| Compound ID |
Compound Name |
Compound Formula |
|
CP0921999
|
cis-(+)-4-(3,4-Dimethoxyphenyl)-2-[4-(morpholinomethyl)benzyl]-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one
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|
C28H34ClN3O4
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0463773
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[(E)-4-imidazol-1-ylbut-2-enyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C23H26N4O3
|
1
|
| 1 |
IC50 = 0.4 nM
|
|
|
|
CP0463774
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-(imidazol-1-ylmethyl)phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C27H28N4O3
|
1
|
| 1 |
IC50 = 0.7 nM
|
|
|
|
CP0458869
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-[(4-oxopiperidin-1-yl)methyl]phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C29H33N3O4
|
1
|
| 1 |
IC50 = 0.9 nM
|
|
|
|
CP0510432
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[2-(morpholin-4-ylmethyl)phenyl]methyl]-4a,5,6,7,8,8a-hexahydrophthalazin-1-one
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|
C28H35N3O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0477286
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylmethyl)phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C31H37N3O5
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0498618
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[2-(morpholin-4-ylmethyl)phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C28H33N3O4
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0463778
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[3-(morpholin-4-ylmethyl)phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C28H33N3O4
|
1
|
| 1 |
IC50 = 1.4 nM
|
|
|
|
CP0430714
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-[(4-methylpiperazin-1-yl)methyl]phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C29H36N4O3
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0498619
|
(1R,6S)-5-(3,4-dimethoxyphenyl)-3-[[4-(morpholin-4-ylmethyl)phenyl]methyl]-3,4-diazabicyclo[4.2.0]oct-4-en-2-one
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|
C26H31N3O4
|
1
|
| 1 |
IC50 = 4.3 nM
|
|
|
|
CP0510431
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[2-(2-imidazol-1-ylethoxy)ethyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C23H28N4O4
|
1
|
| 1 |
IC50 = 5.2 nM
|
|
|
|
CP0513301
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-(piperidin-1-ylmethyl)phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C29H35N3O3
|
1
|
| 1 |
IC50 = 8.2 nM
|
|
|
|
CP0501554
|
(4aS,8aR)-4-(3,4-dimethoxyphenyl)-2-[[4-[(dimethylamino)methyl]phenyl]methyl]-4a,5,8,8a-tetrahydrophthalazin-1-one
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|
C26H31N3O3
|
1
|
| 1 |
IC50 = 9.7 nM
|
|
|
|
CP0477284
|
2-[(4aS,8aR)-4-(3,4-dimethoxyphenyl)-1-oxo-4a,5,8,8a-tetrahydrophthalazin-2-yl]-N-(3-imidazol-1-ylpropyl)acetamide
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|
C24H29N5O4
|
1
|
| 1 |
IC50 = 14.3 nM
|
|
|
|
CP0452131
|
(1R,6S)-5-(3,4-dimethoxyphenyl)-3-[[4-(morpholin-4-ylmethyl)phenyl]methyl]-3,4-diazabicyclo[4.1.0]hept-4-en-2-one
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|
C25H29N3O4
|
1
|
| 1 |
IC50 = 16.4 nM
|
|
|
|
CP0533027
|
6-(3,4-Dimethoxyphenyl)-2-[4-(morpholinomethyl)benzyl]-4,5-dihydropyridazin-3(2H)-one
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|
C24H29N3O4
|
1
|
| 1 |
IC50 = 45.9 nM
|
|
|
|
CP0277281
|
(cis)-4-(3,4-dimethoxyphenyl)-4a,5,8,8a-tetrahydrophthalazin-1(2H)-one
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|
C16H18N2O3
|
1
|
| 1 |
IC50 = 85 nM
|
|
|
