(S)-6-amino-2-((S)-2-amino-3-(1H-indol-3-yl)propanamido)-N-((5R,8S,11S,14S)-5-carbamoyl-15-(4-hydroxyphenyl)-8-isopropyl-11-(2-(methylthio)ethyl)-7,10,13-trioxo-2-thia-6,9,12-triazapentadecan-14-yl)hexanamide

(S)-2-(3-(4-bromophenyl)ureido)-N-(2-oxo-1,3-diazepan-1-yl)-3-phenylpropanamide

ethyl 1-((S)-2-(3-(4-bromophenyl)ureido)-3-phenylpropanoyl)piperidine-3-carboxylate

1-[(2S)-3-(4-cyanophenyl)-1-(2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(S)-1-(4-bromophenyl)-3-(1-oxo-3-phenyl-1-(piperidin-1-yl)propan-2-yl)urea

(S)-1-(4-chlorophenyl)-3-(1-oxo-3-phenyl-1-(piperidin-1-yl)propan-2-yl)urea

(S)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(5-methoxy-2-pyridinyl)cyclohexyl]methyl]propanamide

1-(4-bromophenyl)-3-(4-methoxyphenethyl)urea

(2S)-3-(1H-indol-3-yl)-2-[(4-methoxyphenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]propanamide

(S)-ethyl 1-(2-(3-(4-bromophenyl)ureido)-3-(1H-indol-3-yl)propanoyl)piperidine-4-carboxylate

(S)-1-(4-bromophenyl)-3-(1-oxo-3-phenyl-1-(pyrrolidin-1-yl)propan-2-yl)urea

(S)-ethyl 1-(2-(3-(4-bromophenyl)ureido)-3-phenylpropanoyl)piperidine-4-carboxylate

1-[(2S)-3-(4-cyanophenyl)-1-(2,3-dihydropyrrolo[2,3-b]pyridin-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2S)-3-(4-cyanophenyl)-1-(5-fluoro-2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(2S)-3-(4-cyanophenyl)-2-[(4-fluorophenyl)carbamoylamino]-N-(2-oxoazepan-3-yl)propanamide

(R)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(5-methoxy-2-pyridinyl)cyclohexyl]methyl]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(S)-1-(4-bromophenyl)-3-(1-(indolin-1-yl)-1-oxo-3-phenylpropan-2-yl)urea

1-[(2R)-3-(4-cyanophenyl)-1-(3,4-dihydro-2H-quinolin-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(R)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[(1-phenylcyclohexyl)methyl]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(3,4-dihydro-2H-quinolin-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-((2S)-3-(1H-indol-3-yl)-1-(3-methyl-4-((methylaminooxy)carbonyl)piperidin-1-yl)-1-oxopropan-2-yl)-3-(4-bromophenyl)urea

(S)-1-(4-(methylthio)phenyl)-3-(1-oxo-3-phenyl-1-(piperidin-1-yl)propan-2-yl)urea

(2R)-N-[[1-(3-chloro-4-fluorophenyl)cyclopropyl]methyl]-3-(4-cyanophenyl)-2-[(4-fluorophenyl)carbamoylamino]propanamide

(R)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(2-pyridinyl)cyclohexyl]methyl]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(1,3-dihydroisoindol-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2R)-3-(4-cyanophenyl)-1-(6-fluoro-2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-(4-chlorophenyl)-3-(4-methoxyphenethyl)urea

1-[(2R)-3-(4-cyanophenyl)-1-(5-fluoro-2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(S)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(2-pyridinyl)cyclohexyl]methyl]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(7-fluoro-3,4-dihydro-1H-isoquinolin-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2R)-3-(4-cyanophenyl)-1-(7-fluoro-3,4-dihydro-1H-isoquinolin-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(2S)-3-(4-cyanophenyl)-2-[(4-nitrophenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]propanamide

(S)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(3-pyridinyl)cyclohexyl]methyl]propanamide

(S)-N-[[1-(4-Fluorophenyl)cyclohexyl]methyl]-3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamide

1-(4-fluorophenyl)-3-(4-methoxyphenethyl)urea

1-[(2S)-3-(4-cyanophenyl)-1-oxo-1-piperidin-1-ylpropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-bromophenyl)-2-[5-(3-methoxybenzoyl)-3-methyl-6-oxopyridazin-1-yl]acetamide

(2R)-3-(4-cyanophenyl)-2-[(4-fluorophenyl)carbamoylamino]-N-(2-oxoazepan-3-yl)propanamide

1-[(2R)-3-(4-cyanophenyl)-1-(2,3-dihydropyrrolo[2,3-b]pyridin-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2S)-3-(4-cyanophenyl)-1-(6-fluoro-2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2R)-3-(4-cyanophenyl)-1-(3,4-dihydro-1H-isoquinolin-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(2R)-3-(4-cyanophenyl)-2-[(4-nitrophenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]propanamide

(S)-N-[[(1-(2-Fluoro-4-pyridinyl)cyclohexyl]methyl]-3-(1H-indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(7-fluoro-4,4-dimethyl-1,3-dihydroisoquinolin-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

2-[4-acetyl-5-(4-methoxyanilino)-3-methyl-6-oxopyridazin-1-yl]-N-(4-bromophenyl)acetamide

1-[(2S)-3-(4-cyanophenyl)-1-(5-fluoro-1,3-dihydroisoindol-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(2R)-N-[[1-(3-chloro-4-fluorophenyl)cyclopropyl]methyl]-3-(4-cyanophenyl)-2-[(4-methoxyphenyl)carbamoylamino]propanamide

(2S)-2-[(4-fluorophenyl)carbamoylamino]-3-(1H-indol-3-yl)-N-[(1-phenylcyclopropyl)methyl]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-(3,3-dimethyl-2H-indol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

N-[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]-3-methoxybenzamide

N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(pyridin-3-ylmethyl)pyridazin-1-yl]acetamide

(2R)-2-[(4-nitrophenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]-3-pyridin-3-ylpropanamide

1-(4-methoxyphenethyl)-3-phenylurea

(2S)-3-(4-cyanophenyl)-N-[[1-(3-fluoro-4-methylphenyl)cyclopropyl]methyl]-2-[(4-fluorophenyl)carbamoylamino]propanamide

1-[(2S)-3-(4-cyanophenyl)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-ethylphenyl)-2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetamide

(2S)-N-[[1-(3-chloro-4-fluorophenyl)cyclopropyl]methyl]-3-(4-cyanophenyl)-2-[(4-methoxyphenyl)carbamoylamino]propanamide

N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

(2S)-N-[[1-(3-chloro-4-fluorophenyl)cyclopropyl]methyl]-3-(4-cyanophenyl)-2-[(4-fluorophenyl)carbamoylamino]propanamide

N-(4-chlorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

N-(2-bromophenyl)-2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetamide

N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide

N-(3,4-dimethoxyphenyl)-2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetamide

1-[(2R)-3-(4-cyanophenyl)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-bromophenyl)-3-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]propanamide

2-[3-ethyl-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide

1-[(2R)-3-(4-cyanophenyl)-1-(2,3-dihydroindol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-acetylphenyl)-2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetamide

N-(4-bromophenyl)-2-[5-(furan-3-ylmethyl)-3-methyl-6-oxopyridazin-1-yl]acetamide

(2S)-2-[(4-nitrophenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]-3-pyridin-3-ylpropanamide

(2R)-3-(1H-indol-3-yl)-2-[(4-methoxyphenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]propanamide

(2S)-3-(1H-indol-3-yl)-2-(phenylcarbamoylamino)-N-[(1-phenylcyclopropyl)methyl]propanamide

N-(4-iodophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

1-[(2R)-3-(4-cyanophenyl)-1-(3,3-dimethyl-2H-indol-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-propan-2-ylpyridazin-1-yl]acetamide

1-[(2R)-3-(4-cyanophenyl)-1-(5-fluoro-1,3-dihydroisoindol-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

methyl N-[3-[[2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetyl]amino]phenyl]carbamate

(2S)-3-(1H-indol-3-yl)-2-[(4-nitrophenyl)carbamoylamino]-N-[(1-phenylcyclopropyl)methyl]propanamide

N-(4-bromophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-(4-methoxyanilino)-3-methyl-6-oxopyridazin-1-yl]acetamide

2-[(6-ethoxy-1H-benzimidazol-2-yl)sulfanyl]-N-(2-methylsulfanylphenyl)acetamide

2-[5-(3-Methoxybenzyl)-3-methyl-6-oxo-6H-pyridazin-1-yl]-N-(4-trifluoromethylphenyl)-acetamide

N-(2-chlorophenyl)-2-[(6-methoxy-1H-benzimidazol-2-yl)sulfanyl]acetamide

(2R)-Methyl 2-[(2'S)-[(tert-butoxycarbonyl)amino]-3-(1H-indol-3-yl)propanamido]-3-phenylpropanoate

2-[5-(3-Methoxybenzyl)-3-methyl-6-oxo-6H-pyridazin-1-yl]-N-4-tolyl-acetamide

(2R)-Methyl 2-[(2'S)-2-benzamido-3-(1H-indol-3-yl)propanamido]-4-methylpentanoate

N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(thiophen-2-ylmethyl)pyridazin-1-yl]acetamide

2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)-N-(4-bromophenyl)acetamide

2-[5-(3-Methoxybenzyl)-3-methyl-6-oxo-6H-pyridazin-1-yl]-N-(4-nitrophenyl)-acetamide

1-[(2R)-3-(4-cyanophenyl)-1-oxo-1-piperidin-1-ylpropan-2-yl]-3-(4-fluorophenyl)urea

N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-(thiophen-3-ylmethyl)pyridazin-1-yl]acetamide

2-[5-(3-Methoxybenzyl)-3-methyl-6-oxo-6H-pyridazin-1-yl]-N-(4-methoxyphenyl)-acetamide

(2S)-3-(4-cyanophenyl)-N-[[1-(3-fluoro-4-methylphenyl)cyclopropyl]methyl]-2-[(4-methoxyphenyl)carbamoylamino]propanamide

N-(3,4-dimethoxyphenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

2-[5-[(3-chlorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide

1-[(2R)-3-(4-cyanophenyl)-1-(1,3-dihydroisoindol-2-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

1-[(2S)-3-(4-cyanophenyl)-1-(4,4-difluoropiperidin-1-yl)-1-oxopropan-2-yl]-3-(4-fluorophenyl)urea

(S)-2-[(S)-2-((S)-2-Formylamino-4-methylsulfanyl-butyrylamino)-4-methyl-pentanoylamino]-3-phenyl-propionic acid

4-[[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]methyl]benzamide

2-(5-amino-3-methyl-6-oxopyridazin-1-yl)-N-(4-bromophenyl)acetamide

2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)-N-(4-fluorophenyl)acetamide

N-(4-fluorophenyl)-2-[3-(4-fluorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(1,3-benzodioxol-5-yl)-2-[3-(4-fluorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-[(3-bromophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

2-[3-benzyl-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-bromophenyl)acetamide

N-(4-bromophenyl)-2-[5-[(3,5-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

2-[3-(4-chlorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]-N-(4-fluorophenyl)acetamide

N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-[(4-cyanophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-[(4-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide

N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide

2-[5-[(3,5-dimethoxyphenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]-N-(4-iodophenyl)acetamide

N-(1,3-benzodioxol-5-yl)-2-(5-benzyl-3-methyl-6-oxopyridazin-1-yl)acetamide

N-(4-bromophenyl)-2-[3-methyl-5-(naphthalen-1-ylmethyl)-6-oxopyridazin-1-yl]acetamide

N-(1,3-benzodioxol-5-yl)-2-[3-(4-chlorophenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-thiophen-2-ylpyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[3-cyclohexyl-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[3-(4-chlorophenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-6-oxo-3-phenylpyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-[(3-fluorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

4-bromo-N-[2-[2-(4-bromoanilino)-2-oxoethyl]-6-methyl-3-oxopyridazin-4-yl]benzamide

N-(4-bromophenyl)-2-[3-methyl-6-oxo-5-[[4-(trifluoromethyl)phenyl]methyl]pyridazin-1-yl]acetamide

N-(4-fluorophenyl)-2-[5-[(3-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide

N-(4-iodophenyl)-2-(3-methyl-6-oxo-4,5-dihydropyridazin-1-yl)acetamide

N-(1,3-benzodioxol-5-yl)-2-[3-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[3-(4-methoxyphenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(4-iodophenyl)-2-(3-methyl-6-oxopyridazin-1-yl)acetamide

N-(4-bromophenyl)-2-[3-(4-fluorophenyl)-5-[(4-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

N-(1,3-benzodioxol-5-yl)-2-[5-[(3-methoxyphenyl)methyl]-3-(4-methylphenyl)-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-(4-methoxyphenyl)-3-methyl-6-oxopyridazin-1-yl]acetamide

N-(4-bromophenyl)-2-[5-[(3-chlorophenyl)methyl]-3-methyl-6-oxopyridazin-1-yl]acetamide

N-(4-fluorophenyl)-2-[3-(4-methoxyphenyl)-5-[(3-methoxyphenyl)methyl]-6-oxopyridazin-1-yl]acetamide

1-[(3S,4R)-4-(2,6-difluoro-4-methoxyphenyl)-2-oxopyrrolidin-3-yl]-3-phenylurea

(3S,4R)-3-[[5-(4-chlorophenyl)-1,2-oxazol-3-yl]amino]-4-(2,6-difluoro-4-methoxyphenyl)pyrrolidin-2-one

(3S,4R)-3-[[5-(4-chlorophenyl)-1,3,4-oxadiazol-2-yl]amino]-4-(2,6-difluoro-4-methoxyphenyl)pyrrolidin-2-one

methyl (2S)-2-[[(2S)-2-benzamido-3-(1H-indol-3-yl)propanoyl]amino]-3-phenylpropanoate