| Compound ID |
Compound Name |
Compound Formula |
|
CP0321526
|
(S)-1-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrrolo[1,2-f][1,2,4]triazin-2-yl)-N-(6-fluoropyridin-3-yl)pyrrolidine-2-carboxamide
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|
C22H22FN9O
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0030165
|
US8592579, 104
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|
C23H24FN9O
|
1
|
| 1 |
IC50 = 2.1 nM
|
|
|
|
CP0095643
|
4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-{6-[1-(2-methoxyethyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C29H34ClN5O3
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0347566
|
4-{[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}-3-{6-[1-(2-methoxyethyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C26H32ClN7O2
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0347568
|
4-{[(2S)-2-(3-chloro-4-methoxyphenyl)-2-hydroxyethyl]amino}-3-{6-[1-(3-fluoropropyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C30H35ClFN5O3
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0062475
|
4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-[4-methyl-6-(1-methylpiperidin-4-yl)-1H-1,3-benzodiazol-2-yl]-1,2-dihydropyridin-2-one
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|
C27H30ClN5O2
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0252994
|
4-{[(2S)-2-(3-chloro-4-methoxyphenyl)-2-hydroxyethyl]amino}-3-{6-[1-(2-methoxyethyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C30H36ClN5O4
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
|
CP0347567
|
4-{[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}-3-{6-[1-(2-hydroxyethyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C25H30ClN7O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0247182
|
4-{[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}-3-[4-methyl-6-(1-methylpiperidin-4-yl)-1H-1,3-benzodiazol-2-yl]-1,2-dihydropyridin-2-one
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|
C24H28ClN7O
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0253337
|
4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-{6-[1-(3-fluoropropyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C29H33ClFN5O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0064474
|
4-{[2-(4-chloro-1H-pyrazol-1-yl)ethyl]amino}-3-{6-[1-(3-fluoropropyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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|
C26H31ClFN7O
|
1
|
| 1 |
IC50 = 34 nM
|
|
|
|
CP0303187
|
N-[[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f][1,2,4]triazin-2-yl]methyl]-6-fluoropyridine-3-carboxamide
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|
C19H17FN8O
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0024739
|
4-{[(2S)-2-(3-chlorophenyl)-2-hydroxyethyl]amino}-3-[4-methyl-6-(morpholin-4-yl)-1H-1,3-benzodiazol-2-yl]-1,2-dihydropyridin-2-one
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|
C25H26ClN5O3
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0095974
|
(S)-(2-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrrolo[1,2-f][1,2,4]triazin-2-yl)pyrrolidin-1-yl)(6-fluoropyridin-3-yl)methanone
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|
C22H21FN8O
|
1
|
| 1 |
IC50 = 162 nM
|
|
|
|
CP0308225
|
2-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrrolo[1,2-f][1,2,4]triazin-2-yl)-N-(6-fluoropyridin-3-yl)cyclopent-1-enecarboxamide
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|
C23H21FN8O
|
1
|
| 1 |
IC50 = 237 nM
|
|
|
|
CP0335884
|
(S)-5-(4-(5-cyclopropyl-1H-pyrazol-3-ylamino)pyrrolo[1,2-f][1,2,4]triazin-2-yl)-1-(6-fluoronicotinoyl)pyrrolidin-2-one
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|
C22H19FN8O2
|
1
|
| 1 |
IC50 = 508 nM
|
|
|
