Brief Information of the Compound and Protein
Compound Name
(R)-3-(1H-Indol-3-yl)-2-[3-(4-methoxyphenyl)ureido]-N-[[1-(2-pyridinyl)cyclohexyl]methyl]propanamide
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PubChem ID
CID: 122181323
Canonical SMILES
COc1ccc(NC(=O)N[C@H](Cc2c[nH]c3ccccc23)C(=O)NCC2(c3ccccn3)CCCCC2)cc1
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Compound Formula C31H35N5O3
Compound Structure
Protein Name
N-formyl peptide receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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N-formyl methionyl peptide receptor
Uniprot ID
P25090
Gene Name
FPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000018 HL-60 Homo sapiens (Human)  1
1
EC50 = 310 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 490 nM
2 EC50 = 620 nM