| Compound ID |
Compound Name |
Compound Formula |
|
CP0045636
|
2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C22H22N6O3S
|
1
|
| 1 |
EC50 = 30 nM
|
|
|
|
CP0380424
|
2-(1H-indazol-3-ylamino)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C20H20N8OS
|
1
|
| 1 |
EC50 = 40 nM
|
|
|
|
CP0482421
|
2-indazol-1-yl-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C20H19N7OS
|
1
|
| 1 |
EC50 = 75 nM
|
|
|
|
CP0556355
|
2-(3-oxo-1H-isoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C21H20N6O2S
|
1
|
| 1 |
EC50 = 100 nM
|
|
|
|
CP0529649
|
2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C23H23N5O3S
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0525322
|
2-(1H-indazol-3-ylamino)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C21H21N7OS
|
1
|
| 1 |
EC50 = 350 nM
|
|
|
|
CP0408172
|
2-indazol-1-yl-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C21H20N6OS
|
1
|
| 1 |
EC50 = 750 nM
|
|
|
|
CP0408169
|
2-(1,3-dihydroisoindol-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C21H22N6OS
|
1
|
| 1 |
EC50 = 900 nM
|
|
|
|
CP0409896
|
2-(1-benzothiophen-2-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C21H19N5OS2
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0433813
|
2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-N-(6-methyl-4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C23H24N6O3S
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0482422
|
2-(1H-indol-5-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
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|
C21H20N6OS
|
1
|
| 1 |
EC50 = 1000 nM
|
|
|
|
CP0545841
|
2-(1-benzothiophen-5-yl)-N-(4-piperazin-1-ylpyridin-3-yl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C21H19N5OS2
|
1
|
| 1 |
EC50 = 1250 nM
|
|
|
|
CP0482423
|
2-(1,3-dihydroisoindol-2-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C22H23N5OS
|
1
|
| 1 |
EC50 = 1400 nM
|
|
|
|
CP0450695
|
2-(1-benzothiophen-2-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C22H20N4OS2
|
1
|
| 1 |
EC50 = 1500 nM
|
|
|
|
CP0338384
|
2-(1-benzofuran-5-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C22H20N4O2S
|
1
|
| 1 |
EC50 = 2000 nM
|
|
|
|
CP0114061
|
2-(1-benzothiophen-5-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
Show/Hide
|
C22H20N4OS2
|
1
|
| 1 |
EC50 = 2500 nM
|
|
|
|
CP0123581
|
2-(1H-indol-5-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C22H21N5OS
|
1
|
| 1 |
EC50 = 3500 nM
|
|
|
|
CP0399378
|
2-[[5-(4-methoxyphenyl)-1H-pyrazol-3-yl]amino]-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C24H25N7O2S
|
1
|
| 1 |
EC50 = 3750 nM
|
|
|
|
CP0544608
|
N-(5-fluoro-2-piperazin-1-ylphenyl)-2-(5-methoxy-3-oxo-1H-isoindol-2-yl)-1,3-thiazole-4-carboxamide
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|
C23H22FN5O3S
|
1
|
| 1 |
EC50 = 6000 nM
|
|
|
|
CP0433815
|
2-[(5-phenyl-1H-pyrazol-3-yl)amino]-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C23H23N7OS
|
1
|
| 1 |
EC50 = 7500 nM
|
|
|
|
CP0003092
|
2-(2,3-dihydro-1-benzofuran-5-yl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C22H22N4O2S
|
1
|
| 1 |
EC50 = 10000 nM
|
|
|
|
CP0196834
|
2-(4-phenoxyphenyl)-N-(2-piperazin-1-ylphenyl)-1,3-thiazole-4-carboxamide
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|
C26H24N4O2S
|
1
|
| 1 |
EC50 > 50000 nM
|
|
|
