Compound ID |
Compound Name |
Compound Formula |
CP0423977
|
US10011588, Example 95
Show/Hide
|
C21H21F3N6O
|
1
|
1 |
IC50 = 1067 nM
|
|
|
CP0484845
|
US10011588, Example 96
Show/Hide
|
C21H21F3N6O2
|
1
|
1 |
IC50 = 1356 nM
|
|
|
CP0443731
|
US10011588, Example 83
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 = 1400 nM
|
|
|
CP0523876
|
US10011588, Example 68
Show/Hide
|
C24H28F3N3O3
|
1
|
1 |
IC50 = 1610 nM
|
|
|
CP0424029
|
US10011588, Example 27
Show/Hide
|
C20H22F3N3O3
|
1
|
1 |
IC50 = 2000 nM
|
|
|
CP0478640
|
US10011588, Example 110
Show/Hide
|
C22H24F3N7O
|
1
|
1 |
IC50 = 3549 nM
|
|
|
CP0424035
|
US10011588, Example 92
Show/Hide
|
C20H19ClF3N7O
|
1
|
1 |
IC50 = 5569 nM
|
|
|
CP0531577
|
US10011588, Example 19
Show/Hide
|
C19H17F3N6O2
|
1
|
1 |
IC50 = 6105 nM
|
|
|
CP0523880
|
US10011588, Example 21
Show/Hide
|
C20H21F3N2O4
|
1
|
1 |
IC50 = 6421 nM
|
|
|
CP0529223
|
US10011588, Example 82
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 = 7541 nM
|
|
|
CP0563274
|
US10011588, Example 71
Show/Hide
|
C19H19F4N3O2
|
1
|
1 |
IC50 = 7600 nM
|
|
|
CP0545685
|
US10011588, Example 119
Show/Hide
|
C20H21BrN6O2
|
1
|
1 |
IC50 = 7800 nM
|
|
|
CP0440532
|
US10011588, Example 103
Show/Hide
|
C20H19F4N7O
|
1
|
1 |
IC50 = 7897 nM
|
|
|
CP0443732
|
US10011588, Example 142
Show/Hide
|
C21H21F3N8O
|
1
|
1 |
IC50 = 8827 nM
|
|
|
CP0422561
|
US10011588, Example 99
Show/Hide
|
C20H17F5N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0422563
|
US10011588, Example 122
Show/Hide
|
C19H17ClF3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0423992
|
US10011588, Example 70
Show/Hide
|
C17H16ClF3N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0424030
|
US10011588, Example 57
Show/Hide
|
C22H22F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0424031
|
US10011588, Example 59
Show/Hide
|
C20H18ClF3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0424032
|
US10011588, Example 64
Show/Hide
|
C19H16F5N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0424033
|
US10011588, Example 75
Show/Hide
|
C20H19F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0424034
|
US10011588, Example 86
Show/Hide
|
C19H22F3N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0426337
|
US10011588, Example 108
Show/Hide
|
C21H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0426338
|
US10011588, Example 123
Show/Hide
|
C19H17F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0426370
|
US10011588, Example 127
Show/Hide
|
C19H16F5N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0435055
|
US10011588, Example 124
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0435056
|
US10011588, Example 131
Show/Hide
|
C20H17F5N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0438222
|
US10011588, Example 79
Show/Hide
|
C22H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0440533
|
US10689373, Example 105
Show/Hide
|
C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443726
|
US10011588, Example 11
Show/Hide
|
C21H20F3N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443727
|
US10011588, Example 43
Show/Hide
|
C19H18F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443733
|
US10011588, Example 148
Show/Hide
|
C21H18ClF3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443734
|
US10011588, Example 149
Show/Hide
|
C22H23F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443735
|
US10011588, Example 159
Show/Hide
|
C21H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0443829
|
US10011588, Example 87
Show/Hide
|
C20H19ClF3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450791
|
US10011588, Example 47
Show/Hide
|
C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450792
|
US10011588, Example 97
Show/Hide
|
C20H18ClF3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450793
|
US10011588, Example 111
Show/Hide
|
C21H22F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450794
|
US10011588, Example 112
Show/Hide
|
C21H23N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450795
|
US10011588, Example 49
Show/Hide
|
C18H18BrF3N4O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450796
|
US10011588, Example 61
Show/Hide
|
C19H16F5N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450797
|
US10011588, Example 69
Show/Hide
|
C18H17ClF3N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450798
|
US10011588, Example 141
Show/Hide
|
C21H21F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450818
|
US10011588, Example 51
Show/Hide
|
C21H25F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450819
|
US10011588, Example 67
Show/Hide
|
C21H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0450820
|
US10011588, Example 85
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478630
|
US10011588, Example 32
Show/Hide
|
C19H17F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478632
|
US10011588, Example 38
Show/Hide
|
C21H19F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478633
|
US10011588, Example 42
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478634
|
US10011588, Example 55
Show/Hide
|
C19H17ClF3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478635
|
US10011588, Example 58
Show/Hide
|
C17H15F6N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478638
|
US10011588, Example 89
Show/Hide
|
C20H22F3N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478642
|
US10011588, Example 115
Show/Hide
|
C20H19F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478644
|
US10011588, Example 125
Show/Hide
|
C20H21F3N8O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0478658
|
US10011588, Example 147
Show/Hide
|
C21H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483949
|
US10011588, Example 44
Show/Hide
|
C20H19F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483950
|
US10011588, Example 45
Show/Hide
|
C20H17F6N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483951
|
US10011588, Example 50
Show/Hide
|
C21H21F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483952
|
US10011588, Example 80
Show/Hide
|
C22H20F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483953
|
US10011588, Example 81
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483954
|
US10011588, Example 117
Show/Hide
|
C20H18ClF3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483955
|
US10011588, Example 118
Show/Hide
|
C19H19BrN6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483957
|
US10011588, Example 121
Show/Hide
|
C20H19F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0483958
|
US10011588, Example 2
Show/Hide
|
C19H21F3N4O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0484838
|
US10011588, Example 15
Show/Hide
|
C20H19F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0484839
|
US10011588, Example 29
Show/Hide
|
C20H23F3N4O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0484841
|
US10011588, Example 76
Show/Hide
|
C19H19F3N8O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0484842
|
US10011588, Example 84
Show/Hide
|
C20H19F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0484843
|
US10011588, Example 91
Show/Hide
|
C22H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508962
|
US10011588, Example 17
Show/Hide
|
C19H18F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508963
|
US10011588, Example 28
Show/Hide
|
C16H15BrF3N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508964
|
US10011588, Example 33
Show/Hide
|
C17H15F5N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508965
|
US10011588, Example 34
Show/Hide
|
C19H21F3N4O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508966
|
US10011588, Example 41
Show/Hide
|
C19H17F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508967
|
US10011588, Example 46
Show/Hide
|
C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508968
|
US10011588, Example 54
Show/Hide
|
C20H17F6N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0508978
|
US10011588, Example 160
Show/Hide
|
C21H21F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0514994
|
US10011588, Example 132
Show/Hide
|
C20H16F6N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0514995
|
US10011588, Example 156
Show/Hide
|
C22H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0514996
|
US10011588, Example 157
Show/Hide
|
C20H18F4N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0516756
|
US10011588, Example 151
Show/Hide
|
C23H23F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0516758
|
US10011588, Example 5
Show/Hide
|
C20H21ClN6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0516760
|
US10011588, Example 78
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519849
|
US10011588, Example 7
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519850
|
US10011588, Example 8
Show/Hide
|
C21H20F3N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519851
|
US10011588, Example 16
Show/Hide
|
C20H19F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519852
|
US10011588, Example 26
Show/Hide
|
C22H22F3N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519854
|
US10011588, Example 138
Show/Hide
|
C22H19F4N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0519856
|
US10011588, Example 77
Show/Hide
|
C19H19F3N8O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0520576
|
US10011588, Example 10
Show/Hide
|
C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0520577
|
US10011588, Example 37
Show/Hide
|
C19H21F3N4O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0520578
|
US10011588, Example 114
Show/Hide
|
C20H23N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0520579
|
US10011588, Example 72
Show/Hide
|
C18H16F5N3O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0520583
|
US10011588, Example 106
Show/Hide
|
C20H18ClF3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523297
|
US10011588, Example 31
Show/Hide
|
C20H19F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523298
|
US10011588, Example 145
Show/Hide
|
C21H21F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523300
|
US10011588, Example 88
Show/Hide
|
C18H17F5N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523301
|
US10011588, Example 90
Show/Hide
|
C18H17F6N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523875
|
US10011588, Example 30
Show/Hide
|
C19H22F3N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523878
|
US10011588, Example 153
Show/Hide
|
C21H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523879
|
US10011588, Example 12
Show/Hide
|
C20H19F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523882
|
US10011588, Example 109
Show/Hide
|
C22H22F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0523883
|
US10011588, Example 135
Show/Hide
|
C23H23F3N6O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0525104
|
US10011588, Example 39
Show/Hide
|
C21H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0525105
|
US10011588, Example 52
Show/Hide
|
C19H17ClF3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0525108
|
US10011588, Example 146
Show/Hide
|
C22H20F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0525110
|
US10011588, Example 66
Show/Hide
|
C20H20F4N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529214
|
US10011588, Example 98
Show/Hide
|
C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529217
|
US10011588, Example 40
Show/Hide
|
C19H17ClF3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529218
|
US10011588, Example 48
Show/Hide
|
C21H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529219
|
US10011588, Example 53
Show/Hide
|
C19H17F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529220
|
US10011588, Example 107
Show/Hide
|
C20H18BrF3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529221
|
US10011588, Example 113
Show/Hide
|
C21H25N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0529222
|
US10011588, Example 20
Show/Hide
|
C20H18F3N5O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0531568
|
US10011588, Example 136
Show/Hide
|
C18H18F4N4O2
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0531569
|
US10689373, Example 9
Show/Hide
|
C19H20ClN7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0531575
|
US10011588, Example 3
Show/Hide
|
C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0531576
|
US10011588, Example 6
Show/Hide
|
C21H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0536887
|
US10011588, Example 139
Show/Hide
|
C22H18F5N5O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0538978
|
US10011588, Example 36
Show/Hide
|
C19H17F4N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0538979
|
US10011588, Example 62
Show/Hide
|
C18H16F6N4O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0538980
|
US10011588, Example 1
Show/Hide
|
C20H22F3N3O3
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0538981
|
US10011588, Example 4
Show/Hide
|
C21H25N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0538982
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US10011588, Example 13
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C22H20F3N5O
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1
|
1 |
IC50 > 10000 nM
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CP0538983
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US10011588, Example 18
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C19H18F3N7O
|
1
|
1 |
IC50 > 10000 nM
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CP0538984
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US10011588, Example 63
Show/Hide
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C19H20F3N5O
|
1
|
1 |
IC50 > 10000 nM
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CP0545689
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US10011588, Example 101
Show/Hide
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C20H19F3N6O
|
1
|
1 |
IC50 > 10000 nM
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CP0545691
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US10011588, Example 35
Show/Hide
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C19H18F3N7O
|
1
|
1 |
IC50 > 10000 nM
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CP0545692
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US10011588, Example 65
Show/Hide
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C18H17F5N4O
|
1
|
1 |
IC50 > 10000 nM
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CP0549924
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US10011588, Example 14
Show/Hide
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C22H19F4N5O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0549926
|
US10011588, Example 60
Show/Hide
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C18H20F3N5O2
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0549928
|
US10011588, Example 140
Show/Hide
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C21H19F4N5O2
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0549929
|
US10011588, Example 74
Show/Hide
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C20H19F4N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0549930
|
US10011588, Example 137
Show/Hide
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C22H21F3N6O
|
1
|
1 |
IC50 > 10000 nM
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CP0549931
|
US10011588, Example 143
Show/Hide
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C23H22F3N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0549932
|
US10011588, Example 144
Show/Hide
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C21H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0556922
|
US10011588, Example 102
Show/Hide
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C20H18F4N6O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0561309
|
US10011588, Example 73
Show/Hide
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C20H20F3N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0562277
|
US10011588, Example 158
Show/Hide
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C23H22F4N6O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0562473
|
US10011588, Example 150
Show/Hide
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C22H22F3N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0573859
|
US10011588, Example 56
Show/Hide
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C19H16F5N7O
|
1
|
1 |
IC50 > 10000 nM
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|
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CP0573997
|
US10011588, Example 100
Show/Hide
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C19H18F3N7O
|
1
|
1 |
IC50 > 10000 nM
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