Brief Information of the Compound and Protein
Compound Name
5-(4-{4-[2-Hydroxy-2-(2-oxo-1,2-dihydro-quinolin-5-yloxy)-ethylamino]-piperidin-1-yl}-benzyl)-thiazolidine-2,4-dione
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PubChem ID
CID: 44377535
Canonical SMILES
O=C1NC(=O)C(Cc2ccc(N3CCC(NC[C@H](O)Oc4cccc5nc(O)ccc45)CC3)cc2)S1
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Compound Formula C26H28N4O5S
Compound Structure
Protein Name
Beta-3 adrenergic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Adrenergic receptor
Uniprot ID
P13945
Gene Name
ADRB3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 13 nM
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