General Information of the Compound
Compound ID
CP0573997
Compound Name
US10011588, Example 100
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Structure
Formula
C19H18F3N7O
Molecular Weight
417.395
Canonical SMILES
FC(F)(F)c1ccc(N[C@H]2CCC[C@@H]2NC(=O)c2ncccc2-n2nccn2)nc1
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InChI
InChI=1S/C19H18F3N7O/c20-19(21,22)12-6-7-16(24-11-12)27-13-3-1-4-14(13)28-18(30)17-15(5-2-8-23-17)29-25-9-10-26-29/h2,5-11,13-14H,1,3-4H2,(H,24,27)(H,28,30)/t13-,14-/m0/s1
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InChIKey
KMGNRPCKEDNRLB-KBPBESRZSA-N
Physicochemical Property
logP
2.8391
Rotatable Bonds
5
Heavy Atom Count
30
Polar Areas
97.62
Hydrogen Bond Donor Count
2
Hydrogen Bond Acceptor Count
7
Complexity
30

"RO5" indicates the cutoff set by lipinski's rule of five:

(1) Molecular weight less than 500 Dalton;

(2) xlogp less than 5;

(3) No more than 5 hbonddonor (Hydrogen Bond Donor Count);

(4) No more than 10 hbondacc (Hydrogen Bond Acceptor Count);

(5) No more than 10 rotbonds (Rotatable Bond Count).

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PubChem ID
CID: 118308226
ChEMBL ID
CHEMBL3971206
Map of Molecular Bioactivity Related to the Compound
Map of Molecular Bioactivity Related to the Compound

Compound
Cell Line
Protein

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Compound
Protein ID: PT01132, Orexin receptor type 2
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 > 10000 nM
   TI
   LI
   LO
   TS
Protein ID: PT02001, Orexin/Hypocretin receptor type 1
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000278 RBL-2H3 Rattus norvegicus (Rat)  1
1
IC50 = 128 nM
   TI
   LI
   LO
   TS