General Information of the Compound
Compound ID
CP0514996
Compound Name
US10011588, Example 157
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Structure
Formula
C20H18F4N6O2
Molecular Weight
450.396
Canonical SMILES
FC(F)Oc1ccc(N[C@H]2CC(F)(F)C[C@@H]2NC(=O)c2ccccc2-n2nccn2)nc1
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InChI
InChI=1S/C20H18F4N6O2/c21-19(22)32-12-5-6-17(25-11-12)28-14-9-20(23,24)10-15(14)29-18(31)13-3-1-2-4-16(13)30-26-7-8-27-30/h1-8,11,14-15,19H,9-10H2,(H,25,28)(H,29,31)/t14-,15-/m0/s1
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InChIKey
SQQCTQCNQDPCIH-GJZGRUSLSA-N
Physicochemical Property
logP
3.2719
Rotatable Bonds
7
Heavy Atom Count
32
Polar Areas
93.96
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
32

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118308214
ChEMBL ID
CHEMBL3932153
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 236 nM
   TI
   LI
   LO
   TS