| Compound ID |
Compound Name |
Compound Formula |
|
CP0005166
|
BMS-354825
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|
C22H26ClN7O2S
|
2
|
| 1 |
IC50 = 6 nM
|
|
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| 2 |
Ki = 0.5 nM
|
|
|
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CP0005675
|
2-aminopyrido[2,3-d]pyrimidin-7(8H)-one deriv.
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|
C26H27Cl2N5O2
|
2
|
| 1 |
IC50 = 8 nM
|
|
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| 2 |
Ki = 0.8 nM
|
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|
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CP0021055
|
6-(2,6-dichlorophenyl)-8-methyl-2-{[4-(morpholin-4-yl)phenyl]amino}-7H,8H-pyrido[2,3-d]pyrimidin-7-one
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|
C24H21Cl2N5O2
|
2
|
| 1 |
IC50 = 24 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
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CP0030237
|
6-(2,6-dichlorophenyl)-2-[(4-fluoro-3-methylphenyl)amino]-8-methyl-7H,8H-pyrido[2,3-d]pyrimidin-7-one
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|
C21H15Cl2FN4O
|
2
|
| 1 |
IC50 = 109 nM
|
|
|
| 2 |
Ki = 10.4 nM
|
|
|
|
CP0228501
|
N-methyl-2-[[5-methyl-2-[3-(methylsulfonylmethyl)anilino]pyrimidin-4-yl]amino]benzamide
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|
C21H23N5O3S
|
2
|
| 1 |
IC50 = 115 nM
|
|
|
| 2 |
Ki = 10.94 nM
|
|
|
|
CP0022369
|
4-[(2,4-Dichloro-5-methoxyphenyl)amino]-6-methoxy-7-[3-(4-methyl-1-piperazinyl)propoxy]-3-quinolinecarbonitrile
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|
C26H29Cl2N5O3
|
2
|
| 1 |
IC50 = 133 nM
|
|
|
| 2 |
Ki = 12.7 nM
|
|
|
|
CP0017872
|
3-[(6-methanesulfonylquinolin-4-yl)amino]-4-methylphenol
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|
C17H16N2O3S
|
2
|
| 1 |
IC50 = 177 nM
|
|
|
| 2 |
Ki = 16.85 nM
|
|
|
|
CP0248068
|
2-[[5-chloro-2-(4-morpholin-4-ylanilino)pyrimidin-4-yl]amino]-N-methylbenzamide
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|
C22H23ClN6O2
|
2
|
| 1 |
IC50 = 270 nM
|
|
|
| 2 |
Ki = 25.68 nM
|
|
|
|
CP0554034
|
2-[[5-cyano-2-[3-methoxy-4-(4-methylpiperazin-1-yl)anilino]pyrimidin-4-yl]amino]benzamide
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|
C24H26N8O2
|
2
|
| 1 |
IC50 = 340 nM
|
|
|
| 2 |
Ki = 32.4 nM
|
|
|
|
CP0045281
|
AZD0530
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|
C27H32ClN5O5
|
2
|
| 1 |
IC50 = 418 nM
|
|
|
| 2 |
Ki = 39.8 nM
|
|
|
|
CP0026746
|
2,4-dianilino pyrimidine, 36
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|
C18H15N7O
|
2
|
| 1 |
IC50 = 509 nM
|
|
|
| 2 |
Ki = 48.47 nM
|
|
|
|
CP0141549
|
3-methyl-5-[(7-pyridin-2-ylquinolin-4-yl)amino]phenol
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|
C21H17N3O
|
2
|
| 1 |
IC50 = 543 nM
|
|
|
| 2 |
Ki = 51.73 nM
|
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|
|
CP0239379
|
3-[(7-pyridin-4-ylquinolin-4-yl)amino]phenol
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|
C20H15N3O
|
2
|
| 1 |
IC50 = 706 nM
|
|
|
| 2 |
Ki = 67.19 nM
|
|
|
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CP0096174
|
AZD-1775
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|
C27H32N8O2
|
2
|
| 1 |
IC50 = 4940 nM
|
|
|
| 2 |
Ki = 470 nM
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CP0228499
|
2,6-difluoro-N-[3-[3-[2-(pyridin-3-ylamino)pyrimidin-4-yl]pyrazolo[1,5-b]pyridazin-2-yl]phenyl]benzamide
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|
C28H18F2N8O
|
2
|
| 1 |
IC50 = 7560 nM
|
|
|
| 2 |
Ki = 720.2 nM
|
|
|
|
CP0022401
|
5-[(E)-2-(4-hydroxy-2,6-dimethylphenyl)ethenyl]pyridine-3-carboxamide
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|
C16H16N2O2
|
2
|
| 1 |
IC50 = 14510 nM
|
|
|
| 2 |
Ki = 1380 nM
|
|
|
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CP0016076
|
N-(3-chlorophenyl)-6,7-dimethoxyquinazolin-4-amine
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|
C16H14ClN3O2
|
2
|
| 1 |
IC50 = 19600 nM
|
|
|
| 2 |
Ki = 1870 nM
|
|
|
|
CP0028136
|
2-amino-3-phenyl-5-(pyridin-4-yl)benzamide
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|
C18H15N3O
|
2
|
| 1 |
IC50 = 57990 nM
|
|
|
| 2 |
Ki = 5520 nM
|
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|
