| Compound ID |
Compound Name |
Compound Formula |
|
CP0129530
|
US9090625, 4
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|
C18H16N4S
|
1
|
| 1 |
IC50 = 21.5 nM
|
|
|
|
CP0300059
|
US9090625, 5
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|
C19H16N4S
|
1
|
| 1 |
IC50 = 30.8 nM
|
|
|
|
CP0519620
|
US9090625, 7
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|
C17H14N4S
|
1
|
| 1 |
IC50 = 35.9 nM
|
|
|
|
CP0326838
|
US9090625, 12
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|
C17H14N4S
|
1
|
| 1 |
IC50 = 42.5 nM
|
|
|
|
CP0532071
|
N-[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]-2-(4-propan-2-ylpiperazin-1-yl)pyridin-4-amine
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|
C28H37N7O2
|
1
|
| 1 |
IC50 = 54.9 nM
|
|
|
|
CP0327400
|
US9090625, 13
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|
C19H16N4S
|
1
|
| 1 |
IC50 = 57.5 nM
|
|
|
|
CP0341877
|
5-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]-2-methylbenzenesulfonamide
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|
C23H27N5O4S
|
1
|
| 1 |
IC50 = 69.5 nM
|
|
|
|
CP0352360
|
4-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]-2-(3-hydroxy-3-methylazetidin-1-yl)benzonitrile
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|
C27H30N6O3
|
1
|
| 1 |
IC50 = 85.9 nM
|
|
|
|
CP0484910
|
3-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]-N-methylbenzenesulfonamide
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|
C23H27N5O4S
|
1
|
| 1 |
IC50 = 92.7 nM
|
|
|
|
CP0322659
|
5-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]-2-fluorobenzenesulfonamide
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|
C22H24FN5O4S
|
1
|
| 1 |
IC50 = 126.4 nM
|
|
|
|
CP0479648
|
4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxy-N-[1-(oxan-4-yl)pyrazol-4-yl]pyridin-2-amine
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|
C24H30N6O3
|
1
|
| 1 |
IC50 = 128.3 nM
|
|
|
|
CP0322656
|
4-N-[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]-2-N-(oxan-4-yl)pyridine-2,4-diamine
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|
C26H32N6O3
|
1
|
| 1 |
IC50 = 133.4 nM
|
|
|
|
CP0137007
|
US9090625, 1
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|
C16H12N4S
|
1
|
| 1 |
IC50 = 149 nM
|
|
|
|
CP0367498
|
3-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]benzenesulfonamide
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|
C22H25N5O4S
|
1
|
| 1 |
IC50 = 167.7 nM
|
|
|
|
CP0553100
|
1-[4-[[4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxypyridin-2-yl]amino]pyrazol-1-yl]-2-methylpropan-2-ol
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|
C23H30N6O3
|
1
|
| 1 |
IC50 = 215.2 nM
|
|
|
|
CP0566315
|
US9090625, 6
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|
C18H16N4S
|
1
|
| 1 |
IC50 = 244 nM
|
|
|
|
CP0484909
|
4-[1-cyclopropyl-3-(oxan-4-yl)pyrazol-4-yl]oxy-N-[1-[(3-methyloxetan-3-yl)methyl]pyrazol-4-yl]pyridin-2-amine
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|
C24H30N6O3
|
1
|
| 1 |
IC50 = 338 nM
|
|
|
|
CP0300058
|
US9090625, 3
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|
C18H16N4S
|
1
|
| 1 |
IC50 = 403 nM
|
|
|
|
CP0326837
|
US9090625, 2
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|
C17H14N4S
|
1
|
| 1 |
IC50 = 440 nM
|
|
|
