| Compound ID |
Compound Name |
Compound Formula |
|
CP0503226
|
4-(3,5-Difluorophenyl)-N-(1-[2-chlorophenyl]-3-phenyl-1H-pyrazol-5-yl)picolin-amide
Show/Hide
|
C27H17ClF2N4O
|
1
|
| 1 |
EC50 = 646 nM
|
|
|
|
CP0505427
|
3-Cyano-4-(1-naphthyl)-N-(1-[2-chlorophenyl]-3-phenyl-1H-pyrazol-5-yl)benzamide
Show/Hide
|
C33H21ClN4O
|
1
|
| 1 |
EC50 = 2170 nM
|
|
|
|
CP0510165
|
3-Cyano-4-(4-fluorophenyl)-N-(1-[2-chlorophenyl]-3-phenyl-1H-pyrazol-5-yl)benzamide
Show/Hide
|
C29H18ClFN4O
|
1
|
| 1 |
EC50 = 2430 nM
|
|
|
|
CP0524553
|
3-Cyano-4-phenyl-N-(1-[2-chlorophenyl]-3-phenyl-1H-pyrazol-5-yl)benzamide
Show/Hide
|
C29H19ClN4O
|
1
|
| 1 |
EC50 = 4140 nM
|
|
|
|
CP0505426
|
3-Cyano-4-(3-fluorophenyl)-N-(1-[2-chlorophenyl]-3-phenyl-1H-pyrazol-5-yl)benzamide
Show/Hide
|
C29H18ClFN4O
|
1
|
| 1 |
EC50 > 30000 nM
|
|
|
|
CP0191235
|
2-Methyl-6-(phenylethynyl)pyridine
Show/Hide
|
C14H11N
|
1
|
| 1 |
IC50 = 3.54 nM
|
|
|
|
CP0035762
|
3-Cyano-5-fluoro-N-(6-methylpyridin-2-yl)-benzamide
Show/Hide
|
C14H10FN3O
|
2
|
| 1 |
IC50 = 21.7 nM
|
|
|
| 2 |
Ki = 65.5 nM
|
|
|
|
CP0511307
|
3-Cyano-5-fluoro-N-(6-propylpyridin-2-yl)benzamide
Show/Hide
|
C16H14FN3O
|
1
|
| 1 |
IC50 = 165 nM
|
|
|
|
CP0488892
|
3-cyano-N-(6-ethylpyridin-2-yl)-5-fluorobenzamide
Show/Hide
|
C15H12FN3O
|
1
|
| 1 |
IC50 = 169 nM
|
|
|
|
CP0511308
|
3-Cyano-5-fluoro-N-(6-butylpyridin-2-yl)benzamide
Show/Hide
|
C17H16FN3O
|
1
|
| 1 |
IC50 = 1550 nM
|
|
|
|
CP0528918
|
3-Cyano-5-fluoro-N-(5-methylpyridin-2-yl)benzamide
Show/Hide
|
C14H10FN3O
|
1
|
| 1 |
IC50 = 4170 nM
|
|
|
|
CP0296509
|
3-(6-Methyl-pyridin-2-ylethynyl)-benzonitrile
Show/Hide
|
C15H10N2
|
1
|
| 1 |
Ki = 1.3 nM
|
|
|
|
CP0383634
|
5-((6-Methylpyridin-2-yl)ethynyl)nicotinonitrile
Show/Hide
|
C14H9N3
|
1
|
| 1 |
Ki = 1.5 nM
|
|
|
|
CP0374316
|
2-(4-Fluorophenyl)-5-(6-methylpyridin-2-ylethynyl)benzonitrile
Show/Hide
|
C20H11FN2
|
1
|
| 1 |
Ki = 3 nM
|
|
|
|
CP0382064
|
2-Phenyl-5-(6-methylpyridin-2-ylethynyl)benzonitrile
Show/Hide
|
C20H12N2
|
1
|
| 1 |
Ki = 4 nM
|
|
|
|
CP0098719
|
2-methyl-4-(pyridin-3-ylethynyl)thiazole
Show/Hide
|
C11H8N2S
|
1
|
| 1 |
Ki = 16 nM
|
|
|
|
CP0504493
|
2-(3-Fluorophenyl)-5-(6-methylpyridin-2-ylethynyl)benzonitrile
Show/Hide
|
C20H11FN2
|
1
|
| 1 |
Ki = 17 nM
|
|
|
|
CP0388626
|
5-(2-Methylquinolin-7-yl)-2-(4-fluorophenyl)benzonitrile
Show/Hide
|
C23H15FN2
|
1
|
| 1 |
Ki = 64 nM
|
|
|
|
CP0481731
|
3-Cyano-N-(6-methylpyridin-2-yl)-4-(naphthalen-1-yl)-benzamide
Show/Hide
|
C24H17N3O
|
1
|
| 1 |
Ki = 72 nM
|
|
|
|
CP0383635
|
5-(2-Methylquinolin-7-yl)-2-phenylnicotinonitrile
Show/Hide
|
C22H15N3
|
1
|
| 1 |
Ki = 97 nM
|
|
|
|
CP0388623
|
5-(2-Methylquinolin-7-yl)-2-phenylbenzonitrile
Show/Hide
|
C23H16N2
|
1
|
| 1 |
Ki = 97 nM
|
|
|
|
CP0382060
|
3-Cyano-4-(4'-fluorophenyl)-N-(6-methylpyridin-2-yl)-benzamid
Show/Hide
|
C20H14FN3O
|
1
|
| 1 |
Ki = 134 nM
|
|
|
|
CP0377707
|
3-cyano-N-(6-methylpyridin-2-yl)benzamide
Show/Hide
|
C14H11N3O
|
1
|
| 1 |
Ki = 330 nM
|
|
|
|
CP0374325
|
N-(6-methylpyridin-2-yl)-6-phenylpyridine-3-carboxamide
Show/Hide
|
C18H15N3O
|
1
|
| 1 |
Ki = 356 nM
|
|
|
|
CP0383633
|
2-Phenyl-4-(2-methylbenzo[d]thiazol-5-yl)benzonitrile
Show/Hide
|
C20H12N2S
|
1
|
| 1 |
Ki = 483 nM
|
|
|
|
CP0401712
|
2-Methoxymethoxy-5-(2-methylquinolin-7-yl)benzonitrile
Show/Hide
|
C19H16N2O2
|
1
|
| 1 |
Ki = 596 nM
|
|
|
|
CP0374321
|
5-Fluoro-2'-methyl-N-(6-methylpyridin-2-yl)biphenyl-3-carboxamide
Show/Hide
|
C20H17FN2O
|
1
|
| 1 |
Ki = 610 nM
|
|
|
|
CP0450466
|
3-Fluoro-N-(6-methylpyridin-2-yl)-5-(pyridin-3-yl)-benzamide
Show/Hide
|
C18H14FN3O
|
1
|
| 1 |
Ki = 702 nM
|
|
|
|
CP0383632
|
5-(2-Methylquinolin-7-yl)-2-(pyridin-3-yl)benzonitrile
Show/Hide
|
C22H15N3
|
1
|
| 1 |
Ki = 730 nM
|
|
|
|
CP0388625
|
2-Cyano-4-(2-methylbenzo[d]thiazol-5-yl)phenyl trifluoromethanesulfonate
Show/Hide
|
C16H9F3N2O3S2
|
1
|
| 1 |
Ki = 862 nM
|
|
|
|
CP0373485
|
2-Benzoxy-5-(2-methylquinolin-7-yl)benzonitrile
Show/Hide
|
C24H18N2O
|
1
|
| 1 |
Ki = 1040 nM
|
|
|
|
CP0434337
|
3-chloro-N-(6-methylpyridin-2-yl)benzamide
Show/Hide
|
C13H11ClN2O
|
1
|
| 1 |
Ki = 1730 nM
|
|
|
|
CP0374319
|
3-Cyano-N-(6-methylpyridin-2-yl)-4-(pyridine-3-yl)-benzamid
Show/Hide
|
C19H14N4O
|
1
|
| 1 |
Ki = 2040 nM
|
|
|
|
CP0374324
|
N-(6-methylpyridin-2-yl)-6-pyridin-3-ylpyridine-3-carboxamide
Show/Hide
|
C17H14N4O
|
1
|
| 1 |
Ki = 2480 nM
|
|
|
|
CP0417826
|
3-Chloro-N-(6-methylpyridin-2-yl)-4-(pyridine-3-yl)-benzamid
Show/Hide
|
C18H14ClN3O
|
1
|
| 1 |
Ki = 2780 nM
|
|
|
|
CP0372246
|
4'-fluoro-4-(2-methylbenzo[d]thiazol-5-yl)biphenyl-2-carbonitrile
Show/Hide
|
C21H13FN2S
|
1
|
| 1 |
Ki = 4679 nM
|
|
|
|
CP0383630
|
5-Chloro-2-(2-methylquinolin-7-yl)benzonitrile
Show/Hide
|
C17H11ClN2
|
1
|
| 1 |
Ki = 4720 nM
|
|
|
|
CP0374318
|
5-(2-methoxyphenyl)-N-(6-methylpyridin-2-yl)nicotinamide
Show/Hide
|
C19H17N3O2
|
1
|
| 1 |
Ki = 4920 nM
|
|
|
|
CP0372248
|
2-Benzoxy-5-(2-methylbenzo[d]thiazol-5-yl)benzonitrile
Show/Hide
|
C22H16N2OS
|
1
|
| 1 |
Ki = 7134 nM
|
|
|
|
CP0453859
|
N-(6-methylpyridin-2-yl)-3-phenylbenzamide
Show/Hide
|
C19H16N2O
|
1
|
| 1 |
Ki = 7300 nM
|
|
|
|
CP0377704
|
3-Fluoro-N-(6-methylpyridin-2-yl)-4-(pyridine-3-yl)-benzamide
Show/Hide
|
C18H14FN3O
|
1
|
| 1 |
Ki = 7720 nM
|
|
|
|
CP0382063
|
5-Fluoro-2'-methoxy-N-(6-methylpyridin-2-yl)biphenyl-3-carboxamide
Show/Hide
|
C20H17FN2O2
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0496058
|
N-(6-methylpyridin-2-yl)-5-pyridin-3-ylpyridine-3-carboxamide
Show/Hide
|
C17H14N4O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0372243
|
2-Chloro-5-(2-methylquinolin-7-yl)nicotinonitrile
Show/Hide
|
C16H10ClN3
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0383627
|
2-Hydroxy-5-(2-methylquinolin-7-yl)benzonitrile
Show/Hide
|
C17H12N2O
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
|
CP0388624
|
2-(Pyridin-3-yl)-4-(2-methylbenzo[d]thiazol-5-yl)benzonitrile
Show/Hide
|
C19H11N3S
|
1
|
| 1 |
Ki > 10000 nM
|
|
|
