| Compound ID |
Compound Name |
Compound Formula |
|
CP0224426
|
US10245267, Example 1029
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|
C28H28F4N4O4
|
1
|
| 1 |
EC50 = 5 nM
|
|
|
|
CP0899539
|
N-[5-[6-(4-deuteriotetrahydropyran-4-yl)oxy-5-morpholino-3-pyridyl]-6-methyl-3-pyridyl]-3-(trifluoromethyl)benzamide
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|
C28H29F3N4O4
|
1
|
| 1 |
EC50 = 6 nM
|
|
|
|
CP0177589
|
US10245267, Example 636
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|
C27H28F3N5O4
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0202460
|
N-[3-[2-(2-hydroxyethylamino)-6-morpholin-4-ylpyridin-4-yl]-4-methylphenyl]-2-(trifluoromethyl)pyridine-4-carboxamide
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|
C25H26F3N5O3
|
1
|
| 1 |
EC50 = 8 nM
|
|
|
|
CP0134276
|
US10245267, Example 1156
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|
C25H25F3N4O4
|
1
|
| 1 |
EC50 = 14 nM
|
|
|
|
CP0014402
|
US10245267, Example 131
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|
C28H29F3N4O4
|
2
|
| 1 |
EC50 = 20 nM
|
|
|
| 2 |
EC50 = 100 nM
|
|
|
|
CP0551448
|
N-[5-[6-[(3S,4S)-3-methoxyoxan-4-yl]oxy-5-morpholin-4-ylpyridin-3-yl]-6-methylpyridin-3-yl]-3-(trifluoromethyl)benzamide
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|
C29H31F3N4O5
|
1
|
| 1 |
EC50 = 21 nM
|
|
|
|
CP0557916
|
US10245267, Example 1041
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|
C25H28F2N6O3
|
1
|
| 1 |
EC50 = 27 nM
|
|
|
|
CP0226659
|
US10245267, Example 640
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|
C26H28N6O3
|
1
|
| 1 |
EC50 = 52 nM
|
|
|
|
CP0318226
|
US10245267, Example 31
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|
C25H26F3N5O3
|
1
|
| 1 |
EC50 = 61 nM
|
|
|
|
CP0202928
|
US10245267, Example 988
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|
C23H21F3N4O3
|
1
|
| 1 |
EC50 = 64 nM
|
|
|
|
CP0187401
|
US10245267, Example 117
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|
C25H24F3N3O3
|
1
|
| 1 |
EC50 = 76 nM
|
|
|
|
CP0117616
|
US10245267, Example 1
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|
C23H21F3N4O2
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0243293
|
US10245267, Example 145
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|
C25H25F3N4O4
|
1
|
| 1 |
EC50 = 80 nM
|
|
|
|
CP0346226
|
US10245267, Example 62
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|
C24H22F3N3O2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0474246
|
US10245267, Example 119
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|
C24H23F3N4O3
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0544270
|
N-(3-tert-butylphenyl)-4-methyl-3-(6-morpholin-4-ylpyrimidin-4-yl)benzamide
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|
C26H30N4O2
|
1
|
| 1 |
EC50 = 200 nM
|
|
|
|
CP0107258
|
US10245267, Example 127
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|
C24H23F3N4O3
|
1
|
| 1 |
EC50 = 250 nM
|
|
|
|
CP0117564
|
US10245267, Example 134
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|
C26H27F3N4O3
|
1
|
| 1 |
EC50 = 300 nM
|
|
|
|
CP0226656
|
US10245267, Example 138
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|
C24H23F3N4O3
|
1
|
| 1 |
EC50 = 460 nM
|
|
|
|
CP0573941
|
4-methyl-3-(6-morpholin-4-ylpyrimidin-4-yl)-N-[3-(trifluoromethyl)phenyl]benzamide
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|
C23H21F3N4O2
|
1
|
| 1 |
EC50 = 700 nM
|
|
|
|
CP0566040
|
US10245267, Example 390
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|
C23H22F3N5O3
|
1
|
| 1 |
EC50 = 3960 nM
|
|
|
