| Compound ID |
Compound Name |
Compound Formula |
|
CP0224957
|
N-[2-[2-(dimethylamino)ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C21H24F3N5O2
|
1
|
| 1 |
IC50 = 55 nM
|
|
|
|
CP0553169
|
N-(2-morpholin-4-yl-5-piperidin-1-yl-1,3-benzoxazol-6-yl)-6-(1H-pyrazol-4-yl)pyridine-2-carboxamide
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|
C25H27N7O3
|
1
|
| 1 |
IC50 = 58.5 nM
|
|
|
|
CP0576704
|
N-[2-[2-(dimethylamino)ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-2-(2-methylpyridin-4-yl)-1,3-oxazole-4-carboxamide
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|
C24H28N6O3
|
1
|
| 1 |
IC50 = 58.7 nM
|
|
|
|
CP0471381
|
N-(2-morpholin-4-yl-5-piperidin-1-yl-[1,3]oxazolo[4,5-b]pyridin-6-yl)-6-(1H-pyrazol-4-yl)pyridine-2-carboxamide
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|
C24H26N8O3
|
1
|
| 1 |
IC50 = 102.5 nM
|
|
|
|
CP0575182
|
N-[2-(3-hydroxy-3-methylbutyl)-7-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C20H21F3N4O3
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0469086
|
N-[7-methoxy-2-(1-methylpiperidin-4-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C21H22F3N5O2
|
1
|
| 1 |
IC50 = 125 nM
|
|
|
|
CP0224958
|
N-[2-(3-Hydroxy-3-methylbutyl)-6-(2-hydroxypropan-2-yl)-2H-indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C22H25F3N4O3
|
1
|
| 1 |
IC50 = 128 nM
|
|
|
|
CP0554872
|
N-[2-[2-(dimethylamino)ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-4-(trifluoromethyl)-1,3-thiazole-2-carboxamide
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|
C19H22F3N5O2S
|
1
|
| 1 |
IC50 = 198 nM
|
|
|
|
CP0577954
|
N-[2-[2-(dimethylamino)ethyl]-7-methoxyindazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C19H20F3N5O2
|
1
|
| 1 |
IC50 = 223 nM
|
|
|
|
CP0256659
|
N-[5-[(3S)-3-hydroxypyrrolidin-1-yl]-2-morpholin-4-yl-[1,3]oxazolo[4,5-b]pyridin-6-yl]-2-(2-methylpyridin-4-yl)-1,3-oxazole-4-carboxamide
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|
C24H25N7O5
|
1
|
| 1 |
IC50 = 233 nM
|
|
|
|
CP0573378
|
N-[2-(1-ethylsulfonylazetidin-3-yl)-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C22H24F3N5O4S
|
1
|
| 1 |
IC50 = 256 nM
|
|
|
|
CP0224956
|
N-(7-methoxy-2-piperidin-4-ylindazol-5-yl)-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C20H20F3N5O2
|
1
|
| 1 |
IC50 = 375 nM
|
|
|
|
CP0229603
|
N-[5-[(3R)-3-hydroxypyrrolidin-1-yl]-2-morpholin-4-yl-[1,3]oxazolo[4,5-b]pyridin-6-yl]-2-(2-methylpyridin-4-yl)-1,3-oxazole-4-carboxamide
Show/Hide
|
C24H25N7O5
|
1
|
| 1 |
IC50 = 514 nM
|
|
|
|
CP0552076
|
N-[2-[2-(diethylamino)ethyl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C23H28F3N5O2
|
1
|
| 1 |
IC50 = 514 nM
|
|
|
|
CP0577956
|
N-[6-(2-hydroxypropan-2-yl)-2-[[(2S)-5-oxopyrrolidin-2-yl]methyl]indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
Show/Hide
|
C22H22F3N5O3
|
1
|
| 1 |
IC50 = 730 nM
|
|
|
|
CP0577957
|
N-[2-(azetidin-3-yl)-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C20H20F3N5O2
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0471379
|
6-(6-aminopyridin-3-yl)-N-(2-morpholin-4-yl-[1,3]oxazolo[4,5-b]pyridin-6-yl)pyridine-2-carboxamide
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|
C21H19N7O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0471380
|
6-(6-aminopyridin-3-yl)-N-(2-morpholin-4-yl-[1,3]oxazolo[5,4-b]pyridin-5-yl)pyridine-2-carboxamide
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|
C21H19N7O3
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
|
CP0576705
|
N-[2-[1-(2-cyanoacetyl)azetidin-3-yl]-6-(2-hydroxypropan-2-yl)indazol-5-yl]-6-(trifluoromethyl)pyridine-2-carboxamide
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|
C23H21F3N6O3
|
1
|
| 1 |
IC50 > 2000 nM
|
|
|
