| Compound ID |
Compound Name |
Compound Formula |
|
CP0420680
|
2-[2-oxo-2-[[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]amino]ethyl]sulfanyl-N-(3,4,5-trimethoxyphenyl)acetamide
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|
C31H34N4O5S
|
4
|
| 1 |
IC50 = 0.07 nM
|
|
|
| 2 |
IC50 = 0.64 nM
|
|
|
| 3 |
IC50 = 1.9 nM
|
|
|
| 4 |
IC50 = 185 nM
|
|
|
|
CP0435474
|
N-(1,3-benzothiazol-6-yl)-2-[2-oxo-2-[[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]amino]ethyl]sulfanylacetamide
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|
C29H27N5O2S2
|
4
|
| 1 |
IC50 = 0.78 nM
|
|
|
| 2 |
IC50 = 2.9 nM
|
|
|
| 3 |
IC50 = 34 nM
|
|
|
| 4 |
IC50 = 172 nM
|
|
|
|
CP0484088
|
N-naphthalen-2-yl-2-[2-oxo-2-[[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]amino]ethyl]sulfanylacetamide
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|
C32H30N4O2S
|
4
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 7 nM
|
|
|
| 3 |
IC50 = 46 nM
|
|
|
| 4 |
IC50 = 153 nM
|
|
|
|
CP0476494
|
2-[2-(5,6-dihydrobenzo[b][1]benzazepin-11-yl)-2-oxoethyl]sulfanyl-N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]acetamide
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|
C36H34N4O2S
|
4
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 6 nM
|
|
|
| 3 |
IC50 = 52 nM
|
|
|
| 4 |
IC50 = 164 nM
|
|
|
|
CP0435473
|
5-bromo-N-[3-[2-oxo-2-[[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]amino]ethyl]sulfanylphenyl]pyridine-3-carboxamide
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|
C32H28BrN5O2S
|
4
|
| 1 |
IC50 = 6 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
| 3 |
IC50 = 20 nM
|
|
|
| 4 |
IC50 = 56 nM
|
|
|
|
CP0470736
|
2-[2-(benzhydrylamino)-2-oxoethyl]sulfanyl-N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]acetamide
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|
C35H34N4O2S
|
4
|
| 1 |
IC50 = 11 nM
|
|
|
| 2 |
IC50 = 16 nM
|
|
|
| 3 |
IC50 = 56 nM
|
|
|
| 4 |
IC50 = 160 nM
|
|
|
|
CP0420668
|
2-[2-(1-adamantylamino)-2-oxoethyl]sulfanyl-N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]acetamide
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|
C32H38N4O2S
|
4
|
| 1 |
IC50 = 13 nM
|
|
|
| 2 |
IC50 = 21 nM
|
|
|
| 3 |
IC50 = 109 nM
|
|
|
| 4 |
IC50 = 231 nM
|
|
|
|
CP0435475
|
N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]-2-(5H-[1,2,4]triazino[5,6-b]indol-3-ylsulfanyl)acetamide
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|
C29H25N7OS
|
3
|
| 1 |
IC50 = 17 nM
|
|
|
| 2 |
IC50 = 21 nM
|
|
|
| 3 |
IC50 = 426 nM
|
|
|
|
CP0420667
|
2-[2-(9H-fluoren-2-yl)-2-oxoethyl]sulfanyl-N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]acetamide
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|
C35H31N3O2S
|
4
|
| 1 |
IC50 = 57 nM
|
|
|
| 2 |
IC50 = 62 nM
|
|
|
| 3 |
IC50 = 154 nM
|
|
|
| 4 |
IC50 = 266 nM
|
|
|
|
CP0435472
|
2-[(5-cyclopropyl-1H-1,2,4-triazol-3-yl)sulfanyl]-N-[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]acetamide
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|
C25H26N6OS
|
4
|
| 1 |
IC50 = 59 nM
|
|
|
| 2 |
IC50 = 101 nM
|
|
|
| 3 |
IC50 = 194 nM
|
|
|
| 4 |
IC50 = 629 nM
|
|
|
|
CP0431675
|
N-[(4-fluorophenyl)methyl]-2-[2-oxo-2-[[2-phenyl-5-(2,4,5-trimethylphenyl)pyrazol-3-yl]amino]ethyl]sulfanylacetamide
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|
C29H29FN4O2S
|
4
|
| 1 |
IC50 = 131 nM
|
|
|
| 2 |
IC50 = 192 nM
|
|
|
| 3 |
IC50 = 379 nM
|
|
|
| 4 |
IC50 = 458 nM
|
|
|
