General Information of the Compound
Compound ID
CP0478640
Compound Name
US10011588, Example 110
    Show/Hide
Structure
Formula
C22H24F3N7O
Molecular Weight
459.476
Canonical SMILES
CC(C)c1nc(cnc1N[C@H]1CCC[C@@H]1NC(=O)c1ccccc1-n1nccn1)C(F)(F)F
    Show/Hide
InChI
InChI=1S/C22H24F3N7O/c1-13(2)19-20(26-12-18(31-19)22(23,24)25)29-15-7-5-8-16(15)30-21(33)14-6-3-4-9-17(14)32-27-10-11-28-32/h3-4,6,9-13,15-16H,5,7-8H2,1-2H3,(H,26,29)(H,30,33)/t15-,16-/m0/s1
    Show/Hide
InChIKey
ODRJDAPEFIEULH-HOTGVXAUSA-N
Physicochemical Property
logP
3.9625
Rotatable Bonds
6
Heavy Atom Count
33
Polar Areas
97.62
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
33

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

    Show/Hide
Click to Show/Hide the External Link(s) of This Compound
PubChem ID
CID: 118308270
ChEMBL ID
CHEMBL3966483
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 3549 nM
   TI
   LI
   LO
   TS
Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 43 nM
   TI
   LI
   LO
   TS