| Compound ID |
Compound Name |
Compound Formula |
|
CP0355865
|
N-[6-[4-[(2S)-1,1-difluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3-methoxy-1-methylpyrazole-4-carboxamide
Show/Hide
|
C16H17F2N7O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0569729
|
N-[6-[4-(2,2-difluorocyclobutyl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3-methoxy-1-methylpyrazole-4-carboxamide
Show/Hide
|
C17H17F2N7O2
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0419295
|
1-(cyclopropylmethyl)-3-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C19H20F3N7O2
|
1
|
| 1 |
IC50 = 9 nM
|
|
|
|
CP0163184
|
3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-pyridin-3-ylpyrazole-4-carboxamide
Show/Hide
|
C20H20N8O2
|
1
|
| 1 |
IC50 = 11 nM
|
|
|
|
CP0125694
|
1-(cyclopropylmethyl)-3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
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|
C19H23N7O2
|
1
|
| 1 |
IC50 = 12 nM
|
|
|
|
CP0247995
|
N-[5-(cyclopropylamino)-7-(trifluoromethyl)-[1,2,4]triazolo[1,5-a]pyridin-2-yl]pyridine-3-carboxamide
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|
C16H13F3N6O
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0176881
|
1-ethyl-3-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H18F3N7O2
|
1
|
| 1 |
IC50 = 13 nM
|
|
|
|
CP0555055
|
3-methoxy-1-(2-methoxyethyl)-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C18H20F3N7O3
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
|
CP0564283
|
3-methoxy-1-methyl-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C16H16F3N7O2
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0217203
|
GS-4997
Show/Hide
|
C24H24FN7O
|
1
|
| 1 |
IC50 = 20 nM
|
|
|
|
CP0416385
|
1-[5-(dimethylamino)pyridin-3-yl]-3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C22H25N9O2
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0368691
|
1-ethyl-3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H21N7O2
|
1
|
| 1 |
IC50 = 22 nM
|
|
|
|
CP0519313
|
15-(1-methylpyrazol-4-yl)-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C22H21N7O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0176879
|
5-fluoro-2-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyridine-3-carboxamide
Show/Hide
|
C17H14F4N6O2
|
1
|
| 1 |
IC50 = 25 nM
|
|
|
|
CP0176878
|
2-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyridine-3-carboxamide
Show/Hide
|
C17H15F3N6O2
|
1
|
| 1 |
IC50 = 27 nM
|
|
|
|
CP0326338
|
15-(4-methylimidazol-1-yl)-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C22H21N7O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0354744
|
1-(5-cyclopropylpyridin-3-yl)-3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C23H24N8O2
|
1
|
| 1 |
IC50 = 28 nM
|
|
|
|
CP0176880
|
3-methoxy-1-methyl-N-[6-[4-[1-(trifluoromethyl)cyclopropyl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H16F3N7O2
|
1
|
| 1 |
IC50 = 31 nM
|
|
|
|
CP0125432
|
(7S)-7,14-dimethyl-11-oxa-3,4,6,13,14,18,23-heptazatetracyclo[17.3.1.02,6.012,16]tricosa-1(23),2,4,12,15,19,21-heptaen-17-one
Show/Hide
|
C17H19N7O2
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0354743
|
3-methoxy-1-(2-methoxyethyl)-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C18H23N7O3
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0546434
|
3-methoxy-1-(2,2,2-trifluoroethyl)-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H15F6N7O2
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0326339
|
(8R)-15-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]-14-fluoro-8-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C26H29FN8O2
|
1
|
| 1 |
IC50 = 37 nM
|
|
|
|
CP0558673
|
3-methoxy-1-methyl-N-[6-[4-(1,1,1-trifluoropropan-2-yl)-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C16H16F3N7O2
|
1
|
| 1 |
IC50 = 40 nM
|
|
|
|
CP0402033
|
(7S)-14-fluoro-7-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C19H18FN5O2
|
1
|
| 1 |
IC50 = 43 nM
|
|
|
|
CP0561697
|
3-methoxy-1-pyridazin-3-yl-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C19H16F3N9O2
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0570837
|
N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]quinoxaline-5-carboxamide
Show/Hide
|
C19H14F3N7O
|
1
|
| 1 |
IC50 = 50 nM
|
|
|
|
CP0555056
|
2-methoxy-5-methyl-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyridine-3-carboxamide
Show/Hide
|
C18H17F3N6O2
|
1
|
| 1 |
IC50 = 51 nM
|
|
|
|
CP0546435
|
2-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]benzamide
Show/Hide
|
C18H16F3N5O2
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0444649
|
3-methoxy-1-pyrazin-2-yl-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C19H16F3N9O2
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0565299
|
N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]quinoline-8-carboxamide
Show/Hide
|
C20H15F3N6O
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0402031
|
(7S)-7-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 73 nM
|
|
|
|
CP0125433
|
3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-pyrimidin-5-ylpyrazole-4-carboxamide
Show/Hide
|
C19H19N9O2
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0368689
|
3-methoxy-1-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C16H19N7O2
|
1
|
| 1 |
IC50 = 90 nM
|
|
|
|
CP0354745
|
3-methoxy-1-methyl-N-[6-(3-propan-2-ylimidazol-4-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H20N6O2
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0233898
|
(8R)-14-fluoro-8-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C19H18FN5O2
|
1
|
| 1 |
IC50 = 95 nM
|
|
|
|
CP0259270
|
15-morpholin-4-yl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C22H24N6O3
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0561696
|
3-methoxy-1-methyl-N-[6-[4-[(3R)-oxolan-3-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H19N7O3
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0163191
|
3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-pyrazin-2-ylpyrazole-4-carboxamide
Show/Hide
|
C19H19N9O2
|
1
|
| 1 |
IC50 = 138 nM
|
|
|
|
CP0517074
|
N-[6-[4-[(2R)-1,1-difluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-3-methoxy-1-methylpyrazole-4-carboxamide
Show/Hide
|
C16H17F2N7O2
|
1
|
| 1 |
IC50 = 143 nM
|
|
|
|
CP0561695
|
3-methoxy-1-methyl-N-[6-[4-[(3S)-oxolan-3-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C17H19N7O3
|
1
|
| 1 |
IC50 = 144 nM
|
|
|
|
CP0402034
|
15-[1-[2-(dimethylamino)ethyl]pyrazol-4-yl]-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C25H28N8O2
|
1
|
| 1 |
IC50 = 148 nM
|
|
|
|
CP0552416
|
4-methyl-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-2,3-dihydro-1,4-benzoxazine-8-carboxamide
Show/Hide
|
C20H19F3N6O2
|
1
|
| 1 |
IC50 = 187 nM
|
|
|
|
CP0188712
|
(8R)-8-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 232 nM
|
|
|
|
CP0326337
|
15-(2-oxa-6-azaspiro[3.3]heptan-6-yl)-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C23H24N6O3
|
1
|
| 1 |
IC50 = 253 nM
|
|
|
|
CP0356980
|
N-[4-(6,7-dimethoxyquinolin-4-yl)oxyphenyl]-4-oxo-1-propan-2-ylquinoline-3-carboxamide
Show/Hide
|
C30H27N3O5
|
1
|
| 1 |
IC50 = 277 nM
|
|
|
|
CP0557207
|
2-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
Show/Hide
|
C18H19N5O2
|
1
|
| 1 |
IC50 = 299 nM
|
|
|
|
CP0540783
|
3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-pyridin-2-ylpyrazole-4-carboxamide
Show/Hide
|
C20H20N8O2
|
1
|
| 1 |
IC50 = 299 nM
|
|
|
|
CP0570802
|
4-methoxy-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrimidine-5-carboxamide
Show/Hide
|
C16H14F3N7O2
|
1
|
| 1 |
IC50 = 302 nM
|
|
|
|
CP0517075
|
N-[6-[4-(3,3-difluorocyclobutyl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3-methoxy-1-methylpyrazole-4-carboxamide
Show/Hide
|
C17H17F2N7O2
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0565298
|
3-methoxy-1-methyl-N-[6-[4-[(2R)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C16H16F3N7O2
|
1
|
| 1 |
IC50 = 350 nM
|
|
|
|
CP0384160
|
(9R)-9-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 351 nM
|
|
|
|
CP0561313
|
1-methyl-2-oxo-N-[6-[4-[(2S)-1,1,1-trifluoropropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]pyridine-3-carboxamide
Show/Hide
|
C17H15F3N6O2
|
1
|
| 1 |
IC50 = 363 nM
|
|
|
|
CP0564282
|
3-methoxy-N-[6-[4-[(2R)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-1-methylpyrazole-4-carboxamide
Show/Hide
|
C17H21N7O3
|
1
|
| 1 |
IC50 = 403 nM
|
|
|
|
CP0356982
|
BDBM50505947
Show/Hide
|
C18H16FN5O2
|
1
|
| 1 |
IC50 = 658 nM
|
|
|
|
CP0534062
|
3-methoxy-N-[6-[4-[(2S)-1-methoxypropan-2-yl]-1,2,4-triazol-3-yl]pyridin-2-yl]-1-methylpyrazole-4-carboxamide
Show/Hide
|
C17H21N7O3
|
1
|
| 1 |
IC50 = 793 nM
|
|
|
|
CP0096219
|
BDBM50505948
Show/Hide
|
C18H16FN5O2
|
1
|
| 1 |
IC50 = 867 nM
|
|
|
|
CP0096218
|
N-[4-(6,7-dimethoxycinnolin-4-yl)oxyphenyl]-4-oxo-1-propan-2-ylquinoline-3-carboxamide
Show/Hide
|
C29H26N4O5
|
1
|
| 1 |
IC50 = 869 nM
|
|
|
|
CP0450705
|
(10S)-10-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 969 nM
|
|
|
|
CP0326335
|
11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C18H17N5O2
|
1
|
| 1 |
IC50 = 1210 nM
|
|
|
|
CP0188713
|
15-methylsulfonyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12(17),13,15,20,22-octaen-18-one
Show/Hide
|
C19H19N5O4S
|
1
|
| 1 |
IC50 = 1437 nM
|
|
|
|
CP0557069
|
3-methoxy-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]-1-pyridin-4-ylpyrazole-4-carboxamide
Show/Hide
|
C20H20N8O2
|
1
|
| 1 |
IC50 = 1710 nM
|
|
|
|
CP0356981
|
12-oxa-3,4,6,20,25-pentazatetracyclo[19.3.1.02,6.013,18]pentacosa-1(25),2,4,13,15,17,21,23-octaen-19-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 1776 nM
|
|
|
|
CP0355864
|
N-[6-[4-(1-hydroxypropan-2-yl)-1,2,4-triazol-3-yl]pyridin-2-yl]-3-methoxy-1-methylpyrazole-4-carboxamide
Show/Hide
|
C16H19N7O3
|
1
|
| 1 |
IC50 = 2895 nM
|
|
|
|
CP0491476
|
2-methoxy-N-[6-(4-methyl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
Show/Hide
|
C16H15N5O2
|
1
|
| 1 |
IC50 = 3735 nM
|
|
|
|
CP0469369
|
(7R)-7-methyl-11-oxa-3,4,6,19,24-pentazatetracyclo[18.3.1.02,6.012,17]tetracosa-1(24),2,4,12,14,16,20,22-octaen-18-one
Show/Hide
|
C19H19N5O2
|
1
|
| 1 |
IC50 = 5152 nM
|
|
|
|
CP0326334
|
10-oxa-3,4,6,18,23-pentazatetracyclo[17.3.1.02,6.011,16]tricosa-1(23),2,4,11,13,15,19,21-octaen-17-one
Show/Hide
|
C17H15N5O2
|
1
|
| 1 |
IC50 = 6065 nM
|
|
|
|
CP0416537
|
1-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-4-carboxamide
Show/Hide
|
C15H17N7O
|
1
|
| 1 |
IC50 = 6797 nM
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CP0188711
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2-fluoro-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
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C17H16FN5O
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1
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| 1 |
IC50 = 8164 nM
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CP0127753
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1-methyl-N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]pyrazole-3-carboxamide
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C15H17N7O
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1
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| 1 |
IC50 > 20000 nM
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CP0339225
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3-methoxy-1-methyl-N-[3-(4-propan-2-yl-1,2,4-triazol-3-yl)phenyl]pyrazole-4-carboxamide
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C17H20N6O2
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1
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| 1 |
IC50 > 20000 nM
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CP0559851
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N-[6-(4-propan-2-yl-1,2,4-triazol-3-yl)pyridin-2-yl]benzamide
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C17H17N5O
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1
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| 1 |
IC50 > 20000 nM
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