General Information of the Compound
Compound ID
CP0478635
Compound Name
US10011588, Example 58
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Structure
Formula
C17H15F6N5O2
Molecular Weight
435.328
Canonical SMILES
FC(F)(F)Oc1cccnc1C(=O)N[C@H]1CCC[C@@H]1Nc1cnc(cn1)C(F)(F)F
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InChI
InChI=1S/C17H15F6N5O2/c18-16(19,20)12-7-26-13(8-25-12)27-9-3-1-4-10(9)28-15(29)14-11(5-2-6-24-14)30-17(21,22)23/h2,5-10H,1,3-4H2,(H,26,27)(H,28,29)/t9-,10-/m0/s1
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InChIKey
ZHBMNTVRIQHVHC-UWVGGRQHSA-N
Physicochemical Property
logP
3.552
Rotatable Bonds
5
Heavy Atom Count
30
Polar Areas
89.03
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118308177
ChEMBL ID
CHEMBL3975385
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 934 nM
   TI
   LI
   LO
   TS