Brief Information of the Compound and Protein
Compound Name
(S)-6-(6-(3-(dimethylamino)pyrrolidin-1-yl)pyridin-3-yl)-1-methyl-2-(4-(trifluoromethyl)phenyl)-1H-pyrrolo[2,3-d]pyridazin-7(6H)-one
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PubChem ID
CID: 11641550
SID: 16744813
Canonical SMILES
CN(C)[C@H]1CCN(C1)c1ccc(cn1)-n1ncc2cc(-c3ccc(cc3)C(F)(F)F)n(C)c2c1=O
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Compound Formula C25H25F3N6O
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
P97639
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 14 nM
   TI
   LI
   LO
   TS