Brief Information of the Compound and Protein
Compound Name
4-{[(2S)-2-(3-chloro-4-methoxyphenyl)-2-hydroxyethyl]amino}-3-{6-[1-(3-fluoropropyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazol-2-yl}-1,2-dihydropyridin-2-one
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PubChem ID
CID: 135875712
SID: 56454845
Canonical SMILES
COc1ccc(cc1Cl)[C@H](O)CNc1cc[nH]c(=O)c1-c1nc2c(C)cc(cc2[nH]1)C1CCN(CCCF)CC1
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Compound Formula C30H35ClFN5O3
Compound Structure
Protein Name
Insulin-like growth factor 1 receptor
Protein Classification
Enzyme
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Kinase
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Protein Kinase
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TK protein kinase group
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Tyrosine protein kinase InsR family
Uniprot ID
P08069
Gene Name
IGF1R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000899 IGFSal Homo sapiens (Human)  1
1
IC50 = 20 nM
   TI
   LI
   LO
   TS