP0506002
|
N-[[1-(4-fluorophenyl)indazol-5-yl]methyl]benzamide
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C21H16FN3O
|
1
|
1 |
IC50 = 10000 nM
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|
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CP0504286
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2-propyl-N-[(1-pyrazin-2-ylindazol-5-yl)methyl]pentanamide
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C20H25N5O
|
1
|
1 |
IC50 > 25000 nM
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|
|
CP0416675
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1-(4-methoxyphenyl)-4-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)piperazine
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C22H26N4O
|
1
|
1 |
IC50 > 5000 nM
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|
|
CP0453814
|
1-(4-fluorophenyl)-4-((3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl)piperazine
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|
C21H23FN4
|
1
|
1 |
IC50 > 5000 nM
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|
|