Brief Information of the Compound and Protein
Compound Name
(1R,6S)-5-(3,4-dimethoxyphenyl)-3-[[4-(morpholin-4-ylmethyl)phenyl]methyl]-3,4-diazabicyclo[4.1.0]hept-4-en-2-one
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PubChem ID
CID: 46227306
Canonical SMILES
COc1ccc(cc1OC)C1=NN(Cc2ccc(CN3CCOCC3)cc2)C(=O)[C@@H]2C[C@H]12
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Compound Formula C25H29N3O4
Compound Structure
Protein Name
3',5'-cyclic-AMP phosphodiesterase 4D
Protein Classification
Enzyme
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Phosphodiesterase
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Phosphodiesterase 4
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Phosphodiesterase 4D
Uniprot ID
Q08499
Gene Name
PDE4D
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000018 HL-60 Homo sapiens (Human)  1
1
IC50 = 16.4 nM
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