Compound ID |
Compound Name |
Compound Formula |
CP0276739
|
2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl)carbamoyl)-3-phenylpyrrolidin-1-yl)-2-methylpropanoic acid
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|
C33H38ClN3O4
|
2
|
1 |
IC50 = 1 nM
|
|
|
2 |
Ki = 6 nM
|
|
|
CP0134899
|
2-(4-{1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-ylcarbamoyl}-4-phenyl-piperidin-1-yl)-2-methyl-propionic acid
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|
C34H40ClN3O4
|
2
|
1 |
IC50 = 4 nM
|
|
|
2 |
Ki = 9 nM
|
|
|
CP0186508
|
4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide
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|
C31H37N3O3
|
2
|
1 |
IC50 = 11 nM
|
|
|
2 |
Ki = 62 nM
|
|
|
CP0134896
|
(+/-) 3-phenyl-pyrrolidine-3-carboxylic acid {1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-yl}-amide
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|
C29H32ClN3O2
|
2
|
1 |
IC50 = 22 nM
|
|
|
2 |
Ki = 27 nM
|
|
|
CP0153417
|
1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-yl}-amide
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|
C32H38ClN3O2
|
2
|
1 |
IC50 = 43 nM
|
|
|
2 |
Ki = 15 nM
|
|
|
CP0140912
|
N-[1-[[3-(2-methoxyphenoxy)phenyl]methyl]piperidin-4-yl]-2-phenylacetamide
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|
C27H30N2O3
|
2
|
1 |
IC50 = 55 nM
|
|
|
2 |
Ki = 250 nM
|
|
|
CP0334429
|
1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide
Show/Hide
|
C33H41N3O3
|
2
|
1 |
IC50 = 56 nM
|
|
|
2 |
Ki = 11 nM
|
|
|
CP0511885
|
4-(4-benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester
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|
C25H27N3O5S
|
1
|
1 |
Ki = 0.17 nM
|
|
|
CP0439479
|
N-[4-[(1-butanoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
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|
C27H31N3O4S
|
1
|
1 |
Ki = 0.3 nM
|
|
|
CP0542292
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid methylamide
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|
C25H28N4O4S
|
1
|
1 |
Ki = 0.7 nM
|
|
|
CP0529656
|
2-methyl-N-[4-({[1-(pyrrolidin-1-ylcarbonyl)piperidin-4-yl]-amino}sulfonyl)-1-naphthyl]benzamide
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|
C28H32N4O4S
|
1
|
1 |
Ki = 1.1 nM
|
|
|
CP0535436
|
N-[4-[[1-(azetidine-3-carbonyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C27H30N4O4S
|
1
|
1 |
Ki = 1.5 nM
|
|
|
CP0051222
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethyl ester
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|
C26H29N3O5S
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0372525
|
4-({[4-(benzoylamino)-1-naphthyl]sulfonyl}amino)-N,N-dimethylpiperidine-1-carboxamide
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|
C26H30N4O4S
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0439474
|
N-[4-[[1-(4-aminobutanoyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
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|
C27H32N4O4S
|
1
|
1 |
Ki = 1.6 nM
|
|
|
CP0543727
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethylamide
Show/Hide
|
C26H30N4O4S
|
1
|
1 |
Ki = 2.2 nM
|
|
|
CP0420534
|
ethyl 4-[(5-benzamidonaphthalen-1-yl)sulfonylamino]piperidine-1-carboxylate
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|
C25H27N3O5S
|
1
|
1 |
Ki = 2.3 nM
|
|
|
CP0543731
|
2-methyl-N-[4-(1-propionyl-piperidin-4-ylsulfamoyl)-naphthalen-1-yl]-benzamide
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|
C26H29N3O4S
|
1
|
1 |
Ki = 2.5 nM
|
|
|
CP0435925
|
N-[4-[[1-(azetidine-1-carbonyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C27H30N4O4S
|
1
|
1 |
Ki = 3.5 nM
|
|
|
CP0543730
|
N-[4-[[1-(2-aminoacetyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
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|
C25H28N4O4S
|
1
|
1 |
Ki = 4.1 nM
|
|
|
CP0435924
|
2-methyl-N-{4-[1-(4-methyl-piperazine-1-carbonyl)-piperidin-4-ylsulfamoyl]-aphthalen-1-yl}-benzamide
Show/Hide
|
C29H35N5O4S
|
1
|
1 |
Ki = 4.2 nM
|
|
|
CP0453753
|
2-methyl-N-{4-[1-(piperidine-1-carbonyl)-piperidin-4-ylsulfamoyl]-naphthalen-1-yl}-benzamide
Show/Hide
|
C29H34N4O4S
|
1
|
1 |
Ki = 4.2 nM
|
|
|
CP0543726
|
N-[4-(cyclohexylsulfamoyl)naphthalen-1-yl]benzamide
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|
C23H24N2O3S
|
1
|
1 |
Ki = 4.4 nM
|
|
|
CP0405759
|
4-(4-o-tolylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C26H29N3O5S
|
1
|
1 |
Ki = 5.21 nM
|
|
|
CP0536552
|
N-[4-[[1-(2-hydroxyacetyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C25H27N3O5S
|
1
|
1 |
Ki = 5.4 nM
|
|
|
CP0529655
|
2-methyl-N-[4-({[1-(morpholin-4-ylcarbonyl)piperidin-4-yl]-amino}sulfonyl)-1-naphthyl]benzamide
Show/Hide
|
C28H32N4O5S
|
1
|
1 |
Ki = 6.3 nM
|
|
|
CP0529654
|
N-[4-[(1-acetylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C25H27N3O4S
|
1
|
1 |
Ki = 6.7 nM
|
|
|
CP0453752
|
N-[4-[[1-(cyclopropanecarbonyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
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|
C27H29N3O4S
|
1
|
1 |
Ki = 7.2 nM
|
|
|
CP0439475
|
N-[4-[[1-(cyclopentanecarbonyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
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|
C29H33N3O4S
|
1
|
1 |
Ki = 9.1 nM
|
|
|
CP0448822
|
4-(4-cyclohexylcarbamoyl-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester
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|
C25H33N3O5S
|
1
|
1 |
Ki = 9.5 nM
|
|
|
CP0543729
|
N-[4-[[1-(3-aminopropanoyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C26H30N4O4S
|
1
|
1 |
Ki = 11.3 nM
|
|
|
CP0537859
|
4-(4-benzoylamino-naphthalene-1-sulfonylamino)-piperidine-1-carboxylic acid tert-butyl ester
Show/Hide
|
C27H31N3O5S
|
1
|
1 |
Ki = 15.2 nM
|
|
|
CP0453751
|
N-[4-[[1-(2-methoxyacetyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C26H29N3O5S
|
1
|
1 |
Ki = 15.8 nM
|
|
|
CP0552419
|
ethyl 4-[(4-benzoyloxynaphthalen-1-yl)sulfonylamino]piperidine-1-carboxylate
Show/Hide
|
C25H26N2O6S
|
1
|
1 |
Ki = 16.4 nM
|
|
|
CP0132457
|
1-[3-(2-chlorophenoxy)benzyl]-4-{[(1-ethyl-4-phenylpiperidin-4-yl)carbonyl]amino} piperidine-4-carboxylic acid
Show/Hide
|
C33H38ClN3O4
|
1
|
1 |
Ki = 23 nM
|
|
|
CP0435617
|
4-{4-[(3-phenyl-propylamino)-methyl]-naphthalene-1-sulfonylamino}-piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C27H33N3O4S
|
1
|
1 |
Ki = 32.1 nM
|
|
|
CP0432649
|
((+/-)-N-(4-{[(1-butyrylpyrrolidin-3-yl)amino]sulfonyl}-1-naphthyl)-2-methylbenzamide
Show/Hide
|
C26H29N3O4S
|
1
|
1 |
Ki = 34.3 nM
|
|
|
CP0456889
|
4-[4-(phenethylamino-methyl)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C26H31N3O4S
|
1
|
1 |
Ki = 35.7 nM
|
|
|
CP0525523
|
ethyl 4-[(4-phenylmethoxynaphthalen-1-yl)sulfonylamino]piperidine-1-carboxylate
Show/Hide
|
C25H28N2O5S
|
1
|
1 |
Ki = 37.9 nM
|
|
|
CP0505231
|
N-[4-[(4-methoxyphenyl)sulfamoyl]naphthalen-1-yl]benzamide
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|
C24H20N2O4S
|
1
|
1 |
Ki = 42.6 nM
|
|
|
CP0405757
|
4-[4-(benzylamino-methyl)-naphthalene-1-sulfonylamino]piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C25H29N3O4S
|
1
|
1 |
Ki = 45.6 nM
|
|
|
CP0435921
|
N-[4-[(1-butanoylazetidin-3-yl)sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C25H27N3O4S
|
1
|
1 |
Ki = 50.9 nM
|
|
|
CP0192971
|
1-[3-(2-methoxy-phenoxy)-benzyl]-4-[(4-phenyl-piperidine-4-carbonyl)-amino]-piperidine-4-carboxylic acid
Show/Hide
|
C32H37N3O5
|
1
|
1 |
Ki = 60 nM
|
|
|
CP0524628
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid (3-morpholin-4-yl-propyl)-amide
Show/Hide
|
C31H38N4O5S
|
1
|
1 |
Ki = 71 nM
|
|
|
CP0543732
|
4-[({4-[(2-methylbenzoyl)amino]-1-naphthyl}sulfonyl)amino]-N-propylpiperidine-1-carboxamide
Show/Hide
|
C27H32N4O4S
|
1
|
1 |
Ki = 77.4 nM
|
|
|
CP0439476
|
4-[[4-[(2-methylbenzoyl)amino]naphthalen-1-yl]sulfonylamino]-N-propan-2-ylpiperidine-1-carboxamide
Show/Hide
|
C27H32N4O4S
|
1
|
1 |
Ki = 77.7 nM
|
|
|
CP0435922
|
N-[4-[(1-benzoylpiperidin-4-yl)sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C30H29N3O4S
|
1
|
1 |
Ki = 81.1 nM
|
|
|
CP0529657
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid phenylamide
Show/Hide
|
C30H30N4O4S
|
1
|
1 |
Ki = 108 nM
|
|
|
CP0543728
|
N-[4-[[1-[4-(dimethylamino)benzoyl]piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C32H34N4O4S
|
1
|
1 |
Ki = 114 nM
|
|
|
CP0552418
|
ethyl 4-[[4-(piperidine-1-carbonylamino)naphthalen-1-yl]sulfonylamino]piperidine-1-carboxylate
Show/Hide
|
C24H32N4O5S
|
1
|
1 |
Ki = 125.6 nM
|
|
|
CP0432650
|
N-[4-[[1-(5-aminopentanoyl)piperidin-4-yl]sulfamoyl]naphthalen-1-yl]-2-methylbenzamide
Show/Hide
|
C28H34N4O4S
|
1
|
1 |
Ki = 199 nM
|
|
|
CP0539681
|
N-[4-(benzylsulfamoyl)naphthalen-1-yl]benzamide
Show/Hide
|
C24H20N2O3S
|
1
|
1 |
Ki = 233.1 nM
|
|
|
CP0372526
|
4-(1-(2-methylbenzamido)naphthalene-4-sulfonamido)piperidine-1-carboxamide
Show/Hide
|
C24H26N4O4S
|
1
|
1 |
Ki = 243 nM
|
|
|
CP0166152
|
1-(4-chloro-phenyl)-cyclohexanecarboxylic acid {1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl}-amide
Show/Hide
|
C32H37ClN2O3
|
1
|
1 |
Ki = 250 nM
|
|
|
CP0541871
|
4-[4-(2-methyl-benzoylamino)-naphthalene-1-sulfonylamino]-piperidine-1-carboxylic acid (3-diethylamino-propyl)-amide
Show/Hide
|
C31H40N4O4S
|
1
|
1 |
Ki = 566.5 nM
|
|
|
CP0562405
|
N-[4-(piperidin-4-ylsulfamoyl)naphthalen-1-yl]benzamide
Show/Hide
|
C22H23N3O3S
|
1
|
1 |
Ki = 578 nM
|
|
|
CP0140721
|
N-[1-[(3-phenoxyphenyl)methyl]piperidin-4-yl]-2-phenylacetamide
Show/Hide
|
C26H28N2O2
|
1
|
1 |
Ki = 1400 nM
|
|
|
CP0378509
|
N-[4-(phenylsulfamoyl)naphthalen-1-yl]benzamide
Show/Hide
|
C23H18N2O3S
|
1
|
1 |
Ki = 1760 nM
|
|
|
CP0541872
|
4-(8-benzoylamino-naphthalene-2-sulfonylamino)-piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C25H27N3O5S
|
1
|
1 |
Ki = 2033 nM
|
|
|
CP0166151
|
1-(3-phenoxy-benzyl)-piperidine-4-carboxylic acid ethyl ester
Show/Hide
|
C21H25NO3
|
1
|
1 |
Ki = 2600 nM
|
|
|
CP0525525
|
N-[4-(pyridin-4-ylmethylsulfamoyl)naphthalen-1-yl]benzamide
Show/Hide
|
C23H19N3O3S
|
1
|
1 |
Ki = 3277 nM
|
|
|
CP0453722
|
N-(4-morpholin-4-ylsulfonylnaphthalen-1-yl)benzamide
Show/Hide
|
C21H20N2O4S
|
1
|
1 |
Ki = 7745 nM
|
|
|
CP0134897
|
1-(3-phenoxy-benzyl)-piperidine-4-carboxylic acid ethylamide
Show/Hide
|
C21H26N2O2
|
1
|
1 |
Ki = 9100 nM
|
|
|
CP0153419
|
N-[1-[(3-phenoxyphenyl)methyl]piperidin-4-yl]propanamide
Show/Hide
|
C21H26N2O2
|
1
|
1 |
Ki = 9200 nM
|
|
|
CP0524627
|
N-[4-[(4-methoxyphenyl)sulfamoyl]naphthalen-1-yl]-N-methylbenzamide
Show/Hide
|
C25H22N2O4S
|
1
|
1 |
Ki > 15000 nM
|
|
|
CP0425114
|
N-[4-(4-methylpiperazin-1-yl)sulfonylnaphthalen-1-yl]benzamide
Show/Hide
|
C22H23N3O3S
|
1
|
1 |
Ki > 30000 nM
|
|
|
CP0505233
|
N-(4-piperidin-1-ylsulfonylnaphthalen-1-yl)benzamide
Show/Hide
|
C22H22N2O3S
|
1
|
1 |
Ki > 30000 nM
|
|
|
CP0511884
|
N-[4-(diethylsulfamoyl)naphthalen-1-yl]benzamide
Show/Hide
|
C21H22N2O3S
|
1
|
1 |
Ki > 30000 nM
|
|
|
CP0421193
|
1-(3-phenoxybenzyl)piperidine-4-carboxylic acid
Show/Hide
|
C19H21NO3
|
1
|
1 |
Ki > 30000 nM
|
|
|
CP0378513
|
4-[6-(2-methyl-benzoylamino)-naphthalene-2-sulfonylamino]-piperidine-1-carboxylic acid ethyl ester
Show/Hide
|
C26H29N3O5S
|
1
|
1 |
Ki > 44000 nM
|
|
|
CP0402725
|
N-[4-[methyl(phenyl)sulfamoyl]naphthalen-1-yl]benzamide
Show/Hide
|
C24H20N2O3S
|
1
|
1 |
Ki > 44000 nM
|
|
|
CP0505234
|
4-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-naphthalene-1-sulfonic acid (4-methoxy phenyl)-amide
Show/Hide
|
C25H18N2O5S
|
1
|
1 |
Ki > 44000 nM
|
|
|
CP0373456
|
ethyl 4-[(4-aminonaphthalen-1-yl)sulfonylamino]piperidine-1-carboxylate
Show/Hide
|
C18H23N3O4S
|
1
|
1 |
Ki > 5000 nM
|
|
|
CP0536589
|
ethyl 4-[(4-hydroxynaphthalen-1-yl)sulfonylamino]piperidine-1-carboxylate
Show/Hide
|
C18H22N2O5S
|
1
|
1 |
Ki > 5000 nM
|
|
|