| Compound ID |
Compound Name |
Compound Formula |
|
CP0689386
|
methyl 4-((R)-1-((1S,3R,4S)-3-amino-4-hydroxycyclopentanecarbonyl)piperidin-3-yl)-4-(6-chloro-3'-ethylbiphenyl-2-yl)-4-hydroxybutylcarbamate
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C31H42ClN3O5
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
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CP0567608
|
2-tert-butyl-4-(furan-2-ylmethylamino)-N-(2-methylpropyl)-N-[(3S)-piperidin-3-yl]pyrimidine-5-carboxamide
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|
C23H35N5O2
|
1
|
| 1 |
IC50 = 0.58 nM
|
|
|
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CP0228492
|
methyl N-[4-[(3R)-1-[(1R,3S)-3-aminocyclopentanecarbonyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
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|
C31H42FN3O4
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
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CP0228493
|
methyl N-[4-[3-chloro-2-(3-ethylphenyl)phenyl]-4-hydroxy-4-[(3R)-1-[(1R,3S)-3-(methylamino)cyclopentanecarbonyl]piperidin-3-yl]butyl]carbamate
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|
C32H44ClN3O4
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
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CP0689241
|
methyl 4-(6-chloro-3'-ethylbiphenyl-2-yl)-4-hydroxy-4-((R)-1-(4-(methylamino)butanoyl)piperidin-3-yl)butylcarbamate
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|
C30H42ClN3O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
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CP0865214
|
methyl 4-((R)-1-(4-aminobutanoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
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|
C29H40FN3O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
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CP0445817
|
methyl (3S,5R)-5-[[2-tert-butyl-4-(furan-2-ylmethylamino)pyrimidine-5-carbonyl]-(2-methylpropyl)amino]piperidine-3-carboxylate
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|
C25H37N5O4
|
1
|
| 1 |
IC50 = 1.2 nM
|
|
|
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CP0085985
|
methyl N-[4-[(3R)-1-[(3S)-4-amino-3-hydroxybutanoyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
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|
C29H40FN3O5
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
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CP0673266
|
methyl 4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxy-4-((R)-1-(4-(methylamino)butanoyl)piperidin-3-yl)butylcarbamate
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|
C30H42FN3O4
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
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CP0398673
|
2-tert-butyl-N-[(3S,5R)-5-carbamoylpiperidin-3-yl]-4-(3-methoxypropylamino)-N-(2-methylpropyl)pyrimidine-5-carboxamide
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|
C23H40N6O3
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0074456
|
2-tert-butyl-4-(3-methoxypropylamino)-N-(2-methylpropyl)-N-[(3S,5R)-5-(morpholine-4-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
Show/Hide
|
C27H46N6O4
|
1
|
| 1 |
IC50 = 1.5 nM
|
|
|
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CP0369555
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(2-piperidin-4-ylacetyl)piperidin-3-yl]butyl]carbamate
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|
C32H44FN3O4
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
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CP0766749
|
methyl 4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxy-4-((3R)-1-(2-(morpholin-2-yl)acetyl)piperidin-3-yl)butylcarbamate
Show/Hide
|
C31H42FN3O5
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
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CP0369554
|
methyl N-[4-[(3R)-1-(5-aminopentanoyl)piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
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|
C30H42FN3O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0471782
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(2-piperidin-3-ylacetyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C32H44FN3O4
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0684961
|
methyl 4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxy-4-((3R)-1-(3-hydroxy-4-(methylamino)butanoyl)piperidin-3-yl)butylcarbamate
Show/Hide
|
C30H42FN3O5
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0757362
|
methyl 4-((3R)-1-(4-amino-3-hydroxybutanoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
Show/Hide
|
C29H40FN3O5
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
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CP0965060
|
methyl 4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxy-4-((R)-1-(4-(2-hydroxyethylamino)butanoyl)piperidin-3-yl)butylcarbamate
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|
C31H44FN3O5
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
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CP0477606
|
methyl (3R,5S)-5-[[2-tert-butyl-4-(3-methoxypropylamino)pyrimidine-5-carbonyl]-(2-methylpropyl)amino]piperidine-3-carboxylate
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|
C24H41N5O4
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
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CP0117902
|
methyl N-[4-[(3R)-1-[(1R,3S)-3-aminocyclopentanecarbonyl]piperidin-3-yl]-4-[3-chloro-2-(3-ethylphenyl)phenyl]-4-hydroxybutyl]carbamate
Show/Hide
|
C31H42ClN3O4
|
1
|
| 1 |
IC50 = 3.1 nM
|
|
|
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CP0705220
|
methyl 4-((R)-1-(2-aminoethylcarbamoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
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|
C28H39FN4O4
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
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CP0762386
|
methyl 4-((R)-1-(6-aminohexanoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
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|
C31H44FN3O4
|
1
|
| 1 |
IC50 = 3.2 nM
|
|
|
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CP0507014
|
methyl (3S,5S)-5-[[2-tert-butyl-4-(furan-2-ylmethylamino)pyrimidine-5-carbonyl]-(2-methylpropyl)amino]piperidine-3-carboxylate
Show/Hide
|
C25H37N5O4
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
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CP0110370
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-[3-methoxy-4-(methylamino)butanoyl]piperidin-3-yl]butyl]carbamate
Show/Hide
|
C31H44FN3O5
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
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CP0255937
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-[2-(methylamino)ethylcarbamoyl]piperidin-3-yl]butyl]carbamate
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|
C29H41FN4O4
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
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CP0412181
|
methyl N-[4-[(3R)-1-[(4R)-4-amino-5-hydroxypentanoyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
Show/Hide
|
C30H42FN3O5
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
|
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CP0766748
|
methyl 4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxy-4-((R)-1-(piperidine-4-carbonyl)piperidin-3-yl)butylcarbamate
Show/Hide
|
C31H42FN3O4
|
1
|
| 1 |
IC50 = 6.3 nM
|
|
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CP0541269
|
benzyl (2S)-2-amino-5-[(3R)-3-[1-[2-(3-ethylphenyl)-3-fluorophenyl]-1-hydroxy-4-(methoxycarbonylamino)butyl]piperidin-1-yl]-5-oxopentanoate
Show/Hide
|
C37H46FN3O6
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
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CP0902964
|
methyl 4-((R)-1-((S)-4-amino-5-hydroxypentanoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
Show/Hide
|
C30H42FN3O5
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
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CP0568689
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(pyrrolidine-3-carbonyl)piperidin-3-yl]butyl]carbamate
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|
C30H40FN3O4
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
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CP0725657
|
(2S)-methyl 2-amino-5-((3R)-3-(1-(3'-ethyl-6-fluorobiphenyl-2-yl)-1-hydroxy-4-(methoxycarbonylamino)butyl)piperidin-1-yl)-5-oxopentanoate
Show/Hide
|
C31H42FN3O6
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
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CP0254722
|
2-tert-butyl-4-hexyl-N-(2-methylpropyl)-N-[(3S,5R)-5-(morpholine-4-carbonyl)piperidin-3-yl]pyrimidine-5-carboxamide
Show/Hide
|
C29H49N5O3
|
1
|
| 1 |
IC50 = 29 nM
|
|
|
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CP0117900
|
methyl N-[4-[(3R)-1-[(2S)-4-amino-2-hydroxybutanoyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
Show/Hide
|
C29H40FN3O5
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
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CP0905323
|
methyl 4-((R)-1-(2-aminoacetyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
Show/Hide
|
C27H36FN3O4
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
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CP0476978
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(3-piperidin-4-ylpropanoyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C33H46FN3O4
|
1
|
| 1 |
IC50 = 80 nM
|
|
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CP0965059
|
methyl 4-((R)-1-(3-aminopropanoyl)piperidin-3-yl)-4-(3'-ethyl-6-fluorobiphenyl-2-yl)-4-hydroxybutylcarbamate
Show/Hide
|
C28H38FN3O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
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CP0072456
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(3-piperidin-2-ylpropanoyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C33H46FN3O4
|
1
|
| 1 |
IC50 = 126 nM
|
|
|
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CP0228491
|
methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(piperidine-3-carbonyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C31H42FN3O4
|
1
|
| 1 |
IC50 = 320 nM
|
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CP0412465
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(2S)-2-amino-5-[(3R)-3-[1-[2-(3-ethylphenyl)-3-fluorophenyl]-1-hydroxy-4-(methoxycarbonylamino)butyl]piperidin-1-yl]-5-oxopentanoic acid
Show/Hide
|
C30H40FN3O6
|
1
|
| 1 |
IC50 = 320 nM
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CP0189137
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methyl N-[4-[(3R)-1-[4-(dimethylamino)butanoyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
Show/Hide
|
C31H44FN3O4
|
1
|
| 1 |
IC50 = 630 nM
|
|
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CP0541270
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methyl N-[4-[(3R)-1-[(4S)-4,5-diamino-5-oxopentanoyl]piperidin-3-yl]-4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxybutyl]carbamate
Show/Hide
|
C30H41FN4O5
|
1
|
| 1 |
IC50 = 630 nM
|
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CP0476979
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methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(2-pyrrolidin-2-ylacetyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C31H42FN3O4
|
1
|
| 1 |
IC50 = 800 nM
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CP0396350
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methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(morpholine-2-carbonyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C30H40FN3O5
|
1
|
| 1 |
IC50 = 1000 nM
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CP0230269
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methyl N-[4-[2-(3-ethylphenyl)-3-fluorophenyl]-4-hydroxy-4-[(3R)-1-(piperidine-2-carbonyl)piperidin-3-yl]butyl]carbamate
Show/Hide
|
C31H42FN3O4
|
1
|
| 1 |
IC50 = 2000 nM
|
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