| Compound ID |
Compound Name |
Compound Formula |
|
CP0105792
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C27H30N4O4S
|
2
|
| 1 |
EC50 = 0.02 nM
|
|
|
| 2 |
Ki = 7.3 nM
|
|
|
|
CP0443504
|
(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-(cyclohexyloxy)biphenyl-4-carboxylic acid
Show/Hide
|
C28H33N3O4
|
1
|
| 1 |
EC50 = 0.035 nM
|
|
|
|
CP0418058
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-(cyclohexyloxy)-4-biphenylcarboxylic acid
Show/Hide
|
C28H33N3O4
|
1
|
| 1 |
EC50 = 0.035 nM
|
|
|
|
CP0377225
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(methoxymethyl)phenol
Show/Hide
|
C28H32N4O4S
|
2
|
| 1 |
EC50 = 0.04 nM
|
|
|
| 2 |
Ki = 1 nM
|
|
|
|
CP0699562
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(3-fluorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27FN4O2S
|
1
|
| 1 |
EC50 = 0.04 nM
|
|
|
|
CP0400941
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl)-3-isobutoxy-4-biphenylcarboxylic acid
Show/Hide
|
C28H33NO4
|
1
|
| 1 |
EC50 = 0.041 nM
|
|
|
|
CP0441442
|
4-((2R)-2-{[(2R)-2-Phenyl-2-hydroxyethyl]amino}propyl)-3-cyclohexyloxy-1,1-biphenyl-4-carboxylic acid
Show/Hide
|
C30H35NO4
|
1
|
| 1 |
EC50 = 0.042 nM
|
|
|
|
CP0399010
|
4'-(2-((1R,2S)-1-hydroxy-1-(3-hydroxyphenyl)propan-2-ylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C28H34N2O6S
|
1
|
| 1 |
EC50 = 0.044 nM
|
|
|
|
CP0486915
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethoxy)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C26H31N3O4
|
1
|
| 1 |
EC50 = 0.059 nM
|
|
|
|
CP0375681
|
(3-{2-[(R)-2-((R)-3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-yloxy)-acetic acid
Show/Hide
|
C21H23ClN2O4
|
1
|
| 1 |
EC50 = 0.062 nM
|
|
|
|
CP0851070
|
3-(Cyclohexylamino)-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Trihydrochloride
Show/Hide
|
C29H39Cl3N4O4S
|
1
|
| 1 |
EC50 = 0.062 nM
|
|
|
|
CP0510148
|
4-(2-{[(2R)-2-Hydroxy-2-(3-hydroxyphenyl)ethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H29NO5
|
1
|
| 1 |
EC50 = 0.062 nM
|
|
|
|
CP0440993
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]thiophene-3-carboxylic acid
Show/Hide
|
C22H23ClN2O3S
|
1
|
| 1 |
EC50 = 0.0631 nM
|
|
|
|
CP0375142
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H30N2O4
|
1
|
| 1 |
EC50 = 0.064 nM
|
|
|
|
CP0474560
|
(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
Show/Hide
|
C26H31N3O3
|
1
|
| 1 |
EC50 = 0.066 nM
|
|
|
|
CP0375138
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C26H31N3O3
|
1
|
| 1 |
EC50 = 0.066 nM
|
|
|
|
CP0498018
|
3-(Cyclohexyloxy)-4-((2R)-2-{[(2R)-2-hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-4-biphenylcarboxylic acid
Show/Hide
|
C29H34N2O4
|
1
|
| 1 |
EC50 = 0.069 nM
|
|
|
|
CP0443398
|
4'-[2-[[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino]ethyl]-3-(isopropylthio)-N-(methylsulfonyl)-4-biphenylcarboxamide
Show/Hide
|
C26H32N4O4S2
|
1
|
| 1 |
EC50 = 0.08 nM
|
|
|
|
CP0389986
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 0.091 nM
|
|
|
|
CP0400939
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridyl)ethyl]amino}propyl)-3-isopropyloxy-1,1-biphenyl-4-carboxylic acid
Show/Hide
|
C26H30N2O4
|
1
|
| 1 |
EC50 = 0.099 nM
|
|
|
|
CP0439425
|
3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-4-carboxylic acid
Show/Hide
|
C22H22ClN3O3
|
1
|
| 1 |
EC50 = 0.1 nM
|
|
|
|
CP0466916
|
3-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
EC50 = 0.1 nM
|
|
|
|
CP0404916
|
4'-((R)-2-((R)-2-hydroxy-2-phenylethylamino)propyl)-3-isobutyl-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C29H36N2O4S
|
1
|
| 1 |
EC50 = 0.1 nM
|
|
|
|
CP0071872
|
(3-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-yloxy)-acetic acid
Show/Hide
|
C21H23ClN2O4
|
1
|
| 1 |
EC50 = 0.11 nM
|
|
|
|
CP0900959
|
3-(Cyclohexyloxy)-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C29H37Cl2N3O5S
|
1
|
| 1 |
EC50 = 0.13 nM
|
|
|
|
CP0717837
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(4-fluorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27FN4O2S
|
1
|
| 1 |
EC50 = 0.13 nM
|
|
|
|
CP0877322
|
3-(Cyclohexylamino)-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C30H39Cl2N3O4S
|
1
|
| 1 |
EC50 = 0.14 nM
|
|
|
|
CP0389987
|
4-(2-{[(1S,2R)-2-Hydroxy-2-(4-hydroxyphenyl)-1-methylethyl]-amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO5
|
1
|
| 1 |
EC50 = 0.14 nM
|
|
|
|
CP0444628
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C28H33NO3
|
1
|
| 1 |
EC50 = 0.14 nM
|
|
|
|
CP0469324
|
2-ethyl-4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C28H32N4O3S
|
2
|
| 1 |
EC50 = 0.14 nM
|
|
|
| 2 |
Ki = 9 nM
|
|
|
|
CP0135429
|
(4R)-2-amino-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
EC50 = 0.15 nM
|
|
|
|
CP0765379
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-(3-chlorophenyl)(hydroxy)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27ClN4O2S
|
1
|
| 1 |
EC50 = 0.15 nM
|
|
|
|
CP0217241
|
4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-ylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C28H34N2O6S
|
1
|
| 1 |
EC50 = 0.16 nM
|
|
|
|
CP0440522
|
3-(Cyclohexyloxy)-4-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethoxy)-4-biphenylcarboxylic acid
Show/Hide
|
C29H33NO5
|
1
|
| 1 |
EC50 = 0.16 nM
|
|
|
|
CP0433877
|
4-[(2R)-2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}propyl]-4-biphenylcarboxylic acid
Show/Hide
|
C24H24ClNO3
|
1
|
| 1 |
EC50 = 0.18 nM
|
|
|
|
CP0881856
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)propanamide
Show/Hide
|
C24H28N4O2S
|
1
|
| 1 |
EC50 = 0.18 nM
|
|
|
|
CP0504380
|
(R)-4'-(2-(2-(4-aminopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 = 0.19 nM
|
|
|
|
CP0845123
|
4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-3-(isopropylsulfanyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C26H33Cl2N3O4S2
|
1
|
| 1 |
EC50 = 0.19 nM
|
|
|
|
CP0375143
|
4-((2R)-2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}propyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H30ClNO4
|
1
|
| 1 |
EC50 = 0.19 nM
|
|
|
|
CP0418057
|
4-(2-{[(2R)-2-(6-Amino-3-pyridinyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 = 0.19 nM
|
|
|
|
CP0403283
|
4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzene-1,3-dicarboxylic acid
Show/Hide
|
C25H25ClN2O5
|
1
|
| 1 |
EC50 = 0.1995 nM
|
|
|
|
CP0900958
|
4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-3-(isopropylamino)-N-(methylsulfonyl)biphenyl-4-carboxamide Trihydrochloride
Show/Hide
|
C26H35Cl3N4O4S
|
1
|
| 1 |
EC50 = 0.2 nM
|
|
|
|
CP0039168
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C24H27N3O6S3
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0444691
|
4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethoxy)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H28ClNO5
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0494785
|
4-[(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethyl)amino]-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H29ClN2O4
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0869787
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-4,5,6,7-tetrahydrobenzo[d]-thiazole-4-carboxamide
Show/Hide
|
C26H30N4O2S
|
1
|
| 1 |
EC50 = 0.21 nM
|
|
|
|
CP0488218
|
(R)-4'-(2-(2-(6-acetamidopyridin-3-yl)-2-hydroxyethylamino)ethyl)-3-(cyclohexyloxy)-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C31H38N4O6S
|
1
|
| 1 |
EC50 = 0.23 nM
|
|
|
|
CP0399444
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]furan-3-carboxylic acid
Show/Hide
|
C22H23ClN2O4
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0483335
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
EC50 = 0.2512 nM
|
|
|
|
CP0418060
|
(R)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
Show/Hide
|
C26H30N2O3
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0103438
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] pyridine-3-sulfonate
Show/Hide
|
C28H28N4O6S3
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0417355
|
(R)-4'-(2-(2-hydroxy-2-(4-hydroxy-3-(methylsulfonamido)phenyl)ethylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C28H35N3O8S2
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0389977
|
4-{2-[((2R)-2-Hydroxy-2-{4-hydroxy-3-[(methylsulfonyl)amino]-phenyl}ethyl)amino]ethyl}-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H32N2O7S
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0418059
|
(R)-3-(cyclohexyloxy)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)biphenyl-4-carboxylic acid
Show/Hide
|
C28H32N2O4
|
1
|
| 1 |
EC50 = 0.26 nM
|
|
|
|
CP0510153
|
4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethoxy)-3-(cyclohexyloxy)-4-biphenylcarboxylic acid
Show/Hide
|
C29H32ClNO5
|
1
|
| 1 |
EC50 = 0.27 nM
|
|
|
|
CP0039163
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] octane-1-sulfonate
Show/Hide
|
C31H41N3O6S3
|
1
|
| 1 |
EC50 = 0.28 nM
|
|
|
|
CP0495955
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(isopropylamino)biphenyl-4-carboxylic acid
Show/Hide
|
C26H30N2O3
|
1
|
| 1 |
EC50 = 0.29 nM
|
|
|
|
CP0914180
|
3-Cyclopentyl-4'-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C28H35Cl2N3O4S
|
1
|
| 1 |
EC50 = 0.29 nM
|
|
|
|
CP0381825
|
(R)-3-(cyclohexyloxy)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)biphenyl-4-carboxylic acid
Show/Hide
|
C29H33NO4
|
1
|
| 1 |
EC50 = 0.3 nM
|
|
|
|
CP0375141
|
4-[(2R)-2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}propyl]biphenyl-4-carboxylic acid
Show/Hide
|
C24H25NO3
|
1
|
| 1 |
EC50 = 0.3 nM
|
|
|
|
CP0133084
|
3-Amino-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C25H28N4O5S2
|
1
|
| 1 |
EC50 = 0.31 nM
|
|
|
|
CP0375140
|
3-Ethoxy-4-[(2R)-2-{[(2R)-2-hydroxy-2-phenylethyl]amino}propyl]-biphenyl-4-carboxylic acid
Show/Hide
|
C26H29NO4
|
1
|
| 1 |
EC50 = 0.31 nM
|
|
|
|
CP0382240
|
2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]furan-3-carboxylic acid
Show/Hide
|
C22H23ClN2O4
|
1
|
| 1 |
EC50 = 0.3162 nM
|
|
|
|
CP0845051
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylsulfanyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C27H33ClN2O4S2
|
1
|
| 1 |
EC50 = 0.32 nM
|
|
|
|
CP0851071
|
4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-3-isobutyl-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C27H35Cl2N3O4S
|
1
|
| 1 |
EC50 = 0.32 nM
|
|
|
|
CP0495906
|
4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethoxy)-3-isobutoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H30ClNO5
|
1
|
| 1 |
EC50 = 0.32 nM
|
|
|
|
CP0851074
|
3-Cyclohexyl-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C30H37ClN2O4S
|
1
|
| 1 |
EC50 = 0.33 nM
|
|
|
|
CP0433178
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-phenoxybiphenyl-4-carboxylic acid
Show/Hide
|
C29H27NO4
|
1
|
| 1 |
EC50 = 0.34 nM
|
|
|
|
CP0514692
|
3-(cyclohexyloxy)-4'-(2-((1R,2S)-1-hydroxy-1-(4-hydroxyphenyl)propan-2-ylamino)ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C31H38N2O6S
|
1
|
| 1 |
EC50 = 0.35 nM
|
|
|
|
CP0374720
|
(R)-1-((R)-3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
EC50 = 0.36 nM
|
|
|
|
CP0881884
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C24H27N5O2S
|
1
|
| 1 |
EC50 = 0.37 nM
|
|
|
|
CP0877323
|
3-(Cycloheptyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C31H39ClN2O5S
|
1
|
| 1 |
EC50 = 0.38 nM
|
|
|
|
CP0493893
|
4-((S)-7-((R)-2-(4-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
|
C25H24ClNO3
|
1
|
| 1 |
EC50 = 0.38 nM
|
|
|
|
CP0382241
|
2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]thiophene-3-carboxylic acid
Show/Hide
|
C22H23ClN2O3S
|
1
|
| 1 |
EC50 = 0.3981 nM
|
|
|
|
CP0849244
|
3-Cyclopentyl-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C29H35ClN2O4S
|
1
|
| 1 |
EC50 = 0.41 nM
|
|
|
|
CP0474707
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 0.43 nM
|
|
|
|
CP0399122
|
(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-(cyclohexyloxy)biphenyl-4-carboxylic acid
Show/Hide
|
C29H32ClNO4
|
1
|
| 1 |
EC50 = 0.46 nM
|
|
|
|
CP0882007
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-isobutyl-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C28H35ClN2O4S
|
1
|
| 1 |
EC50 = 0.46 nM
|
|
|
|
CP0133061
|
3-Amino-N-(3-{(R)-1-hydroxy-2-[(R)-2-(7-methanesulfonyl-1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C26H30N4O5S2
|
1
|
| 1 |
EC50 = 0.47 nM
|
|
|
|
CP0869783
|
(R)-N-(4-(((2S,5R)-5-((R)-Hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-2-methyl-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
Show/Hide
|
C26H29N3O2S
|
1
|
| 1 |
EC50 = 0.48 nM
|
|
|
|
CP0484987
|
4-((2R)-2-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}propyl)-1,1-biphenyl-4-carboxylic acid
Show/Hide
|
C23H24N2O3
|
1
|
| 1 |
EC50 = 0.49 nM
|
|
|
|
CP0224385
|
ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate
Show/Hide
|
C27H32N2O4
|
1
|
| 1 |
EC50 = 0.49 nM
|
|
|
|
CP0851072
|
3-(Cyclohexylsulfanyl)-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C30H37ClN2O4S2
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0849414
|
1-(4-{(S)-3-Hydroxy-2-[2-hydroxy-3-((S)-phenoxy)-propylamino]-propyl}-phenyl)-3-phenyl-urea
Show/Hide
|
C25H29N3O4
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0399009
|
4'-(2-{[(2R)-2-(4-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-(cyclohexyloxy)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C30H37N3O5S
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0458514
|
4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethoxy)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H28ClNO5
|
1
|
| 1 |
EC50 = 0.5 nM
|
|
|
|
CP0406244
|
4-(2-hydroxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C25H28N4O4S2
|
2
|
| 1 |
EC50 = 0.5 nM
|
|
|
| 2 |
Ki = 62 nM
|
|
|
|
CP0118799
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] propane-2-sulfonate
Show/Hide
|
C26H31N3O6S3
|
1
|
| 1 |
EC50 = 0.51 nM
|
|
|
|
CP0915150
|
3-(Cyclohexylmethyl)-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C31H39ClN2O4S
|
1
|
| 1 |
EC50 = 0.54 nM
|
|
|
|
CP0477828
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-2-(2-methylpropyl)benzoic acid
Show/Hide
|
C27H30ClNO3
|
1
|
| 1 |
EC50 = 0.54 nM
|
|
|
|
CP0469284
|
[3-[(2R)-2-[[(2R)-2-[3-(benzenesulfonamido)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C26H29N3O6S2
|
1
|
| 1 |
EC50 = 0.54 nM
|
|
|
|
CP0071878
|
N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-methoxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
|
C24H27N3O4S2
|
1
|
| 1 |
EC50 = 0.55 nM
|
|
|
|
CP0433878
|
4-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethoxy)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO5
|
1
|
| 1 |
EC50 = 0.55 nM
|
|
|
|
CP0372880
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-(isopropylthio)biphenyl-4-carboxylic acid
Show/Hide
|
C26H29NO3S
|
1
|
| 1 |
EC50 = 0.56 nM
|
|
|
|
CP0279836
|
Butane-1-sulfonic acid 3-(2-{(R)-(R)-2-hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yl ester
Show/Hide
|
C27H33N3O6S3
|
1
|
| 1 |
EC50 = 0.59 nM
|
|
|
|
CP0405175
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-2-(2-methylpropoxy)benzoic acid
Show/Hide
|
C27H30ClNO4
|
1
|
| 1 |
EC50 = 0.59 nM
|
|
|
|
CP0375139
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isobutylbiphenyl-4-carboxylic acid
Show/Hide
|
C27H31NO3
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0845050
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-(isopropylamino)-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C27H35Cl2N3O4S
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0849245
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)-3-phenoxybiphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C30H31ClN2O5S
|
1
|
| 1 |
EC50 = 0.6 nM
|
|
|
|
CP0882008
|
3-(Cyclopentyloxy)-4'-(2-{[(2R)-2-hydroxy-2-phenylethyl]amino}-ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C29H35ClN2O5S
|
1
|
| 1 |
EC50 = 0.62 nM
|
|
|
|
CP0373026
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-3-methoxybenzoic acid
Show/Hide
|
C24H24ClNO4
|
1
|
| 1 |
EC50 = 0.62 nM
|
|
|
|
CP0377226
|
3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C26H28N4O3S
|
2
|
| 1 |
EC50 = 0.62 nM
|
|
|
| 2 |
Ki = 8.5 nM
|
|
|
|
CP0105653
|
(3S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5-oxo-2,3-dihydro-1H-indolizine-3-carboxamide
Show/Hide
|
C27H29N3O3
|
1
|
| 1 |
EC50 = 0.62 nM
|
|
|
|
CP0118781
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] thiophene-2-sulfonate
Show/Hide
|
C27H27N3O6S4
|
1
|
| 1 |
EC50 = 0.64 nM
|
|
|
|
CP0908527
|
(R)-N-(4-(((2S,5R)-5-((R)-Hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C25H27N3O2S
|
1
|
| 1 |
EC50 = 0.64 nM
|
|
|
|
CP0535263
|
N-[4-[2-[[(2S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl]amino]ethyl]phenyl]-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O5S
|
1
|
| 1 |
EC50 = 0.65 nM
|
|
|
|
CP0058502
|
(R)-1-(3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
EC50 = 0.67 nM
|
|
|
|
CP0881853
|
(S)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-propanamide
Show/Hide
|
C24H28N4O2S
|
1
|
| 1 |
EC50 = 0.67 nM
|
|
|
|
CP0443397
|
4'-(2-{[(2R)-2-(6-Aminopyridin-3-yl)-2-hydroxyethyl]amino}ethyl)-3-ethoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C25H30N4O5S
|
1
|
| 1 |
EC50 = 0.68 nM
|
|
|
|
CP0433879
|
4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}ethoxy)-3-isobutyl-4-biphenylcarboxylic acid
Show/Hide
|
C27H30ClNO4
|
1
|
| 1 |
EC50 = 0.68 nM
|
|
|
|
CP0372776
|
4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-2-isopropoxybenzoic Acid
Show/Hide
|
C28H30ClNO4
|
1
|
| 1 |
EC50 = 0.7 nM
|
|
|
|
CP0458352
|
4-(3-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}propyl)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H30ClNO4
|
1
|
| 1 |
EC50 = 0.7 nM
|
|
|
|
CP0393665
|
N-octyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C23H31N3O3S
|
1
|
| 1 |
EC50 = 0.73 nM
|
|
|
|
CP0071879
|
N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-phenylmethoxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
|
C30H31N3O4S2
|
1
|
| 1 |
EC50 = 0.76 nM
|
|
|
|
CP0381356
|
3-{[(7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydronaphthalen-2-yl]oxy}-5-(propylamino)benzoicAcid
Show/Hide
|
C28H31ClN2O4
|
1
|
| 1 |
EC50 = 0.77 nM
|
|
|
|
CP0394124
|
3-{[(7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydronaphthalen-2-yl]oxy}-5-(cyclohexylamino)benzoicAcid
Show/Hide
|
C31H35ClN2O4
|
1
|
| 1 |
EC50 = 0.78 nM
|
|
|
|
CP0456747
|
4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-2-methoxybenzoic Acid
Show/Hide
|
C26H26ClNO4
|
1
|
| 1 |
EC50 = 0.78 nM
|
|
|
|
CP0372777
|
4-((7S)-7-{[(2R)-2-Hydroxy-2-(4-methylphenyl)ethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)benzoic Acid
Show/Hide
|
C26H27NO3
|
1
|
| 1 |
EC50 = 0.79 nM
|
|
|
|
CP0400938
|
4-((2R)-2-{[(2R)-2-Phenyl-2-hydroxyethyl]amino}propyl)-3-methoxy-1,1-biphenyl-4-carboxylic acid
Show/Hide
|
C25H27NO4
|
1
|
| 1 |
EC50 = 0.79 nM
|
|
|
|
CP0441102
|
N-(benzenesulfonyl)-2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetamide
Show/Hide
|
C25H28ClN3O4S
|
1
|
| 1 |
EC50 = 0.7943 nM
|
|
|
|
CP0457573
|
2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C21H22ClN3O3S
|
1
|
| 1 |
EC50 = 0.7943 nM
|
|
|
|
CP0460849
|
4-[(4-octyl-1,3-thiazol-2-yl)amino]-N-phenylbenzene-1-sulfonamide
Show/Hide
|
C23H29N3O2S2
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0500795
|
1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-(3-methoxyphenyl)urea
Show/Hide
|
C26H31N3O5
|
1
|
| 1 |
EC50 = 0.8 nM
|
|
|
|
CP0372881
|
4-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-2-(2-methylpropoxy)benzoic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 0.81 nM
|
|
|
|
CP0437888
|
4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-2-fluorobenzoic Acid
Show/Hide
|
C25H23ClFNO3
|
1
|
| 1 |
EC50 = 0.81 nM
|
|
|
|
CP0484975
|
4-(2-{[(1S,2R)-2-Hydroxy-1-methyl-2-phenylethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO4
|
1
|
| 1 |
EC50 = 0.81 nM
|
|
|
|
CP0404917
|
3-(cyclohexyloxy)-4'-((S)-3-hydroxy-2-((R)-2-hydroxy-2-phenylethylamino)propyl)-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C31H38N2O6S
|
1
|
| 1 |
EC50 = 0.82 nM
|
|
|
|
CP0869756
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)butanamide
Show/Hide
|
C25H30N4O2S
|
1
|
| 1 |
EC50 = 0.83 nM
|
|
|
|
CP0381359
|
4-((S)-7-((R)-2-(6-chloropyridin-3-yl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
|
C24H23ClN2O3
|
1
|
| 1 |
EC50 = 0.85 nM
|
|
|
|
CP0103437
|
Benzenesulfonic acid 3-(2-{(R)-(R)-2-hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yl ester
Show/Hide
|
C29H29N3O6S3
|
1
|
| 1 |
EC50 = 0.87 nM
|
|
|
|
CP0071873
|
N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
|
C23H25N3O3S2
|
1
|
| 1 |
EC50 = 0.88 nM
|
|
|
|
CP0869758
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)pentanamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
EC50 = 0.88 nM
|
|
|
|
CP0378009
|
1-(4-hexyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C23H27N3O2S2
|
1
|
| 1 |
EC50 = 0.9 nM
|
|
|
|
CP0051719
|
2-(2-aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)acetamide
Show/Hide
|
C23H26N4O2S
|
2
|
| 1 |
EC50 = 0.9 nM
|
|
|
| 2 |
EC50 = 0.98 nM
|
|
|
|
CP0400940
|
4-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}-2-methylpropyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C28H33NO4
|
1
|
| 1 |
EC50 = 0.91 nM
|
|
|
|
CP0503319
|
(3-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-yloxy)-acetic acid methyl ester
Show/Hide
|
C22H25ClN2O4
|
1
|
| 1 |
EC50 = 0.92 nM
|
|
|
|
CP0395300
|
1-(4-octyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H31N3O2S2
|
1
|
| 1 |
EC50 = 0.93 nM
|
|
|
|
CP0445493
|
N-[3-[(1R)-1-hydroxy-2-[2-(7-methylsulfonyl-1H-indol-3-yl)ethylamino]ethyl]phenyl]-3-methoxybenzenesulfonamide
Show/Hide
|
C26H29N3O6S2
|
1
|
| 1 |
EC50 = 0.94 nM
|
|
|
|
CP0529838
|
(R)-1-(3-Chloro-phenyl)-2-[2-(7-ethoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C21H25ClN2O2
|
1
|
| 1 |
EC50 = 0.96 nM
|
|
|
|
CP0068209
|
4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;hydrochloride
Show/Hide
|
C11H17NO3
|
11
|
| 1 |
EC50 = 0.97 nM
|
|
|
| 2 |
EC50 = 2 nM
|
|
|
| 3 |
EC50 = 3.162 nM
|
|
|
| 4 |
EC50 = 3.9 nM
|
|
|
| 5 |
EC50 = 5.8 nM
|
|
|
| 6 |
EC50 = 12 nM
|
|
|
| 7 |
EC50 = 39.81 nM
|
|
|
| 8 |
EC50 = 86 nM
|
|
|
| 9 |
EC50 = 100 nM
|
|
|
| 10 |
EC50 = 1000 nM
|
|
|
| 11 |
Ki = 18620.87 nM
|
|
|
|
CP0432925
|
1-(6-octylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C27H33N3O2S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0460123
|
4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-3-methanesulfonylamino-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,5-difluoro-benzylamide
Show/Hide
|
C31H39F2N5O6S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0047480
|
(S)-4-(3-hexylureido)-N-(4-(2-(1-hydroxy-2-(4-hydroxyphenoxy)ethylamino)ethyl)phenyl)benzenesulfonamide
Show/Hide
|
C30H40N4O6S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0431156
|
N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[1-[4-[(Z)-(4-oxo-2-piperidin-1-yl-1,3-thiazol-5-ylidene)methyl]phenyl]piperidin-4-yl]amino]propoxy]phenyl]methanesulfonamide
Show/Hide
|
C30H39N5O6S2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0399929
|
1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2S)-2-hydroxy-3-[4-hydroxy-3-(methanesulfonamido)phenoxy]propyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
|
C30H37F2N5O8S2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0420107
|
3-Chloro-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C25H26ClN3O5S2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0851069
|
4'-(2-{[(2R)-2-Hydroxy-2-pyridin-3-ylethyl]amino}ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
|
C26H33Cl2N3O5S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0378083
|
N-[3-[(1R)-2-[[(2R)-1-(7-ethoxy-1H-indol-3-yl)propan-2-yl]amino]-1-hydroxyethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
|
C25H29N3O4S2
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0404637
|
1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-(3-nitrophenyl)urea
Show/Hide
|
C25H28N4O6
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0405841
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-[[(E)-3-phenylprop-2-enyl]amino]phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C29H33N3O4S
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0393170
|
3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-(tetrahydro-2H-pyran-4-ylamino)benzoic Acid
Show/Hide
|
C30H33ClN2O5
|
1
|
| 1 |
EC50 = 1 nM
|
|
|
|
CP0388516
|
4-(2-hydroxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C24H26N4O3S2
|
2
|
| 1 |
EC50 = 1 nM
|
|
|
| 2 |
Ki = 76 nM
|
|
|
|
CP0037154
|
(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C26H28ClNO4
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0467150
|
4-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxysulfonyl]-benzoic acid
Show/Hide
|
C30H29N3O8S3
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0497042
|
1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-(2-methoxyphenyl)urea
Show/Hide
|
C26H31N3O5
|
1
|
| 1 |
EC50 = 1.1 nM
|
|
|
|
CP0071877
|
(+/-)-2-(4-((R)-2-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)propyl)phenoxy)acetic acid
Show/Hide
|
C19H22ClNO4
|
5
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
EC50 = 5.9 nM
|
|
|
| 3 |
EC50 = 21 nM
|
|
|
| 4 |
Ki = 660 nM
|
|
|
| 5 |
Ki = 960 nM
|
|
|
|
CP0105650
|
KRP-114V
Show/Hide
|
C26H28N4O3
|
2
|
| 1 |
EC50 = 1.1 nM
|
|
|
| 2 |
EC50 = 1.6 nM
|
|
|
|
CP0135425
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-methyl-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C25H28N4O2S
|
1
|
| 1 |
EC50 = 1.15 nM
|
|
|
|
CP0448240
|
1-(6-hexylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0492498
|
4-[4-(4-Hexyl-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C36H40N4O3S2
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0497035
|
4-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxysulfonyl]-benzoic acid ethyl ester
Show/Hide
|
C32H33N3O8S3
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0510295
|
4-[[4-(4-hexylphenyl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C38H43N3O3S2
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0039162
|
[3-[(2R)-2-[[(2R)-2-[3-[[(E)-but-2-enyl]amino]phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C24H31N3O4S
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0505776
|
(R)-4'-(2-(2-(3-aminophenyl)-2-hydroxyethylamino)ethyl)-3-(cyclohexyloxy)-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
|
C30H37N3O5S
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0495997
|
4-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethoxy)-3-propoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H29NO5
|
1
|
| 1 |
EC50 = 1.2 nM
|
|
|
|
CP0377224
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzene-1,2-diol
Show/Hide
|
C26H28N4O4S
|
2
|
| 1 |
EC50 = 1.2 nM
|
|
|
| 2 |
Ki = 932 nM
|
|
|
|
CP0378418
|
2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(4-methylphenyl)sulfonylacetamide
Show/Hide
|
C26H30ClN3O4S
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0405573
|
2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(1,3-thiazol-2-yl)acetamide
Show/Hide
|
C22H25ClN4O2S
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0440991
|
2-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]thiophene-3-carboxylic acid
Show/Hide
|
C21H21ClN2O3S
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0457575
|
5-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
|
C21H22ClN3O4
|
1
|
| 1 |
EC50 = 1.259 nM
|
|
|
|
CP0374130
|
1-(3-octylphenyl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C28H34N2O2S
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0486040
|
2-[3-(2-{(R)-(R)-2-Hydroxy-2-[3-(thiophene-2-sulfonylamino)-phenyl]-ethylamino}-propyl)-1H-indol-7-yloxy]-N,N-dimethyl-acetamide
Show/Hide
|
C27H32N4O5S2
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0374421
|
3-(Acetylamino)-5-[((7S)-7-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoicAcid
Show/Hide
|
C27H27ClN2O5
|
1
|
| 1 |
EC50 = 1.3 nM
|
|
|
|
CP0135426
|
(4R)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-cyclopenta[d][1,3]thiazole-4-carboxamide
Show/Hide
|
C24H26N4O2S
|
2
|
| 1 |
EC50 = 1.36 nM
|
|
|
| 2 |
EC50 = 1.4 nM
|
|
|
|
CP0851073
|
4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)-3-(propylsulfanyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
|
C27H33ClN2O4S2
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0472167
|
4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-3-fluorobenzoic Acid
Show/Hide
|
C25H23ClFNO3
|
1
|
| 1 |
EC50 = 1.4 nM
|
|
|
|
CP0393173
|
6-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]nicotinic Acid
Show/Hide
|
C24H23ClN2O4
|
1
|
| 1 |
EC50 = 1.47 nM
|
|
|
|
CP0442243
|
3-[[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]carbamoylamino]benzoic acid
Show/Hide
|
C26H29N3O6
|
1
|
| 1 |
EC50 = 1.5 nM
|
|
|
|
CP0399297
|
(R)-4'-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C25H28N2O4
|
1
|
| 1 |
EC50 = 1.5 nM
|
|
|
|
CP0371725
|
N-[2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethylsulfonyl]benzenesulfonamide
Show/Hide
|
C25H30ClN3O5S2
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0464671
|
4-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-2-carboxylic acid
Show/Hide
|
C21H22ClN3O3S
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0386624
|
3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]-4-methylbenzoic acid
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
EC50 = 1.585 nM
|
|
|
|
CP0409911
|
1-(5-hexylpyridin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C25H29N3O2S
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0440280
|
1-[4-[2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethyl]phenyl]-3-phenylurea
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0374122
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C26H28N4O3S
|
2
|
| 1 |
EC50 = 1.6 nM
|
|
|
| 2 |
Ki = 148 nM
|
|
|
|
CP0901747
|
(R)-2-(2-Aminothiazol-4-yl)-N-(4-(((2S,5R)-5-((R)-hydroxy-(phenyl)methyl)pyrrolidin-2-yl)methyl)phenyl)-3-methylbutanamide
Show/Hide
|
C26H32N4O2S
|
1
|
| 1 |
EC50 = 1.6 nM
|
|
|
|
CP0403534
|
1-[6-(3-cyclopentylpropyl)pyridin-2-yl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C27H31N3O2S
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0460908
|
3-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-ol
Show/Hide
|
C19H21ClN2O2
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0505780
|
1-(3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C20H23ClN2O2
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0307131
|
[3-[2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]ethyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C23H25N3O6S3
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0075978
|
2-[[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl]oxy]acetic acid
Show/Hide
|
C25H27N3O6S2
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0406249
|
4-(2-hydroxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
|
C21H26N4O4S
|
2
|
| 1 |
EC50 = 1.7 nM
|
|
|
| 2 |
Ki = 670 nM
|
|
|
|
CP0406252
|
4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-3-(hydroxymethyl)phenol
Show/Hide
|
C27H30N4O4S
|
2
|
| 1 |
EC50 = 1.7 nM
|
|
|
| 2 |
Ki = 72 nM
|
|
|
|
CP0407116
|
[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-[(1R,5S)-6-(1,3,4-oxadiazol-2-yl)-3-azabicyclo[3.1.0]hexan-3-yl]methanone
Show/Hide
|
C26H28N4O3
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0074648
|
N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(4-oxoquinazolin-3-yl)acetamide
Show/Hide
|
C28H28N4O3
|
1
|
| 1 |
EC50 = 1.7 nM
|
|
|
|
CP0409506
|
1-(3-hexylphenyl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C26H30N2O2S
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0500725
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-3-methylbenzoic acid
Show/Hide
|
C24H24ClNO3
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0374332
|
3-[((7S)-7-{[(2R)-2-(6-Chloro-3-pyridinyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-(dimethylamino)benzoicAcid
Show/Hide
|
C26H28ClN3O4
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0472168
|
4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-2-methylbenzoic Acid
Show/Hide
|
C26H26ClNO3
|
1
|
| 1 |
EC50 = 1.8 nM
|
|
|
|
CP0903641
|
(R)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6,7,8-tetrahydro-4Hcyclohepta[d]thiazole-4-carboxamide
Show/Hide
|
C27H32N4O2S
|
1
|
| 1 |
EC50 = 1.86 nM
|
|
|
|
CP0522726
|
3-(3-((R)-2-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)propyl)phenoxy)benzoic acid
Show/Hide
|
C24H24ClNO4
|
1
|
| 1 |
EC50 = 1.9 nM
|
|
|
|
CP0417917
|
2-(2-aminothiazol-4-yl)-N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
|
C21H25N5O2S
|
1
|
| 1 |
EC50 = 1.9 nM
|
|
|
|
CP0452014
|
8-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3,3-dimethyl-2-oxa-8-azaspiro[4.5]decan-1-one
Show/Hide
|
C29H36N2O4
|
1
|
| 1 |
EC50 = 1.9 nM
|
|
|
|
CP0869757
|
(R)-2-Ethyl-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
Show/Hide
|
C27H31N3O2S
|
1
|
| 1 |
EC50 = 1.95 nM
|
|
|
|
CP0382239
|
4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-2-carboxylic acid
Show/Hide
|
C21H22ClN3O3S
|
1
|
| 1 |
EC50 = 1.995 nM
|
|
|
|
CP0375151
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-pyridin-2-ylphenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C35H32N6O4S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0492342
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(3,4,5-trifluorophenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C30H26F3N5O4S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0421404
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-naphthalen-2-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C34H30N4O3S2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0880613
|
N'-[5-(4-{4-[(S)-2-Hydroxy-3-(8-hydroxy-2-oxo-1,2,3,4-tetrahydro-quinolin-5-yloxy)-propylamino]-piperidin-1-yl}-benzylidene)-4-oxo-4,5-dihydro-thiazol-2-yl]-N,N-dimethyl-guanidine
Show/Hide
|
C30H37N7O5S
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0491848
|
N-[3-[(1R)-1-hydroxy-2-[2-(7-methylsulfonyl-1H-indol-3-yl)ethylamino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C25H27N3O5S2
|
1
|
| 1 |
EC50 = 2 nM
|
|
|
|
CP0137177
|
(R)-4'-(2-(2-hydroxy-2-phenylethylamino)ethyl)-3-isopropoxybiphenyl-4-carboxylic acid
Show/Hide
|
C26H29NO4
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1
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| 1 |
EC50 = 2 nM
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CP0378084
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N-[3-[(1R)-1-hydroxy-2-[[(2R)-1-(7-propan-2-yloxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C26H31N3O4S2
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1
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| 1 |
EC50 = 2 nM
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CP0392099
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-naphthalen-2-yl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
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C36H33N3O3S2
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1
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| 1 |
EC50 = 2 nM
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CP0405176
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3-chloro-4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]benzoic acid
Show/Hide
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C23H21Cl2NO3
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1
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| 1 |
EC50 = 2 nM
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CP0381358
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4-((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-3-methylbenzoic Acid
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C26H26ClNO3
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1
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| 1 |
EC50 = 2 nM
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CP0406256
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4-(2-hydroxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C21H26N4O4S
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2
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| 1 |
EC50 = 2 nM
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| 2 |
Ki = 600 nM
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CP0156740
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-(4-(4-(trifluoromethyl)phenyl)thiazol-2-yl)benzenesulfonamide
Show/Hide
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C31H27F3N4O3S2
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5
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| 1 |
EC50 = 2 nM
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| 2 |
EC50 = 3 nM
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| 3 |
EC50 = 3.6 nM
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| 4 |
EC50 = 7.9 nM
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| 5 |
IC50 = 46 nM
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CP0442303
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1-cyclohexyl-3-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]urea
Show/Hide
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C25H35N3O4
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1
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| 1 |
EC50 = 2.1 nM
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CP0418061
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4-(2-{[(2R)-2-(3-Fluorophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-1,1-biphenyl-4-carboxylic acid
Show/Hide
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C26H28FNO4
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1
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| 1 |
EC50 = 2.1 nM
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CP0156745
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(2S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)propanamide
Show/Hide
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C25H28N4O3
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2
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| 1 |
EC50 = 2.1 nM
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| 2 |
EC50 = 2.7 nM
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CP0373027
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4-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-2-propan-2-ylsulfonylbenzoic acid
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C26H29NO5S
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1
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| 1 |
EC50 = 2.2 nM
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CP0406254
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3-ethyl-4-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C28H32N4O3S
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2
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| 1 |
EC50 = 2.2 nM
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| 2 |
Ki = 30 nM
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CP0140965
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N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(2-oxopyrimidin-1-yl)acetamide
Show/Hide
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C24H26N4O3
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1
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| 1 |
EC50 = 2.2 nM
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CP0429158
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1-(4-octylpyrimidin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C26H32N4O2S
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1
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| 1 |
EC50 = 2.4 nM
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CP0402246
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4-[4-(4-tert-Butyl-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C34H36N4O3S2
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1
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| 1 |
EC50 = 2.4 nM
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CP0442308
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3-Fluoro-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
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C25H26FN3O5S2
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1
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| 1 |
EC50 = 2.4 nM
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CP0493222
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4-[[4-(4-tert-butylphenyl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
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C36H39N3O3S2
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1
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| 1 |
EC50 = 2.4 nM
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CP0417774
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5-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)-2-thiophenecarboxylic Acid
Show/Hide
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C23H22ClNO3S
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1
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| 1 |
EC50 = 2.4 nM
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CP0440523
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4-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethoxy)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
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C26H29NO5
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1
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| 1 |
EC50 = 2.4 nM
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CP0491158
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4-(2-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
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C26H28ClNO4
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1
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| 1 |
EC50 = 2.4 nM
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CP0379214
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1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-(4-methoxyphenyl)urea
Show/Hide
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C26H31N3O5
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1
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| 1 |
EC50 = 2.5 nM
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CP0374173
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1-(2-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C27H30N4O3S
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2
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| 1 |
EC50 = 2.5 nM
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| 2 |
Ki = 11 nM
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CP0851888
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(R)-1-cyclohexyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
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C34H53N3O7
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1
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| 1 |
EC50 = 2.512 nM
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CP0389978
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4-(2-{[(2R)-2-(4-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
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C26H30N2O4
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1
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| 1 |
EC50 = 2.6 nM
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CP0140960
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(2S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)propanamide
Show/Hide
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C24H27N5O3
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1
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| 1 |
EC50 = 2.6 nM
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CP0480430
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-quinolin-6-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
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C33H29N5O3S2
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1
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| 1 |
EC50 = 2.7 nM
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CP0448044
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-quinolin-6-yl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
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C35H32N4O3S2
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1
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| 1 |
EC50 = 2.7 nM
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CP0458653
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(S)-6-(4-(2-(3-(3,3-diethyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C31H38N4O5
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1
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| 1 |
EC50 = 2.7 nM
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CP0386223
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(2S)-2-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]propanoic acid
Show/Hide
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C19H23NO4
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1
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| 1 |
EC50 = 2.7 nM
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CP0507313
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(R)-1-(3-Chloro-phenyl)-2-[2-(7-isopropoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C22H27ClN2O2
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1
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| 1 |
EC50 = 2.8 nM
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CP0445499
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5-Bromo-thiophene-2-sulfonic acid (3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-amide
Show/Hide
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C23H24BrN3O5S3
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1
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| 1 |
EC50 = 2.8 nM
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CP0882009
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4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-N-(methylsulfonyl)-3-(pentyloxy)biphenyl-4-carboxamide Hydrochloride
Show/Hide
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C29H37ClN2O5S
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1
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| 1 |
EC50 = 2.8 nM
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CP0387764
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4-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)benzoic Acid
Show/Hide
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C25H24ClNO3
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1
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| 1 |
EC50 = 2.8 nM
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CP0388617
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1-phenoxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C20H24N4O2S
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2
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| 1 |
EC50 = 2.8 nM
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| 2 |
Ki = 41 nM
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CP0198056
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(naphthalen-2-ylmethylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C31H33N3O4S
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1
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| 1 |
EC50 = 2.9 nM
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CP0469323
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4-(2-hydroxy-3-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C22H28N4O4S
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2
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| 1 |
EC50 = 2.9 nM
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| 2 |
Ki = 989 nM
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CP0409587
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4-{5-[(4-Fluoro-phenyl)-(3-methyl-ureido)-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C32H32FN7O5S
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1
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| 1 |
EC50 = 3 nM
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CP0440122
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-methylsulfanylphenyl)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
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C31H31N5O4S2
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1
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| 1 |
EC50 = 3 nM
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CP0849868
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N-[(R)-5-(2-{1-[4-(2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethoxy)-2-hydroxy-phenyl]-methanesulfonamide
Show/Hide
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C24H30N4O7S2
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1
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| 1 |
EC50 = 3 nM
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CP0918555
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N-{5-[(R)-2-(1-{4-[2-(N',N'-Dimethyl-guanidino)-4-oxo-4H-thiazol-5-ylidenemethyl]-phenyl}-piperidin-4-ylamino)-1-hydroxy-ethyl]-2-hydroxy-phenyl}-methanesulfonamide
Show/Hide
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C27H35N7O5S2
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1
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| 1 |
EC50 = 3 nM
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CP0496883
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2-Amino-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
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C25H28N4O5S2
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1
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| 1 |
EC50 = 3 nM
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CP0447745
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethyl)phenyl]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C31H29F3N6O3S
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1
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| 1 |
EC50 = 3.1 nM
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CP0388613
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4-(2-hydroxy-3-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C28H32N4O4S
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2
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| 1 |
EC50 = 3.1 nM
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| 2 |
Ki = 300 nM
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CP0412012
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4-(3-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-2-hydroxypropoxy)phenol
Show/Hide
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C26H27FN4O3S
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2
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| 1 |
EC50 = 3.1 nM
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| 2 |
Ki = 75 nM
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CP0452015
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[(1R,5S)-6-(5-ethyl-1,3,4-oxadiazol-2-yl)-3-azabicyclo[3.1.0]hexan-3-yl]-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]methanone
Show/Hide
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C28H32N4O3
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1
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| 1 |
EC50 = 3.1 nM
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CP0402511
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1-[4-(3-cyclopentylpropyl)-1,3-thiazol-2-yl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
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C25H29N3O2S2
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1
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| 1 |
EC50 = 3.2 nM
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CP0467168
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(prop-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C23H29N3O4S
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1
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| 1 |
EC50 = 3.2 nM
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CP0387892
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3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-(dimethylamino)benzoicAcid
Show/Hide
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C27H29ClN2O4
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1
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| 1 |
EC50 = 3.2 nM
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CP0387893
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3-Amino-5-[((7S)-7-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
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C25H25ClN2O4
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1
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| 1 |
EC50 = 3.2 nM
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CP0509904
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4-{4-[(4-Fluoro-phenyl)-hydroxy-methyl]-[1,2,3]triazol-2-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H29FN6O4S
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1
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| 1 |
EC50 = 3.3 nM
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CP0225356
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8-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-2-oxa-8-azaspiro[4.5]decan-1-one
Show/Hide
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C27H32N2O4
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1
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| 1 |
EC50 = 3.3 nM
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CP0467666
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(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-isopropoxybenzoic acid
Show/Hide
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C26H28ClNO5
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1
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| 1 |
EC50 = 3.4 nM
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CP0382376
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2-[4-[2-[[(2S)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C20H25NO4
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1
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| 1 |
EC50 = 3.4 nM
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CP0387894
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4-((S)-7-((R)-2-hydroxy-2-(4-(trifluoromethyl)phenyl)ethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
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C26H24F3NO3
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1
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| 1 |
EC50 = 3.5 nM
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CP0372774
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5-[((7S)-7-{[(2R)-2-(6-Chloro-3-pyridinyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
Show/Hide
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C25H25ClN2O5
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1
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| 1 |
EC50 = 3.6 nM
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CP0459230
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1-(5-octyl-1,3-oxazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
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C25H31N3O3S
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1
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| 1 |
EC50 = 3.7 nM
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CP0105651
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(6S)-N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide
Show/Hide
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C24H27N5O2
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1
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| 1 |
EC50 = 3.7 nM
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CP0407115
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N-[4-[[(2S,5R)-5-[(R)-hydroxy(pyridin-3-yl)methyl]pyrrolidin-2-yl]methyl]phenyl]-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazole-6-carboxamide
Show/Hide
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C24H27N5O2
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1
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| 1 |
EC50 = 3.7 nM
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CP0845194
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(+/-)-2-{4-[2-(2-hydroxy-2-phenylethylamino)ethyl]-phenoxy}propanoic acid
Show/Hide
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C19H23NO4
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1
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| 1 |
EC50 = 3.8 nM
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CP0373306
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2-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]-2-methylpropanoic acid
Show/Hide
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C20H25NO4
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1
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| 1 |
EC50 = 3.9 nM
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CP0105654
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N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyrimidin-1-yl)acetamide
Show/Hide
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C24H26N4O3
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1
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| 1 |
EC50 = 3.9 nM
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CP0216696
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]benzenesulfonamide
Show/Hide
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C24H26N4O4S
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1
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| 1 |
EC50 = 3.9 nM
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CP0449742
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5-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 3.981 nM
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CP0403282
|
Solabegron
Show/Hide
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C23H23ClN2O3
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1
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| 1 |
EC50 = 3.981 nM
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CP0399813
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4-[5-(3,4-Difluoro-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H27F2N5O5S
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1
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| 1 |
EC50 = 4 nM
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CP0431268
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4-[5-(4-Fluoro-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H28FN5O5S
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1
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| 1 |
EC50 = 4 nM
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CP0136837
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-phenyl-propionic acid
Show/Hide
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C30H36N4O7S
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1
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| 1 |
EC50 = 4 nM
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CP0448512
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2-[butyl-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]phenyl]sulfamoyl]acetic acid
Show/Hide
|
C26H38N4O8S2
|
1
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| 1 |
EC50 = 4 nM
|
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CP0405174
|
4-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-2-(oxan-4-yloxy)benzoic acid
Show/Hide
|
C28H31NO5
|
1
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| 1 |
EC50 = 4 nM
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CP0854281
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(3S,5R)-3,5-Dimethyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
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C24H38Cl2N4O3S
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1
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| 1 |
EC50 = 4 nM
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CP0424633
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethoxy)phenyl]methyl]triazol-2-yl]benzenesulfonamide
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C31H29F3N6O4S
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1
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| 1 |
EC50 = 4.1 nM
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CP0372773
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3-[((7S)-7-{[(2R)-2-(6-Chloro-3-pyridinyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
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C24H23ClN2O4
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1
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| 1 |
EC50 = 4.1 nM
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CP0393191
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethoxy)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
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C31H27F3N4O4S2
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2
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| 1 |
EC50 = 4.3 nM
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| 2 |
IC50 = 30 nM
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CP0435558
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N-[3-[(1R)-2-[[(2R)-1-[7-(2-aminoethoxy)-1H-indol-3-yl]propan-2-yl]amino]-1-hydroxyethyl]phenyl]thiophene-2-sulfonamide
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C25H30N4O4S2
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1
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| 1 |
EC50 = 4.3 nM
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CP0427871
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2-(2-ethoxyethoxy)-4-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzoic acid
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C27H31NO5
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1
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| 1 |
EC50 = 4.3 nM
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CP0140955
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N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(2-oxopyridin-1-yl)acetamide
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C25H27N3O3
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1
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| 1 |
EC50 = 4.3 nM
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CP0504227
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3-[((8S)-8-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-yl)oxy]benzoic Acid
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C26H26ClNO4
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1
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| 1 |
EC50 = 4.5 nM
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CP0422399
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4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]anilino]benzoic acid
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C23H23ClN2O3
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1
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| 1 |
EC50 = 4.6 nM
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CP0459677
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(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-pivalamidobenzoic acid
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C28H31ClN2O5
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1
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| 1 |
EC50 = 4.6 nM
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CP0456745
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5-[((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
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C26H26ClNO5
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1
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| 1 |
EC50 = 4.7 nM
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CP0435325
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1-phenoxy-3-(1-(5-(thiophen-2-yl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
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C24H26N4O2S2
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2
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| 1 |
EC50 = 4.7 nM
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| 2 |
Ki = 11 nM
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CP0381824
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(R)-4'-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)-3-methoxybiphenyl-4-carboxylic acid
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C24H24ClNO4
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1
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| 1 |
EC50 = 4.8 nM
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CP0381354
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3-[((7S)-7-{[(2R)-2-(4-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
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C25H24ClNO4
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1
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| 1 |
EC50 = 4.8 nM
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CP0105652
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N-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-2-(6-oxopyridazin-1-yl)acetamide
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C24H26N4O3
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2
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| 1 |
EC50 = 4.8 nM
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| 2 |
EC50 = 5.9 nM
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CP0383393
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(1H-indol-3-yl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
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C32H29N5O3S2
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1
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| 1 |
EC50 = 4.9 nM
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CP0433171
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4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-3-fluorobenzoic acid
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C23H21ClFNO3
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1
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| 1 |
EC50 = 4.9 nM
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CP0421178
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1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-propan-2-ylurea
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C22H31N3O4
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1
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| 1 |
EC50 = 4.9 nM
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CP0412418
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2-[4-[2-[(2-hydroxy-2-phenylethyl)amino]ethyl]phenoxy]-2-methylpropanoic acid
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C20H25NO4
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1
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| 1 |
EC50 = 4.9 nM
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CP0395094
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1-[3-(3-cyclopentylpropyl)phenyl]-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C28H32N2O2S
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1
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| 1 |
EC50 = 5 nM
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CP0414877
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(naphthalen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
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C34H31N5O4S
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1
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| 1 |
EC50 = 5 nM
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CP0499569
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]benzenesulfonamide
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C35H32N4O3S2
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1
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| 1 |
EC50 = 5 nM
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CP0524320
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4-(4-{2-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,5-difluoro-benzylamide
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C30H37F2N5O5S
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1
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| 1 |
EC50 = 5 nM
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CP0375236
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1-[4-(4-{[(S)-2-Hydroxy-3-(8-hydroxy-2-oxo-1,2,3,4-tetrahydro-quinolin-5-yloxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-octyl-urea
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C33H49N5O7S
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1
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| 1 |
EC50 = 5 nM
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CP0467627
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1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
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C29H35F2N5O7S2
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1
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| 1 |
EC50 = 5 nM
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CP0401269
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4-[[4-(1-benzofuran-2-yl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
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C34H31N3O4S2
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1
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| 1 |
EC50 = 5 nM
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CP0166797
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1-hexyl-3-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]sulfonylphenyl]urea
Show/Hide
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C27H41N5O7S2
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1
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| 1 |
EC50 = 5 nM
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CP0430587
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-methylsulfonylacetamide
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C20H26ClN3O4S
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1
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| 1 |
EC50 = 5.012 nM
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CP0853347
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2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({2-[(1-naphthalenylmethyl)oxy]ethyl}oxy)hexyl]amino}ethyl)phenolAcetate Salt
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C30H41NO7
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1
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| 1 |
EC50 = 5.012 nM
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CP0906725
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4-[(1R)-2-({6-[(2-{[(3,5-Dimethylphenyl)methyl]oxy}ethyl)oxy]-hexyl}-amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol Acetate Salt
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C28H43NO7
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1
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| 1 |
EC50 = 5.012 nM
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CP0383247
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1-(4-hexylpyrimidin-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C24H28N4O2S
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1
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| 1 |
EC50 = 5.1 nM
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CP0409159
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(S)-6-(4-(2-(3-(3-ethyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C28H33N5O5
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1
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| 1 |
EC50 = 5.2 nM
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CP0419619
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(S)-6-(4-(2-(2-hydroxy-3-(2-oxo-3-propyl-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C29H35N5O5
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1
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| 1 |
EC50 = 5.2 nM
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CP0458654
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(S)-6-(4-(2-(3-(3,3-dimethyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
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C29H34N4O5
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1
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| 1 |
EC50 = 5.2 nM
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CP0500727
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3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-5-methoxybenzoic Acid
Show/Hide
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C26H26ClNO5
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1
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| 1 |
EC50 = 5.3 nM
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CP0198066
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(R)-1-((R)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
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1
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| 1 |
EC50 = 5.4 nM
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CP0424777
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(S)-6-(4-(2-(3-(3-(2-cyclopropylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C31H37N5O5
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1
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| 1 |
EC50 = 5.4 nM
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CP0148856
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[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]-[(1R,5S)-6-(2-methyltetrazol-5-yl)-3-azabicyclo[3.1.0]hexan-3-yl]methanone
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C26H30N6O2
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1
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| 1 |
EC50 = 5.4 nM
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CP0448298
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4-[methyl(4-octyl-1,3-thiazol-2-yl)amino]-N-phenylbenzene-1-sulfonamide
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C24H31N3O2S2
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1
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| 1 |
EC50 = 5.5 nM
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CP0405177
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3-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]anilino]benzoic acid
Show/Hide
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C23H23ClN2O3
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1
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| 1 |
EC50 = 5.5 nM
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CP0039930
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(-)-arterenol
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C8H11NO3
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2
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| 1 |
EC50 = 5.5 nM
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| 2 |
EC50 = 6.3 nM
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CP0399007
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4'-(2-{[(2R)-2-(4-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide Dihydrochloride
Show/Hide
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C27H33N3O5S
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1
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| 1 |
EC50 = 5.5 nM
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CP0399816
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5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-thiophenecarboxylic Acid
Show/Hide
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C23H22ClNO4S
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1
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| 1 |
EC50 = 5.7 nM
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CP0455443
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4-(4-Benzo[b]thiophen-2-yl-thiazol-2-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C32H28N4O3S3
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1
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| 1 |
EC50 = 5.8 nM
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CP0441804
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4-[[4-(1-benzothiophen-2-yl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
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C34H31N3O3S3
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1
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| 1 |
EC50 = 5.8 nM
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CP0393188
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4-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)phenoxy]acetic Acid
Show/Hide
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C26H26ClNO4
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1
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| 1 |
EC50 = 5.8 nM
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CP0403739
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[(4-methoxyphenoxy)methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
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C31H31N5O6S
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1
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| 1 |
EC50 = 6 nM
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CP0409613
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4-[5-(3,4-Difluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H27F2N5O4S
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1
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| 1 |
EC50 = 6 nM
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CP0502500
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4-[5-(2-Hydroxy-phenoxymethyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H29N5O6S
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1
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| 1 |
EC50 = 6 nM
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CP0857860
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N-[5-(2-{1-[4-((R)-2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-benzenesulfonamide
Show/Hide
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C29H32N4O6S2
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1
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| 1 |
EC50 = 6 nM
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CP0462341
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8-Hydroxy-5-((S)-2-hydroxy-3-{1-[4-(4-oxo-2-piperidin-1-yl-4H-thiazol-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-propoxy)-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C32H39N5O5S
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1
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| 1 |
EC50 = 6 nM
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CP0874997
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N-[5-(2-{1-[4-(2,4-Dioxo-thiazolidin-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide
Show/Hide
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C24H28N4O6S2
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1
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| 1 |
EC50 = 6 nM
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CP0189834
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N-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]nonanamide
Show/Hide
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C30H46N4O7S2
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1
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| 1 |
EC50 = 6 nM
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CP0383083
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4-Aminomethylpiperidine substituted analogue
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C26H34N4O9S
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1
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| 1 |
EC50 = 6 nM
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CP0417354
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(R)-4'-(2-(2-(3-aminophenyl)-2-hydroxyethylamino)ethyl)-3-isopropoxy-N-(methylsulfonyl)biphenyl-4-carboxamide
Show/Hide
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C27H33N3O5S
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1
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| 1 |
EC50 = 6 nM
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CP0372799
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5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methoxybenzoic Acid
Show/Hide
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C26H26ClNO5
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1
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| 1 |
EC50 = 6 nM
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CP0399139
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4-[(2S)-2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}propyl]-4-biphenylcarboxylic acid
Show/Hide
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C24H24ClNO3
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1
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| 1 |
EC50 = 6 nM
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CP0392506
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4-[4-(4-Fluoro-benzyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C31H29FN4O3S2
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1
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| 1 |
EC50 = 6.2 nM
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CP0498169
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4-[[4-[(4-fluorophenyl)methyl]-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
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C33H32FN3O3S2
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1
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| 1 |
EC50 = 6.2 nM
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CP0279585
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4-(3-Hexyl-ureido)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C28H37N5O4S
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1
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| 1 |
EC50 = 6.3 nM
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CP0448737
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(3,4,5-trifluorophenyl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
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C30H25F3N4O3S2
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1
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| 1 |
EC50 = 6.3 nM
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CP0419581
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-(4-methylphenyl)sulfonylacetamide
Show/Hide
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C26H30ClN3O4S
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1
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| 1 |
EC50 = 6.31 nM
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CP0457574
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-thiazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O3S
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1
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| 1 |
EC50 = 6.31 nM
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CP0404004
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4-[4-(3-Fluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H29FN6O3S
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1
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| 1 |
EC50 = 6.4 nM
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CP0495476
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4-[4-(4-Fluoro-benzoyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H27FN6O4S
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1
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| 1 |
EC50 = 6.4 nM
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CP0484626
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(R)-3-acetamido-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C25H25ClN2O5
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1
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| 1 |
EC50 = 6.5 nM
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CP0442324
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[3-[(2R)-2-[[(2R)-2-[3-(but-2-ynylamino)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H29N3O4S
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1
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| 1 |
EC50 = 6.5 nM
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CP0393355
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]propane-1-sulfonamide
Show/Hide
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C21H28N4O4S
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1
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| 1 |
EC50 = 6.5 nM
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CP0434354
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6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclopropane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
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C29H32N4O5
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1
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| 1 |
EC50 = 6.6 nM
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CP0504190
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(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-(2-oxopyrrolidin-1-yl)benzoic acid
Show/Hide
|
C27H27ClN2O5
|
1
|
| 1 |
EC50 = 6.6 nM
|
|
|
|
CP0491847
|
4,5-Dichloro-thiophene-2-sulfonic acid (3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-amide
Show/Hide
|
C23H23Cl2N3O5S3
|
1
|
| 1 |
EC50 = 6.7 nM
|
|
|
|
CP0373035
|
4'-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-ethyl}-biphenyl-4-carboxylic acid
Show/Hide
|
C23H22ClNO3
|
1
|
| 1 |
EC50 = 6.7 nM
|
|
|
|
CP0428928
|
(R)-2-(2-aminothiazol-4-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C20H23N5O2S
|
1
|
| 1 |
EC50 = 6.8 nM
|
|
|
|
CP0488859
|
N-hexyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
|
C21H27N3O3S
|
1
|
| 1 |
EC50 = 6.9 nM
|
|
|
|
CP0486017
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[3-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
|
C31H27F3N4O3S2
|
1
|
| 1 |
EC50 = 6.9 nM
|
|
|
|
CP0428936
|
(R)-3-(2-(1H-pyrrol-1-yl)ethyl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
|
C28H30N4O2
|
1
|
| 1 |
EC50 = 6.9 nM
|
|
|
|
CP0393663
|
1-nonanoyl-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C23H30N2O3S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0447728
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-(naphthalen-2-yloxymethyl)-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C34H31N5O5S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0918027
|
N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}-2-methylpropyl)phenyl]N-phenylsulfamide; 2HCl
Show/Hide
|
C23H30Cl2N4O3S
|
1
|
| 1 |
EC50 = 7 nM
|
|
|
|
CP0377642
|
4-[4-(3,4-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26F2N4O3S2
|
2
|
| 1 |
EC50 = 7.1 nM
|
|
|
| 2 |
IC50 = 20 nM
|
|
|
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CP0401271
|
4-[[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C32H29F2N3O3S2
|
1
|
| 1 |
EC50 = 7.1 nM
|
|
|
|
CP0437372
|
(S)-6-(4-(2-(2-hydroxy-3-(3-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C27H31N5O5
|
1
|
| 1 |
EC50 = 7.1 nM
|
|
|
|
CP0503536
|
3-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
|
C25H24ClNO4
|
1
|
| 1 |
EC50 = 7.1 nM
|
|
|
|
CP0377153
|
1-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
|
C21H26N4O2S
|
2
|
| 1 |
EC50 = 7.1 nM
|
|
|
| 2 |
Ki = 151 nM
|
|
|
|
CP0451356
|
4-[4-(3,4-Difluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28F2N6O3S
|
1
|
| 1 |
EC50 = 7.2 nM
|
|
|
|
CP0459675
|
(R)-2-acetamido-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
|
C25H25ClN2O5
|
1
|
| 1 |
EC50 = 7.2 nM
|
|
|
|
CP0399955
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-quinolin-3-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C33H29N5O3S2
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0439416
|
N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-quinolin-3-yl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
|
C35H32N4O3S2
|
1
|
| 1 |
EC50 = 7.3 nM
|
|
|
|
CP0510149
|
4-((2S)-3-Hydroxy-2-{[(2R)-2-hydroxy-2-phenylethyl]amino}propyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C27H31NO5
|
1
|
| 1 |
EC50 = 7.4 nM
|
|
|
|
CP0471180
|
5-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]thiophene-2-carboxylic acid
Show/Hide
|
C21H20ClNO3S
|
1
|
| 1 |
EC50 = 7.5 nM
|
|
|
|
CP0501622
|
4-[4-(2,3-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26F2N4O3S2
|
1
|
| 1 |
EC50 = 7.6 nM
|
|
|
|
CP0540290
|
N-[3-[(1R)-1-hydroxy-2-[2-(7-phenylmethoxy-1H-indol-3-yl)ethylamino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
|
C29H29N3O4S2
|
1
|
| 1 |
EC50 = 7.6 nM
|
|
|
|
CP0388612
|
4-(2-hydroxy-3-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
EC50 = 7.8 nM
|
|
|
| 2 |
Ki = 499 nM
|
|
|
|
CP0457572
|
2-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]furan-3-carboxylic acid
Show/Hide
|
C21H21ClN2O4
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0874631
|
4-[(1R)-2-({6-[(2-{[(2,5-Dichlorophenyl)methyl]oxy}ethyl)oxy]-hexyl}-amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
|
C26H37Cl2NO7
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0903932
|
(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
|
C28H43N3O7
|
1
|
| 1 |
EC50 = 7.943 nM
|
|
|
|
CP0375247
|
4-{5-[(4-Fluoro-phenyl)-hydroxy-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O5S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0376678
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O5S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0403717
|
4-[3-(4-Fluoro-phenoxymethyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28FN5O5S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0406150
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethoxy)phenoxy]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
|
C31H28F3N5O6S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0440071
|
4-{5-[Amino-(4-fluoro-phenyl)-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H29FN6O4S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0383760
|
4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid octylamide
Show/Hide
|
C31H48N4O4
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0208046
|
2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-4-methyl-pentanoic acid
Show/Hide
|
C27H38N4O7S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0861088
|
(2R,6S)-2,6-Dimethyl-morpholine-4-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
Show/Hide
|
C23H36Cl2N4O4S
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0373722
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(5-phenyl-4H-1,2,4-triazol-3-yl)acetamide
Show/Hide
|
C25H26N6O2
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0535177
|
1-(4-methyl-1,3-thiazol-2-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
|
C18H17N3O2S2
|
1
|
| 1 |
EC50 = 8.1 nM
|
|
|
|
CP0399127
|
4-(2-{[(2R)-2-(3-Aminophenyl)-2-hydroxyethyl]amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
Show/Hide
|
C26H30N2O4
|
1
|
| 1 |
EC50 = 8.1 nM
|
|
|
|
CP0371757
|
6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclohexane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
|
C32H38N4O5
|
1
|
| 1 |
EC50 = 8.3 nM
|
|
|
|
CP0522562
|
1-[4-[(2S)-3-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]propyl]phenyl]-3-propylurea
Show/Hide
|
C22H31N3O4
|
1
|
| 1 |
EC50 = 8.3 nM
|
|
|
|
CP0406259
|
1-(2-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C26H27FN4O2S
|
2
|
| 1 |
EC50 = 8.3 nM
|
|
|
| 2 |
Ki = 14 nM
|
|
|
|
CP0501656
|
4-Amino-N-(3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-benzenesulfonamide
Show/Hide
|
C25H28N4O5S2
|
1
|
| 1 |
EC50 = 8.4 nM
|
|
|
|
CP0522724
|
(R)-2-benzamido-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
|
C30H27ClN2O5
|
1
|
| 1 |
EC50 = 8.6 nM
|
|
|
|
CP0505158
|
6-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenoxy]pyridine-3-carboxylic acid
Show/Hide
|
C22H21ClN2O4
|
1
|
| 1 |
EC50 = 8.7 nM
|
|
|
|
CP0856438
|
(R)-2-(4-Fluorophenyl)-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
|
C30H29FN4O2S
|
1
|
| 1 |
EC50 = 8.78 nM
|
|
|
|
CP0373717
|
(R)-2-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C24H25N5O2
|
1
|
| 1 |
EC50 = 8.8 nM
|
|
|
|
CP0213665
|
3-[N-butyl-4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]anilino]-3-oxopropanoic acid
Show/Hide
|
C27H38N4O7S
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0453894
|
N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[1-[4-[(Z)-(4-oxo-2-piperidin-1-yl-1,3-thiazol-5-ylidene)methyl]phenyl]piperidin-4-yl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C29H37N5O5S2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0849759
|
4-((S)-2-Hydroxy-3-{1-[4-(4-oxo-2-piperidin-1-yl-4H-thiazol-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-propoxy)-1,3-dihydro-benzoimidazol-2-one
Show/Hide
|
C30H36N6O4S
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0889554
|
N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(2-imino-4-oxo-thiazolidin-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-ethyl)-phenyl]-methanesulfonamide
Show/Hide
|
C24H29N5O5S2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0463273
|
1-[4-(4-{[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-1H-indole-4-carboxylic acid
Show/Hide
|
C30H34N4O8S2
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0431043
|
[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-[[(E)-pent-2-enyl]amino]phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C25H33N3O4S
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0472165
|
5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]-2-methylbenzoic Acid
Show/Hide
|
C26H26ClNO4
|
1
|
| 1 |
EC50 = 9 nM
|
|
|
|
CP0492302
|
4-(4-Benzofuran-2-yl-thiazol-2-yl)-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C32H28N4O4S2
|
1
|
| 1 |
EC50 = 9.1 nM
|
|
|
|
CP0493221
|
N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[[4-(1H-indol-3-yl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
|
C34H32N4O3S2
|
1
|
| 1 |
EC50 = 9.1 nM
|
|
|
|
CP0515394
|
(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-fluorobenzoic acid
Show/Hide
|
C23H21ClFNO4
|
1
|
| 1 |
EC50 = 9.4 nM
|
|
|
|
CP0404462
|
4-[4-(4-Fluoro-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H27FN4O3S2
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0495302
|
4-[[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
|
C32H30FN3O3S2
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0459676
|
(R)-2-chloro-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
|
C23H21Cl2NO4
|
1
|
| 1 |
EC50 = 9.5 nM
|
|
|
|
CP0393175
|
6-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)nicotinic Acid
Show/Hide
|
C24H23ClN2O3
|
1
|
| 1 |
EC50 = 9.6 nM
|
|
|
|
CP0373025
|
4-[2-chloro-4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]benzoic acid
Show/Hide
|
C23H21Cl2NO3
|
1
|
| 1 |
EC50 = 9.7 nM
|
|
|
|
CP0203142
|
(4-ethylsulfonylpiperidin-1-yl)-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]phenyl]methanone
Show/Hide
|
C26H34N2O4S
|
1
|
| 1 |
EC50 = 9.7 nM
|
|
|
|
CP0406380
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[(4-octyl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
|
C33H42N4O3S2
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0436017
|
N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[2-(4-octyl-1,3-thiazol-2-yl)ethyl]benzenesulfonamide
Show/Hide
|
C35H45N3O3S2
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0422398
|
4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-2-fluorobenzoic acid
Show/Hide
|
C23H21ClFNO3
|
1
|
| 1 |
EC50 = 9.8 nM
|
|
|
|
CP0408753
|
methyl N-[(4-fluorophenyl)-[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methyl]carbamate
Show/Hide
|
C32H31FN6O6S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0454388
|
4-[5-(4-Fluoro-benzoyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H26FN5O5S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0393166
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-octyl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
|
C32H40N4O3S2
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0471480
|
4-[4-(3,4-Difluoro-phenoxymethyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28F2N6O4S
|
1
|
| 1 |
EC50 = 10 nM
|
|
|
|
CP0889313
|
N-[5-(2-{1-[4-((R)-2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide
Show/Hide
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C24H30N4O6S2
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1
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| 1 |
EC50 = 10 nM
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CP0654243
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N'-[5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo-2,3-dihydro-1H-benzoimidazol-4-yloxy)-propylamino]-piperidin-1-yl}-benzylidene)-4-oxo-4,5-dihydro-thiazol-2-yl]-N,N-dimethyl-guanidine
Show/Hide
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C28H34N8O4S
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1
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| 1 |
EC50 = 10 nM
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CP0921865
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N-[5-((R)-2-{1-[4-(2-Cyanoamino-4-oxo-4H-thiazol-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-2-hydroxy-phenyl]-methanesulfonamide
Show/Hide
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C25H28N6O5S2
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1
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| 1 |
EC50 = 10 nM
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CP0384274
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1-Hexyl-3-[4-(4-{[(S)-2-hydroxy-3-(2-oxo-2,3-dihydro-1H-benzoimidazol-4-yloxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-urea
Show/Hide
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C29H42N6O6S
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1
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| 1 |
EC50 = 10 nM
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CP0374848
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N-[2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethylsulfonyl]benzamide
Show/Hide
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C26H30ClN3O4S
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1
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| 1 |
EC50 = 10 nM
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CP0463635
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4-Aminomethylpiperidine substituted analogue
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C28H40N4O7S
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1
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| 1 |
EC50 = 10 nM
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CP0448984
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(3-{2-[(R)-2-((S)-3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-1H-indol-7-yloxy)-acetic acid
Show/Hide
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C21H23ClN2O4
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1
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| 1 |
EC50 = 10 nM
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CP0378227
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-octyl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
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C34H43N3O3S2
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1
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| 1 |
EC50 = 10 nM
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CP0058497
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(prop-2-ynylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C23H27N3O4S
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1
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| 1 |
EC50 = 10 nM
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CP0919461
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4-Methyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
Show/Hide
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C23H36Cl2N4O3S
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1
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| 1 |
EC50 = 10 nM
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CP0428937
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-(1H-imidazol-2-yl)benzamide
Show/Hide
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C25H25N5O2
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1
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| 1 |
EC50 = 10 nM
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CP0845306
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N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-pyrazol-1-yl)propanamide hydrochloride
Show/Hide
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C21H26ClN5O2
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1
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| 1 |
EC50 = 10 nM
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CP0495940
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2-[3-[(7S)-7-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-5,6,7,8-tetrahydronaphthalen-2-yl]phenoxy]acetic acid
Show/Hide
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C26H26ClNO4
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1
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| 1 |
EC50 = 10 nM
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CP0388522
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1-(1-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
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C26H27FN4O2S
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2
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| 1 |
EC50 = 10 nM
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| 2 |
Ki = 23 nM
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CP0409669
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(S)-6-(4-(2-(3-(3-(2-cyclobutylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C32H39N5O5
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1
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| 1 |
EC50 = 10.1 nM
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CP0434351
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6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclopentane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
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C31H36N4O5
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1
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| 1 |
EC50 = 10.6 nM
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CP0416046
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4-{5-[(4-Fluoro-phenyl)-methanesulfonylamino-methyl]-[1,2,4]oxadiazol-3-yl}-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C31H31FN6O6S2
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1
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| 1 |
EC50 = 11 nM
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CP0372587
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethyl)phenoxy]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C31H29F3N6O4S
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1
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| 1 |
EC50 = 11 nM
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CP0318599
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2-[1-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]indol-3-yl]acetic acid
Show/Hide
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C31H36N4O8S2
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1
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| 1 |
EC50 = 11 nM
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CP0418812
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(R)-2-[2-(7-Benzyloxy-1H-indol-3-yl)-1-methyl-ethylamino]-1-(3-chloro-phenyl)-ethanol
Show/Hide
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C26H27ClN2O2
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1
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| 1 |
EC50 = 11 nM
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CP0514765
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(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-methoxybenzoic acid
Show/Hide
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C24H24ClNO5
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1
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| 1 |
EC50 = 11 nM
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CP0461634
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[3-[(2R)-2-[[(2R)-2-[3-(benzylamino)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C27H31N3O4S
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1
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| 1 |
EC50 = 11 nM
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CP0409670
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(S)-6-(4-(2-(3-(3-(2-cyclopentylethyl)-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C33H41N5O5
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1
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| 1 |
EC50 = 11.7 nM
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CP0383690
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4-[5-(4-Fluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H28FN5O4S
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1
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| 1 |
EC50 = 12 nM
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CP0399921
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4-[3-(3,4-Difluoro-benzyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H27F2N5O4S
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1
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| 1 |
EC50 = 12 nM
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CP0447792
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4-[5-(3-Fluoro-benzyl)-[1,2,4]oxadiazol-3-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H28FN5O4S
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1
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| 1 |
EC50 = 12 nM
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CP0453406
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4-[3-(3,4-Difluoro-phenoxymethyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H27F2N5O5S
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1
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| 1 |
EC50 = 12 nM
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CP0460921
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
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C36H34N4O3S2
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1
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| 1 |
EC50 = 12 nM
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CP0906407
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5-(4-{4-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-piperidin-1-yl}-benzyl)-thiazolidine-2,4-dione
Show/Hide
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C24H29N3O5S
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1
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| 1 |
EC50 = 12 nM
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CP0496418
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1-(3-Chloro-phenyl)-2-[1-methyl-2-(6-methyl-1H-indol-3-yl)-ethylamino]-ethanol
Show/Hide
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C20H23ClN2O
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1
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| 1 |
EC50 = 12 nM
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CP0375678
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1-(3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
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1
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| 1 |
EC50 = 12 nM
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CP0493219
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[2-[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]ethyl]benzenesulfonamide
Show/Hide
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C38H37N3O3S2
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1
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| 1 |
EC50 = 12 nM
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CP0417209
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6-(4-(2-((S)-2-hydroxy-3-(3-methyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C28H32N4O5
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1
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| 1 |
EC50 = 12 nM
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CP0412628
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4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]-2-methoxyphenyl]benzoic acid
Show/Hide
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C24H24ClNO4
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1
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| 1 |
EC50 = 12 nM
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CP0870007
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(4-{[4-(2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-ethyl)phenyl]amino}phenoxy)acetic acid hydrochloride
Show/Hide
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C24H26Cl2N2O4
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1
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| 1 |
EC50 = 12 nM
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CP0515392
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(R)-2-acetamido-5-(3-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C24H25N3O5
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1
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| 1 |
EC50 = 12 nM
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CP0371753
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6-(4-(2-((S)-3-(3-benzyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C34H36N4O5
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1
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| 1 |
EC50 = 12.3 nM
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CP0869784
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(R)-2-Cyclopropyl-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
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C27H30N4O2S
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1
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| 1 |
EC50 = 12.4 nM
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CP0404412
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N-[[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]acetamide
Show/Hide
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C20H26ClN3O2
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1
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| 1 |
EC50 = 12.59 nM
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CP0849999
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(R)-N-cyclopentyl-2-(3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)ureido)acetamide acetate
Show/Hide
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C35H54N4O8
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1
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| 1 |
EC50 = 12.59 nM
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CP0852279
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(R)-1-ethyl-3-(4-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
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C30H47N3O7
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1
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| 1 |
EC50 = 12.59 nM
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CP0530370
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1-(5-hexyl-1,2,4-oxadiazol-3-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
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C22H26N4O3S
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1
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| 1 |
EC50 = 13 nM
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CP0885826
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5-(4-{4-[2-Hydroxy-2-(2-oxo-1,2-dihydro-quinolin-5-yloxy)-ethylamino]-piperidin-1-yl}-benzyl)-thiazolidine-2,4-dione
Show/Hide
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C26H28N4O5S
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1
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| 1 |
EC50 = 13 nM
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CP0382297
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N-[3-[(1R)-1-hydroxy-2-[2-(7-methoxy-1H-indol-3-yl)ethylamino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C23H25N3O4S2
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1
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| 1 |
EC50 = 13 nM
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CP0497039
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1-[4-[(2S)-2-hydroxy-2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethyl]phenyl]-3-phenylurea
Show/Hide
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C24H27N3O4
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1
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| 1 |
EC50 = 13 nM
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CP0481422
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(R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)-2-methylbenzoic acid
Show/Hide
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C24H24ClNO4
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1
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| 1 |
EC50 = 13 nM
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CP0473749
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4-((7S)-7-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)benzoic Acid
Show/Hide
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C24H24N2O3
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1
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| 1 |
EC50 = 13 nM
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CP0155749
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-propan-2-yl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C21H28N4O4S
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1
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| 1 |
EC50 = 13 nM
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CP0869699
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(R)-2-Ethyl-N-(4-(((2S,5R)-5-((R)-hydroxy(pyridin-3-yl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
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C26H30N4O2S
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1
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| 1 |
EC50 = 13.6 nM
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CP0424778
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6-(4-(2-((S)-2-hydroxy-3-(3-isopropyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C30H36N4O5
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1
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| 1 |
EC50 = 13.9 nM
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CP0277683
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4-(3-Hexyl-2-oxo-2,3-dihydro-imidazol-1-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H37N5O4S
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1
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| 1 |
EC50 = 14 nM
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CP0376057
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4-[4-(3,4-Difluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C29H26F2N6O3S
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1
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| 1 |
EC50 = 14 nM
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CP0376379
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4-[4-(4-Fluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H29FN6O3S
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1
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| 1 |
EC50 = 14 nM
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CP0439361
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[[4-(trifluoromethoxy)phenoxy]methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C31H29F3N6O5S
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1
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| 1 |
EC50 = 14 nM
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CP0453458
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethyl)phenyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C30H27F3N6O3S
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1
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| 1 |
EC50 = 14 nM
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CP0487318
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(R)-1-(3-Chloro-phenyl)-2-[1-methyl-2-(7-propoxy-1H-indol-3-yl)-ethylamino]-ethanol
Show/Hide
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C22H27ClN2O2
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1
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| 1 |
EC50 = 14 nM
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CP0436369
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6-(4-(2-((S)-2-hydroxy-3-(3-isobutyl-2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C31H38N4O5
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1
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| 1 |
EC50 = 14 nM
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CP0515393
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(R)-3-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C23H22ClNO4
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1
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| 1 |
EC50 = 14 nM
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CP0373726
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2H-indazol-2-yl)acetamide
Show/Hide
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C24H25N5O2
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1
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| 1 |
EC50 = 14 nM
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CP0382115
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N-[3-[(1R)-2-[2-[(3-ethyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
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C20H26N4O4S
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1
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| 1 |
EC50 = 14 nM
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CP0454745
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(trifluoromethyl)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
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C31H28F3N5O4S
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1
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| 1 |
EC50 = 15 nM
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CP0438096
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-acetic acid ethyl ester
Show/Hide
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C25H34N4O7S
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1
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| 1 |
EC50 = 15 nM
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CP0424821
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4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]-2-methylbenzoic acid
Show/Hide
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C24H24ClNO3
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1
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| 1 |
EC50 = 15 nM
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CP0492962
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-(3-phenylmethoxyphenyl)ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C27H30N2O5S
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1
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| 1 |
EC50 = 15 nM
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CP0388524
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1-phenoxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C20H24N4O2S
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2
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| 1 |
EC50 = 15 nM
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| 2 |
Ki = 113 nM
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CP0382237
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetic acid
Show/Hide
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C19H23ClN2O3
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1
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| 1 |
EC50 = 15.85 nM
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CP0449854
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1-(benzenesulfonyl)-3-[[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]urea
Show/Hide
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C25H29ClN4O4S
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1
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| 1 |
EC50 = 15.85 nM
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CP0382242
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 15.85 nM
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CP0464672
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-1,3-oxazole-4-carboxylic acid
Show/Hide
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C21H22ClN3O4
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1
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| 1 |
EC50 = 15.85 nM
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CP0888674
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(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)benzyl)urea acetate
Show/Hide
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C29H45N3O7
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1
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| 1 |
EC50 = 15.85 nM
|
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CP0288880
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ethyl 2-[[(6S)-6-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-6,7,8,9-tetrahydro-5H-benzo[7]annulen-3-yl]oxy]acetate
Show/Hide
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C23H28ClNO4
|
1
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| 1 |
EC50 = 16 nM
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CP0373724
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(R)-2-(5,6-dimethyl-4-oxothieno[2,3-d]pyrimidin-3(4H)-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C25H27N5O3S
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1
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| 1 |
EC50 = 16 nM
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CP0422957
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2-Chloro-5-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
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C25H23Cl2NO4
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1
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| 1 |
EC50 = 16 nM
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CP0893924
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(S)-N-(4-(((2S,5R)-5-((R)-Hydroxy(pyridin-3-yl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-2-(1H-pyrazol-1-yl)-propanamide
Show/Hide
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C23H27N5O2
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1
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| 1 |
EC50 = 16.7 nM
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CP0433172
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2-chloro-4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]benzoic acid
Show/Hide
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C23H21Cl2NO3
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1
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| 1 |
EC50 = 17 nM
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CP0378048
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(2-methylprop-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C24H31N3O4S
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1
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| 1 |
EC50 = 17 nM
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CP0382114
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N-[3-[(1R)-2-[2-[(3-cyclopropyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
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C21H26N4O4S
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1
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| 1 |
EC50 = 17 nM
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CP0434352
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6-[4-(2-{[(2S)-2-hydroxy-3-{2'-oxo-1',2'-dihydrospiro[cyclobutane-1,3'-indole]-4'-yloxy}propyl]amino}-2-methylpropyl)phenoxy]pyridine-3-carboxamide
Show/Hide
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C30H34N4O5
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1
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| 1 |
EC50 = 17.6 nM
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CP0529098
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N-methyl-N-octyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
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C24H33N3O3S
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1
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| 1 |
EC50 = 18 nM
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CP0506458
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4-[3-(4-Fluoro-benzyl)-[1,2,4]oxadiazol-5-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H28FN5O4S
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1
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| 1 |
EC50 = 18 nM
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CP0498929
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[4-(trifluoromethoxy)phenyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C30H27F3N6O4S
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1
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| 1 |
EC50 = 18 nM
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CP0497812
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N-[3-[(1R)-1-hydroxy-2-[2-(7-methylsulfonyl-1H-indol-3-yl)ethylamino]ethyl]phenyl]ethanesulfonamide
Show/Hide
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C21H27N3O5S2
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1
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| 1 |
EC50 = 18 nM
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CP0872817
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4'-(2-{[(2R)-2-Hydroxy-2-phenylethyl]amino}ethyl)-3-methoxy-N-(methylsulfonyl)biphenyl-4-carboxamide Hydrochloride
Show/Hide
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C25H29ClN2O5S
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1
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| 1 |
EC50 = 18 nM
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CP0513757
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2-[4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]phenoxy]acetic acid
Show/Hide
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C24H24ClNO4
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1
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| 1 |
EC50 = 18 nM
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CP0921625
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4-Benzyl-piperazine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
Show/Hide
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C28H39Cl2N5O3S
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1
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| 1 |
EC50 = 18 nM
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CP0388489
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1-phenoxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C26H28N4O2S
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2
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| 1 |
EC50 = 18 nM
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| 2 |
Ki = 17 nM
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CP0085893
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]cyclobutanesulfonamide
Show/Hide
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C22H28N4O4S
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1
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| 1 |
EC50 = 18 nM
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CP0396232
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[3-[2-[[(2R)-2-[3-(ethylsulfonylamino)phenyl]-2-hydroxyethyl]amino]ethyl]-1H-indol-7-yl] methanesulfonate
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C21H27N3O6S2
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1
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| 1 |
EC50 = 18 nM
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CP0431336
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4-[4-(2,4-Difluoro-phenyl)-thiazol-2-yl]-N-{4-[2-(2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H26F2N4O3S2
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1
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| 1 |
EC50 = 19 nM
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CP0373982
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-oxoquinazolin-3(4H)-yl)acetamide
Show/Hide
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C25H25N5O3
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1
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| 1 |
EC50 = 19 nM
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CP0428924
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-oxoquinazolin-1(2H)-yl)acetamide
Show/Hide
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C25H25N5O3
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1
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| 1 |
EC50 = 19 nM
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CP0429905
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-indazol-3-yl)acetamide
Show/Hide
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C24H25N5O2
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1
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| 1 |
EC50 = 19 nM
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CP0374871
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N-[[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]methyl]methanesulfonamide
Show/Hide
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C19H26ClN3O3S
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1
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| 1 |
EC50 = 19.95 nM
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CP0448280
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(1R)-2-[[(2R)-1-anilinopropan-2-yl]amino]-1-(3-chlorophenyl)ethanol
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C17H21ClN2O
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1
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| 1 |
EC50 = 19.95 nM
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CP0488117
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N-[2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]ethyl]-4-methylbenzenesulfonamide
Show/Hide
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C26H32ClN3O3S
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1
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| 1 |
EC50 = 19.95 nM
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CP0460647
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4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzamide
Show/Hide
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C21H28N4O5S
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1
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| 1 |
EC50 = 20 nM
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CP0137653
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N-[5-[(1R)-2-[[1-[4-[(3,5-dioxo-1,2,4-oxadiazolidin-2-yl)methyl]phenyl]piperidin-4-yl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C23H29N5O7S
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1
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| 1 |
EC50 = 20 nM
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CP0504145
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1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-(3-thiophen-2-yl-propyl)-urea
Show/Hide
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C29H38N4O6S2
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1
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| 1 |
EC50 = 20 nM
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CP0515790
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3-Chloro-propane-1-sulfonic acid (3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-amide
Show/Hide
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C22H28ClN3O5S2
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1
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| 1 |
EC50 = 20 nM
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CP0378407
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(R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C18H19N3O3
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1
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| 1 |
EC50 = 20 nM
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CP0139363
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(S)-1-(9H-Carbazol-4-yloxy)-3-[1-(3,4-dimethoxy-benzenesulfonyl)-piperidin-4-ylamino]-propan-2-ol
Show/Hide
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C28H33N3O6S
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1
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| 1 |
EC50 = 20 nM
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CP0422958
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3-[((7S)-7-{[(2R)-2-Hydroxy-2-(3-pyridinyl)ethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
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C24H24N2O4
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1
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| 1 |
EC50 = 20 nM
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CP0377155
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4-(2-hydroxy-3-(1-(5-methylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C21H26N4O3S
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2
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| 1 |
EC50 = 20 nM
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| 2 |
Ki = 1390 nM
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CP0490790
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N-[3-[(1R)-1-hydroxy-2-[2-(1H-indol-3-yl)ethylamino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C22H23N3O3S2
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1
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| 1 |
EC50 = 21 nM
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CP0452654
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(R)-3-benzamido-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C30H27ClN2O5
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1
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| 1 |
EC50 = 21 nM
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CP0373743
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-imidazol-2-yl)benzamide
Show/Hide
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C25H25N5O2
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1
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| 1 |
EC50 = 21 nM
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CP0400357
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(R)-2-(benzo[d]oxazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C24H24N4O3
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1
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| 1 |
EC50 = 21 nM
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CP0374193
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1-(3-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C27H30N4O3S
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2
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| 1 |
EC50 = 21 nM
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| 2 |
Ki = 42 nM
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CP0059008
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C19H24N4O4S
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1
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| 1 |
EC50 = 21 nM
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CP0449007
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-pyridin-2-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
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C29H27N5O3S2
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1
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| 1 |
EC50 = 22 nM
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CP0384184
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4-[4-(3-Fluoro-4-methoxy-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H29FN6O4S
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1
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| 1 |
EC50 = 22 nM
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CP0479820
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1-(3-Chloro-phenyl)-2-[2-(6-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C20H23ClN2O2
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1
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| 1 |
EC50 = 22 nM
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CP0505688
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-pyridin-2-yl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
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C31H30N4O3S2
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1
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| 1 |
EC50 = 22 nM
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CP0464629
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1-[4-[(2S)-2-[[(2S)-3-(9H-carbazol-4-yloxy)-2-hydroxypropyl]amino]-3-hydroxypropyl]phenyl]-3-phenylurea
Show/Hide
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C31H32N4O4
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1
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| 1 |
EC50 = 22 nM
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CP0373721
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(R)-2-(3-amino-1H-1,2,4-triazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C19H23N7O2
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1
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| 1 |
EC50 = 22 nM
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CP0387765
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2-[3-[[(7S)-7-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-5,6,7,8-tetrahydronaphthalen-2-yl]oxy]phenoxy]acetic acid
Show/Hide
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C26H26ClNO5
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1
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| 1 |
EC50 = 22 nM
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CP0460285
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,5-difluoro-benzylamide
Show/Hide
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C30H36F2N4O4
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1
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| 1 |
EC50 = 23 nM
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CP0869578
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4-Phenyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide dihydrochloride
Show/Hide
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C26H34Cl2N4O3S
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1
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| 1 |
EC50 = 23 nM
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CP0419359
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4-[4-(2,6-Difluoro-benzyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H28F2N6O3S
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1
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| 1 |
EC50 = 24 nM
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CP0495477
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4-[4-(4-Fluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C29H27FN6O3S
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1
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| 1 |
EC50 = 24 nM
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CP0850027
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5-(4-{4-[(S)-2-Hydroxy-3-(2-oxo-2H-benzoimidazol-4-yloxy)-propylamino]-piperidin-1-yl}-benzyl)-thiazolidine-2,4-dione
Show/Hide
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C25H27N5O5S
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1
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| 1 |
EC50 = 24 nM
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CP0926692
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(3S,5R)-3,5-Dimethyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide dihydrochloride
Show/Hide
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C22H34Cl2N4O3S
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1
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| 1 |
EC50 = 24 nM
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CP0428926
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(R)-2-(2H-benzo[d][1,2,3]triazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C23H24N6O2
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1
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| 1 |
EC50 = 24 nM
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CP0428933
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(R)-2-(2-(1H-pyrrol-1-yl)ethyl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
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C28H30N4O2
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1
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| 1 |
EC50 = 24 nM
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CP0423023
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2-[4-[[(7S)-7-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-5,6,7,8-tetrahydronaphthalen-2-yl]oxy]phenoxy]acetic acid
Show/Hide
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C26H26ClNO5
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1
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| 1 |
EC50 = 24 nM
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CP0388618
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4-(2-hydroxy-3-(1-(thieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C20H24N4O3S
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2
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| 1 |
EC50 = 24 nM
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| 2 |
Ki = 1300 nM
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CP0100405
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N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzamide
Show/Hide
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C23H26N4O2S
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1
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| 1 |
EC50 = 24 nM
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CP0371758
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(S)-6-(4-(2-(2-hydroxy-3-(2-oxoindolin-4-yloxy)propylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
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C27H30N4O5
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1
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| 1 |
EC50 = 24.4 nM
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CP0442313
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N-[3-[(1R)-1-hydroxy-2-[2-(7-methyl-1H-indol-3-yl)ethylamino]ethyl]phenyl]thiophene-2-sulfonamide
Show/Hide
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C23H25N3O3S2
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1
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| 1 |
EC50 = 25 nM
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CP0897953
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N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}-2-methylpropyl)phenyl]N-cyclohexylsulfamide; 2HCl
Show/Hide
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C23H36Cl2N4O3S
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1
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| 1 |
EC50 = 25 nM
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CP0382238
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3-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]propanoic acid
Show/Hide
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C20H25ClN2O3
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1
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| 1 |
EC50 = 25.12 nM
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CP0386623
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sodium;2-[4-[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]phenoxy]acetate
Show/Hide
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C19H21ClNO4-
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1
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| 1 |
EC50 = 25.12 nM
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CP0066323
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CAS_73573-87-2
Show/Hide
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C19H24N2O4
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1
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| 1 |
EC50 = 25.12 nM
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CP0708203
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(R,R)-formoterol fumarate
Show/Hide
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C23H28N2O8
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1
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| 1 |
EC50 = 25.12 nM
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CP0917315
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1-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4,5-imidazolidinetrione formate salt
Show/Hide
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C30H41N3O9
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1
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| 1 |
EC50 = 25.12 nM
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CP0850450
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Formoterol fumarate
Show/Hide
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C23H30N2O9
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1
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| 1 |
EC50 = 25.12 nM
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CP0888673
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(R)-1-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)-5-(trifluoromethyl)phenyl)urea acetate
Show/Hide
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C29H42F3N3O7
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1
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| 1 |
EC50 = 25.12 nM
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CP0467467
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4-[4-(3-Cyclopentyl-propyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C32H38N4O3S2
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1
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| 1 |
EC50 = 26 nM
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CP0345975
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-3-methyl-butyric acid
Show/Hide
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C26H36N4O7S
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1
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| 1 |
EC50 = 26 nM
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CP0559881
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1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-pyridin-2-yl-urea
Show/Hide
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C27H33N5O6S
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1
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| 1 |
EC50 = 26 nM
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CP0439415
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4-[[4-(2-cyclopentylethyl)-1,3-thiazol-2-yl]methyl]-N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]benzenesulfonamide
Show/Hide
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C33H39N3O3S2
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1
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| 1 |
EC50 = 26 nM
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CP0377154
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1-(3-(hydroxymethyl)phenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
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2
|
| 1 |
EC50 = 26 nM
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| 2 |
Ki = 49 nM
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CP0458862
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1-[(2,5-difluorophenyl)methyl]-3-[4-[4-[[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]piperidin-1-yl]sulfonylphenyl]-1-propan-2-ylurea
Show/Hide
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C32H41F2N5O7S2
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1
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| 1 |
EC50 = 27 nM
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CP0229485
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(R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy)ethylamino)ethanol
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C18H19N3O2S
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1
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| 1 |
EC50 = 27 nM
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CP0373733
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-pyrazol-1-ylpropanamide
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C21H25N5O2
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1
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| 1 |
EC50 = 27 nM
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CP0397769
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2-[2-(6-Chloro-1H-indol-3-yl)-1-methyl-ethylamino]-1-(3-chloro-phenyl)-ethanol
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C19H20Cl2N2O
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1
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| 1 |
EC50 = 28 nM
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CP0417356
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3-(cyclohexyloxy)-4'-(2-((1R,2S)-1-hydroxy-1-(4-methoxyphenyl)propan-2-ylamino)ethyl)-N-(methylsulfonyl)biphenyl-4-carboxamide
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C32H40N2O6S
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1
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| 1 |
EC50 = 28 nM
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CP0381357
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4-((S)-7-((R)-2-(4-cyanophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
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C26H24N2O3
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1
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| 1 |
EC50 = 28 nM
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CP0483633
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[3-(trifluoromethoxy)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
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C31H28F3N5O5S
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1
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| 1 |
EC50 = 29 nM
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CP0408895
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1-(2,5-Difluoro-benzyl)-3-[4-(4-{[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-urea
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C29H34F2N4O6S
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1
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| 1 |
EC50 = 29 nM
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CP0371987
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3-((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)benzoic Acid
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C25H24ClNO3
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1
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| 1 |
EC50 = 29 nM
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CP0403508
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid amide
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C23H32N4O4
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1
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| 1 |
EC50 = 30 nM
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CP0409519
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,4-difluoro-benzylamide
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C30H36F2N4O4
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1
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| 1 |
EC50 = 30 nM
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CP0036332
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4-{(R)-2-[1-(4-Butoxy-benzenesulfonyl)-azetidin-3-ylamino]-1-hydroxy-ethyl}-phenol
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C21H28N2O5S
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1
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| 1 |
EC50 = 30 nM
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CP0456117
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4-(2-{[(2R)-2-(3-Methansulfonylaminophenyl)-2-hydroxyethyl]-amino}ethyl)-3-isopropoxy-4-biphenylcarboxylic acid
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C27H32N2O6S
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1
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| 1 |
EC50 = 30 nM
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CP0409910
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1-(5-octyl-1,2,4-oxadiazol-3-yl)-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
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C24H30N4O3S
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1
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| 1 |
EC50 = 31 nM
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CP0441693
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N-[4-[[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methoxy]phenyl]acetamide
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C32H32N6O6S
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1
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| 1 |
EC50 = 31 nM
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CP0401690
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4-Aminomethylpiperidine substituted analogue
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C31H39N5O9S2
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1
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| 1 |
EC50 = 31 nM
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CP0432795
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4-Aminomethylpiperidine substituted analogue
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C31H38N4O7S
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1
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| 1 |
EC50 = 31 nM
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CP0522725
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(R)-2-fluoro-5-(3-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenoxy)benzoic acid
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C22H21FN2O4
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1
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| 1 |
EC50 = 31 nM
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CP0042352
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2,3-bis(oxidanyl)butanedioic acid;4-[(1R)-2-(methylamino)-1-oxidanyl-ethyl]benzene-1,2-diol
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C9H13NO3
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2
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| 1 |
EC50 = 31 nM
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| 2 |
EC50 = 49 nM
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CP0441823
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]pyridine-3-carboxylic acid
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C23H24ClN3O3
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1
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| 1 |
EC50 = 31.62 nM
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CP0451649
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4-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]benzoic acid
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C24H25ClN2O3
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1
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| 1 |
EC50 = 31.62 nM
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CP0847188
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4-[(1R)-1-Hydroxy-2-({6-[(2-{[(3-hydroxyphenyl)methyl]oxy}-ethyl)oxy]-hexyl}amino)ethyl]-2-(hydroxymethyl)phenol Acetate Salt
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C26H39NO8
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1
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| 1 |
EC50 = 31.62 nM
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CP0890908
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3-[4-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione acetate salt
Show/Hide
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C30H43N3O8
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1
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| 1 |
EC50 = 31.62 nM
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CP0870890
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(R)-1-ethyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)benzyl)urea acetate
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C31H49N3O7
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1
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| 1 |
EC50 = 31.62 nM
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CP0399662
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,6-difluoro-benzylamide
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C30H36F2N4O4
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1
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| 1 |
EC50 = 32 nM
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CP0403166
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2-[4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]phenyl]acetic acid
Show/Hide
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C24H24ClNO3
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1
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| 1 |
EC50 = 32 nM
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CP0379227
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Benzenesulfonic acid 3-{(R)-1-hydroxy-2-[(R)-2-(7-methanesulfonyloxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethyl}-phenyl ester
Show/Hide
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C26H28N2O7S2
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1
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| 1 |
EC50 = 32 nM
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CP0428934
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-phenethylbenzamide
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C30H31N3O2
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1
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| 1 |
EC50 = 32 nM
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CP0377145
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-(2-phenylethyl)-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
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C32H32N4O3S2
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1
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| 1 |
EC50 = 33 nM
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CP0371935
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[[4-(2-phenylethyl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
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C34H35N3O3S2
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1
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| 1 |
EC50 = 33 nM
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CP0378228
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[[4-(naphthalen-2-ylmethyl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
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C37H35N3O3S2
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1
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| 1 |
EC50 = 33 nM
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CP0422410
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6-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]pyridine-3-carboxylic acid
Show/Hide
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C22H21ClN2O3
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1
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| 1 |
EC50 = 33 nM
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CP0387867
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4-((S)-7-((R)-2-(3,4-dichlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
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C25H23Cl2NO3
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1
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| 1 |
EC50 = 33 nM
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CP0472744
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4-(2-hydroxy-3-(1-(thieno[3,2-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenol
Show/Hide
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C20H24N4O3S
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2
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| 1 |
EC50 = 33 nM
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| 2 |
Ki = 1385 nM
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CP0741529
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[5-(4-{4-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzyl)-2,4-dioxo-thiazolidin-3-yl]-acetic acid
Show/Hide
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C26H32N4O8S2
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1
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| 1 |
EC50 = 34 nM
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CP0850065
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N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(2-imino-5-oxo-imidazolidin-4-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-ethyl)-phenyl]-methanesulfonamide
Show/Hide
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C24H30N6O5S
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1
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| 1 |
EC50 = 34 nM
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CP0429875
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(R)-2-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
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C29H27N5O2
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1
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| 1 |
EC50 = 35 nM
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CP0377227
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3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzonitrile
Show/Hide
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C27H27N5O2S
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2
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| 1 |
EC50 = 35 nM
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| 2 |
Ki = 47 nM
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CP0498840
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid diethylamide
Show/Hide
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C27H40N4O4
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1
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| 1 |
EC50 = 36 nM
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CP0454822
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2-[butyl-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]benzoyl]amino]acetic acid
Show/Hide
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C27H38N4O7S
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1
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| 1 |
EC50 = 36 nM
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CP0039161
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[3-[(2R)-2-[[(2R)-2-hydroxy-2-[3-(3-methylbut-2-enylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
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C25H33N3O4S
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1
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| 1 |
EC50 = 36 nM
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CP0230988
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1-Hexyl-3-(4-{4-[(S)-2-hydroxy-3-(2-oxo-2,3-dihydro-1H-benzoimidazol-4-yloxy)-propylamino]-piperidine-1-sulfonyl}-phenyl)-urea
Show/Hide
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C28H40N6O6S
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1
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| 1 |
EC50 = 36 nM
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CP0853728
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4-Methyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide dihydrochloride
Show/Hide
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C21H32Cl2N4O3S
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1
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| 1 |
EC50 = 36 nM
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CP0373744
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(R)-2-(benzo[d]thiazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
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C29H26N4O2S
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1
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| 1 |
EC50 = 36 nM
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CP0384229
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2-fluoro-benzylamide
Show/Hide
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C30H37FN4O4
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1
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| 1 |
EC50 = 37 nM
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CP0378414
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(R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3O3
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1
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| 1 |
EC50 = 37 nM
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CP0428932
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(R)-2-(2,5-dimethylthiazol-4-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C22H26N4O2S
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1
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| 1 |
EC50 = 37 nM
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CP0428938
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-phenethylbenzamide
Show/Hide
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C30H31N3O2
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1
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| 1 |
EC50 = 37 nM
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CP0479015
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4-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]benzoic Acid
Show/Hide
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C25H24ClNO4
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1
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| 1 |
EC50 = 37 nM
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CP0480615
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2-[2-(6-Bromo-1H-indol-3-yl)-1-methyl-ethylamino]-1-(3-chloro-phenyl)-ethanol
Show/Hide
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C19H20BrClN2O
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1
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| 1 |
EC50 = 38 nM
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CP0932600
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N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}-2-methylpropyl)phenyl]N,N-dimethylsulfamide; 2HCl
Show/Hide
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C19H30Cl2N4O3S
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1
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| 1 |
EC50 = 38 nM
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CP0456746
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4-((S)-7-((R)-2-(2-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yl)benzoic acid
Show/Hide
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C25H24ClNO3
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1
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| 1 |
EC50 = 38 nM
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CP0420451
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3-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-phenyl)-propionic acid
Show/Hide
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C23H31N3O6S
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1
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| 1 |
EC50 = 39 nM
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CP0393172
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(R)-3-(4-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C23H22ClNO4
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1
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| 1 |
EC50 = 39 nM
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CP0422403
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2-[4-[[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]methyl]phenoxy]acetic acid
Show/Hide
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C25H26ClNO4
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1
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| 1 |
EC50 = 39 nM
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CP0423025
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2-((S)-7-((R)-2-(3-chlorophenyl)-2-hydroxyethylamino)-5,6,7,8-tetrahydronaphthalen-2-yloxy)acetic acid
Show/Hide
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C20H22ClNO4
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1
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| 1 |
EC50 = 39 nM
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CP0456857
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6-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-2-carboxylic acid
Show/Hide
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C22H22ClN3O3
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1
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| 1 |
EC50 = 39.81 nM
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CP0874619
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2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({2-[(phenylmethyl)-oxy]ethyl}oxy)hexyl]amino}ethyl)phenol
Show/Hide
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C26H39NO7
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1
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| 1 |
EC50 = 39.81 nM
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CP0884855
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3-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4-imidazolidinedione acetate salt
Show/Hide
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C31H45N3O8
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1
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| 1 |
EC50 = 39.81 nM
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CP0851887
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N-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)-5-methylphenyl]urea acetate salt
Show/Hide
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C29H45N3O7
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1
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| 1 |
EC50 = 39.81 nM
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CP0106025
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(-)ISOPROTERENOL
Show/Hide
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C11H17NO3
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1
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| 1 |
EC50 = 39.81 nM
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CP0376537
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-(4-pyridin-3-yl-1,3-thiazol-2-yl)benzenesulfonamide
Show/Hide
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C29H27N5O3S2
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1
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| 1 |
EC50 = 40 nM
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CP0885547
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5-{4-[4-((S)-2-Hydroxy-3-phenoxy-propylamino)-piperidin-1-yl]-benzyl}-thiazolidine-2,4-dione
Show/Hide
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C24H29N3O4S
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1
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| 1 |
EC50 = 40 nM
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CP0495316
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[(4-pyridin-3-yl-1,3-thiazol-2-yl)methyl]benzenesulfonamide
Show/Hide
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C31H30N4O3S2
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1
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| 1 |
EC50 = 40 nM
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CP0382117
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methoxy-1H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C19H24N4O5S
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1
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| 1 |
EC50 = 40 nM
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CP0404367
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 4-fluoro-benzylamide
Show/Hide
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C30H37FN4O4
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1
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| 1 |
EC50 = 41 nM
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CP0921819
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4-Methyl-piperazine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
Show/Hide
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C22H35Cl2N5O3S
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1
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| 1 |
EC50 = 41 nM
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CP0377222
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1-(3-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C26H27FN4O2S
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2
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| 1 |
EC50 = 41 nM
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| 2 |
Ki = 17 nM
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CP0378409
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(R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3O4
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1
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| 1 |
EC50 = 42 nM
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CP0452934
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(R)-2-cyclohexyl-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
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C28H33N3O2
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1
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| 1 |
EC50 = 42 nM
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CP0403823
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1-[4-(4-{[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-1H-pyrazole-4-carboxylic acid
Show/Hide
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C25H31N5O8S2
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1
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| 1 |
EC50 = 43 nM
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CP0382118
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N-[3-[(1R)-2-[2-[(3-chloro-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
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C18H21ClN4O4S
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1
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| 1 |
EC50 = 43 nM
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CP0408383
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]cyclopropanesulfonamide
Show/Hide
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C21H26N4O4S
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1
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| 1 |
EC50 = 43 nM
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CP0937943
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(S)-2-Amino-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)methyl)-pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4H-cyclopenta[d]-thiazole-4-carboxamide
Show/Hide
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C25H28N4O2S
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1
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| 1 |
EC50 = 44.2 nM
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CP0383394
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4-[4-(4-Hydroxy-phenyl)-thiazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
|
C30H28N4O4S2
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1
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| 1 |
EC50 = 45 nM
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CP0421152
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N-[4-[2-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,3-thiazol-4-yl]phenyl]acetamide
Show/Hide
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C32H31N5O4S2
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1
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| 1 |
EC50 = 45 nM
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CP0460775
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1-(2,5-Difluoro-benzyl)-3-[4-(4-{[(S)-3-(3-fluoro-4-hydroxy-phenoxy)-2-hydroxy-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-urea
Show/Hide
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C29H33F3N4O6S
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1
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| 1 |
EC50 = 45 nM
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CP0436006
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[[4-(4-hydroxyphenyl)-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
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C32H31N3O4S2
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1
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| 1 |
EC50 = 45 nM
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CP0486675
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N-[4-[2-[[4-[[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]methyl]-1,3-thiazol-4-yl]phenyl]acetamide
Show/Hide
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C34H34N4O4S2
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1
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| 1 |
EC50 = 45 nM
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CP0383192
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N-hexyl-N-methyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
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C22H29N3O3S
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1
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| 1 |
EC50 = 47 nM
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CP0391295
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid methylamide
Show/Hide
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C24H34N4O4
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1
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| 1 |
EC50 = 47 nM
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CP0378413
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(R)-2-(2-(4-(2-(methoxymethyl)oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C20H23N3O4
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1
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| 1 |
EC50 = 47 nM
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CP0950698
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4-Phenyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-2-methyl-propyl]-phenyl}-amide dihydrochloride
Show/Hide
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C28H38Cl2N4O3S
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1
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| 1 |
EC50 = 47 nM
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CP0428935
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(phenoxymethyl)benzamide
Show/Hide
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C29H29N3O3
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1
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| 1 |
EC50 = 47 nM
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CP0432468
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[(2,4,6-trifluorophenyl)methyl]triazol-2-yl]benzenesulfonamide
Show/Hide
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C30H27F3N6O3S
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1
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| 1 |
EC50 = 48 nM
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CP0430919
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1-[(S)-4-(4-{[3-(9H-Carbazol-4-yloxy)-2-hydroxy-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-hexyl-urea
Show/Hide
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C34H45N5O5S
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1
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| 1 |
EC50 = 48 nM
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CP0496882
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2,2,2-Trifluoro-ethanesulfonic acid (3-{(R)-1-hydroxy-2-[2-(7-methanesulfonyl-1H-indol-3-yl)-ethylamino]-ethyl}-phenyl)-amide
Show/Hide
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C21H24F3N3O5S2
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1
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| 1 |
EC50 = 48 nM
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CP0876201
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{4-[4-(2-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-ethyl)phenoxy]phenoxy}acetic acid hydrochloride
Show/Hide
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C24H25Cl2NO5
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1
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| 1 |
EC50 = 48 nM
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CP0417913
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-indazol-1-yl)acetamide
Show/Hide
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C24H25N5O2
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1
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| 1 |
EC50 = 48 nM
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CP0375239
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1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-octyl-urea
Show/Hide
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C30H46N4O6S
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1
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| 1 |
EC50 = 49 nM
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CP0371984
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2-[((7S)-7-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-5,6,7,8-tetrahydro-2-naphthalenyl)oxy]nicotinic Acid
Show/Hide
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C24H23ClN2O4
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1
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| 1 |
EC50 = 49 nM
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CP0377641
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N-[5-[2-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,3-thiazol-4-yl]pentyl]acetamide
Show/Hide
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C31H37N5O4S2
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1
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| 1 |
EC50 = 50 nM
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CP0506166
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid (3-cyclopentyl-propyl)-amide
Show/Hide
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C31H46N4O4
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1
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| 1 |
EC50 = 50 nM
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CP0527866
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N-[5-[2-[[4-[[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]methyl]-1,3-thiazol-4-yl]pentyl]acetamide
Show/Hide
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C33H40N4O4S2
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1
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| 1 |
EC50 = 50 nM
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CP0850211
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N-Cyclohexyl-3-(4-{[6-({(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
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C33H52N2O8S
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1
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| 1 |
EC50 = 50.12 nM
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CP0851858
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1-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4(1H,3H)-pyrimidinedione acetate salt
Show/Hide
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C31H43N3O8
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1
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| 1 |
EC50 = 50.12 nM
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CP0434375
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4-(4-Hexyl-thiazol-2-yl)-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C30H36N4O3S2
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1
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| 1 |
EC50 = 51 nM
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CP0378231
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N-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenyl]-4-[[4-[(1E,5E)-octa-1,5-dienyl]-1,3-thiazol-2-yl]methyl]benzenesulfonamide
Show/Hide
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C34H39N3O3S2
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1
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| 1 |
EC50 = 51 nM
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CP0404091
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4-[4-(3-Fluoro-phenyl)-[1,2,3]triazol-2-yl]-N-{4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-benzenesulfonamide
Show/Hide
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C29H27FN6O3S
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1
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| 1 |
EC50 = 52 nM
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CP0469299
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[3-[(2R)-2-[[(2R)-2-[3-[benzenesulfonyl(methyl)amino]phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
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C27H31N3O6S2
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1
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| 1 |
EC50 = 52 nM
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CP0377071
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[4-[2-(trifluoromethyl)phenyl]-1,3-thiazol-2-yl]benzenesulfonamide
Show/Hide
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C31H27F3N4O3S2
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1
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| 1 |
EC50 = 53 nM
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CP0378309
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N-methyl-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
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C16H17N3O3S
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1
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| 1 |
EC50 = 55 nM
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CP0429222
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N-methyl-N-(2-phenylethyl)-5-(phenylsulfamoyl)-2,3-dihydroindole-1-carboxamide
Show/Hide
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C24H25N3O3S
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1
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| 1 |
EC50 = 55 nM
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CP0392923
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1-[4-(4-{[(S)-2-Hydroxy-3-(2-oxo-2,3-dihydro-1H-indol-4-yloxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-octyl-urea
Show/Hide
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C32H47N5O6S
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1
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| 1 |
EC50 = 55 nM
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CP0388094
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(6-chloro-2-pyridyl)acetanilide
Show/Hide
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C24H26ClN3O3
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1
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| 1 |
EC50 = 55 nM
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CP0044683
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4-{(S)-2-Hydroxy-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propoxy}-phenol
Show/Hide
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C21H28N2O6S
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1
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| 1 |
EC50 = 55 nM
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CP0377150
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(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenyl)(morpholino)methanone
Show/Hide
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C31H35N5O4S
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2
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| 1 |
EC50 = 55 nM
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| 2 |
Ki = 149 nM
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CP0401170
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(R)-5-(3-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenoxy)-2-methoxybenzoic acid
Show/Hide
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C23H24N2O5
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1
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| 1 |
EC50 = 56 nM
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CP0378410
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(R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C21H25N3O3
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1
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| 1 |
EC50 = 57 nM
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CP0434384
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(R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C20H23N3O3
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1
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| 1 |
EC50 = 57 nM
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CP0501735
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1-Hexyl-3-[4-(4-{[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-urea
Show/Hide
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C28H42N4O6S
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1
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| 1 |
EC50 = 58 nM
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CP0135421
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-acetic acid
Show/Hide
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C23H30N4O7S
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1
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| 1 |
EC50 = 60 nM
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CP0440221
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1-Cyclohexyl-3-[4-(4-{[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-urea
Show/Hide
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C28H40N4O6S
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1
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| 1 |
EC50 = 60 nM
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CP0491317
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(R)-4-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C23H22ClNO4
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1
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| 1 |
EC50 = 60 nM
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CP0094903
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(S)-1-(9H-Carbazol-4-yloxy)-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propan-2-ol
Show/Hide
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C27H31N3O5S
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1
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| 1 |
EC50 = 60 nM
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CP0403165
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2-[4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]benzoyl]phenoxy]acetic acid
Show/Hide
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C25H24ClNO5
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1
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| 1 |
EC50 = 61 nM
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CP0231692
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ethyl 1-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]piperidine-4-carboxylate
Show/Hide
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C27H34N2O4
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1
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| 1 |
EC50 = 63 nM
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CP0449097
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2-[4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]-N-[(4-methylphenyl)methyl]acetamide
Show/Hide
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C27H32ClN3O2
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1
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| 1 |
EC50 = 63.1 nM
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CP0420505
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5-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]pyridine-3-carboxylic acid
Show/Hide
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C22H22ClN3O3
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1
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| 1 |
EC50 = 63.1 nM
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CP0482973
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4-[(1R)-1-hydroxy-2-[6-[2-[(4-hydroxyphenyl)methoxy]ethoxy]hexylamino]ethyl]-2-(hydroxymethyl)phenol
Show/Hide
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C24H35NO6
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1
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| 1 |
EC50 = 63.1 nM
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CP0884854
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3-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-5,5-dimethyl-2,4-imidazolidinedione acetate salt
Show/Hide
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C32H47N3O8
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1
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| 1 |
EC50 = 63.1 nM
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CP0913516
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1-{[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]methyl}-2,4-imidazolidinedione acetate salt
Show/Hide
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C31H45N3O8
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1
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| 1 |
EC50 = 63.1 nM
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CP0860176
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N-{4-[2-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-4-{5-[4-(5H-tetrazol-5-yl)-phenoxymethyl]-[1,2,4]oxadiazol-3-yl}-benzenesulfonamide
Show/Hide
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C31H29N9O5S
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1
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| 1 |
EC50 = 64 nM
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CP0373723
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N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
Show/Hide
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C27H30N4O3
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1
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| 1 |
EC50 = 64 nM
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CP0433203
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N-[3-[(1R)-1-hydroxy-2-[2-[[3-(trifluoromethyl)-2H-indazol-6-yl]oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C19H21F3N4O4S
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1
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| 1 |
EC50 = 64 nM
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CP0424751
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(R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thiazol-4-yl)phenoxy)ethylamino)ethanol
Show/Hide
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C23H22N4O2S
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1
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| 1 |
EC50 = 65 nM
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CP0376758
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4-(4-{2-[(S)-2-Hydroxy-3-(8-hydroxy-2-oxo-1,2,3,4-tetrahydro-quinolin-5-yloxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid octylamide
Show/Hide
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C34H51N5O5
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1
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| 1 |
EC50 = 66 nM
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CP0422142
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzyloxy)-acetic acid
Show/Hide
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C23H31N3O7S
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1
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| 1 |
EC50 = 66 nM
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CP0382113
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N-[3-[(1R)-2-[2-[(3-cyclobutyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
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C22H28N4O4S
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1
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| 1 |
EC50 = 66 nM
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CP0373741
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(pyrrolidin-1-yl)benzamide
Show/Hide
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C26H30N4O2
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1
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| 1 |
EC50 = 67 nM
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CP0475694
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1-(3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-ethylamino]-ethanol
Show/Hide
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C18H19ClN2O
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1
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| 1 |
EC50 = 69 nM
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CP0372414
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(2-naphtylmethyl)imidazol-2-yl]acetanilide
Show/Hide
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C33H34N4O3
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1
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| 1 |
EC50 = 69 nM
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CP0472259
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3-[((S)-4-{[3-(9H-Carbazol-4-yloxy)-2-hydroxy-propylamino]-methyl}-piperidine-1-carbonyl)-amino]-benzoic acid
Show/Hide
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C29H32N4O5
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1
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| 1 |
EC50 = 70 nM
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CP0437512
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1-(3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1,1-dimethyl-ethylamino]-ethanol
Show/Hide
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C20H23ClN2O
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1
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| 1 |
EC50 = 70 nM
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CP0101006
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4-{(S)-3-[1-(Dibenzofuran-2-sulfonyl)-piperidin-4-ylamino]-2-hydroxy-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
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C27H28N4O6S
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1
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| 1 |
EC50 = 70 nM
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CP0464884
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N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]propane-2-sulfonamide
Show/Hide
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C21H28N4O4S
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1
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| 1 |
EC50 = 70 nM
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CP0388095
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(4-bromobenzyl)imidazol-2-yl]acetanilide
Show/Hide
|
C29H31BrN4O3
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1
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| 1 |
EC50 = 71 nM
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CP0445254
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N-[3-[(1R)-2-[2-[(3-ethoxy-1H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
|
C20H26N4O5S
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1
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| 1 |
EC50 = 71 nM
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CP0373746
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-5-methyl-2-(pyrrolidin-1-yl)benzamide
Show/Hide
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C27H32N4O2
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1
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| 1 |
EC50 = 73 nM
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CP0388090
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-[1-(4-chlorobenzyl)imidazol-2-yl]acetanilide
Show/Hide
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C29H31ClN4O3
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1
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| 1 |
EC50 = 74 nM
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CP0499962
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1-[4-[(2S)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]-3-hydroxypropyl]phenyl]-3-phenylurea
Show/Hide
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C24H26ClN3O3
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1
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| 1 |
EC50 = 74 nM
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CP0400358
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-methylthiazol-2-yl)acetamide
Show/Hide
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C21H24N4O2S
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1
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| 1 |
EC50 = 74 nM
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CP0383926
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5-{4-[4-((S)-2-Hydroxy-3-phenoxy-propylamino)-piperidin-1-yl]-benzylidene}-2-piperidin-1-yl-thiazol-4-one
Show/Hide
|
C29H36N4O3S
|
1
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| 1 |
EC50 = 75 nM
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CP0472576
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ethyl (1S,5R)-3-[4-[[(2S,5R)-5-[(R)-hydroxy(phenyl)methyl]pyrrolidin-2-yl]methyl]benzoyl]-3-azabicyclo[3.1.0]hexane-6-carboxylate
Show/Hide
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C27H32N2O4
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1
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| 1 |
EC50 = 75 nM
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CP0430396
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-methyl-2-(pyrrolidin-1-yl)benzamide
Show/Hide
|
C27H32N4O2
|
1
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| 1 |
EC50 = 76 nM
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CP0429887
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2H-1,2,3-triazol-2-yl)benzamide
Show/Hide
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C24H24N6O2
|
1
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| 1 |
EC50 = 76.2 nM
|
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CP0869700
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N-(4-(((2S,5R)-5-((R)-Hydroxy(pyridin-3-yl)methyl)pyrrolidin-2-yl)methyl)phenyl)-2-(1H-pyrazol-1-yl)acetamide
Show/Hide
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C22H25N5O2
|
1
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| 1 |
EC50 = 76.7 nM
|
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CP0279642
|
(S)-N-(4-(2-(2-hydroxy-3-(4-hydroxyphenoxy)propylamino)ethyl)phenyl)benzenesulfonamide
Show/Hide
|
C23H26N2O5S
|
1
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| 1 |
EC50 = 78 nM
|
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CP0440078
|
N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]-4-[5-[[4-(methanesulfonamido)phenyl]methyl]-1,2,4-oxadiazol-3-yl]benzenesulfonamide
Show/Hide
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C31H32N6O6S2
|
1
|
| 1 |
EC50 = 79 nM
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CP0435332
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1-(2-allylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C29H32N4O2S
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2
|
| 1 |
EC50 = 79 nM
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| 2 |
Ki = 86 nM
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CP0853348
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N-(3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]-ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}phenyl)methanesulfonamideAcetate Salt
Show/Hide
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C27H42N2O9S
|
1
|
| 1 |
EC50 = 79.43 nM
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CP0871785
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2-{3-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,5-dioxo-1-imidazolidinyl}acetamide acetate salt
Show/Hide
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C32H46N4O9
|
1
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| 1 |
EC50 = 79.43 nM
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CP0404342
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid cyclohexylamide
Show/Hide
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C29H42N4O4
|
1
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| 1 |
EC50 = 80 nM
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CP0871261
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N-[2-Hydroxy-5-((R)-1-hydroxy-2-{1-[4-(2-hydroxyamino-4-oxo-4H-thiazol-5-ylidenemethyl)-phenyl]-piperidin-4-ylamino}-ethyl)-phenyl]-methanesulfonamide
Show/Hide
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C24H29N5O6S2
|
1
|
| 1 |
EC50 = 80 nM
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CP0387789
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(pyrazin-2-yl)acetanilide
Show/Hide
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C23H26N4O4
|
1
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| 1 |
EC50 = 83 nM
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CP0471185
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2-[4-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]sulfanylphenoxy]acetic acid
Show/Hide
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C24H24ClNO4S
|
1
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| 1 |
EC50 = 85 nM
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CP0915960
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N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(2-imino-4-oxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-ethyl)-phenyl]-methanesulfonamide
Show/Hide
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C24H31N5O5S2
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1
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| 1 |
EC50 = 86 nM
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CP0373718
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(4-phenylthiazol-2-yl)acetamide
Show/Hide
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C26H26N4O2S
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1
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| 1 |
EC50 = 86 nM
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CP0373745
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(R)-2-(furan-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)benzamide
Show/Hide
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C26H25N3O3
|
1
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| 1 |
EC50 = 86 nM
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CP0403724
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1-heptanoyl-N-phenyl-2,3-dihydro-1H-indole-5-sulfonamide
Show/Hide
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C21H26N2O3S
|
1
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| 1 |
EC50 = 88 nM
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CP0437394
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid isopropylamide
Show/Hide
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C26H38N4O4
|
1
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| 1 |
EC50 = 90 nM
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CP0959403
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N-{5-[(R)-2-(1-{4-[2-(1-Benzyl-piperidin-4-ylamino)-4-oxo-4H-thiazol-5-ylidenemethyl]-phenyl}-piperidin-4-ylamino)-1-hydroxy-ethyl]-2-hydroxy-phenyl}-methanesulfonamide
Show/Hide
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C36H44N6O5S2
|
1
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| 1 |
EC50 = 90 nM
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CP0130252
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4-{(S)-3-[1-(3,4-Dimethoxy-benzenesulfonyl)-piperidin-4-ylamino]-2-hydroxy-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
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C23H30N4O7S
|
1
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| 1 |
EC50 = 90 nM
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CP0403167
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3-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]benzoic acid
Show/Hide
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C23H22ClNO3
|
1
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| 1 |
EC50 = 91 nM
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CP0378013
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2-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoylamino)-pentanedioic acid
Show/Hide
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C26H34N4O9S
|
1
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| 1 |
EC50 = 92 nM
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CP0374195
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1-(4-fluorophenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C26H27FN4O2S
|
2
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| 1 |
EC50 = 92 nM
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| 2 |
Ki = 88 nM
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CP0417912
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2,5-dimethylbenzamide
Show/Hide
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C24H27N3O2
|
1
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| 1 |
EC50 = 95 nM
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CP0503582
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1-(3-Chloro-phenyl)-2-[1-methyl-2-(4-methyl-1H-indol-3-yl)-ethylamino]-ethanol
Show/Hide
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C20H23ClN2O
|
1
|
| 1 |
EC50 = 96 nM
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CP0388603
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1-(1-(5-methyl-6-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-phenoxypropan-2-ol
Show/Hide
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C27H30N4O2S
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2
|
| 1 |
EC50 = 96 nM
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| 2 |
Ki = 90 nM
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CP0388503
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5-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-2-(hydroxymethyl)phenol
Show/Hide
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C27H30N4O4S
|
2
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| 1 |
EC50 = 97 nM
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| 2 |
Ki = 620 nM
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CP0478306
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1-(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoyl)-pyrrolidine-2-carboxylic acid
Show/Hide
|
C26H34N4O7S
|
1
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| 1 |
EC50 = 98 nM
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CP0845333
|
Piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethyl]-phenyl}-amide dihydrochloride
Show/Hide
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C20H30Cl2N4O3S
|
1
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| 1 |
EC50 = 99 nM
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CP0428111
|
(R)-4-(4-(2-(2-(3-chlorophenyl)-2-hydroxyethylamino)ethyl)phenoxy)benzoic acid
Show/Hide
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C23H22ClNO4
|
1
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| 1 |
EC50 = 100 nM
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CP0429988
|
[3-[(2R)-2-[[(2R)-2-[3-(benzenesulfonylmethyl)phenyl]-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C27H30N2O6S2
|
1
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| 1 |
EC50 = 100 nM
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CP0851797
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(3-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
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| 1 |
EC50 = 100 nM
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CP0873012
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
|
| 1 |
EC50 = 100 nM
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CP0377223
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1-(2-isopropylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C29H34N4O2S
|
2
|
| 1 |
EC50 = 100 nM
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| 2 |
Ki = 64 nM
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CP0451500
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2-[[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]carbamoylamino]acetic acid
Show/Hide
|
C28H41N3O7
|
1
|
| 1 |
EC50 = 100 nM
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CP0917314
|
3-[3-(4-{[6-([(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino)hexyl]oxy}butyl)phenyl]imidazolidine-2,4-dione acetate
Show/Hide
|
C30H43N3O8
|
1
|
| 1 |
EC50 = 100 nM
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CP0851889
|
(R)-2-(3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)ureido)acetamide formate
Show/Hide
|
C29H44N4O8
|
1
|
| 1 |
EC50 = 100 nM
|
|
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CP0428927
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-methylthiazol-4-yl)acetamide
Show/Hide
|
C21H24N4O2S
|
1
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| 1 |
EC50 = 103 nM
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CP0447499
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-4-phenethylbenzamide
Show/Hide
|
C30H31N3O2
|
1
|
| 1 |
EC50 = 105 nM
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CP0388477
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(pyrimidin-2-yl)acetanilide
Show/Hide
|
C23H26N4O4
|
1
|
| 1 |
EC50 = 110 nM
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CP0545377
|
N-[3-[(1R)-1-hydroxy-2-[2-[[3-(hydroxymethyl)-2H-indazol-6-yl]oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C19H24N4O5S
|
1
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| 1 |
EC50 = 111 nM
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CP0388490
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1-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)-3-(3-(trifluoromethoxy)phenoxy)propan-2-ol
Show/Hide
|
C27H27F3N4O3S
|
2
|
| 1 |
EC50 = 113 nM
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| 2 |
Ki = 59 nM
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CP0144775
|
(4-{(R)-2-[(S)-2-Hydroxy-3-(4-hydroxy-3-methanesulfonylamino-phenoxy)-propylamino]-propyl}-phenoxymethyl)-phenyl-phosphinic acid
Show/Hide
|
C26H33N2O8PS
|
1
|
| 1 |
EC50 = 120 nM
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CP0397942
|
(R)-1-((S)-3-Chloro-phenyl)-2-[2-(7-methoxy-1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C20H23ClN2O2
|
1
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| 1 |
EC50 = 120 nM
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CP0431167
|
(S)-1-[(2-{1-[(1-Benzylimidazol-2-yl)acetyl]-1,2,3,4-tetrahydroquinolin-6-yl}ethyl)-amino]-3-phenoxy-2-propanol
Show/Hide
|
C32H36N4O3
|
1
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| 1 |
EC50 = 120 nM
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CP0407832
|
(1R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-3-yl)thiazol-4-yl)phenoxy)ethylamino)ethanol
Show/Hide
|
C23H22N4O2S
|
1
|
| 1 |
EC50 = 120 nM
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CP0097140
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4-{(S)-2-Hydroxy-3-[1-(4-methoxy-benzenesulfonyl)-piperidin-4-ylamino]-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
|
C22H28N4O6S
|
1
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| 1 |
EC50 = 120 nM
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CP0246496
|
N-[5-[(1R)-2-[(1-dibenzofuran-2-ylsulfonylpiperidin-4-yl)amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H29N3O7S2
|
1
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| 1 |
EC50 = 120 nM
|
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CP0372784
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2,2-diphenylacetanilide
Show/Hide
|
C31H32N2O4
|
1
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| 1 |
EC50 = 120 nM
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|
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CP0388508
|
1-(4-methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
EC50 = 120 nM
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| 2 |
Ki = 460 nM
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CP0417833
|
(R)-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
|
C22H27N5O2
|
1
|
| 1 |
EC50 = 123 nM
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CP0859375
|
3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]-ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}benzenesulfonamideacetate salt
Show/Hide
|
C26H40N2O9S
|
1
|
| 1 |
EC50 = 125.89 nM
|
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CP0492697
|
1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-isobutyl-urea
Show/Hide
|
C26H38N4O6S
|
1
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| 1 |
EC50 = 126 nM
|
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CP0437478
|
3-[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]anilino]-3-oxopropanoic acid
Show/Hide
|
C23H30N4O7S
|
1
|
| 1 |
EC50 = 130 nM
|
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CP0372411
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-benzylimidazol-2-yl)-acetanilide
Show/Hide
|
C29H32N4O3
|
1
|
| 1 |
EC50 = 130 nM
|
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CP0378399
|
(R)-N-(5-(2-(4-(2-ethylthiazol-4-yl)phenethylamino)-1-hydroxyethyl)-2-chlorophenyl)methanesulfonamide
Show/Hide
|
C22H26ClN3O3S2
|
1
|
| 1 |
EC50 = 130 nM
|
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CP0409487
|
1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-phenyl-urea
Show/Hide
|
C28H34N4O6S
|
1
|
| 1 |
EC50 = 135 nM
|
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CP0412417
|
(2R)-2-[4-[2-[[(2S)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]propanoic acid
Show/Hide
|
C19H23NO4
|
1
|
| 1 |
EC50 = 136 nM
|
|
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CP0377688
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(isoquinolin-3-yl)acetanilide
Show/Hide
|
C28H29N3O4
|
1
|
| 1 |
EC50 = 140 nM
|
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CP0374199
|
1-(3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)phenyl)urea
Show/Hide
|
C27H30N6O3S
|
2
|
| 1 |
EC50 = 150 nM
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| 2 |
Ki = 37 nM
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CP0388525
|
5-(phenoxymethyl)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)oxazolidin-2-one
Show/Hide
|
C27H26N4O3S
|
1
|
| 1 |
EC50 = 150 nM
|
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CP0411906
|
1-(benzyl(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)amino)-3-phenoxypropan-2-ol
Show/Hide
|
C33H34N4O2S
|
1
|
| 1 |
EC50 = 150 nM
|
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CP0470421
|
N-(2-hydroxy-3-phenoxypropyl)-N-[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]acetamide
Show/Hide
|
C28H30N4O3S
|
1
|
| 1 |
EC50 = 150 nM
|
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CP0470422
|
2-(phenoxymethyl)-4-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)morpholine
Show/Hide
|
C28H30N4O2S
|
1
|
| 1 |
EC50 = 150 nM
|
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CP0500002
|
1-((2-hydroxyethyl)(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)amino)-3-phenoxypropan-2-ol
Show/Hide
|
C28H32N4O3S
|
1
|
| 1 |
EC50 = 150 nM
|
|
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CP0501001
|
1-(methyl(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)amino)-3-phenoxypropan-2-ol
Show/Hide
|
C27H30N4O2S
|
1
|
| 1 |
EC50 = 150 nM
|
|
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CP0501002
|
1-((3-morpholinopropyl)(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl)amino)-3-phenoxypropan-2-ol
Show/Hide
|
C33H41N5O3S
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
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CP0526492
|
N-(2-methoxy-3-phenoxypropyl)-N-methyl-1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-amine
Show/Hide
|
C28H32N4O2S
|
1
|
| 1 |
EC50 = 150 nM
|
|
|
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CP0386625
|
methyl 3-[3-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethylamino]phenyl]benzoate
Show/Hide
|
C24H25ClN2O3
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
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CP0850324
|
2-(Hydroxymethyl)-4-{(1R)-1-hydroxy-2-[(6-{4-[3-(piperidin-1-ylsulfonyl)phenyl]butoxy}hexyl)amino]ethyl}phenol
Show/Hide
|
C32H50N2O8S
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
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CP0851886
|
(R)-1-ethyl-3-(3-(4-(6-(2-hydroxy-2-(4-hydroxy-3-(hydroxymethyl)phenyl)ethylamino)hexyloxy)butyl)phenyl)urea acetate
Show/Hide
|
C30H47N3O7
|
1
|
| 1 |
EC50 = 158.49 nM
|
|
|
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CP0429984
|
[3-[(2R)-2-[[(2R)-2-(3-benzamidophenyl)-2-hydroxyethyl]amino]propyl]-1H-indol-7-yl] methanesulfonate
Show/Hide
|
C27H29N3O5S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
|
CP0858640
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(3-methoxyphenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O3S
|
1
|
| 1 |
EC50 = 160 nM
|
|
|
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CP0897966
|
N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}-2-methylpropyl)phenyl]N-2-Methoxy-ethylaminesulfamide; 2HCl
Show/Hide
|
C20H32Cl2N4O4S
|
1
|
| 1 |
EC50 = 165 nM
|
|
|
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CP0870184
|
5-(4-{4-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-piperidin-1-yl}-benzyl)-thiazolidine-2,4-dione
Show/Hide
|
C23H26ClN3O3S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0309024
|
(R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C19H21N3O2S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
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CP0371720
|
(R)-2-(2-(4-(2-ethylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C20H23N3O2S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0844962
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-methoxycarbonylphenyl)thiourea hydrochloride
Show/Hide
|
C26H30ClN3O4S
|
1
|
| 1 |
EC50 = 170 nM
|
|
|
|
CP0373719
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(5-methyl-4H-1,2,4-triazol-3-yl)acetamide
Show/Hide
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C20H24N6O2
|
1
|
| 1 |
EC50 = 171 nM
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CP0428922
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-phenylthiazol-4-yl)acetamide
Show/Hide
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C26H26N4O2S
|
1
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| 1 |
EC50 = 174 nM
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CP0373737
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-2-carboxamide
Show/Hide
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C28H27N3O2
|
1
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| 1 |
EC50 = 179 nM
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CP0918992
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N'-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)phenyl]-N-methyl,N-cyclohexylsulfamide; 2HCl
Show/Hide
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C22H34Cl2N4O3S
|
1
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| 1 |
EC50 = 180 nM
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CP0412419
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(2S)-2-[4-[2-[[(2S)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]propanoic acid
Show/Hide
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C19H23NO4
|
1
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| 1 |
EC50 = 181 nM
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CP0373738
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-3-carboxamide
Show/Hide
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C28H27N3O2
|
1
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| 1 |
EC50 = 184 nM
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CP0893925
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(R)-2-(4-Fluorophenyl)-N-(4-(((2S,5R)-5-((R)-hydroxy(phenyl)-methyl)pyrrolidin-2-yl)methyl)phenyl)-5,6-dihydro-4Hcyclopenta[d]thiazole-4-carboxamide
Show/Hide
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C31H30FN3O2S
|
1
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| 1 |
EC50 = 186 nM
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CP0403918
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1-(9H-Carbazol-4-yloxy)-3-{[1-(3,3,3-trifluoro-propyl)-piperidin-4-ylmethyl]-amino}-propan-2-ol
Show/Hide
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C24H30F3N3O2
|
1
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| 1 |
EC50 = 187 nM
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CP0373740
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)biphenyl-4-carboxamide
Show/Hide
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C28H27N3O2
|
1
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| 1 |
EC50 = 187 nM
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CP0380788
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N-[4-[[3-[4-[[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]sulfamoyl]phenyl]-1,2,4-oxadiazol-5-yl]methyl]phenyl]acetamide
Show/Hide
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C32H32N6O5S
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1
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| 1 |
EC50 = 190 nM
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CP0847406
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3-(4-{[6-({(2R)-2-[3-(Formylamino)-4-hydroxyphenyl]-2-hydroxyethyl}amino)hexyl]oxy}butyl)benzenesulfonamide fumarate salt
Show/Hide
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C29H41N3O10S
|
1
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| 1 |
EC50 = 199.53 nM
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CP0884853
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3-[2-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione
Show/Hide
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C28H39N3O6
|
1
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| 1 |
EC50 = 199.53 nM
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CP0403527
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-3-methanesulfonylamino-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid octylamide
Show/Hide
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C32H51N5O6S
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1
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| 1 |
EC50 = 200 nM
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CP0443473
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(6-benzyloxy-2-pyridyl)-acetanilide
Show/Hide
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C31H33N3O4
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1
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| 1 |
EC50 = 200 nM
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CP0378404
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(R)-1-(pyridin-3-yl)-2-(2-(4-(2-(trifluoromethyl)thiazol-4-yl)phenoxy)ethylamino)ethanol
Show/Hide
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C19H18F3N3O2S
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1
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| 1 |
EC50 = 200 nM
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CP0378406
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(R)-2-(2-(4-(oxazol-5-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C18H19N3O3
|
1
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| 1 |
EC50 = 200 nM
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CP0861820
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-methoxyphenyl)thiourea hydrochloride
Show/Hide
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C25H30ClN3O3S
|
1
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| 1 |
EC50 = 200 nM
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CP0373730
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-pyrazol-1-yl)acetamide
Show/Hide
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C20H23N5O2
|
1
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| 1 |
EC50 = 218 nM
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CP0451328
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4-(4-{(R)-2-Hydroxy-2-[4-hydroxy-3-(methanesulfonyl-methyl-amino)-phenyl]-ethylamino}-piperidin-1-yl)-benzoic acid
Show/Hide
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C22H29N3O6S
|
1
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| 1 |
EC50 = 220 nM
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CP0460947
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4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-benzoic acid
Show/Hide
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C21H27N3O6S
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1
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| 1 |
EC50 = 220 nM
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CP0039165
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(S)-1-((R)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
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C19H21ClN2O
|
1
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| 1 |
EC50 = 220 nM
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CP0378415
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(R)-2-(2-(4-(2-(benzyloxymethyl)oxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C26H27N3O4
|
1
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| 1 |
EC50 = 220 nM
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CP0428923
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-phenylacetamide
Show/Hide
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C23H25N3O2
|
1
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| 1 |
EC50 = 225 nM
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CP0847475
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N-[2-Hydroxy-5-(1-hydroxy-2-{1-[4-(2-imino-5-oxo-imidazolidin-4-ylmethyl)-phenyl]-piperidin-4-ylamino}-ethyl)-phenyl]-methanesulfonamide
Show/Hide
|
C24H32N6O5S
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1
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| 1 |
EC50 = 230 nM
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CP0457905
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(R)-N-(5-(2-(4-(2-methylthiazol-4-yl)phenethylamino)-1-hydroxyethyl)-2-chlorophenyl)methanesulfonamide
Show/Hide
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C21H24ClN3O3S2
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1
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| 1 |
EC50 = 230 nM
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CP0844967
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(S)-1-(4-Bromophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27BrClN3O2S
|
1
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| 1 |
EC50 = 230 nM
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CP0873014
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(S)-1-(4-Fluorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClFN3O2S
|
1
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| 1 |
EC50 = 230 nM
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CP0373304
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(2R)-2-[4-[2-[[(2R)-2-hydroxy-2-phenylethyl]amino]ethyl]phenoxy]propanoic acid
Show/Hide
|
C19H23NO4
|
1
|
| 1 |
EC50 = 235 nM
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CP0375498
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(R)-1-((S)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C19H21ClN2O
|
1
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| 1 |
EC50 = 240 nM
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CP0377700
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-naphthyl)acetanilide
Show/Hide
|
C29H30N2O4
|
1
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| 1 |
EC50 = 240 nM
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CP0373731
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(3-methyl-1H-pyrazol-1-yl)acetamide
Show/Hide
|
C21H25N5O2
|
1
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| 1 |
EC50 = 241 nM
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CP0490225
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4-(4-{2-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid 2,4-dichloro-benzylamide
Show/Hide
|
C30H36Cl2N4O4
|
1
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| 1 |
EC50 = 250 nM
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CP0875711
|
4-((1R)-2-{[6-({4-[3-(Cyclohexylsulfonyl)phenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
|
C33H51NO8S
|
1
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| 1 |
EC50 = 251.19 nM
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CP0532365
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3-[[4-[4-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]piperidin-1-yl]benzoyl]amino]propanoic acid
Show/Hide
|
C24H32N4O7S
|
1
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| 1 |
EC50 = 260 nM
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CP0428931
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)pyrazolo[1,5-a]pyridine-7-carboxamide
Show/Hide
|
C23H23N5O2
|
1
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| 1 |
EC50 = 261 nM
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CP0388475
|
1-(3-ethylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
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C28H32N4O2S
|
2
|
| 1 |
EC50 = 264 nM
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| 2 |
Ki = 63 nM
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CP0919819
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N'-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)phenyl]-N,N-dimethylsulfamide; 2HCl
Show/Hide
|
C17H26Cl2N4O3S
|
1
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| 1 |
EC50 = 265 nM
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CP0424781
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(S)-6-(4-(2-(3-(3,3-dibenzyl-2-oxoindolin-4-yloxy)-2-hydroxypropylamino)-2-methylpropyl)phenoxy)nicotinamide
Show/Hide
|
C41H42N4O5
|
1
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| 1 |
EC50 = 268.1 nM
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CP0438189
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(4-{4-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-piperidin-1-yl}-phenyl)-acetic acid
Show/Hide
|
C22H29N3O6S
|
1
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| 1 |
EC50 = 270 nM
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CP0851807
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(S)-1-(3-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27Cl2N3O2S
|
1
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| 1 |
EC50 = 270 nM
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CP0861819
|
(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-methoxyphenyl)thiourea hydrochloride
Show/Hide
|
C25H30ClN3O3S
|
1
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| 1 |
EC50 = 270 nM
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CP0388089
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-benzylimidazol-4-yl)-acetanilide
Show/Hide
|
C29H32N4O3
|
1
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| 1 |
EC50 = 280 nM
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CP0861800
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(S)-1-(4-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
|
C24H27Cl2N3O2S
|
1
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| 1 |
EC50 = 280 nM
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CP0373727
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-1H-benzo[d]imidazole-2-carboxamide
Show/Hide
|
C23H23N5O2
|
1
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| 1 |
EC50 = 283 nM
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CP0457023
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hexyl-[[4-[2-[[(2S)-2-hydroxy-3-[(8-hydroxy-2-oxo-3,4-dihydro-1H-quinolin-5-yl)oxy]propyl]amino]ethyl]phenoxy]methyl]phosphinic acid
Show/Hide
|
C27H39N2O7P
|
1
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| 1 |
EC50 = 290 nM
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CP0496221
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4-(4-{2-[(S)-3-(6-Amino-pyridin-3-yloxy)-2-hydroxy-propylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid octylamide
Show/Hide
|
C30H48N6O3
|
1
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| 1 |
EC50 = 290 nM
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CP0493505
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1-(9H-Carbazol-4-yloxy)-3-[(1-isopropyl-piperidin-4-ylmethyl)-amino]-propan-2-ol
Show/Hide
|
C24H33N3O2
|
1
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| 1 |
EC50 = 290 nM
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CP0378403
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(R)-2-(2-(4-(2-cyclopentylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C23H27N3O2S
|
1
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| 1 |
EC50 = 290 nM
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CP0372413
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C24H27N3O4
|
2
|
| 1 |
EC50 = 290 nM
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| 2 |
EC50 = 2700 nM
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CP0447473
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-methylbenzamide
Show/Hide
|
C23H25N3O2
|
1
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| 1 |
EC50 = 297 nM
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CP0503252
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1-chloro-3-[(1R)-2-[2-[4-(dimethylsulfamoylamino)phenyl]ethylamino]-1-hydroxyethyl]benzene
Show/Hide
|
C18H24ClN3O3S
|
1
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| 1 |
EC50 = 299 nM
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CP0406160
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1-[4-(4-{[(S)-2-Hydroxy-3-(4-hydroxy-3-methyl-phenoxy)-propylamino]-methyl}-piperidine-1-sulfonyl)-phenyl]-3-octyl-urea
Show/Hide
|
C31H48N4O6S
|
1
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| 1 |
EC50 = 306 nM
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CP0378412
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(R)-2-(2-(4-(5-methyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C19H21N3O3
|
1
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| 1 |
EC50 = 309 nM
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CP0464883
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-methyl-2H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]cyclopentanesulfonamide
Show/Hide
|
C23H30N4O4S
|
1
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| 1 |
EC50 = 309 nM
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CP0372204
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(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(4,6-dimethyl-2-pyridyl)-acetanilide
Show/Hide
|
C26H31N3O3
|
1
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| 1 |
EC50 = 310 nM
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CP0412042
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2-hydroxy-5-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzoic acid
Show/Hide
|
C27H28N4O5S
|
2
|
| 1 |
EC50 = 310 nM
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| 2 |
Ki = 3500 nM
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CP0455408
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2-[3-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]phenyl]acetic acid
Show/Hide
|
C19H23ClN2O3
|
1
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| 1 |
EC50 = 316.23 nM
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CP0847408
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3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N-isopropylbenzenesulfonamide acetate salt
Show/Hide
|
C30H48N2O8S
|
1
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| 1 |
EC50 = 316.23 nM
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CP0850210
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3-(3-{[7-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)heptyl]oxy}propyl)benzenesulfonamide sulfamate salt
Show/Hide
|
C25H41N3O9S2
|
1
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| 1 |
EC50 = 316.23 nM
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CP0924345
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N-(3-{[(2-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}ethyl)oxy]methyl}phenyl)urea Acetate salt
Show/Hide
|
C27H41N3O8
|
1
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| 1 |
EC50 = 316.23 nM
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CP0917316
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1-[3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)hexyl]oxy}butyl)phenyl]-2,4-imidazolidinedione acetate salt
Show/Hide
|
C30H43N3O8
|
1
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| 1 |
EC50 = 316.23 nM
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CP0898259
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4-((1R)-2-{[6-({4-[3-(Cyclopentylsulfonyl)-5-methylphenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetic acid salt
Show/Hide
|
C33H51NO8S
|
1
|
| 1 |
EC50 = 316.23 nM
|
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CP0399928
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1-(9H-Carbazol-4-yloxy)-3-[(1-pentyl-piperidin-4-ylmethyl)-amino]-propan-2-ol
Show/Hide
|
C26H37N3O2
|
1
|
| 1 |
EC50 = 319 nM
|
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CP0858641
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-sulfamoylphenyl)thiourea hydrochloride
Show/Hide
|
C24H29ClN4O4S2
|
1
|
| 1 |
EC50 = 320 nM
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CP0891546
|
(S)-N-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)benzamide hydrochloride
Show/Hide
|
C24H27ClN2O3
|
1
|
| 1 |
EC50 = 330 nM
|
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CP0433202
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N-[3-[(1R)-2-[2-[(3-tert-butyl-2H-indazol-6-yl)oxy]ethylamino]-1-hydroxyethyl]phenyl]methanesulfonamide
Show/Hide
|
C22H30N4O4S
|
1
|
| 1 |
EC50 = 338 nM
|
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CP0858644
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-nitrophenyl)thiourea hydrochloride
Show/Hide
|
C24H27ClN4O4S
|
1
|
| 1 |
EC50 = 340 nM
|
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CP0150115
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N-[5-[(1R)-2-[[1-(4-butoxyphenyl)sulfonylpyrrolidin-3-yl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C23H33N3O7S2
|
1
|
| 1 |
EC50 = 360 nM
|
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CP0375775
|
(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-methoxyphenyl)acetanilide
Show/Hide
|
C26H30N2O5
|
1
|
| 1 |
EC50 = 360 nM
|
|
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CP0885471
|
N-[(R)-5-(2-{1-[4-(2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethoxy)-2-hydroxy-phenyl]-benzenesulfonamide
Show/Hide
|
C29H32N4O7S2
|
1
|
| 1 |
EC50 = 380 nM
|
|
|
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CP0504897
|
1-(9H-Carbazol-4-yloxy)-3-{[1-(naphthalene-2-sulfonyl)-piperidin-4-ylmethyl]-amino}-propan-2-ol
Show/Hide
|
C31H33N3O4S
|
1
|
| 1 |
EC50 = 380 nM
|
|
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CP0388092
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(3-methyl-2-pyridyl)acetanilide
Show/Hide
|
C25H29N3O3
|
1
|
| 1 |
EC50 = 390 nM
|
|
|
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CP0390982
|
4-[2-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]ethoxymethyl]benzenesulfonamide
Show/Hide
|
C24H36N2O7S
|
1
|
| 1 |
EC50 = 398.11 nM
|
|
|
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CP0499227
|
3-[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]-1H-pyrimidine-2,4-dione
Show/Hide
|
C29H39N3O6
|
1
|
| 1 |
EC50 = 398.11 nM
|
|
|
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CP0875710
|
4-((1R)-2-{[6-({4-[3-(3-Cyclopenten-1-ylsulfonyl)phenyl]butyl}oxy)hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
|
C32H47NO8S
|
1
|
| 1 |
EC50 = 398.11 nM
|
|
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CP0875712
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4-{(1R)-2-[(6-{4-[4-(Cyclopentylsulfonyl)phenyl]butoxy}hexyl)amino]-1-hydroxyethyl}-2-(hydroxymethyl)phenol acetate salt
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C32H49NO8S
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1
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| 1 |
EC50 = 398.11 nM
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CP0528758
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[2-(4-methoxyphenyl)ethylamino]propoxy]phenyl]methanesulfonamide
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C19H26N2O6S
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1
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| 1 |
EC50 = 400 nM
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CP0916906
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N'-[5-(4-{4-[(S)-2-Hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-piperidin-1-yl}-benzylidene)-4-oxo-4,5-dihydro-thiazol-2-yl]-N,N-dimethyl-guanidine
Show/Hide
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C27H34N6O4S
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1
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| 1 |
EC50 = 400 nM
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CP0858643
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(S)-1-(2-Chlorophenyl)-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)thiourea hydrochloride
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C24H27Cl2N3O2S
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1
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| 1 |
EC50 = 400 nM
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CP0404751
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(S)-N-(4-(2-(2-hydroxy-3-phenoxypropylamino)ethyl)phenyl)benzenesulfonamide
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C23H26N2O4S
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1
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| 1 |
EC50 = 410 nM
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CP0844961
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-phenylthiourea hydrochloride
Show/Hide
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C24H28ClN3O2S
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1
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| 1 |
EC50 = 440 nM
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CP0429908
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-3-(1-methyl-1H-benzo[d]imidazol-2-yl)propanamide
Show/Hide
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C26H29N5O2
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1
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| 1 |
EC50 = 454 nM
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CP0383868
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(1R)-1-(3-chlorophenyl)-2-[2-[4-(cyclohexylsulfamoylamino)phenyl]ethylamino]ethanol
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C22H30ClN3O3S
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1
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| 1 |
EC50 = 464 nM
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CP0844968
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(S)-1-Benzyl-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]-ethyl}phenyl)thiourea hydrochloride
Show/Hide
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C25H30ClN3O2S
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1
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| 1 |
EC50 = 470 nM
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CP0851798
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-iodophenyl)thiourea hydrochloride
Show/Hide
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C24H27ClIN3O2S
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1
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| 1 |
EC50 = 470 nM
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CP0504027
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(1-naphthyl)acetanilide
Show/Hide
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C29H30N2O4
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1
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| 1 |
EC50 = 470 nM
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CP0412715
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(R)-N-(5-(2-(4-(2-phenylthiazol-4-yl)phenethylamino)-1-hydroxyethyl)-2-methylphenyl)methanesulfonamide
Show/Hide
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C27H29N3O3S2
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1
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| 1 |
EC50 = 490 nM
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CP0851904
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(indol-3-yl)acetanilide
Show/Hide
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C27H29N3O4
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1
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| 1 |
EC50 = 490 nM
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CP0490952
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(R)-2-(3,5-diphenyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C32H31N5O2
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1
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| 1 |
EC50 = 498 nM
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CP0431469
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-thenyl)acetanilide
Show/Hide
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C23H26N2O4S
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1
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| 1 |
EC50 = 500 nM
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CP0871038
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2-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 501.19 nM
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CP0372199
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(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1H-imidazol-2-yl)acetanilide
Show/Hide
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C22H26N4O3
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1
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| 1 |
EC50 = 510 nM
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CP0873011
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(2-phenylethyl)thiourea hydrochloride
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C26H32ClN3O2S
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1
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| 1 |
EC50 = 510 nM
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CP0454126
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(R)-2-(2-(4-(oxazol-2-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C18H19N3O3
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1
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| 1 |
EC50 = 520 nM
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CP0372785
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-pyridyl)acetanilide
Show/Hide
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C24H27N3O4
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1
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| 1 |
EC50 = 520 nM
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CP0515540
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1-chloro-3-[(1R)-2-[2-[4-[[cyclohexyl(methyl)sulfamoyl]amino]phenyl]ethylamino]-1-hydroxyethyl]benzene
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C23H32ClN3O3S
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1
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| 1 |
EC50 = 537 nM
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CP0377701
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-thenyl)acetanilide
Show/Hide
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C23H26N2O4S
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1
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| 1 |
EC50 = 550 nM
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CP0454784
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8-Hydroxy-5-{2-hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-3,4-dihydro-1H-quinolin-2-one
Show/Hide
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C21H26N2O5
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1
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| 1 |
EC50 = 560 nM
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CP0431466
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-methoxyphenyl)acetanilide
Show/Hide
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C26H30N2O5
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1
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| 1 |
EC50 = 560 nM
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CP0378402
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(R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
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C24H23N3O2S
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1
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| 1 |
EC50 = 580 nM
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CP0452933
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(R)-2-(4,5-diphenyl-1H-pyrazol-1-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)acetamide
Show/Hide
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C32H31N5O2
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1
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| 1 |
EC50 = 580 nM
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CP0378408
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(R)-2-(2-(4-(2,5-dimethyloxazol-4-yl)phenoxy)ethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C20H23N3O3
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1
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| 1 |
EC50 = 606 nM
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CP0440315
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N-[4-[2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]ethyl]phenyl]piperidine-1-sulfonamide
Show/Hide
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C21H28ClN3O3S
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1
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| 1 |
EC50 = 617 nM
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CP0877391
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2-(Hydroxymethyl)-4-{(1R)-1-hydroxy-2-[(6-{4-[3-(morpholin-4-ylsulfonyl)phenyl]butoxy}hexyl)amino]ethyl}phenol acetate salt
Show/Hide
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C31H48N2O9S
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1
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| 1 |
EC50 = 630.96 nM
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CP0888635
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3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N,N-dimethylbenzenesulfonamide acetate salt
Show/Hide
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C29H46N2O8S
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1
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| 1 |
EC50 = 630.96 nM
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CP0851799
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-phenyl)-3-(4-methylphenyl)thiourea hydrochloride
Show/Hide
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C25H30ClN3O2S
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1
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| 1 |
EC50 = 650 nM
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CP0377697
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(quinolin-2-yl)acetanilide
Show/Hide
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C28H29N3O4
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1
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| 1 |
EC50 = 650 nM
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CP0855839
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N-[2-Chloro-5-(2-{1-[4-((R)-2,4-dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-phenyl]-methanesulfonamide
Show/Hide
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C24H29ClN4O5S2
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1
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| 1 |
EC50 = 660 nM
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CP0403861
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1-(9H-Carbazol-4-yloxy)-3-[(1-hexyl-piperidin-4-ylmethyl)-amino]-propan-2-ol
Show/Hide
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C27H39N3O2
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1
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| 1 |
EC50 = 665 nM
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CP0428929
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
Show/Hide
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C19H22N6O2
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1
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| 1 |
EC50 = 693 nM
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CP0387792
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(2-chlorophenyl)acetanilide
Show/Hide
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C25H27ClN2O4
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1
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| 1 |
EC50 = 740 nM
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CP0401348
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4-[[(2R)-2-[[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino]propyl]amino]benzoic acid
Show/Hide
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C18H21ClN2O3
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1
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| 1 |
EC50 = 794.33 nM
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CP0847407
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3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)-N-methylbenzenesulfonamide acetate salt
Show/Hide
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C28H44N2O8S
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1
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| 1 |
EC50 = 794.33 nM
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CP0708199
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Vilanterol
Show/Hide
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C26H37Cl2NO7
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1
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| 1 |
EC50 = 794.33 nM
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CP0708202
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4-((1R)-2-{[6-({4-[3-(Cyclopentylsulfonyl)phenyl]butyl}oxy)-hexyl]amino}-1-hydroxyethyl)-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C32H49NO8S
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1
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| 1 |
EC50 = 794.33 nM
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CP0530060
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4-{2-Hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-benzene-1,2-diol
Show/Hide
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C18H23NO5
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1
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| 1 |
EC50 = 820 nM
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CP0167484
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4-{(S)-3-[1-(Benzo[1,2,5]thiadiazole-4-sulfonyl)-piperidin-4-ylamino]-2-hydroxy-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
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C21H24N6O5S2
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1
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| 1 |
EC50 = 850 nM
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CP0270078
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(S)-1-[1-(4-Butoxy-benzenesulfonyl)-piperidin-4-ylamino]-3-(9H-carbazol-4-yloxy)-propan-2-ol
Show/Hide
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C30H37N3O5S
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1
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| 1 |
EC50 = 850 nM
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CP0505610
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1-(9H-Carbazol-4-yloxy)-3-[(1-propyl-piperidin-4-ylmethyl)-amino]-propan-2-ol
Show/Hide
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C24H33N3O2
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1
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| 1 |
EC50 = 870 nM
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CP0375758
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-chlorophenyl)acetanilide
Show/Hide
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C25H27ClN2O4
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1
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| 1 |
EC50 = 890 nM
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CP0855866
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5-{4-[4-((R)-2-Hydroxy-2-pyridin-3-yl-ethylamino)-piperidin-1-yl]-benzyl}-thiazolidine-2,4-dione
Show/Hide
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C22H26N4O3S
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1
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| 1 |
EC50 = 900 nM
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CP0149971
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(S)-1-(9H-Carbazol-4-yloxy)-3-{1-[4-(2,2-dimethyl-propyl)-benzenesulfonyl]-piperidin-4-ylamino}-propan-2-ol
Show/Hide
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C31H39N3O4S
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1
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| 1 |
EC50 = 920 nM
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CP0932642
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N'-(5-{4-[4-((S)-2-Hydroxy-3-phenoxy-propylamino)-piperidin-1-yl]-benzylidene}-4-oxo-4,5-dihydro-thiazol-2-yl)-N,N-dimethyl-guanidine
Show/Hide
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C27H34N6O3S
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1
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| 1 |
EC50 = 940 nM
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CP0919873
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N'-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethoxy)phenyl]-N,N-dimethylsulfamide; 2HCl
Show/Hide
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C17H26Cl2N4O4S
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1
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| 1 |
EC50 = 943 nM
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CP0377695
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-amino-2-phenylacetanilide
Show/Hide
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C25H29N3O4
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1
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| 1 |
EC50 = 960 nM
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CP0377702
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-hydroxy-2-phenylacetanilide
Show/Hide
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C25H28N2O5
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1
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| 1 |
EC50 = 960 nM
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CP0373736
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(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-(2-(methylamino)thiazol-4-yl)acetamide
Show/Hide
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C21H25N5O2S
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1
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| 1 |
EC50 = 978 nM
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CP0463712
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4-{2-Hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-phenol
Show/Hide
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C18H23NO4
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1
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| 1 |
EC50 = 1000 nM
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CP0511407
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4-(4-{2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-ethyl}-phenylamino)-piperidine-1-carboxylic acid octylamide
Show/Hide
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C30H45ClN4O2
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1
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| 1 |
EC50 = 1020 nM
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CP0554964
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2-Fluoro-5-{2-hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-phenol
Show/Hide
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C18H22FNO4
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1
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| 1 |
EC50 = 1100 nM
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CP0097141
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N-[5-[(1R)-2-[[1-(4-butoxyphenyl)sulfonylazetidin-3-yl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C22H31N3O7S2
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1
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| 1 |
EC50 = 1100 nM
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CP0718208
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SID50106054
Show/Hide
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C20H18ClNNa2O7
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2
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| 1 |
EC50 = 1150 nM
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| 2 |
Ki = 20000 nM
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CP0384329
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(1R)-2-(4-(2-(pyridin-3-yl)thiazol-4-yl)phenethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C23H22N4OS
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1
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| 1 |
EC50 = 1190 nM
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CP0474045
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-chlorophenyl)acetanilide
Show/Hide
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C25H27ClN2O4
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1
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| 1 |
EC50 = 1200 nM
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CP0065062
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1-hydroxy-2-naphthoic acid;4-[1-hydroxy-2-[6-(4-phenylbutoxy)hexylamino]ethyl]-2-methylol-phenol
Show/Hide
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C25H37NO4
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1
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| 1 |
EC50 = 1258.93 nM
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CP0910906
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4-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 1258.93 nM
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CP0412716
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(R)-2-(4-(2-methylthiazol-4-yl)phenethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
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C19H21N3OS
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1
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| 1 |
EC50 = 1360 nM
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CP0847311
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4-Methyl-piperidine-1-sulfonic acid {4-[2-((R)-2-hydroxy-2-pyridin-3-yl-ethylamino)-ethoxy]-phenyl}-amide dihydrochloride
Show/Hide
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C21H32Cl2N4O4S
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1
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| 1 |
EC50 = 1360 nM
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CP0858642
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(S)-1-Cyclohexyl-3-(4-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}phenyl)thiourea hydrochloride
Show/Hide
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C24H34ClN3O2S
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1
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| 1 |
EC50 = 1400 nM
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CP0373735
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2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(4-(2-((R)-2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
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C23H29N5O2
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1
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| 1 |
EC50 = 1404 nM
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CP0889558
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N'-[4-(2-{[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino}ethyl)phenyl]-N-cyclohexylsulfamide; 2HCl
Show/Hide
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C21H32Cl2N4O3S
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1
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| 1 |
EC50 = 1460 nM
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CP0375759
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(3-pyridyl)acetanilide
Show/Hide
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C24H27N3O4
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1
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| 1 |
EC50 = 1500 nM
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CP0859379
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3-(4-{[6-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl}amino)-hexyl]oxy}butyl)benzenesulfonamide cinnamate salt
Show/Hide
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C34H46N2O8S
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1
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| 1 |
EC50 = 1584.89 nM
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CP0375760
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-phenylacetanilide
Show/Hide
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C25H28N2O4
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1
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| 1 |
EC50 = 1700 nM
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CP0387797
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(S)-4'-(2-{[2-Hydroxy-3-(4-hydroxyphenoxy)propyl]amino}ethyl)-2-(4-methoxyphenyl)acetanilide
Show/Hide
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C26H30N2O5
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1
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| 1 |
EC50 = 1700 nM
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CP0861821
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(S)-1-(4-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)-3-phenylurea hydrochloride
Show/Hide
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C24H28ClN3O3
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1
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| 1 |
EC50 = 1900 nM
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CP0850325
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3-{6-[4-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)butoxy]hexyl}benzenesulfonamide acetate salt
Show/Hide
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C27H42N2O8S
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1
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| 1 |
EC50 = 1995.26 nM
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CP0853673
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4-[(1R)-2-({6-[4-(1,1-Dioxo-2,3-dihydro-1-benzothien-6-yl)butoxy]hexyl}amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol acetate salt
Show/Hide
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C29H43NO8S
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1
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| 1 |
EC50 = 1995.26 nM
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CP0383039
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4-[3-(tert-butylamino)-2-hydroxypropoxy]-2,3-dihydro-1H-1,3-benzodiazol-2-one hydrochloride
Show/Hide
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C14H21N3O3
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1
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| 1 |
EC50 = 2000 nM
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CP0525995
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3-{2-Hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-phenol
Show/Hide
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C18H23NO4
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1
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| 1 |
EC50 = 2000 nM
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CP0861826
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(S)-N-Phenyl-4-{2-[(2-hydroxy-3-phenoxypropyl)amino]-ethyl}benzenesulfonamide hydrochloride
Show/Hide
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C23H27ClN2O4S
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1
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| 1 |
EC50 = 2000 nM
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CP0463701
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4-{2-Hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-1,3-dihydro-benzoimidazol-2-one
Show/Hide
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C19H23N3O4
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1
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| 1 |
EC50 = 2200 nM
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CP0378400
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(R)-2-(4-(2-ethylthiazol-4-yl)phenethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C20H23N3OS
|
1
|
| 1 |
EC50 = 2250 nM
|
|
|
|
CP0388502
|
3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzoic acid
Show/Hide
|
C27H28N4O4S
|
2
|
| 1 |
EC50 = 2410 nM
|
|
|
| 2 |
Ki = 2646 nM
|
|
|
|
CP0481594
|
[3-[4-[6-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(hydroxymethyl)phenyl]ethyl]amino]hexoxy]butyl]phenyl]methanesulfonamide
Show/Hide
|
C26H40N2O6S
|
1
|
| 1 |
EC50 = 2511.89 nM
|
|
|
|
CP0871071
|
3-(5-{[5-({(2R)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)pentyl]oxy}pentyl)benzenesulfonamide acetate salt
Show/Hide
|
C27H42N2O8S
|
1
|
| 1 |
EC50 = 2511.89 nM
|
|
|
|
CP0853672
|
4-[(1R)-2-({6-[4-(1,1-Dioxido-3,4-dihydro-2H-thiochromen-7-yl)butoxy]hexyl}amino)-1-hydroxyethyl]-2-(hydroxymethyl)phenol formate salt
Show/Hide
|
C29H43NO8S
|
1
|
| 1 |
EC50 = 2511.89 nM
|
|
|
|
CP0428930
|
(R)-3-(1H-benzo[d]imidazol-2-yl)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)propanamide
Show/Hide
|
C25H27N5O2
|
1
|
| 1 |
EC50 = 2647 nM
|
|
|
|
CP0378286
|
(R)-2-(4-(2-phenylthiazol-4-yl)phenethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C24H23N3OS
|
1
|
| 1 |
EC50 = 2740 nM
|
|
|
|
CP0410079
|
(S)-1-((S)-3-Chloro-phenyl)-2-[2-(1H-indol-3-yl)-1-methyl-ethylamino]-ethanol
Show/Hide
|
C19H21ClN2O
|
1
|
| 1 |
EC50 = 3300 nM
|
|
|
|
CP0373734
|
(R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenyl)-2-methyl-2-(1H-pyrazol-1-yl)propanamide
Show/Hide
|
C22H27N5O2
|
1
|
| 1 |
EC50 = 3768 nM
|
|
|
|
CP0853659
|
2-(Hydroxymethyl)-4-((1R)-1-hydroxy-2-{[6-({4-[4-(methylsulfonyl)phenyl]butyl}oxy)hexyl]amino}ethyl)phenol acetate salt
Show/Hide
|
C28H43NO8S
|
1
|
| 1 |
EC50 = 3981.07 nM
|
|
|
|
CP0371714
|
(R)-2-(4-(2-(trifluoromethyl)thiazol-4-yl)phenethylamino)-1-(pyridin-3-yl)ethanol
Show/Hide
|
C19H18F3N3OS
|
1
|
| 1 |
EC50 = 4490 nM
|
|
|
|
CP0530609
|
4-{2-Hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-2-hydroxymethyl-phenol
Show/Hide
|
C19H25NO5
|
1
|
| 1 |
EC50 = 4700 nM
|
|
|
|
CP0454884
|
2-Fluoro-4-{2-hydroxy-3-[2-(4-methoxy-phenyl)-ethylamino]-propoxy}-phenol
Show/Hide
|
C18H22FNO4
|
1
|
| 1 |
EC50 = 7900 nM
|
|
|
|
CP0851810
|
Phenyl (S)-(4-{2-[(2-hydroxy-3-phenoxypropyl)amino]ethyl}phenyl)carbamate hydrochloride
Show/Hide
|
C24H27ClN2O4
|
1
|
| 1 |
EC50 = 9300 nM
|
|
|
|
CP0509682
|
(1R)-1-(3-chlorophenyl)-2-[2-[4-[dimethylsulfamoyl(methyl)amino]phenyl]ethylamino]ethanol
Show/Hide
|
C19H26ClN3O3S
|
1
|
| 1 |
EC50 = 9900 nM
|
|
|
|
CP0863135
|
N-[3-(2-{1-[4-((R)-2,4-Dioxo-thiazolidin-5-ylmethyl)-phenyl]-piperidin-4-ylamino}-1-hydroxy-ethyl)-phenyl]-methanesulfonamide
Show/Hide
|
C24H30N4O5S2
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0433204
|
N-[3-[(1R)-1-hydroxy-2-[2-[(3-phenyl-1H-indazol-6-yl)oxy]ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C24H26N4O4S
|
1
|
| 1 |
EC50 > 10000 nM
|
|
|
|
CP0851800
|
(S)-1-Phenoxy-3-({2-[4-(phenylamino)phenyl]ethyl}amino)-2-propanol hydrochloride
Show/Hide
|
C23H27ClN2O2
|
1
|
| 1 |
EC50 = 12000 nM
|
|
|
|
CP0853349
|
4-[(1R)-1-Hydroxy-2-({6-[(2-hydroxyethyl)oxy]hexyl}amino)-ethyl]-2-(hydroxymethyl)phenol Acetate Salt
Show/Hide
|
C19H33NO7
|
1
|
| 1 |
EC50 = 12589.25 nM
|
|
|
|
CP0847405
|
3-(4-{[6-({(2S)-2-Hydroxy-2-[4-hydroxy-3-(hydroxymethyl)-phenyl]ethyl}amino)hexyl]oxy}butyl)benzenesulfonamide acetate salt
Show/Hide
|
C27H42N2O8S
|
1
|
| 1 |
EC50 = 19952.62 nM
|
|
|
|
CP0844965
|
(S)-2-Cyano-1-(4-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}phenyl)-3-phenylguanidine hydrochloride
Show/Hide
|
C25H28ClN5O2
|
1
|
| 1 |
EC50 = 33000 nM
|
|
|
|
CP0372205
|
(S)-N-Propyl-4'-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}-2-(1-benzylimidazol-2-yl)acetanilide
Show/Hide
|
C32H38N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372410
|
(S)-4'-(2-{[2-Hydroxy-3-(4-methylsulfonamidophenoxy)-propyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C25H30N4O5S
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0372412
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(1-benzyl-benzimidazol-2-yl)-acetanilide
Show/Hide
|
C33H34N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0382049
|
(S)-N-Methyl-4'-{2-[(2-hydroxy-3-phenoxypropyl)-amino]ethyl}-2-(1-benzylimidazol-2-yl)acetanilide
Show/Hide
|
C30H34N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0427161
|
(S)-4'-(2-{[2-Hydroxy-3-(carbazol-4-yloxy)propyl]-amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C26H28N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0431169
|
(S)-4'-{2-[(2-Hydroxy-3-phenoxypropyl)amino]ethyl}-2-(1-phenylimidazol-2-yl)-acetanilide
Show/Hide
|
C28H30N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0439488
|
(S)-4'-(2-{[2-Hydroxy-3-(carbazol-4-yloxy)propyl]-amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C30H30N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0439490
|
(S)-4'-(2-{[2-Hydroxy-3-(indol-4-yloxy)propyl]amino}-ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C25H27N5O4
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0443470
|
(S)-4'-(2-{[2-Hydroxy-3-phenoxypropyl]amino}ethyl)-2-(2-pyridyl)acetanilide
Show/Hide
|
C24H27N3O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0443472
|
(S)-4'-(2-{[2-Hydroxy-3-(2-benzimidazolon-4-yloxy)-propyl]amino}ethyl)-2-(2-pyridyl)-acetanilide
Show/Hide
|
C23H26N4O3
|
1
|
| 1 |
EC50 > 100000 nM
|
|
|
|
CP0373729
|
(R)-(1H-benzo[d]imidazol-2-yl)methyl 4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)ethyl)phenylcarbamate
Show/Hide
|
C24H25N5O3
|
1
|
| 1 |
EC50 > 10 nM
|
|
|
|
CP0870010
|
{4-[[4-(2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-ethyl)phenyl](methyl)-amino]phenoxy}acetic acid hydrochloride
Show/Hide
|
C25H28Cl2N2O4
|
1
|
| 1 |
EC50 > 100 nM
|
|
|
|
CP0371992
|
4-[(8S)-8-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-6,7,8,9-tetrahydro-5H-benzo[7]annulen-2-yl]benzoic Acid
Show/Hide
|
C26H26ClNO3
|
1
|
| 1 |
EC50 > 100 nM
|
|
|
|
CP0521941
|
4-[((8S)-8-{[(2R)-2-(3-Chlorophenyl)-2-hydroxyethyl]amino}-6,7,8,9-tetrahydro-5H-benzo[a]cyclohepten-2-yl)oxy]benzoic Acid
Show/Hide
|
C26H26ClNO4
|
1
|
| 1 |
EC50 > 100 nM
|
|
|
|
CP0036425
|
1-Hexyl-3-(4-{4-[(S)-2-hydroxy-3-(4-hydroxy-phenoxy)-propylamino]-piperidine-1-sulfonyl}-phenyl)-urea
Show/Hide
|
C27H40N4O6S
|
1
|
| 1 |
EC50 > 2000 nM
|
|
|
|
CP0044564
|
(S)-1-[1-(4-Butoxy-benzenesulfonyl)-pyrrolidin-3-ylamino]-3-(9H-carbazol-4-yloxy)-propan-2-ol
Show/Hide
|
C29H35N3O5S
|
1
|
| 1 |
EC50 > 2000 nM
|
|
|
|
CP0194012
|
(S)-1-[1-(4-Butoxy-benzenesulfonyl)-azetidin-3-ylamino]-3-(9H-carbazol-4-yloxy)-propan-2-ol
Show/Hide
|
C28H33N3O5S
|
1
|
| 1 |
EC50 > 2000 nM
|
|
|
|
CP0271556
|
4-{(S)-3-[1-(4-Butoxy-benzenesulfonyl)-piperidin-4-ylamino]-2-hydroxy-propoxy}-phenol
Show/Hide
|
C24H34N2O6S
|
1
|
| 1 |
EC50 > 2000 nM
|
|
|
|
CP0388476
|
N-[3-[2-hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenyl]acetamide
Show/Hide
|
C28H31N5O3S
|
2
|
| 1 |
IC50 = 107 nM
|
|
|
| 2 |
Ki = 85 nM
|
|
|
|
CP0388521
|
1-(4-(hydroxymethyl)phenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C27H30N4O3S
|
2
|
| 1 |
IC50 = 162 nM
|
|
|
| 2 |
Ki = 290 nM
|
|
|
|
CP0412043
|
3-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)-N-methylbenzamide
Show/Hide
|
C28H31N5O3S
|
2
|
| 1 |
IC50 = 402 nM
|
|
|
| 2 |
Ki = 331 nM
|
|
|
|
CP0388474
|
1-(4-ethylphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-ol
Show/Hide
|
C28H32N4O2S
|
2
|
| 1 |
IC50 = 8064 nM
|
|
|
| 2 |
Ki = 107 nM
|
|
|
|
CP0530624
|
N-[5-[(1R)-2-[[(1R)-1-[4-(difluoromethoxy)naphthalen-1-yl]-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C28H28F2N2O5S
|
1
|
| 1 |
Ki = 2 nM
|
|
|
|
CP0522849
|
N-[5-[(3R)-4-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-3-hydroxybutanoyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H32N2O7S
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0522847
|
N-[5-[(3R)-4-[[(1R)-1-[4-(difluoromethoxy)phenyl]-2-phenylethyl]amino]-3-hydroxybutanoyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H28F2N2O6S
|
1
|
| 1 |
Ki = 5 nM
|
|
|
|
CP0309177
|
N-[5-[(2S)-3-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H32N2O6S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0522850
|
N-[5-[(2S)-3-[[(1R)-2-(3-chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H31ClN2O6S
|
1
|
| 1 |
Ki = 6 nM
|
|
|
|
CP0452776
|
N-[5-[(2R)-3-[[(1S)-3-(2-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H33ClN2O6S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0490314
|
N-[5-[(2S)-3-[[(1R)-2-(2-chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H31ClN2O6S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0536377
|
(R)-N-(2-hydroxy-5-(1-hydroxy-2-(2-(4-methoxyphenyl)propan-2-ylamino)ethyl)phenyl)methanesulfonamide
Show/Hide
|
C19H26N2O5S
|
1
|
| 1 |
Ki = 7 nM
|
|
|
|
CP0405739
|
N-[5-[(1R)-2-[[(1R)-1-(1,3-benzodioxol-5-yl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C24H26N2O6S
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0461704
|
N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-hydroxy-4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C25H30N2O6S
|
1
|
| 1 |
Ki = 8 nM
|
|
|
|
CP0453349
|
(S)-N-(4-Chloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H28ClN3O6S
|
1
|
| 1 |
Ki = 8.8 nM
|
|
|
|
CP0573386
|
N-[5-[(1R)-2-[[(2R)-2-[4-(difluoromethoxy)phenyl]-1-phenylpropan-2-yl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C25H28F2N2O5S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0091266
|
N-[5-[(2S)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H32N2O6S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0538610
|
N-[5-[(2R)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-3-phenylpropyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H34N2O6S
|
1
|
| 1 |
Ki = 9 nM
|
|
|
|
CP0467189
|
N-[5-[(1R)-2-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C25H30N2O6S
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0303127
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(2-methyl-benzothiazol-5-yl)-propionamide
Show/Hide
|
C27H30N4O6S2
|
1
|
| 1 |
Ki = 11 nM
|
|
|
|
CP0467205
|
N-[5-[(2R)-3-[[(1S)-3-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H33ClN2O6S
|
1
|
| 1 |
Ki = 12 nM
|
|
|
|
CP0505802
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(4-phenoxy-phenyl)-propionamide
Show/Hide
|
C31H33N3O7S
|
1
|
| 1 |
Ki = 14 nM
|
|
|
|
CP0454829
|
N-[5-[(1R)-2-[[(1R)-1-(2,6-dimethoxypyridin-3-yl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C24H29N3O6S
|
1
|
| 1 |
Ki = 15 nM
|
|
|
|
CP0272451
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2,N-bis-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C26H31N3O7S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0343989
|
(S)-N-(3-Chloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H28ClN3O6S
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0490367
|
N-[5-[(2S)-3-[[(1R)-1-[3,4-bis(difluoromethoxy)phenyl]-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H28F4N2O6S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0317098
|
(S)-N-(3-Bromo-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H28BrN3O6S
|
1
|
| 1 |
Ki = 19 nM
|
|
|
|
CP0530870
|
N-[5-[(1R)-2-[1,1-bis(4-methoxyphenyl)ethylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C25H30N2O6S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0455464
|
4-[(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionylamino]-N-propyl-benzamide
Show/Hide
|
C29H36N4O7S
|
1
|
| 1 |
Ki = 20 nM
|
|
|
|
CP0184780
|
BMS-196085
Show/Hide
|
C24H26F2N2O5S
|
1
|
| 1 |
Ki = 21 nM
|
|
|
|
CP0039258
|
TMQ, 3',5'-Diiodo
Show/Hide
|
C17H17I2NO3
|
1
|
| 1 |
Ki = 21.38 nM
|
|
|
|
CP0111515
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-N-(4-hydroxy-phenyl)-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H29N3O7S
|
1
|
| 1 |
Ki = 23 nM
|
|
|
|
CP0530322
|
N-[5-[(2S)-3-[[(1R)-2-(4-chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H31ClN2O6S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0316404
|
(S)-N-(3,4-Dichloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H27Cl2N3O6S
|
1
|
| 1 |
Ki = 24 nM
|
|
|
|
CP0460930
|
N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[(1R)-1-(6-methoxypyridin-3-yl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C23H27N3O5S
|
1
|
| 1 |
Ki = 25 nM
|
|
|
|
CP0364380
|
N-[5-[(2R)-3-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C26H32N2O6S
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1
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| 1 |
Ki = 25 nM
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CP0540131
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N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[(1R)-1-(4-methoxynaphthalen-1-yl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C28H30N2O5S
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1
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| 1 |
Ki = 26 nM
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CP0225172
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-p-tolyl-propionamide
Show/Hide
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C26H31N3O6S
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1
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| 1 |
Ki = 28 nM
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CP0453931
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N-[5-[(2R)-3-[[(1S)-3-(3-chlorophenyl)-1-(3,4-dimethoxyphenyl)propyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H33ClN2O6S
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1
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| 1 |
Ki = 29 nM
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CP0453908
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1S)-1-(4-methoxyphenyl)-3-phenylpropyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C26H32N2O5S
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1
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| 1 |
Ki = 31 nM
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CP0487315
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N-[5-[2-[[1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H30N2O6S
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1
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| 1 |
Ki = 33 nM
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CP0421486
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N-[5-[(1R)-2-[[(1R)-1-[3,4-bis(difluoromethoxy)phenyl]-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H26F4N2O6S
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1
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| 1 |
Ki = 38 nM
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CP0420397
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N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[(1R)-1-naphthalen-1-yl-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C27H28N2O4S
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1
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| 1 |
Ki = 43 nM
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CP0460728
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N-[2-hydroxy-5-[1-hydroxy-2-[[1-(4-methoxyphenyl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C24H28N2O5S
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1
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| 1 |
Ki = 44 nM
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CP0372928
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(R)-N-((R)-2-Hydroxy-5-{1-hydroxy-2-[(R)-1-(4-methoxy-phenyl)-2-phenyl-ethylamino]-ethyl}-phenyl)-methanesulfonamide
Show/Hide
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C24H28N2O5S
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1
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| 1 |
Ki = 44 nM
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CP0287189
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(S)-N-(3,4-Dimethoxy-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
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C27H33N3O8S
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1
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| 1 |
Ki = 46 nM
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CP0288494
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(S)-N-(4-Chloro-2-fluoro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
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C25H27ClFN3O6S
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1
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| 1 |
Ki = 47 nM
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CP0092359
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(3,4,5-trichloro-phenyl)-propionamide
Show/Hide
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C25H26Cl3N3O6S
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1
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| 1 |
Ki = 51 nM
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CP0457458
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N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 53 nM
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CP0510848
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N-[5-[(2R)-3-[[(1S)-1-[3,4-bis(difluoromethoxy)phenyl]-3-phenylpropyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H30F4N2O6S
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1
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| 1 |
Ki = 59 nM
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CP0316290
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-m-tolyl-propionamide
Show/Hide
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C26H31N3O6S
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1
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| 1 |
Ki = 61 nM
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CP0461454
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N-[5-[(1R)-2-[[(1R)-1-[4-(difluoromethoxy)-3-methylphenyl]-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H28F2N2O5S
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1
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| 1 |
Ki = 69 nM
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CP0494752
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N-[5-[2-[[1-(2,4-dimethoxyphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H30N2O6S
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1
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| 1 |
Ki = 70 nM
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CP0401705
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N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[2-phenyl-1-(4-phenylmethoxyphenyl)ethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C30H32N2O5S
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1
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| 1 |
Ki = 70 nM
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CP0448524
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4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-benzamide
Show/Hide
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C24H27N3O5S
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1
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| 1 |
Ki = 70 nM
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CP0237359
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(S)-N-(3,5-Dichloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
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C25H27Cl2N3O6S
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1
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| 1 |
Ki = 71 nM
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CP0373313
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2-(4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-phenyl)-acetamide
Show/Hide
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C25H29N3O5S
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1
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| 1 |
Ki = 74 nM
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CP0289271
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(R)-(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-phenyl-acetamide
Show/Hide
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C24H27N3O6S
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1
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| 1 |
Ki = 77 nM
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CP0401220
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(R)-N-(5-(2-(bis(4-methoxyphenyl)methylamino)-1-hydroxyethyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C24H28N2O6S
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1
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| 1 |
Ki = 81 nM
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CP0506622
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(R)-N-(5-(2-(1,1-bis(4-(difluoromethoxy)phenyl)ethylamino)-1-hydroxyethyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C25H26F4N2O6S
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1
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| 1 |
Ki = 81 nM
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CP0468143
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N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[2-phenyl-1-[4-(2,2,2-trifluoroethoxy)phenyl]ethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C25H27F3N2O5S
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1
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| 1 |
Ki = 84 nM
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CP0454778
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4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-benzoic acid methyl ester
Show/Hide
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C25H28N2O6S
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1
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| 1 |
Ki = 85 nM
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CP0430949
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(S)-N-(4-Chloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-acetamide
Show/Hide
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C24H26ClN3O6S
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1
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| 1 |
Ki = 89 nM
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CP0267721
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(2S)-N-[4-(diethoxyphosphorylmethyl)phenyl]-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)propanamide
Show/Hide
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C30H40N3O9PS
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1
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| 1 |
Ki = 93 nM
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CP0535407
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N-[2-hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C25H30N2O5S
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1
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| 1 |
Ki = 110 nM
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CP0046414
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(2S)-N-[3-(aminomethyl)phenyl]-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)propanamide
Show/Hide
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C26H32N4O6S
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1
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| 1 |
Ki = 115 nM
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CP0465000
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4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-N-methyl-benzamide
Show/Hide
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C25H29N3O5S
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1
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| 1 |
Ki = 120 nM
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CP0565825
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N-[2-hydroxy-5-[1-hydroxy-2-[(2-phenyl-1-thiophen-3-ylethyl)amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C21H24N2O4S2
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1
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| 1 |
Ki = 129 nM
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CP0494740
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N-[5-[2-[[1-(3,4-dimethylphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H30N2O4S
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1
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| 1 |
Ki = 133 nM
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CP0536378
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N-[5-[(2S)-3-[[(1R)-1-(3,4-dichlorophenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C24H26Cl2N2O4S
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1
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| 1 |
Ki = 133 nM
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CP0279593
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(3-methoxy-phenyl)-propionamide
Show/Hide
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C26H31N3O7S
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1
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| 1 |
Ki = 142 nM
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CP0530720
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N-hydroxy-4-[(1R)-1-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-phenylethyl]benzamide
Show/Hide
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C24H27N3O6S
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1
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| 1 |
Ki = 147 nM
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CP0333937
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N-[5-[(2R)-3-[[(1S)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C26H32N2O6S
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1
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| 1 |
Ki = 150 nM
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CP0420759
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(R)-N-(5-(2-(bis(4-(difluoromethoxy)phenyl)methylamino)-1-hydroxyethyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C24H24F4N2O6S
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1
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| 1 |
Ki = 160 nM
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CP0522848
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N-[5-[(3R)-4-[[(1R)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-3-hydroxybutyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C27H34N2O6S
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1
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| 1 |
Ki = 160 nM
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CP0457459
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(S)-N-(5-(3-(1,3-bis(3,4-dimethoxyphenyl)propan-2-ylamino)-2-hydroxypropyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C29H38N2O8S
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1
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| 1 |
Ki = 170 nM
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CP0430646
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(S)-2-(4-Difluoromethoxy-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-N-phenyl-propionamide
Show/Hide
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C25H27F2N3O6S
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1
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| 1 |
Ki = 190 nM
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CP0467227
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(R)-N-(2-fluoro-6-hydroxy-3-(1-hydroxy-2-(2-(4-methoxyphenyl)propan-2-ylamino)ethyl)phenyl)methanesulfonamide
Show/Hide
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C19H25FN2O5S
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1
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| 1 |
Ki = 200 nM
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CP0453343
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N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[2-phenyl-1-[4-(trifluoromethoxy)phenyl]ethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C24H25F3N2O5S
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1
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| 1 |
Ki = 210 nM
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CP0528978
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N-[5-[(1R)-2-[[(1R)-1-(4-cyanophenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C24H25N3O4S
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1
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| 1 |
Ki = 210 nM
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CP0494792
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2-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2,2-bis-(4-methoxy-phenyl)-acetamide
Show/Hide
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C25H29N3O7S
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1
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| 1 |
Ki = 220 nM
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CP0420862
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N-[2-hydroxy-5-[1-hydroxy-2-[[1-(3-methoxyphenyl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C24H28N2O5S
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1
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| 1 |
Ki = 230 nM
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CP0534330
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N-[5-[2-[[1-(1-benzothiophen-5-yl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H26N2O4S2
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1
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| 1 |
Ki = 230 nM
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CP0511598
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(S)-N-[4-(2-Dimethylamino-ethoxy)-phenyl]-2-[(R)-2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
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C29H38N4O7S
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1
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| 1 |
Ki = 260 nM
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CP0553062
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N-[3-[(1R)-2-[[(1R)-1-[4-(difluoromethoxy)phenyl]-2-phenylethyl]amino]-1-hydroxyethyl]-2-fluoro-6-hydroxyphenyl]methanesulfonamide
Show/Hide
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C24H25F3N2O5S
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1
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| 1 |
Ki = 270 nM
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CP0425929
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N-[4-[(4-acetamidophenyl)-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]methyl]phenyl]acetamide
Show/Hide
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C26H30N4O6S
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1
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| 1 |
Ki = 300 nM
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CP0449878
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N-[5-[(1R)-2-[[(1S)-1-(3,4-dimethoxyphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C25H30N2O6S
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1
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| 1 |
Ki = 320 nM
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CP0464372
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N-[2-hydroxy-5-[1-hydroxy-2-(1-phenylheptan-2-ylamino)ethyl]phenyl]methanesulfonamide
Show/Hide
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C22H32N2O4S
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1
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| 1 |
Ki = 320 nM
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CP0399394
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(S)-N-(5-(3-(bis(4-(difluoromethoxy)phenyl)methylamino)-2-hydroxypropyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C25H26F4N2O6S
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1
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| 1 |
Ki = 340 nM
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CP0258516
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-N-(3-hydroxy-phenyl)-2-(4-methoxy-phenyl)-propionamide
Show/Hide
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C25H29N3O7S
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1
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| 1 |
Ki = 340 nM
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CP0406503
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N-[5-[2-(1,2-diphenylethylamino)-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
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C23H26N2O4S
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1
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| 1 |
Ki = 360 nM
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CP0510851
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(R)-N-(5-(4-(4-methoxybenzylamino)-3-hydroxybutanoyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
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C19H24N2O6S
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1
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| 1 |
Ki = 360 nM
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CP0284397
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2-[4-[[(2S)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)propanoyl]amino]phenoxy]acetic acid
Show/Hide
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C27H31N3O9S
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1
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| 1 |
Ki = 370 nM
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CP0343459
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(3,4,5-trimethoxy-phenyl)-propionamide
Show/Hide
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C28H35N3O9S
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1
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| 1 |
Ki = 370 nM
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CP0470423
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1-(4-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-ylamino)piperidin-1-yl)-3-phenoxypropan-2-ol
Show/Hide
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C26H27FN4O2S
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1
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| 1 |
Ki = 370 nM
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CP0493866
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(S)-N-(2-Chloro-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C25H28ClN3O6S
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1
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| 1 |
Ki = 380 nM
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CP0392741
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5-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-pentanoic acid
Show/Hide
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C20H28N2O4S
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1
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| 1 |
Ki = 390 nM
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CP0452808
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1S)-1-(3-methoxyphenyl)-3-phenylpropyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
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C26H32N2O5S
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1
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| 1 |
Ki = 390 nM
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CP0457421
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4-{(S)-1-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-1-phenylcarbamoyl-ethyl}-benzamide
Show/Hide
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C25H28N4O6S
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1
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| 1 |
Ki = 400 nM
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CP0511094
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N-[5-[2-[[1-(3,4-dichlorophenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C23H24Cl2N2O4S
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1
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| 1 |
Ki = 414 nM
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CP0377985
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N-[2-hydroxy-5-[1-hydroxy-2-[[1-(4-methylsulfonylphenyl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
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C24H28N2O6S2
|
1
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| 1 |
Ki = 440 nM
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CP0317085
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2-[3-[[(2S)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)propanoyl]amino]phenoxy]acetic acid
Show/Hide
|
C27H31N3O9S
|
1
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| 1 |
Ki = 450 nM
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CP0490366
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N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C25H30N2O5S
|
1
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| 1 |
Ki = 460 nM
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CP0447765
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N-[2-hydroxy-5-[1-hydroxy-2-[2-(4-methoxyphenyl)ethylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C18H24N2O5S
|
1
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| 1 |
Ki = 480 nM
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CP0502929
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N-[2-hydroxy-5-[1-hydroxy-2-[(7-hydroxy-1-phenylheptan-2-yl)amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C22H32N2O5S
|
1
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| 1 |
Ki = 480 nM
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CP0516073
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(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(3-phenoxy-phenyl)-propionamide
Show/Hide
|
C31H33N3O7S
|
1
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| 1 |
Ki = 490 nM
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CP0440458
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2-[4-[2-[[(2S)-2-hydroxy-3-phenoxypropyl]amino]ethoxy]phenoxy]acetic acid
Show/Hide
|
C19H23NO6
|
1
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| 1 |
Ki = 520 nM
|
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CP0449899
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N-[5-[2-[[1-(3,4-diethylphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C27H34N2O4S
|
1
|
| 1 |
Ki = 520 nM
|
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CP0320565
|
(S)-N-[3-(2-Dimethylamino-ethoxy)-phenyl]-2-[(R)-2-hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionamide
Show/Hide
|
C29H38N4O7S
|
1
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| 1 |
Ki = 520 nM
|
|
|
|
CP0514359
|
N-[5-[2-[2-(3,4-dimethoxyphenyl)ethylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C19H26N2O6S
|
1
|
| 1 |
Ki = 550 nM
|
|
|
|
CP0515029
|
6-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-7-phenyl-heptanoic acid methyl ester
Show/Hide
|
C23H32N2O6S
|
1
|
| 1 |
Ki = 570 nM
|
|
|
|
CP0496356
|
N-[2-hydroxy-5-[1-hydroxy-2-[(2-phenyl-1-pyridin-4-ylethyl)amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C22H25N3O4S
|
1
|
| 1 |
Ki = 700 nM
|
|
|
|
CP0373483
|
4-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-butyric acid
Show/Hide
|
C19H26N2O4S
|
1
|
| 1 |
Ki = 760 nM
|
|
|
|
CP0486224
|
1-(4-((5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-ylamino)methyl)piperidin-1-yl)-3-phenoxypropan-2-ol
Show/Hide
|
C27H29FN4O2S
|
1
|
| 1 |
Ki = 770 nM
|
|
|
|
CP0463560
|
4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-N,N-dimethyl-benzamide
Show/Hide
|
C26H31N3O5S
|
1
|
| 1 |
Ki = 800 nM
|
|
|
|
CP0144828
|
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-methanesulfonic acid
Show/Hide
|
C18H22ClNO5S
|
1
|
| 1 |
Ki = 806 nM
|
|
|
|
CP0420396
|
N-[5-[2-[[1-(4-fluorophenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C23H25FN2O4S
|
1
|
| 1 |
Ki = 836 nM
|
|
|
|
CP0510852
|
N-[5-[(3R)-4-[[(1R)-1-[4-(difluoromethoxy)phenyl]-2-phenylethyl]amino]-3-hydroxybutyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H30F2N2O5S
|
1
|
| 1 |
Ki = 880 nM
|
|
|
|
CP0472738
|
4-hydroxy-2-(2-hydroxy-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propoxy)benzoic acid
Show/Hide
|
C27H28N4O5S
|
1
|
| 1 |
Ki = 919 nM
|
|
|
|
CP0475885
|
(S)-2-(4-Bromo-phenyl)-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-N-phenyl-propionamide
Show/Hide
|
C24H26BrN3O5S
|
1
|
| 1 |
Ki = 950 nM
|
|
|
|
CP0502793
|
N-[5-[(1R)-2-[bis[4-(methoxymethyl)phenyl]methylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C26H32N2O6S
|
1
|
| 1 |
Ki = 980 nM
|
|
|
|
CP0463730
|
N-[2-hydroxy-5-[(1R)-1-hydroxy-2-[[1-(4-phenoxyphenyl)-2-phenylethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C29H30N2O5S
|
1
|
| 1 |
Ki = 990 nM
|
|
|
|
CP0497770
|
N-[2-hydroxy-5-[1-hydroxy-2-(2-phenylethylamino)ethyl]phenyl]methanesulfonamide
Show/Hide
|
C17H22N2O4S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0333936
|
N-[2-hydroxy-5-[(2R)-2-hydroxy-3-[[(1R)-1-(3-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C25H30N2O5S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0461726
|
N-[2-hydroxy-5-[2-hydroxy-3-[(4-methoxyphenyl)methylamino]propyl]phenyl]methanesulfonamide
Show/Hide
|
C18H24N2O5S
|
1
|
| 1 |
Ki = 1100 nM
|
|
|
|
CP0520584
|
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetic acid methyl ester
Show/Hide
|
C20H24ClNO4
|
1
|
| 1 |
Ki = 1150 nM
|
|
|
|
CP0406365
|
4-(3,5-Diiodo-4-methoxy-benzyl)-4,5,6,7-tetrahydro-thiazolo[5,4-c]pyridin-2-ylamine
Show/Hide
|
C14H15I2N3OS
|
1
|
| 1 |
Ki = 1479.11 nM
|
|
|
|
CP0453389
|
N-[5-[2-(1,3-diphenylpropan-2-ylamino)-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C24H28N2O4S
|
1
|
| 1 |
Ki = 1500 nM
|
|
|
|
CP0522320
|
N-[2-hydroxy-5-[1-hydroxy-2-[(4-methoxyphenyl)methylamino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C17H22N2O5S
|
1
|
| 1 |
Ki = 1550 nM
|
|
|
|
CP0533015
|
6-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-7-phenyl-heptanoic acid methylamide
Show/Hide
|
C23H33N3O5S
|
1
|
| 1 |
Ki = 1600 nM
|
|
|
|
CP0490365
|
(R)-N-(3-(2-(bis(4-methoxyphenyl)methylamino)-1-hydroxyethyl)-2-fluoro-6-hydroxyphenyl)methanesulfonamide
Show/Hide
|
C24H27FN2O6S
|
1
|
| 1 |
Ki = 1700 nM
|
|
|
|
CP0402240
|
3-[(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-propionylamino]-benzoic acid
Show/Hide
|
C26H29N3O8S
|
1
|
| 1 |
Ki = 1800 nM
|
|
|
|
CP0375479
|
2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-N-hydroxy-acetamide
Show/Hide
|
C19H23ClN2O4
|
1
|
| 1 |
Ki = 1960 nM
|
|
|
|
CP0416729
|
(R)-1-(3-Chloro-phenyl)-2-{(R)-2-[4-(2-hydroxy-ethoxy)-phenyl]-1-methyl-ethylamino}-ethanol
Show/Hide
|
C19H24ClNO3
|
1
|
| 1 |
Ki = 2140 nM
|
|
|
|
CP0529584
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-o-tolyl-propionamide
Show/Hide
|
C26H31N3O6S
|
1
|
| 1 |
Ki = 2200 nM
|
|
|
|
CP0534329
|
N-[2-hydroxy-5-[1-hydroxy-2-[[2-phenyl-1-(1,3-thiazol-2-yl)ethyl]amino]ethyl]phenyl]methanesulfonamide
Show/Hide
|
C20H23N3O4S2
|
1
|
| 1 |
Ki = 2400 nM
|
|
|
|
CP0483832
|
(S,R)-(-)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol
Show/Hide
|
C18H25BrN2O3
|
1
|
| 1 |
Ki = 2485 nM
|
|
|
|
CP0498228
|
N-[5-[(1R)-2-[bis(4-fluorophenyl)methylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C22H22F2N2O4S
|
1
|
| 1 |
Ki = 2800 nM
|
|
|
|
CP0492228
|
(R)-(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-acetamide
Show/Hide
|
C18H23N3O6S
|
1
|
| 1 |
Ki = 2910 nM
|
|
|
|
CP0303758
|
(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-(2-methoxy-phenyl)-propionamide
Show/Hide
|
C26H31N3O7S
|
1
|
| 1 |
Ki = 3100 nM
|
|
|
|
CP0497506
|
(S)-(S)-N-Benzyl-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-acetamide
Show/Hide
|
C25H29N3O6S
|
1
|
| 1 |
Ki = 3100 nM
|
|
|
|
CP0466591
|
(4-{2-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-ethyl}-phenoxy)-acetic acid methyl ester
Show/Hide
|
C20H26N2O7S
|
1
|
| 1 |
Ki = 3300 nM
|
|
|
|
CP0522697
|
1-(4-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)-1,4-diazepan-1-yl)-3-phenoxypropan-2-ol
Show/Hide
|
C26H27FN4O2S
|
1
|
| 1 |
Ki = 3300 nM
|
|
|
|
CP0480559
|
3-{2-[(R)-2-((S)-2-Hydroxy-3-phenoxy-propylamino)-propyl]-thiazol-5-yl}-propionic acid
Show/Hide
|
C18H24N2O4S
|
1
|
| 1 |
Ki = 3530 nM
|
|
|
|
CP0515032
|
N-[2-hydroxy-5-[1-hydroxy-2-(2-methylbutan-2-ylamino)ethyl]phenyl]methanesulfonamide
Show/Hide
|
C14H24N2O4S
|
1
|
| 1 |
Ki = 3700 nM
|
|
|
|
CP0457460
|
(R)-N-(5-(4-(4-methoxybenzylamino)-3-hydroxybutyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
|
C19H26N2O5S
|
1
|
| 1 |
Ki = 3700 nM
|
|
|
|
CP0498432
|
2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetamide
Show/Hide
|
C19H23ClN2O3
|
1
|
| 1 |
Ki = 3700 nM
|
|
|
|
CP0044877
|
1-(3,4,5-Trimethoxy-benzyl)-1,2,3,4-tetrahydro-isoquinoline-6,7-diol
Show/Hide
|
C19H23NO5
|
1
|
| 1 |
Ki = 3715.35 nM
|
|
|
|
CP0169504
|
N-[2-hydroxy-5-[1-hydroxy-2-(propan-2-ylamino)ethyl]phenyl]methanesulfonamide
Show/Hide
|
C12H20N2O4S
|
1
|
| 1 |
Ki = 4100 nM
|
|
|
|
CP0559749
|
N-[5-[2-[(1-cyclohexyl-2-phenylethyl)amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C23H32N2O4S
|
1
|
| 1 |
Ki = 4300 nM
|
|
|
|
CP0375808
|
N-[5-[(1R)-2-(benzhydrylamino)-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C22H24N2O4S
|
1
|
| 1 |
Ki = 5800 nM
|
|
|
|
CP0398915
|
(S)-(S)-N-Cyclohexyl-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-acetamide
Show/Hide
|
C24H33N3O6S
|
1
|
| 1 |
Ki = 7000 nM
|
|
|
|
CP0490315
|
N-[5-[3-[2-(3,4-dimethoxyphenyl)ethylamino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C20H28N2O6S
|
1
|
| 1 |
Ki = 7300 nM
|
|
|
|
CP0411907
|
1-(4-(5-(4-fluorophenyl)thieno[2,3-d]pyrimidin-4-yl)piperazin-1-yl)-3-phenoxypropan-2-ol
Show/Hide
|
C25H25FN4O2S
|
1
|
| 1 |
Ki = 8000 nM
|
|
|
|
CP0480421
|
2-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-N-phenyl-acetamide
Show/Hide
|
C17H21N3O5S
|
1
|
| 1 |
Ki = 8200 nM
|
|
|
|
CP0454617
|
4-{(R)-1-[(R)-2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-phenyl-ethyl}-benzoic acid
Show/Hide
|
C24H26N2O6S
|
1
|
| 1 |
Ki = 8600 nM
|
|
|
|
CP0492801
|
(S)-(S)-N-tert-Butyl-2-[2-hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-acetamide
Show/Hide
|
C22H31N3O6S
|
1
|
| 1 |
Ki = 9600 nM
|
|
|
|
CP0393025
|
(S)-N-((R)-2-Hydroxy-5-{1-hydroxy-2-[(S)-1-(4-methoxy-phenyl)-2-oxo-2-piperidin-1-yl-ethylamino]-ethyl}-phenyl)-methanesulfonamide
Show/Hide
|
C23H31N3O6S
|
1
|
| 1 |
Ki = 10000 nM
|
|
|
|
CP0483868
|
(S,R)-(-)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate
Show/Hide
|
C18H23BrN2O5
|
1
|
| 1 |
Ki = 10100 nM
|
|
|
|
CP0454267
|
(R,R)-(+)-1-(3-bromoisoxazol-5-yl)-2-{[2-(4-butoxyphenyl)-1-methylethyl]amino}ethanol
Show/Hide
|
C18H25BrN2O3
|
1
|
| 1 |
Ki = 10700 nM
|
|
|
|
CP0403638
|
N-[5-[2-(1-adamantylamino)-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C19H28N2O4S
|
1
|
| 1 |
Ki = 11000 nM
|
|
|
|
CP0404156
|
2-(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-malonic acid
Show/Hide
|
C20H22ClNO6
|
1
|
| 1 |
Ki = 11100 nM
|
|
|
|
CP0428592
|
N-[5-[2-(benzylamino)-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C16H20N2O4S
|
1
|
| 1 |
Ki = 12700 nM
|
|
|
|
CP0492458
|
(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)acetamide
Show/Hide
|
C18H23N3O6S
|
1
|
| 1 |
Ki = 14100 nM
|
|
|
|
CP0510853
|
(R)-N-(5-(4-amino-3-hydroxybutanoyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
|
C11H16N2O5S
|
1
|
| 1 |
Ki = 15000 nM
|
|
|
|
CP0439278
|
N-[5-(2-amino-1-hydroxyethyl)-2-hydroxyphenyl]methanesulfonamide
Show/Hide
|
C9H14N2O4S
|
1
|
| 1 |
Ki = 17000 nM
|
|
|
|
CP0490313
|
(R)-N-(5-(2-amino-1-hydroxyethyl)-2-hydroxyphenyl)methanesulfonamide
Show/Hide
|
C9H14N2O4S
|
1
|
| 1 |
Ki = 17000 nM
|
|
|
|
CP0518305
|
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid monoisopropyl ester
Show/Hide
|
C21H29ClNO5P
|
1
|
| 1 |
Ki = 18800 nM
|
|
|
|
CP0448909
|
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-methyl-phosphinic acid
Show/Hide
|
C19H25ClNO4P
|
1
|
| 1 |
Ki = 19900 nM
|
|
|
|
CP0457725
|
(R,R)-(+)-ethyl {4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]amino}propyl]phenoxy} acetate
Show/Hide
|
C18H23BrN2O5
|
1
|
| 1 |
Ki = 21800 nM
|
|
|
|
CP0439745
|
(S,R)-(-)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid
Show/Hide
|
C16H19BrN2O5
|
1
|
| 1 |
Ki = 22000 nM
|
|
|
|
CP0437626
|
(2R)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)-N-phenylacetamide
Show/Hide
|
C24H27N3O6S
|
1
|
| 1 |
Ki = 30000 nM
|
|
|
|
CP0500303
|
(S)-(S)-2-[2-Hydroxy-2-((R)-4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-2-(4-methoxy-phenyl)-N-methyl-N-phenyl-acetamide
Show/Hide
|
C25H29N3O6S
|
1
|
| 1 |
Ki = 33000 nM
|
|
|
|
CP0412982
|
4-(2-{(R)-2-[2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-thiazol-5-yl)-butyric acid
Show/Hide
|
C18H23ClN2O3S
|
1
|
| 1 |
Ki = 36500 nM
|
|
|
|
CP0464443
|
(4-{2-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-ethyl}-phenoxy)-acetic acid
Show/Hide
|
C19H24N2O7S
|
1
|
| 1 |
Ki = 49000 nM
|
|
|
|
CP0501137
|
(R,R)-(+)-{4-[2-{[2-(3-bromoisoxazol-5-yl)-2-hydroxyethyl]-amino}propyl]phenoxy}acetic acid
Show/Hide
|
C16H19BrN2O5
|
1
|
| 1 |
Ki > 50000 nM
|
|
|
|
CP0374790
|
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxymethyl)-phosphonic acid
Show/Hide
|
C18H23ClNO5P
|
1
|
| 1 |
Ki = 55300 nM
|
|
|
|
CP0403859
|
4-[(3,4,5-trimethoxyphenyl)methyl]-4,5,6,7-tetrahydro-[1,3]thiazolo[5,4-c]pyridin-2-amine
Show/Hide
|
C16H21N3O3S
|
1
|
| 1 |
Ki = 67608.3 nM
|
|
|
|
CP0409182
|
6-[2-Hydroxy-2-(4-hydroxy-3-methanesulfonylamino-phenyl)-ethylamino]-7-phenyl-heptanoic acid
Show/Hide
|
C22H30N2O6S
|
1
|
| 1 |
Ki = 87000 nM
|
|
|
|
CP0461669
|
(+/-)-N-[5-(2-bromo-1-hydroxyethyl)isoxazol-3-yl]methanesulfonamide
Show/Hide
|
C10H19N3O4S
|
1
|
| 1 |
Ki > 100000 nM
|
|
|
