Compound ID |
Compound Name |
Compound Formula |
CP0545727
|
2-amino-5-(1-methyl-1H-pyrazol-4-yl)-N-((1S,2S)-2-((4′-((4-methylpiperazin-1-yl)methyl)-[1,1′-biphenyl]-4-yl)methoxy)cyclopentyl)nicotinamide
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C34H41N7O2
|
1
|
1 |
IC50 = 31.62 nM
|
|
|
CP0514791
|
N-methyl-N-[[3-(1-methylpyrazol-4-yl)imidazo[1,2-a]pyridin-6-yl]methyl]-5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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C28H29N9O
|
1
|
1 |
IC50 = 63.1 nM
|
|
|
CP0552479
|
N-[[3-[4-[(dimethylamino)methyl]phenyl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C32H35N9O
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0480273
|
N-[[3-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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|
C31H36N10O
|
1
|
1 |
IC50 = 125.89 nM
|
|
|
CP0527506
|
N-[[3-[5-[(dimethylamino)methyl]pyridin-2-yl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C31H34N10O
|
1
|
1 |
IC50 = 125.89 nM
|
|
|
CP0480272
|
N-methyl-5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-N-[(3-phenylimidazo[1,2-a]pyridin-6-yl)methyl]-1,3,4-oxadiazol-2-amine
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|
C30H29N7O
|
1
|
1 |
IC50 = 199.53 nM
|
|
|
CP0514792
|
N-[[3-[3-[(dimethylamino)methyl]phenyl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C32H35N9O
|
1
|
1 |
IC50 = 316.23 nM
|
|
|
CP0245111
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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|
C24H25N7O
|
1
|
1 |
IC50 = 398.11 nM
|
|
|
CP0480271
|
N,N-dimethyl-6-[[methyl-[5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-yl]amino]methyl]imidazo[1,2-a]pyridine-3-carboxamide
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|
C27H30N8O2
|
1
|
1 |
IC50 = 398.11 nM
|
|
|
CP0545741
|
4-[4-[5-[imidazo[1,2-a]pyridin-6-ylmethyl(methyl)amino]-1,3,4-oxadiazol-2-yl]-3-methylphenyl]-2,5-dimethylpyrazole-3-carbonitrile
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|
C24H22N8O
|
1
|
1 |
IC50 = 398.11 nM
|
|
|
CP0354548
|
5-[4-(1,5-dimethylpyrazol-4-yl)-2-methylphenyl]-N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
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|
C23H23N7O
|
1
|
1 |
IC50 = 794.33 nM
|
|
|
CP0494149
|
5-[2-chloro-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
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|
C23H22ClN7O
|
1
|
1 |
IC50 = 794.33 nM
|
|
|
CP0548059
|
N-[[3-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C30H35N11O
|
1
|
1 |
IC50 = 1000 nM
|
|
|
CP0494150
|
N-methyl-N-[[3-(1-methylpiperidin-4-yl)imidazo[1,2-a]pyridin-6-yl]methyl]-5-[2-methyl-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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|
C30H36N8O
|
1
|
1 |
IC50 = 1258.93 nM
|
|
|
CP0494159
|
N-[[3-[6-[(dimethylamino)methyl]pyridin-3-yl]imidazo[1,2-a]pyridin-6-yl]methyl]-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C31H34N10O
|
1
|
1 |
IC50 = 1584.89 nM
|
|
|
CP0257794
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-5-[2-methoxy-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-N-methyl-1,3,4-oxadiazol-2-amine
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|
C24H25N7O2
|
1
|
1 |
IC50 = 1995.26 nM
|
|
|
CP0343136
|
5-[2-fluoro-4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
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|
C23H22FN7O
|
1
|
1 |
IC50 = 3162.28 nM
|
|
|
CP0553528
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[4-(1,3,5-trimethylpyrazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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|
C23H23N7O
|
1
|
1 |
IC50 = 3162.28 nM
|
|
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CP0480275
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[2-methyl-4-(2,3,5-trimethylimidazol-4-yl)phenyl]-1,3,4-oxadiazol-2-amine
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|
C24H25N7O
|
1
|
1 |
IC50 = 5011.87 nM
|
|
|
CP0487262
|
4-[4-[5-[imidazo[1,2-a]pyridin-6-ylmethyl(methyl)amino]-1,3,4-oxadiazol-2-yl]-3-methylphenyl]-1,5-dimethylpyrazole-3-carbonitrile
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|
C24H22N8O
|
1
|
1 |
IC50 = 6309.57 nM
|
|
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CP0554525
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[3-methyl-5-(1,3,5-trimethylpyrazol-4-yl)pyridin-2-yl]-1,3,4-oxadiazol-2-amine
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|
C23H24N8O
|
1
|
1 |
IC50 = 6309.57 nM
|
|
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CP0245112
|
5-[4-[1-(difluoromethyl)-3,5-dimethylpyrazol-4-yl]-2-methylphenyl]-N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
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|
C24H23F2N7O
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0368045
|
N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-5-[2-methyl-6-(1,3,5-trimethylpyrazol-4-yl)pyridin-3-yl]-1,3,4-oxadiazol-2-amine
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|
C23H24N8O
|
1
|
1 |
IC50 = 10000 nM
|
|
|
CP0271463
|
5-[4-(3,5-dimethyl-1H-pyrazol-4-yl)-2-methylphenyl]-N-(imidazo[1,2-a]pyridin-6-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
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|
C23H23N7O
|
1
|
1 |
IC50 = 15848.93 nM
|
|
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CP0540377
|
2-[5-[imidazo[1,2-a]pyridin-6-ylmethyl(methyl)amino]-1,3,4-oxadiazol-2-yl]-5-(1,3,5-trimethylpyrazol-4-yl)benzonitrile
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|
C24H22N8O
|
1
|
1 |
IC50 > 31622.78 nM
|
|
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