1-(6-{13-[4-(trifluoromethyl)phenyl]tridecanamido}quinolin-2-yl)-1-azabicyclo[2.2.2]octan-1-ylium

N-[2-[3-(methylcarbamoylamino)pyrrolidin-1-yl]quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)quinolin-2-yl)pyrrolidin-3-ylsulfamic acid

N-[2-(azetidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

2-methyl-N-[1-[6-[3-[4-(trifluoromethyl)phenyl]propanoylamino]quinolin-2-yl]pyrrolidin-3-yl]propanamide

N-[1-[6-[3-[4-(trifluoromethyl)phenyl]propanoylamino]quinolin-2-yl]pyrrolidin-3-yl]benzamide

N-[2-(dimethylamino)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-(2-piperidin-1-ylquinolin-6-yl)-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-[methyl(propyl)amino]quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2,7-diazaspiro[4.4]nonan-2-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-[methyl(propan-2-yl)amino]quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2-azabicyclo[2.2.1]heptan-2-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2-azabicyclo[2.2.2]octan-2-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(3-aminopyrrolidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2-methylpyrrolidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-(2-pyrrolidin-1-ylquinolin-6-yl)-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(methylamino)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-[cyclopentyl(methyl)amino]quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(3-methylpyrrolidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(3-acetamidopyrrolidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

methyl 1-[6-[3-[4-(trifluoromethyl)phenyl]propanoylamino]quinolin-2-yl]pyrrolidine-2-carboxylate

N-(2-aminoquinolin-6-yl)-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(diethylamino)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-[cyclohexyl(methyl)amino]quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(3-phenylpyrrolidin-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

N-[2-(azepan-1-yl)quinolin-6-yl]-3-[4-(trifluoromethyl)phenyl]propanamide

1-{6-[6-(trifluoromethyl)pyridine-3-amido]quinolin-2-yl}-1-azabicyclo[2.2.2]octan-1-ylium

1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-phenylurea

1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea

(4aR,11R,11aS)-11-methyl-2-[3-(oxan-4-yl)propyl]-9-(trifluoromethyl)-1,3,4,4a,5,6,11,11a-octahydropyrido[4,3-b]carbazole

1-(4-bromophenyl)-3-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)urea

1-(2-(4-fluoro-3-methylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea

1-(5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)-2-(m-tolyloxy)phenyl)-3-(3-fluorophenyl)urea

N-[3-[1-[3-[[2,2-bis(4-fluorophenyl)acetyl]amino]propyl]piperidin-4-yl]phenyl]-2-methylpropanamide

1-(2-chlorophenyl)-3-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)urea

N-[3-[1-[3-[(2,2-diphenylacetyl)amino]propyl]piperidin-4-yl]phenyl]-2-methylpropanamide

(2S)-2-(4-fluorophenyl)-N-(3-{4-[5-(isobutyrylamino)-2-methylphenyl]-1-piperidinyl}propyl)propanamide

N-[3-[1-[3-[(2-hydroxy-2,2-diphenylacetyl)amino]propyl]piperidin-4-yl]-4-methylphenyl]-2-methylpropanamide

N-[3-[1-[3-[[2,2-bis(4-fluorophenyl)acetyl]amino]propyl]piperidin-4-yl]-4-methylphenyl]-2-methylpropanamide

N-[3-[1-[3-[(2,2-diphenylacetyl)amino]propyl]piperidin-4-yl]-4-methylphenyl]-2-methylpropanamide

1-(2-(3,4-difluorophenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea

1-(5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)-2-(p-tolyloxy)phenyl)-3-(3-fluorophenyl)urea

N-[5-[1-[3-[[2,2-bis(4-fluorophenyl)acetyl]amino]propyl]piperidin-4-yl]-2,4-difluorophenyl]-2-methylpropanamide

1-(2-(3-fluorophenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(3-fluorophenyl)urea

1-(4-fluorophenyl)-N-(3-{4-[5-(isobutylamino)-2-methylphenyl]-1-piperidinyl}propyl)cyclohexanecarboxamide

N-[3-[1-[2-[(2,2-diphenylacetyl)amino]ethyl]piperidin-4-yl]phenyl]-2-methylpropanamide

(2R)-2-(4-fluorophenyl)-N-(3-{4-[5-(isobutyrylamino)-2-methylphenyl]-1-piperidinyl}propyl)propanamide

2-methyl-N-{4-methyl-3-[1-(3-{[(2R)-2-phenylpropanoyl]-amino}propyl)-4-piperidinyl]phenyl}propanamide

N-[3-[1-[4-(4-chlorophenyl)-4-oxobutyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[[4-(3,4-difluorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

2-methyl-N-{4-methyl-3-[1-(3-{[(2S)-2-phenylpropanoyl]-amino}propyl)-4-piperidinyl]phenyl}propanamide

N-[3-[1-[3-(2,2-diphenylpropanoylamino)propyl]piperidin-4-yl]phenyl]-2-methylpropanamide

3-cinnamamido-4-(3,4-dimethylphenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

N-[3-[4-[3-(2-methylpropanoylamino)phenyl]piperidin-1-yl]propyl]-2,2-diphenylbutanamide

1-(4-fluorophenyl)-N-(3-{4-[5-(isobutyrylamino)-2-methylphenyl]-1-piperidinyl}propyl)cyclopentanecarboxamide

N-[3-[1-[[4-(3,4-difluorophenoxy)phenyl]methyl]piperidin-4-yl]-4-methylphenyl]-2-methylpropanamide

4-(3,4-dimethylphenoxy)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

3-(3-biphenyl-4-yl-ureido)-4-(3,4-dimethyl-phenoxy)-N-(2-pyrrolidin-1-yl-ethyl)-benzamide

4-(3,4-dimethylphenoxy)-3-((1R,2R)-2-phenylcyclopropanecarboxamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

2-methyl-N-{3-[1-(4-phenoxybenzyl)-4-piperidinyl]phenyl}-propanamide

N-[3-[1-[[4-(4-chlorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[5-[1-[[4-(3,4-difluorophenoxy)phenyl]methyl]piperidin-4-yl]-2-methylphenyl]-2-methylpropanamide

4-(naphthalen-2-yloxy)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

N-[3-[1-[4-(4-chlorophenyl)-4-oxobutyl]piperidin-4-yl]phenyl]acetamide

N-[3-[1-[6-[(2,2-diphenylacetyl)amino]hexyl]piperidin-4-yl]phenyl]-2-methylpropanamide

1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(4-phenoxyphenyl)urea

N-[3-[1-[4-[(2,2-diphenylacetyl)amino]butyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[[4-(3,4-dichlorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[[4-(4-methoxyphenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[4-(3,4-dimethylphenyl)-4-oxobutyl]piperidin-4-yl]phenyl]acetamide

N-[3-[1-[[3-(3,5-dichlorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[[3-(4-chlorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-[4-(4-methylphenyl)-4-oxobutyl]piperidin-4-yl]phenyl]acetamide

N-[3-[1-[[3-(3,4-dichlorophenoxy)phenyl]methyl]piperidin-4-yl]phenyl]-2-methylpropanamide

N-[3-[1-(4-oxo-4-phenylbutyl)piperidin-4-yl]phenyl]acetamide

2-methyl-N-[3-(1-{3-[3-(trifluoromethyl)phenoxy]benzyl}-4-piperidinyl)phenyl]-propanamide

N-[3-[1-[4-oxo-4-(4-phenoxyphenyl)butyl]piperidin-4-yl]phenyl]acetamide

3-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-1-methyl-1-phenylurea

4-(3,4-dimethylphenylthio)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

phenyl N-[2-(3,4-dimethylphenoxy)-5-(2-pyrrolidin-1-ylethylcarbamoyl)phenyl]carbamate

3-acetamido-4-(3,4-dimethylphenoxy)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

1-(2-(3,4-dimethylphenoxy)-5-((2-(pyrrolidin-1-yl)ethyl)carbamoyl)phenyl)-3-(pyridin-2-yl)urea

4-(3,4-dimethylphenoxy)-3-propionamido-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

4-(3,4-dimethylphenoxy)-3-(2-phenylacetamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

N-(2-aminoethyl)-4-(3,4-dimethylphenoxy)-3-(3-phenylpropanoylamino)benzamide

4-(3,4-dimethylphenylamino)-3-(3-phenylpropanamido)-N-(2-(pyrrolidin-1-yl)ethyl)benzamide

N-[5-[1-[3-[(2,2-diphenylacetyl)amino]propyl]piperidin-4-yl]-2-methylphenyl]-2-methylpropanamide

(S)-3-{3-[4-(3-Acetylamino-phenyl)-piperidin-1-yl]-propylcarbamoyl}-4-(3,4-difluoro-phenyl)-6-methoxymethyl-2-oxo-1,2,3,4-tetrahydro-pyrimidine-5-carboxylic acid methyl ester

(S)-6-(4-chlorophenyl)-2-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(R)-6-(4-chlorophenyl)-2-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(S)-6-(4-chlorophenyl)-2-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(R)-2-(4-methoxyphenyl)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)thieno[2,3-d]pyridazin-7(6H)-one

(R)-6-(4-chlorophenyl)-2-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(S)-6-(4-chlorophenyl)-2-(6-(3-(pyrrolidin-1-ylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(R)-2-(4-chlorophenyl)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)thieno[2,3-d]pyridazin-7(6H)-one

(S)-6-(4-chlorophenyl)-2-(6-(3-(ethylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(S)-2-(4-fluorophenyl)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)thieno[2,3-d]pyridazin-7(6H)-one

N-[3-[1-[3-[[2,2-bis(4-chlorophenyl)acetyl]amino]propyl]piperidin-4-yl]phenyl]-2-methylpropanamide

(R)-2-(4-fluorophenyl)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)thieno[2,3-d]pyridazin-7(6H)-one

(R)-2-(4-ethylphenyl)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)thieno[2,3-d]pyridazin-7(6H)-one

N-[3-[1-[3-[[2,2-bis(4-fluorophenyl)acetyl]amino]propyl]piperidin-4-yl]-2,4,6-trifluorophenyl]-2-methylpropanamide

(S)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)-2-(4-(trifluoromethyl)phenyl)thieno[2,3-d]pyridazin-7(6H)-one

(R)-6-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)-2-(4-(trifluoromethyl)phenyl)thieno[2,3-d]pyridazin-7(6H)-one

(S)-6-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-2-(4-(trifluoromethyl)phenyl)thieno[2,3-d]pyridazin-7(6H)-one

(S)-2-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)-6-(4-(trifluoromethyl)phenyl)phthalazin-1(2H)-one

N-[3-[4-[3-(2-methylpropanoylamino)phenyl]piperidin-1-yl]propyl]-2,2-diphenylheptanamide

(R)-2-(6-(3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)-6-(4-(trifluoromethyl)phenyl)phthalazin-1(2H)-one

6-(4-methoxy-2-methylphenyl)-2-(6-((S)-3-(methylamino)pyrrolidin-1-yl)pyridin-3-yl)phthalazin-1(2H)-one

(S)-6-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-1-methyl-2-(4-(trifluoromethyl)phenyl)-1H-pyrrolo[2,3-d]pyridazin-7(6H)-one

(S)-6-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-2-(4-(trifluoromethyl)phenyl)furo[2,3-d]pyridazin-7(6H)-one

N-[3-[1-[5-[(2,2-diphenylacetyl)amino]pentyl]piperidin-4-yl]phenyl]-2-methylpropanamide