General Information of the Compound
Compound ID
CP0523301
Compound Name
US10011588, Example 90
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Structure
Formula
C18H17F6N5O2
Molecular Weight
449.355
Canonical SMILES
C[C@@]1(CCC[C@@H]1NC(=O)c1ncccc1OC(F)(F)F)Nc1cnc(cn1)C(F)(F)F
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InChI
InChI=1S/C18H17F6N5O2/c1-16(29-13-9-26-12(8-27-13)17(19,20)21)6-2-5-11(16)28-15(30)14-10(4-3-7-25-14)31-18(22,23)24/h3-4,7-9,11H,2,5-6H2,1H3,(H,27,29)(H,28,30)/t11-,16-/m0/s1
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InChIKey
SJAGXZSCDINIMC-ZBEGNZNMSA-N
Physicochemical Property
logP
3.9421
Rotatable Bonds
5
Heavy Atom Count
31
Polar Areas
89.03
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
6
Complexity
31

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118308224
ChEMBL ID
CHEMBL3985601
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 68 nM
   TI
   LI
   LO
   TS