(NE)-N-[6-(2-morpholin-4-ylethoxy)-2-pyrrolo[1,2-c]pyrimidin-3-ylchromen-4-ylidene]hydroxylamine

(S)-2-Amino-4-phosphono-butyric acid

sodium;2-[2-[7-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]heptylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

sodium;2-[2-[8-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]octylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

sodium;2-[2-[6-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]hexylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

sodium;2-[2-[4-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]butylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

(3R)-N-(3-bromo-5-chlorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-[4-[(2-chlorobenzoyl)amino]-3-methoxy-phenyl]picolinamide

sodium;2-[2-[5-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]pentylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

(3R)-N-(3,5-dibromophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

sodium;2-[2-[3-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]propylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

(NE)-N-[6-(3-morpholin-4-ylpropyl)-2-thieno[3,2-c]pyridin-6-ylchromen-4-ylidene]hydroxylamine

7-fluoro-3-methyl-N-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1,2-benzoxazol-5-amine

US9212196, Derivative 20

(3S)-N-(3-bromo-5-chlorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

3-methyl-N-(2H-pyrazolo[3,4-b]pyrazin-3-yl)-1,2-benzoxazol-5-amine

(3S)-N-(3,5-dibromophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-[3-(difluoromethoxy)phenyl]pyridine-2-carboxamide

US9212196, Derivative 6

6-((1H-pyrazolo[3,4-b] pyrazin-3- yl)amino)-N-(3,3- difluorocyclobutyl) benzo[d] isothiazole-3- carboxamide

6-((1H-pyrazolo[4,3-b] pyridin- 3-yl)amino)-N-(3,3- difluorocyclobutyl)benzo[d] isothiazole-3-carboxamide

3-methyl-N-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1,2-benzoxazol-5-amine

US9212196, Derivative 3

N-(4-chloro-3-methoxyphenyl)pyridine-2-carboxamide

US9212196, Derivative 2

(3R)-N-(3-bromo-5-iodophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-(6-fluoro-1H-pyrazolo[4,3-b]pyridin-3-yl)-3-methyl-1,2-benzoxazol-5-amine

(1R,2R)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid

D-AP4

US9212196, Derivative 7

(6-((1H-pyrazolo[4,3-b] pyridin-3-yl)amino) benzo[d]isothiazol-3-yl) (4,4-difluoropiperidin-1-yl) methanone

(3R)-N-(3-chlorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

US9212196, Derivative 8

3-(2,2-dimethylpropyl)-N-(2H-pyrazolo[3,4-b]pyrazin-3-yl)-[1,2]thiazolo[4,5-b]pyridin-6-amine

1-(4-(6-((1H- pyrazolo[4,3-b] pyridin-3-yl)amino) benzo[d] isothiazol-3-yl)piperidin- 1-yl)ethan-1-one

7-fluoro-3-methyl-N-(2H-pyrazolo[3,4-b]pyridin-3-yl)-1,2-benzoxazol-5-amine

N-(5-fluoro-2H-pyrazolo[3,4-b]pyridin-3-yl)-3-methyl-1,2-benzoxazol-5-amine

3-methyl-N-(2H-pyrazolo[3,4-b]pyridin-3-yl)-1,2-benzoxazol-5-amine

N-(3-methoxy-4-methylphenyl)pyridine-2-carboxamide

US9212196, Derivative 26

US9212196, Derivative 24

(3R)-N-(3,5-dichlorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

(3R)-N-(3-chloro-5-fluorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

US9212196, Derivative 5

N-(3-chlorophenyl)pyridine-2-carboxamide

US9212196, Derivative 28

(1S,2S)-1-amino-2-fluoro-2-(phosphonomethyl)cyclopropane-1-carboxylic acid

(3R)-N-(3-bromo-5-fluorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-(4-fluoro-3-methoxyphenyl)pyridine-2-carboxamide

US9212196, Derivative 14

US9212196, Derivative 9

US9212196, Derivative 11

N-(1,3-benzodioxol-5-yl)pyridine-2-carboxamide

US9212196, Derivative 4

3-(2,2-dimethylpropyl)-N-(2H-pyrazolo[3,4-b]pyrazin-3-yl)-1,2-benzoxazol-6-amine

3-cyclopentyl-N-(2H-pyrazolo[3,4-b]pyrazin-3-yl)-1,2-benzoxazol-6-amine

US9212196, Derivative 10

3-(2,2-dimethylpropyl)-N-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1,2-benzoxazol-6-amine

(3R)-N-(3-fluoro-5-iodophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

sodium;2-[2-[2-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]ethylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

3-cyclopentyl-N-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1,2-benzoxazol-6-amine

N-(3-chloro-4-methoxyphenyl)pyridine-2-carboxamide

US9212196, Derivative 21

US9212196, Derivative 29

(3R)-N-[3,5-bis(trifluoromethyl)phenyl]-5-oxo-1,4-thiazepane-3-carboxamide

US9212196, Derivative 12

(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-chloropropanoic Acid

(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]propenoic acid

N-[4-fluoro-3-(trifluoromethyl)phenyl]pyridine-2-carboxamide

US9212196, Derivative 30

(3R)-N-(3-chloro-5-methylphenyl)-5-oxo-1,4-thiazepane-3-carboxamide

2-(2-bromophenoxy)-1-(2,4-dihydroxyphenyl)ethanone

US9212196, Derivative 25

US9212196, Derivative 22

US9212196, Derivative 32

3-(1,1-difluoroethyl)-N-(1H-pyrazolo[4,3-b]pyridin-3-yl)-1,2-benzoxazol-6-amine

US9212196, Derivative 19

N-[4-chloro-3-(trifluoromethyl)phenyl]pyridine-2-carboxamide

(1R,2S)-4-aminocyclopentane-1,2,4-tricarboxylic acid

N-[3-(trifluoromethyl)phenyl]pyridine-2-carboxamide

(1aS,7E,7aS)-7-hydroxyimino-N-phenyl-1,7a-dihydrocyclopropa[b]chromene-1a-carboxamide

(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)-methyl]butan-1,4-dioic Acid

(3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]ethanoic Acid

N-(3,4-dimethoxyphenyl)pyridine-2-carboxamide

(1S,2S)-1-[(2S)-2-amino-2-carboxyethyl]cyclopropane-1,2-dicarboxylic acid

US9212196, Derivative 18

(2S)-2-aminopentanedioic acid

US9212196, Derivative 34

US9212196, Derivative 23

(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)hydroxymethyl]cyclopropane-1-carboxylic Acid

(S)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid

US9212196, Derivative 35

(3R)-N-(3-bromophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

(+/-)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid

(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-(hydroxymethyl)ethanoic Acid

US9212196, Derivative 31

(3S)-4-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-butanoic Acid

4-((S)-Amino-carboxy-methyl)-phthalic acid

(3R)-N-(3,5-difluorophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-[4-cyano-3-(trifluoromethyl)phenyl]pyridine-2-carboxamide

N-(6-methoxypyrimidin-4-yl)pyridine-2-carboxamide

N-[6-(trifluoromethyl)pyridin-2-yl]pyridine-2-carboxamide

sodium;2-[2-[12-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]dodecylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

sodium;2-[2-[10-[[2-[2-[3-chloro-4-[[2-methoxy-4-(pyridine-2-carbonylamino)phenyl]carbamoyl]anilino]-2-oxoethoxy]acetyl]amino]decylamino]-2-oxoethoxy]-5-[3-[(2-cyclopentyl-6,7-dimethyl-1-oxo-2,3-dihydroinden-5-yl)oxymethyl]phenyl]benzoate

(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-2-methylpropanoic Acid

US9212196, Derivative 13

(R)-3-amino-3-carboxypropyl-2'-carboxyethyl phosphinic acid

(3S)-2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)hydroxymethyl]cyclopropane-1-carboxylic Acid hydrochloride

(3S)-3-[((3-Amino-3-carboxylate)propyl)(hydroxy)phosphinate]-2-(2-hydroxyethyl)propanoate

(3S)-3-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-3-trifluoromethypropanoic Acid

(+/-)-(Z)-1-Amino-2-fluoro-2-(hydroxy(phosphono)methyl)cyclopropanecarboxylic acid hydrochloride

3-[3-[(2-cyclopentyl-1-oxo-3H-isoindol-5-yl)oxymethyl]phenyl]-4-methoxybenzoic acid

2-chloro-5-[3-(2-cyclopentyl-1-oxo-3H-isoindol-5-yl)phenyl]benzoic acid

2-chloro-5-[3-[(2-cyclopropyl-3-oxo-1,2-benzothiazol-6-yl)oxymethyl]phenyl]benzoic acid

(3S)-N-(3-bromophenyl)-5-oxo-1,4-thiazepane-3-carboxamide

2-[(((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl)]butan-1,4-dioic Acid

US9212196, Derivative 33

(+/-)-(Z)-1-Amino-2-fluoro-2-(sulfomethyl)cyclopropane carboxylic acid hydrochloride

(3S)-2-[((3-Amino-3-carboxy)propyl)(hydroxy)phosphinyl]-ethylphosphonate

(1S,3R)-1-aminocyclopentane-1,3-dicarboxylic acid;hydrate

(2S)-amino(3,5-dihydroxyphenyl)ethanoic acid

(S)-3-(amino(carboxy)methyl)bicyclo[1.1.1]pentane-1-carboxylic acid

(+/-)-trans-ACPD

(1S,2S,5R,6S)-2-Amino-bicyclo[3.1.0]hexane-2,6-dicarboxylic acid

(S)-4-(amino(carboxy)methyl)-2-hydroxybenzoic acid

(2R,4R)-4-aminopyrrolidine-2,4-dicarboxylic acid

(2R,4S)-2-Amino-4-methyl-pentanedioic acid

(2R)-2-amino-4-methylidenepentanedioic acid4-methylidene-D-glutamic acid

(S)-2-Amino-4-(3,5-dioxo-[1,2,4]oxadiazolidin-2-yl)-butyric acid

2-Amino-4-phosphono-butyric acid

(1S,3R)-1-aminopentane-1,3,5-tricarboxylic acid

(3R)-N-(3,5-dimethylphenyl)-5-oxo-1,4-thiazepane-3-carboxamide

N-[3-(trifluoromethoxy)phenyl]pyridine-2-carboxamide

(2S)-2-amino-3-(phosphonooxy)propanoic acid

(2R)-2-aminopentanedioic acid

(S)-2-amino-4-sulfobutanoic acid

(1S,2S)-4-Amino-cyclopentane-1,2,4-tricarboxylic acid

Amino-(4-phosphono-phenyl)-acetic acid

2-Amino-bicyclo[2.1.1]hexane-2,5-dicarboxylic acid

(1R,2R)-2-((S)-Amino-carboxy-methyl)-cyclopropanecarboxylic acid

2-[4-(4-butanoyl-3-hydroxy-2-methylphenoxy)butoxy]-3-methoxybenzoic acid

7-(4-fluorophenyl)-2-[[2-(trifluoromethyl)pyridin-4-yl]oxymethyl]pyrazolo[1,5-a]pyrimidine-5-carboxamide

2-[[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl]-7-(4-fluorophenyl)thieno[3,2-b]pyridine-5-carboxamide