| Compound ID |
Compound Name |
Compound Formula |
|
CP0542929
|
2-[[(3aS,9R,9aR)-4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-ethylamino]-1,3-thiazole-4-carboxylic acid
Show/Hide
|
C26H27N3O4S
|
3
|
| 1 |
EC50 = 12 nM
|
|
|
| 2 |
IC50 = 2920 nM
|
|
|
| 3 |
Ki = 51 nM
|
|
|
|
CP0461747
|
(S)-2-(2-((4-(2-(4-fluorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)-4-(trifluoromethyl)phenoxy)acetic acid
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|
C23H24F4N2O4
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0498085
|
2-[4-chloro-2-[[(3S)-4-[2-(4-chlorophenyl)acetyl]-3-methylpiperazin-1-yl]methyl]phenoxy]acetic acid
Show/Hide
|
C22H24Cl2N2O4
|
1
|
| 1 |
IC50 = 0.5 nM
|
|
|
|
CP0447086
|
(S)-2-(2-((4-(benzylsulfonyl)-3-methylpiperazin-1-yl)methyl)-4-chlorophenyl)acetic acid
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|
C21H25ClN2O4S
|
1
|
| 1 |
IC50 = 0.6 nM
|
|
|
|
CP0399932
|
(S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0444397
|
2-[[(2aS,8R,8aR)-3-(3-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid
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|
C24H23FN2O5
|
2
|
| 1 |
IC50 = 0.8 nM
|
|
|
| 2 |
Ki = 4.1 nM
|
|
|
|
CP0416496
|
2-[[(2aS,8R,8aR)-3-[4-(trifluoromethoxy)benzoyl]-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid
Show/Hide
|
C25H23F3N2O6
|
2
|
| 1 |
IC50 = 0.9 nM
|
|
|
| 2 |
Ki = 2.5 nM
|
|
|
|
CP0417719
|
2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-4'-fluoro-6-methoxybiphenyl-3-yl)acetic acid
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|
C26H26FNO5
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
|
CP0424092
|
(S)-2-(4-chloro-2-((4-(2-(4-fluorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H24ClFN2O4
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0499693
|
2-[4-methoxy-3-[2-[[(1S)-1-phenylethyl]carbamoyl]-4-(propanoylamino)phenoxy]phenyl]acetic acid
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|
C27H28N2O6
|
2
|
| 1 |
IC50 = 1 nM
|
|
|
| 2 |
IC50 = 6 nM
|
|
|
|
CP0498086
|
(S)-2-(4-chloro-2-((4-(phenylsulfonyl)-3-propylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H27ClN2O5S
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0531436
|
(S)-2-(4-chloro-2-(((S)-4-(2-(4-chlorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)propanoic acid
Show/Hide
|
C23H26Cl2N2O4
|
1
|
| 1 |
IC50 = 1.3 nM
|
|
|
|
CP0523739
|
4-bromo-2-[1-(4-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid
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|
C18H12Br2N2O4
|
2
|
| 1 |
IC50 = 1.4 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
|
CP0035019
|
4-bromo-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
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|
C18H13BrN2O4
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 24 nM
|
|
|
|
CP0425386
|
4-bromo-2-[1-(4-chlorophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid
Show/Hide
|
C18H12BrClN2O4
|
2
|
| 1 |
IC50 = 1.5 nM
|
|
|
| 2 |
IC50 = 17 nM
|
|
|
|
CP0487270
|
2-[2-[(5-benzoyl-2-methoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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|
C24H19FN2O4S
|
2
|
| 1 |
IC50 = 1.7 nM
|
|
|
| 2 |
IC50 = 4 nM
|
|
|
|
CP0453604
|
4-bromo-2-[1-(2-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid
Show/Hide
|
C18H12Br2N2O4
|
2
|
| 1 |
IC50 = 1.9 nM
|
|
|
| 2 |
IC50 = 12 nM
|
|
|
|
CP0392938
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3,5-dimethoxyphenyl)acetic acid
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|
C25H24Cl2N2O8S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 16 nM
|
|
|
|
CP0415000
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(propylcarbamoyl)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C25H24Cl2N2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0508252
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(isopropylcarbamoyl)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C25H24Cl2N2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0534326
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3-fluorophenyl)acetic acid
Show/Hide
|
C23H19Cl2FN2O6S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0535115
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3-ethoxyphenyl)acetic acid
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|
C25H24Cl2N2O7S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0399063
|
2-[3-[2-[[1-(4-fluorophenyl)-2-methylpropan-2-yl]carbamoyl]-4-(propanoylamino)phenoxy]-4-methoxyphenyl]acetic acid
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|
C29H31FN2O6
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 15 nM
|
|
|
|
CP0403514
|
2-[3-[2-[[(1S)-1-(4-chlorophenyl)ethyl]carbamoyl]-4-(propanoylamino)phenoxy]-4-methoxyphenyl]acetic acid
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|
C27H27ClN2O6
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 15 nM
|
|
|
|
CP0499694
|
2-[3-[2-[2-(4-fluorophenyl)ethylcarbamoyl]-4-(propanoylamino)phenoxy]-4-methoxyphenyl]acetic acid
Show/Hide
|
C27H27FN2O6
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 13 nM
|
|
|
|
CP0400765
|
2-[4-[2-[(2,4-dichlorophenyl)sulfonylamino]-4-(5-propyl-1H-pyrazol-3-yl)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C27H25Cl2N3O6S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
|
CP0400766
|
2-[4-[[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]methyl]-3-methoxyphenyl]acetic acid
Show/Hide
|
C27H28Cl2N2O6S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0403549
|
2-[5-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]indol-1-yl]acetic acid
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|
C27H25Cl2N3O6S
|
1
|
| 1 |
IC50 = 2 nM
|
|
|
|
CP0476525
|
2-[4-[2-[(2,4-dichlorophenyl)sulfonylamino]-4-(2-propyl-1H-imidazol-5-yl)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C27H25Cl2N3O6S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 20 nM
|
|
|
|
CP0050067
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C19H18N2O4S
|
3
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
| 3 |
IC50 = 25 nM
|
|
|
|
CP0126760
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C19H17FN2O4S
|
3
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 5 nM
|
|
|
| 3 |
IC50 = 14 nM
|
|
|
|
CP0504939
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-nitrobenzimidazol-1-yl]acetic acid
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|
C19H17N3O6S
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
IC50 = 3 nM
|
|
|
|
CP0466068
|
2-[[(2aS,8R,8aR)-3-(4-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylcarbamoyl]oxyacetic acid
Show/Hide
|
C24H23FN2O5
|
2
|
| 1 |
IC50 = 2 nM
|
|
|
| 2 |
Ki = 3.5 nM
|
|
|
|
CP0522682
|
2-[4-chloro-2-[[(3S)-4-[2-(4-chlorophenyl)acetyl]-3-methylpiperazin-1-yl]methyl]phenyl]acetic acid
Show/Hide
|
C22H24Cl2N2O3
|
1
|
| 1 |
IC50 = 2.2 nM
|
|
|
|
CP0495921
|
2-(3-(8-chloroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid
Show/Hide
|
C21H17ClN2O2
|
1
|
| 1 |
IC50 = 2.3 nM
|
|
|
|
CP0055602
|
(R)-2-(4-fluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H20F2N2O4S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0081599
|
(R)-2-(3,4-difluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H19F3N2O4S
|
1
|
| 1 |
IC50 = 2.5 nM
|
|
|
|
CP0082341
|
2-(2,5-dimethyl-3-(8-methylquinolin-4-yl)-1H-indol-1-yl)acetic acid
Show/Hide
|
C22H20N2O2
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0145080
|
(R)-2-(3-fluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H20F2N2O4S
|
1
|
| 1 |
IC50 = 2.6 nM
|
|
|
|
CP0086262
|
4-(((2S,4R)-1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-4-oxobutanoic acid
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|
C27H26N2O4
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 130 nM
|
|
|
|
CP0388282
|
2-(4-(4-(butylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C26H26Cl2N2O7S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 21 nM
|
|
|
|
CP0414997
|
2-(3-chloro-5-(2-(4-chlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
Show/Hide
|
C23H20Cl2N2O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0415001
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(isobutylcarbamoyl)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C26H26Cl2N2O7S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0415003
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C24H22Cl2N2O7S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0491157
|
2-(4-(4-(cyclobutylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C26H24Cl2N2O7S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0496650
|
2-(3-chloro-5-(4-(ethylcarbamoyl)-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C23H21ClN2O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0032668
|
(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H21FN2O4S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
Ki = 2.5 nM
|
|
|
|
CP0117323
|
(R)-2-(2-fluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H20F2N2O4S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0243368
|
(R)-2-(3-chloro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H20ClFN2O4S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0473196
|
2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-4'-(4-chlorophenylsulfonamido)-6-methoxybiphenyl-3-yl)acetic acid
Show/Hide
|
C32H31ClN2O7S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 90 nM
|
|
|
|
CP0107693
|
2-[4-[4-(tert-butylcarbamoyl)-2-[(2-chloro-4-cyclopropylphenyl)sulfonylamino]phenoxy]-5-chloro-2-fluorophenyl]acetic acid
Show/Hide
|
C28H27Cl2FN2O6S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 8 nM
|
|
|
|
CP0391761
|
2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-methylphenyl]acetic acid
Show/Hide
|
C26H26Cl2N2O6S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 26 nM
|
|
|
|
CP0405871
|
2-[6-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-1H-indol-3-yl]acetic acid
Show/Hide
|
C27H25Cl2N3O6S
|
1
|
| 1 |
IC50 = 3 nM
|
|
|
|
CP0093475
|
2-[3-[1-[(4-fluorophenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]-4-methoxyphenyl]acetic acid
Show/Hide
|
C25H21FN2O4
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 9 nM
|
|
|
|
CP0154070
|
2-[2-[[5-(2,3-dihydroindole-1-carbonyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C26H22FN3O4S
|
3
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 4 nM
|
|
|
| 3 |
IC50 = 8 nM
|
|
|
|
CP0462640
|
2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-(trifluoromethyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C20H17F3N2O4S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 5 nM
|
|
|
|
CP0469001
|
2-[4-[[4-[(2,4-dichlorophenyl)sulfonylamino]-2-oxo-1,3-dihydroindol-5-yl]oxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C23H18Cl2N2O7S
|
2
|
| 1 |
IC50 = 3 nM
|
|
|
| 2 |
IC50 = 31 nM
|
|
|
|
CP0426598
|
(R)-2-(2-chloro-8-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C20H19ClFN3O4S
|
2
|
| 1 |
IC50 = 3.2 nM
|
|
|
| 2 |
Ki = 1.8 nM
|
|
|
|
CP0500985
|
(S)-2-(4-chloro-2-((3-methyl-4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H25ClN2O4
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0522846
|
4-bromo-2-[1-(3-bromophenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid
Show/Hide
|
C18H12Br2N2O4
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
IC50 = 31 nM
|
|
|
|
CP0143839
|
(R)-2-(8-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C20H20FN3O4S
|
2
|
| 1 |
IC50 = 3.4 nM
|
|
|
| 2 |
Ki = 3.3 nM
|
|
|
|
CP0501728
|
(R)-2-(8-(2-(4-fluorophenyl)-N,2-dimethylpropanamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C24H26FN3O3
|
2
|
| 1 |
IC50 = 3.5 nM
|
|
|
| 2 |
Ki = 4.7 nM
|
|
|
|
CP0445961
|
4-bromo-2-[1-(4-methoxyphenyl)-1H-pyrazole-4-carbonyl]phenoxyacetic acid
Show/Hide
|
C19H15BrN2O5
|
2
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
IC50 = 53 nM
|
|
|
|
CP0478525
|
(R)-2-(8-(4-fluoro-N-methylphenylsulfonamido)-2-(4-fluorophenyl)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C26H23F2N3O4S
|
2
|
| 1 |
IC50 = 3.6 nM
|
|
|
| 2 |
Ki = 1.9 nM
|
|
|
|
CP0055829
|
(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-(trifluoromethyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C22H20F4N2O4S
|
1
|
| 1 |
IC50 = 3.6 nM
|
|
|
|
CP0225635
|
(R)-2-(2,3-difluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H19F3N2O4S
|
1
|
| 1 |
IC50 = 3.8 nM
|
|
|
|
CP0398264
|
2-(4-(4-(cyclopropylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C25H22Cl2N2O7S
|
2
|
| 1 |
IC50 = 4 nM
|
|
|
| 2 |
IC50 = 28 nM
|
|
|
|
CP0496651
|
2-(3-chloro-5-(2-(2-chlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
Show/Hide
|
C23H20Cl2N2O6S
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1
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| 1 |
IC50 = 4 nM
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CP0502788
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2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
Show/Hide
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C23H20Cl2N2O6S
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1
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| 1 |
IC50 = 4 nM
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CP0535114
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2-(3-chloro-5-(2-(3-chloro-4-methylphenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
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C24H22Cl2N2O6S
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1
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| 1 |
IC50 = 4 nM
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CP0403512
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2-[4-[4-(butylcarbamoyl)-2-[(4-chlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
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C26H27ClN2O7S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 100 nM
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CP0391756
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2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-2,5-difluorophenyl]acetic acid
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C25H22Cl2F2N2O6S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 32 nM
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CP0406437
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2-[4-[2-[[2-chloro-4-(trifluoromethyl)phenyl]sulfonylamino]-4-(cyclobutylcarbamoyl)phenoxy]-3-methoxyphenyl]acetic acid
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C27H24ClF3N2O7S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 13 nM
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CP0496379
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2-[4-[4-(butylcarbamoyl)-2-[[2-chloro-4-(trifluoromethyl)phenyl]sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
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C27H26ClF3N2O7S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 47 nM
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CP0476524
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2-[4-[2-[(2,4-dichlorophenyl)sulfonylamino]-4-(5-propyl-1H-1,2,4-triazol-3-yl)phenoxy]-3-methoxyphenyl]acetic acid
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C26H24Cl2N4O6S
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1
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| 1 |
IC50 = 4 nM
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CP0487251
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2-[2-[(5-acetyl-2-ethoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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C20H19FN2O4S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 5 nM
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CP0494078
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2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-formylbenzimidazol-1-yl]acetic acid
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C20H18N2O5S
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2
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 9 nM
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CP0042409
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2-[2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C28H26N2O3
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4
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 7 nM
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| 3 |
IC50 = 190 nM
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| 4 |
IC50 = 320 nM
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CP0042410
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2-[8-chloro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C24H19ClN2O3
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4
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 30 nM
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| 3 |
IC50 = 65 nM
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| 4 |
IC50 = 110 nM
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CP0055874
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2-[8-fluoro-2-(thiophene-2-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C18H15FN2O3S
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4
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 12 nM
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| 3 |
IC50 = 40 nM
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| 4 |
IC50 = 70 nM
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CP0086409
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2-[8-fluoro-2-(2-naphthalen-1-ylacetyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C25H21FN2O3
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4
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| 1 |
IC50 = 4 nM
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| 2 |
IC50 = 70 nM
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| 3 |
IC50 = 160 nM
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| 4 |
IC50 = 180 nM
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CP0511770
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4-[[(3aS,9R,9aR)-6-fluoro-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
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C27H26F4N2O5
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2
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| 1 |
IC50 = 4 nM
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| 2 |
Ki = 3 nM
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CP0410062
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2-((8R)-8-(1-(4-fluorophenyl)-N,2,2-trimethylcyclopropanecarboxamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
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C26H28FN3O3
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2
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| 1 |
IC50 = 4.4 nM
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| 2 |
Ki = 5.1 nM
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CP0410064
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(R)-2-(8-(1-(4-fluorophenyl)-N-methylcyclopentanecarboxamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
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C26H28FN3O3
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2
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| 1 |
IC50 = 4.5 nM
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| 2 |
Ki = 3.9 nM
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CP0081597
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(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-phenyl-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C27H25FN2O4S
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1
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| 1 |
IC50 = 4.5 nM
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CP0447087
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(S)-2-(4-chloro-2-((3-ethyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
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C21H25ClN2O5S
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1
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| 1 |
IC50 = 4.5 nM
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CP0906028
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rac-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
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C20H23ClN2O5S
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1
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| 1 |
IC50 = 4.5 nM
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CP0503601
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(R)-2-(8-(1-(4-fluorophenyl)-N-methylcyclobutanecarboxamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
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C25H26FN3O3
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2
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| 1 |
IC50 = 4.7 nM
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| 2 |
Ki = 3.4 nM
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CP0443728
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5-[3-(4-fluorophenyl)-7-[(5S)-5-[(S)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
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C30H28FN3O5
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1
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| 1 |
IC50 = 4.7 nM
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CP0055126
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(R)-2-(7-(4-fluoro-N-pentylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C25H29FN2O4S
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1
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| 1 |
IC50 = 4.9 nM
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CP0501857
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(+/-)-4-((1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-4-oxobutanoic acid
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C27H26N2O4
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 28 nM
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CP0544208
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2-(3-chloro-5-(4-(ethylcarbamoyl)-2-(4-methylphenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
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C24H23ClN2O6S
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1
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| 1 |
IC50 = 5 nM
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CP0487311
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2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-6-methoxy-4'-(methylsulfonyl)biphenyl-3-yl)acetic acid
Show/Hide
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C27H29NO7S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 7 nM
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CP0427658
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2-[4-[4-(cyclobutylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylmethyl]phenoxy]-3-methoxyphenyl]acetic acid
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C27H25Cl2NO7S
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1
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| 1 |
IC50 = 5 nM
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CP0391763
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2-[4-[4-(tert-butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-chlorophenyl]acetic acid
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C25H23Cl3N2O6S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 12 nM
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CP0391765
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2-[3-chloro-4-[4-(cyclobutylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]phenyl]acetic acid
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C25H21Cl3N2O6S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 19 nM
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CP0392767
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2-[5-chloro-4-[2-[[2-chloro-4-(trifluoromethoxy)phenyl]sulfonylamino]-4-(cyclobutylcarbamoyl)phenoxy]-2-fluorophenyl]acetic acid
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C26H20Cl2F4N2O7S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 8 nM
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CP0496381
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2-[4-[4-(butylcarbamoyl)-2-[(3,4-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
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C26H26Cl2N2O7S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 23 nM
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CP0476522
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2-[6-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-1-benzofuran-3-yl]acetic acid
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C27H24Cl2N2O7S
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1
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| 1 |
IC50 = 5 nM
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CP0327130
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2-[3-(1-benzyl-2-oxo-3H-1,4-benzodiazepin-5-yl)-4-methoxyphenyl]acetic acid
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C25H22N2O4
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 60 nM
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CP0432249
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2-[2-[(5-acetyl-2-propoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
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C21H21FN2O4S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 9 nM
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CP0475880
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2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-4-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
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C19H17FN2O4S
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2
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 10 nM
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CP0055873
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2-[8-fluoro-2-[2-(1H-indol-3-yl)acetyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C23H20FN3O3
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4
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 15 nM
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| 3 |
IC50 = 35 nM
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| 4 |
IC50 = 40 nM
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CP0130562
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2-[8-methyl-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
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C25H22N2O3
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3
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| 1 |
IC50 = 5 nM
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| 2 |
IC50 = 60 nM
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| 3 |
IC50 = 190 nM
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CP0240867
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2-(2-benzoyl-8-chloro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C20H17ClN2O3
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1
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| 1 |
IC50 = 5 nM
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CP0443723
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5-[7-[(5S)-5-(3-cyanophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
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C30H25FN4O4
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1
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| 1 |
IC50 = 5.2 nM
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CP0381943
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2-(2,5-dimethyl-3-(7-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid
Show/Hide
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C22H17F3N2O2
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1
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| 1 |
IC50 = 5.4 nM
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CP0234514
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(R)-2-(7-(4-methoxy-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C22H24N2O5S
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1
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| 1 |
IC50 = 5.5 nM
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CP0459722
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2-[3-[3-[3,3-diphenylpropyl-(4-methoxybenzoyl)amino]propyl]phenoxy]acetic acid
Show/Hide
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C34H35NO5
|
1
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| 1 |
IC50 = 5.5 nM
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CP0399934
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(S)-2-(4-chloro-2-((4-(2-(2-chlorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
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C22H24Cl2N2O4
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1
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| 1 |
IC50 = 5.6 nM
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CP0287896
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2-((R)-8-((R)-2-(4-fluorophenyl)-N-methylpropanamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
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C23H24FN3O3
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2
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| 1 |
IC50 = 5.7 nM
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| 2 |
Ki = 3.4 nM
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CP0081606
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(R)-2-(7-(4-fluoro-N-(4-fluorobenzyl)phenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C27H24F2N2O4S
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1
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| 1 |
IC50 = 5.7 nM
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CP0332328
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(R)-2-(3-chloro-2-fluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H19ClF2N2O4S
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1
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| 1 |
IC50 = 5.7 nM
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CP0443724
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5-[3-(4-fluorophenyl)-7-[(5S)-5-[(R)-hydroxy(phenyl)methyl]-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O5
|
1
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| 1 |
IC50 = 5.7 nM
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CP0509308
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2-[3-[3-[5-[bis(4-methoxyphenyl)methyl]-2-oxopyridin-1-yl]propyl]phenoxy]acetic acid
Show/Hide
|
C31H31NO6
|
1
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| 1 |
IC50 = 5.8 nM
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CP0433527
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2-(2,5-dimethyl-3-(8-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid
Show/Hide
|
C22H17F3N2O2
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1
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| 1 |
IC50 = 6 nM
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CP0415002
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2-(4-(4-(cyclopentylcarbamoyl)-2-(2,4-dichlorophenylsulfonamido)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C27H26Cl2N2O7S
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1
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| 1 |
IC50 = 6 nM
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CP0695948
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Sodium [2'-[(cyclopropanecarbonyl-ethyl-amino)-methyl]-4'-(6-ethoxy-pyridin-3-yl)-6-methoxy-biphenyl-3-yl]-acetate
Show/Hide
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C29H31N2NaO5
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 31 nM
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CP0506025
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2-(2-((4-(benzylsulfonyl)piperazin-1-yl)methyl)-4-chlorophenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
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| 1 |
IC50 = 6 nM
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CP0391759
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2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-chlorophenyl]acetic acid
Show/Hide
|
C25H23Cl3N2O6S
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 90 nM
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CP0496380
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2-[3-chloro-4-[2-[(4-chlorophenyl)sulfonylamino]-4-(cyclobutylcarbamoyl)phenoxy]phenyl]acetic acid
Show/Hide
|
C25H22Cl2N2O6S
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 12 nM
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CP0417155
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2-[4-[2-[(2,4-dichlorophenyl)sulfonylamino]-4-(5-ethyl-1H-1,2,4-triazol-3-yl)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C25H22Cl2N4O6S
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1
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| 1 |
IC50 = 6 nM
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CP0348730
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2-[3-[1-[(3,4-difluorophenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]-4-methoxyphenyl]acetic acid
Show/Hide
|
C25H20F2N2O4
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2
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| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 15 nM
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CP0087804
|
ACT-129968
Show/Hide
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C24H19FN2O3
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4
|
| 1 |
IC50 = 6 nM
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| 2 |
IC50 = 30 nM
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| 3 |
IC50 = 80 nM
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| 4 |
IC50 = 340 nM
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CP0401618
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2-[3-[3-[5-[bis(4-methylphenyl)methyl]-2-oxopyridin-1-yl]propyl]phenoxy]acetic acid
Show/Hide
|
C31H31NO4
|
1
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| 1 |
IC50 = 6.2 nM
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CP0371087
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(R)-2-(7-(N-(cyclopropylmethyl)-4-fluorophenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C24H25FN2O4S
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1
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| 1 |
IC50 = 6.7 nM
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CP0447088
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(S)-2-(4-chloro-2-((4-(2-(3-chlorophenyl)acetyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C22H24Cl2N2O4
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1
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| 1 |
IC50 = 6.8 nM
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CP0257988
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(R)-2-(7-(4-fluoro-N-(2,2,2-trifluoroethyl)phenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C22H20F4N2O4S
|
1
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| 1 |
IC50 = 6.9 nM
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CP0495695
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2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(pentylcarbamoyl)phenoxy)-3-methoxyphenyl)acetic acid
Show/Hide
|
C27H28Cl2N2O7S
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1
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| 1 |
IC50 = 7 nM
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CP0496655
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2-(3-(2-(4-chlorophenylsulfonamido)-4-propionamidophenoxy)phenyl)acetic acid
Show/Hide
|
C23H21ClN2O6S
|
1
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| 1 |
IC50 = 7 nM
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CP0502785
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2-(3-(4-(ethylcarbamoyl)-2-(4-methylphenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C24H24N2O6S
|
1
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| 1 |
IC50 = 7 nM
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CP0379723
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(R)-2-(8-(4-(4-fluorophenyl)-N-methyltetrahydro-2H-pyran-4-carboxamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C26H28FN3O4
|
2
|
| 1 |
IC50 = 7 nM
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| 2 |
Ki = 11.5 nM
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CP0499526
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2-(4'-acetamido-2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-6-methoxybiphenyl-3-yl)acetic acid
Show/Hide
|
C28H30N2O6
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2
|
| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 60 nM
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CP0505623
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2-(2'-((N-ethylcyclopropanecarboxamido)methyl)-6-methoxy-4'-(quinolin-3-yl)biphenyl-3-yl)acetic acid
Show/Hide
|
C31H30N2O4
|
2
|
| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 52 nM
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CP0390767
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2-[3-[2-[(4-chlorophenyl)methylcarbamoyl]-4-(propanoylamino)phenoxy]-4-methoxyphenyl]acetic acid
Show/Hide
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C26H25ClN2O6
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 65 nM
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CP0406440
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2-[3-chloro-4-[4-(cyclopropylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]phenyl]acetic acid
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C24H19Cl3N2O6S
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 25 nM
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CP0510763
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2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-fluorophenyl]acetic acid
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C25H23Cl2FN2O6S
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 110 nM
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CP0327131
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2-[3-[1-[(4-chlorophenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]-4-methoxyphenyl]acetic acid
Show/Hide
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C25H21ClN2O4
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2
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| 1 |
IC50 = 7 nM
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| 2 |
IC50 = 22 nM
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CP0156971
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2-(2-benzoyl-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C20H17FN2O3
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1
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| 1 |
IC50 = 7 nM
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CP0444403
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4-[[(2aS,8R,8aR)-3-[4-(trifluoromethoxy)benzoyl]-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C26H25F3N2O5
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2
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| 1 |
IC50 = 7 nM
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| 2 |
Ki = 4 nM
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CP0390633
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2-(3-(8-fluoroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid
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C21H17FN2O2
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1
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| 1 |
IC50 = 7.1 nM
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CP0410061
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(R)-2-(8-(1-(4-fluorophenyl)-N-methylcyclopropanecarboxamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
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C24H24FN3O3
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2
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| 1 |
IC50 = 7.5 nM
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| 2 |
Ki = 3.6 nM
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CP0481765
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5-[7-[(5S)-5-(3,5-difluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
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C29H24F3N3O4
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1
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| 1 |
IC50 = 7.8 nM
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CP0274942
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2-(3-(7-chloroquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid
Show/Hide
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C21H17ClN2O2
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1
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| 1 |
IC50 = 8 nM
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CP0473345
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2-(((benzyloxycarbonyl)(ethyl)amino)methyl)-5'-(carboxymethyl)-2'-methoxybiphenyl-4-carboxylic acid
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C27H27NO7
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 254 nM
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CP0392770
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2-[4-[4-(butylcarbamoyl)-2-[(2,5-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
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C26H26Cl2N2O7S
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 69 nM
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CP0163597
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2-[3-[1-[(3-chlorophenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]-4-methoxyphenyl]acetic acid
Show/Hide
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C25H21ClN2O4
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 78 nM
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CP0469000
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2-[4-[[2-cyclopropyl-4-[(2,4-dichlorophenyl)sulfonylamino]-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
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C26H22Cl2N2O6S
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2
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| 1 |
IC50 = 8 nM
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| 2 |
IC50 = 25 nM
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CP0063174
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4-[[(3aS,9R,9aR)-7-fluoro-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C27H26F4N2O5
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2
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| 1 |
IC50 = 8 nM
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| 2 |
Ki = 5 nM
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CP0162672
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(R)-2-(7-(N-ethyl-4-fluorophenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C22H23FN2O4S
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1
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| 1 |
IC50 = 8.1 nM
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CP0395524
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5-[3-(4-fluorophenyl)-7-[(5S)-5-methyl-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
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C29H26FN3O4
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1
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| 1 |
IC50 = 8.1 nM
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CP0117321
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(R)-2-(7-(4-chloro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C21H21ClN2O4S
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1
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| 1 |
IC50 = 8.5 nM
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CP0384322
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(+/-)-N-(1-(4-methoxybenzoyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
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C26H26N2O3
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 28 nM
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CP0225634
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(R)-2-(3-cyano-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C22H20FN3O4S
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1
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| 1 |
IC50 = 9 nM
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CP0470311
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2-(2'-((N-ethylcyclopropanecarboxamido)methyl)-4'-(5-fluoropyridin-2-yl)-6-methoxybiphenyl-3-yl)acetic acid
Show/Hide
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C27H27FN2O4
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 60 nM
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CP0391758
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2-[4-[4-(tert-butylcarbamoyl)-2-[(4-chlorophenyl)sulfonylamino]phenoxy]-3-chlorophenyl]acetic acid
Show/Hide
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C25H24Cl2N2O6S
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 15 nM
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CP0504138
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2-[4-[4-(tert-butylcarbamoyl)-2-[[2-chloro-4-(trifluoromethoxy)phenyl]sulfonylamino]phenoxy]-5-chloro-2-fluorophenyl]acetic acid
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C26H22Cl2F4N2O7S
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 19 nM
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CP0432248
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2-[2-[(5-acetyl-2-butoxyphenyl)methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
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C22H23FN2O4S
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2
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| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 12 nM
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CP0045673
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2-[2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H16ClFN2O3
|
4
|
| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 40 nM
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| 3 |
IC50 = 60 nM
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| 4 |
IC50 = 95 nM
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CP0055416
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2-[2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H20N2O3
|
4
|
| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 30 nM
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| 3 |
IC50 = 140 nM
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| 4 |
IC50 = 420 nM
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CP0055877
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2-[2-benzoyl-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C21H17F3N2O3
|
4
|
| 1 |
IC50 = 9 nM
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| 2 |
IC50 = 50 nM
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| 3 |
IC50 = 60 nM
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| 4 |
IC50 = 160 nM
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CP0401617
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2-[3-[3-[5-[bis(4-chlorophenyl)methyl]-2-oxopyridin-1-yl]propyl]phenoxy]acetic acid
Show/Hide
|
C29H25Cl2NO4
|
1
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| 1 |
IC50 = 9.2 nM
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CP0401620
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2-[3-[3-[benzoyl(3,3-diphenylpropyl)amino]propyl]phenoxy]acetic acid
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C33H33NO4
|
1
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| 1 |
IC50 = 9.7 nM
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CP0073144
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5-[7-[(5S)-5-(1,3-benzoxazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H25FN4O5
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1
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| 1 |
IC50 = 9.7 nM
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CP0234517
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(R)-2-(2,4-difluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H19F3N2O4S
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1
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| 1 |
IC50 = 9.9 nM
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CP0475043
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2-(3-chloro-5-(2-(2,4-dichloro-5-methylphenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
Show/Hide
|
C24H21Cl3N2O6S
|
1
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| 1 |
IC50 = 10 nM
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CP0441306
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2-(6-(2-chloro-4-(methylsulfonyl)benzyl)-5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
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C17H16ClNO4S2
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2
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| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 45000 nM
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CP0506024
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2-(4-chloro-2-((4-(4-fluorophenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
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C19H20ClFN2O5S
|
1
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| 1 |
IC50 = 10 nM
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CP0417114
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2-[5-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]pyridin-2-yl]acetic acid
Show/Hide
|
C24H23Cl2N3O6S
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1
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| 1 |
IC50 = 10 nM
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CP0055420
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2-[2-(3-chlorobenzoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H17ClN2O3
|
4
|
| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 30 nM
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| 3 |
IC50 = 40 nM
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| 4 |
IC50 = 70 nM
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CP0083568
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2-[8-fluoro-2-(3-naphthalen-1-ylpropanoyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C26H23FN2O3
|
4
|
| 1 |
IC50 = 10 nM
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| 2 |
IC50 = 30 nM
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| 3 |
IC50 = 65 nM
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| 4 |
IC50 = 160 nM
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CP0389632
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5-[3-(4-fluorophenyl)-7-[(5S)-5-(4-fluorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H25F2N3O4
|
1
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| 1 |
IC50 = 10.2 nM
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CP0478950
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5-[7-[(5S)-5-(4-chlorophenyl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H25ClFN3O4
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1
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| 1 |
IC50 = 10.5 nM
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CP0421158
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2-(3-(8-methoxyquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid
Show/Hide
|
C22H20N2O3
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1
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| 1 |
IC50 = 11 nM
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CP0459813
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2-[3-[3-[5-[bis(4-fluorophenyl)methyl]-2-oxopyridin-1-yl]propyl]phenoxy]acetic acid
Show/Hide
|
C29H25F2NO4
|
1
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| 1 |
IC50 = 11 nM
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CP0476535
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4-[3-[3-(5-benzhydryl-2-oxopyridin-1-yl)propyl]phenoxy]butanoic acid
Show/Hide
|
C31H31NO4
|
1
|
| 1 |
IC50 = 11 nM
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CP0261961
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2-[2-(naphthalene-1-carbonyl)-8-(trifluoromethyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C25H19F3N2O3
|
4
|
| 1 |
IC50 = 11 nM
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| 2 |
IC50 = 20 nM
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| 3 |
IC50 = 70 nM
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| 4 |
IC50 = 380 nM
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CP0283176
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2-(2-benzoyl-8-methyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C21H20N2O3
|
1
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| 1 |
IC50 = 11 nM
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CP0475053
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2-(3-chloro-5-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
Show/Hide
|
C23H19Cl3N2O6S
|
1
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| 1 |
IC50 = 12 nM
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CP0117319
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(R)-2-(7-(N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H22N2O4S
|
1
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| 1 |
IC50 = 12 nM
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CP0490691
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2-(2'-(((benzyloxycarbonyl)(ethyl)amino)methyl)-4'-(2-hydroxypropan-2-yl)-6-methoxybiphenyl-3-yl)acetic acid
Show/Hide
|
C29H33NO6
|
2
|
| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 24 nM
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CP0439418
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2-[4-[4-(butylcarbamoyl)-2-[(2,6-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C26H26Cl2N2O7S
|
2
|
| 1 |
IC50 = 12 nM
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| 2 |
IC50 = 1180 nM
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CP0516002
|
4-[[(3aS,9R,9aR)-7-fluoro-4-[4-(trifluoromethylsulfanyl)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
|
C27H26F4N2O4S
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2
|
| 1 |
IC50 = 12 nM
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| 2 |
Ki = 8.4 nM
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CP0441808
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2-[4-(3,5-difluorophenyl)-2-(1-phenylpyrazole-4-carbonyl)phenoxy]acetic acid
Show/Hide
|
C24H16F2N2O4
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2
|
| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 147 nM
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CP0539417
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(+/-)-N-(2-methyl-1-(4-phenoxybenzoyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C31H28N2O3
|
1
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| 1 |
IC50 = 13 nM
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CP0414998
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2-(3-(4-(ethylcarbamoyl)-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C23H22N2O6S
|
1
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| 1 |
IC50 = 13 nM
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CP0055129
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(R)-2-(7-(N,3-dimethylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C22H24N2O4S
|
1
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| 1 |
IC50 = 13 nM
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CP0332329
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(R)-2-(7-(5-chloro-N-methylthiophene-2-sulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C19H19ClN2O4S2
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1
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| 1 |
IC50 = 13 nM
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CP0405857
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4-[3-[3-(3-benzhydryl-6-oxopyridazin-1-yl)propyl]phenoxy]butanoic acid
Show/Hide
|
C30H30N2O4
|
1
|
| 1 |
IC50 = 13 nM
|
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CP0406441
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2-[4-[2-[[2-chloro-4-(trifluoromethyl)phenyl]sulfonylamino]-4-(cyclobutylcarbamoyl)phenoxy]-2,5-difluorophenyl]acetic acid
Show/Hide
|
C26H20ClF5N2O6S
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2
|
| 1 |
IC50 = 13 nM
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| 2 |
IC50 = 41 nM
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CP0432909
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5-[7-[(5S)-5-benzyl-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O4
|
1
|
| 1 |
IC50 = 13.7 nM
|
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|
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CP0399062
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2-[3-[2-[[(1R)-1-(4-chlorophenyl)ethyl]carbamoyl]-4-(propanoylamino)phenoxy]-4-methoxyphenyl]acetic acid
Show/Hide
|
C27H27ClN2O6
|
2
|
| 1 |
IC50 = 14 nM
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| 2 |
IC50 = 260 nM
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CP0371875
|
4-chloro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
Show/Hide
|
C18H13ClN2O4
|
2
|
| 1 |
IC50 = 15 nM
|
|
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| 2 |
IC50 = 185 nM
|
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CP0417941
|
N-[(2S,4R)-1-(3-methoxybenzoyl)-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N-phenylacetamide
Show/Hide
|
C26H26N2O3
|
2
|
| 1 |
IC50 = 15 nM
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| 2 |
IC50 > 10000 nM
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CP0053453
|
(R)-2-(7-(4-ethyl-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C23H26N2O4S
|
1
|
| 1 |
IC50 = 15 nM
|
|
|
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CP0327132
|
2-[4-methoxy-3-[1-[(4-methylphenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]phenyl]acetic acid
Show/Hide
|
C26H24N2O4
|
2
|
| 1 |
IC50 = 15 nM
|
|
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| 2 |
IC50 = 104 nM
|
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|
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CP0115424
|
2-[2-[[5-(butylcarbamoyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C22H24FN3O4S
|
3
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
IC50 = 16 nM
|
|
|
| 3 |
IC50 = 81 nM
|
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CP0378064
|
2-[2-[[5-(ethylcarbamoyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C20H20FN3O4S
|
2
|
| 1 |
IC50 = 15 nM
|
|
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| 2 |
IC50 = 16 nM
|
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|
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CP0070143
|
2-(2-benzoyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C20H18N2O3
|
4
|
| 1 |
IC50 = 15 nM
|
|
|
| 2 |
IC50 = 17 nM
|
|
|
| 3 |
IC50 = 170 nM
|
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| 4 |
IC50 = 190 nM
|
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|
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CP0461375
|
5-[7-[(5R)-5-benzyl-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O4
|
1
|
| 1 |
IC50 = 15.2 nM
|
|
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CP0392937
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2-(3-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
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C23H20Cl2N2O6S
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1
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| 1 |
IC50 = 16 nM
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CP0495694
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2-(3-(2-(4-chlorophenylsulfonamido)-4-(3-ethylureido)phenoxy)phenyl)acetic acid
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C23H22ClN3O6S
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1
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| 1 |
IC50 = 16 nM
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CP0511333
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2-[2-[[4-(benzenesulfonyl)piperazin-1-yl]methyl]-4-chlorophenoxy]acetic acid
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C19H21ClN2O5S
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1
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| 1 |
IC50 = 16 nM
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CP0392761
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2-[3-[3-(5-benzhydryl-2-oxopyridin-1-yl)propyl]phenoxy]propanoic acid
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C30H29NO4
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1
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| 1 |
IC50 = 17 nM
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CP0388965
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5-[7-[(5S)-5-(1,3-benzothiazol-2-yl)-5-methyl-4H-1,2-oxazol-3-yl]-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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C30H25FN4O4S
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1
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| 1 |
IC50 = 17.2 nM
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CP0376268
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2-(2,5-dimethyl-3-(2-methylquinolin-4-yl)-1H-indol-1-yl)acetic acid
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C22H20N2O2
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1
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| 1 |
IC50 = 18 nM
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CP0395339
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2-(3-(8-cyanoquinolin-4-yl)-2,5-dimethyl-1H-indol-1-yl)acetic acid
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C22H17N3O2
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1
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| 1 |
IC50 = 18 nM
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CP0461748
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2-(2-((4-(phenylsulfonyl)piperazin-1-yl)methyl)-4-(trifluoromethyl)phenoxy)acetic acid
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C20H21F3N2O5S
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1
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| 1 |
IC50 = 18 nM
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CP0392760
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2-[3-[3-(3-benzhydryl-6-oxopyridazin-1-yl)propyl]phenoxy]acetic acid
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C28H26N2O4
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1
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| 1 |
IC50 = 18 nM
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CP0492399
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2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-cyanophenyl]acetic acid
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C26H23Cl2N3O6S
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2
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| 1 |
IC50 = 18 nM
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| 2 |
IC50 = 210 nM
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CP0447102
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2-[4-[4-[(2,4-dichlorophenyl)sulfonylamino]-1-methylindol-5-yl]oxy-3-methoxyphenyl]acetic acid
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C24H20Cl2N2O6S
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2
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| 1 |
IC50 = 18 nM
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| 2 |
IC50 = 56 nM
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CP0444401
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4-[[(3aS,9R,9aR)-6-chloro-7-fluoro-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
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C27H25ClF4N2O5
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2
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| 1 |
IC50 = 18 nM
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| 2 |
Ki = 3.4 nM
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CP0388963
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5-[3-(4-fluorophenyl)-7-(5-methyl-5-phenyl-4H-1,2-oxazol-3-yl)-4-oxoquinazolin-2-yl]pentanoic acid
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C29H26FN3O4
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1
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| 1 |
IC50 = 18.6 nM
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CP0441307
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2-(6-(4-(N-cyclohexyl-N-methylsulfamoyl)benzyl)-5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
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C23H28N2O4S2
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2
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| 1 |
IC50 = 20 nM
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| 2 |
IC50 = 31000 nM
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CP0425641
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(S)-2-(4-chloro-2-((4-(2-(4-chlorophenyl)-2-methylpropanoyl)-3-methylpiperazin-1-yl)methyl)phenoxy)acetic acid
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C24H28Cl2N2O4
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1
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| 1 |
IC50 = 20 nM
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CP0478535
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4-[[(2aS,8R,8aR)-3-(4-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid
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C25H25FN2O4
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2
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| 1 |
IC50 = 20 nM
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| 2 |
Ki = 7.3 nM
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CP0391088
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2-(2,5-dimethyl-3-(quinolin-4-yl)-1H-indol-1-yl)acetic acid
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C21H18N2O2
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1
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| 1 |
IC50 = 21 nM
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CP0476523
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2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]sulfanylphenyl]acetic acid
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C25H24Cl2N2O5S2
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1
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| 1 |
IC50 = 21 nM
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CP0529079
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(+/-)-5-((1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-5-oxopentanoic acid
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C28H28N2O4
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1
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| 1 |
IC50 = 22 nM
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CP0117316
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(R)-2-(7-(2-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C21H21FN2O4S
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1
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| 1 |
IC50 = 22 nM
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CP0499518
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2-[4-[4-[(2,4-dichlorophenyl)sulfonylamino]-1,2-dimethylindol-5-yl]oxy-3-methoxyphenyl]acetic acid
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C25H22Cl2N2O6S
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2
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| 1 |
IC50 = 22 nM
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| 2 |
IC50 = 56 nM
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CP0433528
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2-(2,5-dimethyl-3-(8-(methylsulfonyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid
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C22H20N2O4S
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1
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| 1 |
IC50 = 23 nM
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CP0086399
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2-[6-chloro-2-[4-(4-ethylphenyl)benzoyl]-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
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C28H25ClN2O3
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3
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| 1 |
IC50 = 23 nM
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| 2 |
IC50 = 90 nM
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| 3 |
IC50 = 2600 nM
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CP0081601
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(R)-2-(1,3-dichloro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C21H19Cl2FN2O4S
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1
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| 1 |
IC50 = 24 nM
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CP0382771
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N-[(2S,4R)-2-methyl-1-[3-(trifluoromethoxy)benzoyl]-3,4-dihydro-2H-quinolin-4-yl]-N-phenylacetamide
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C26H23F3N2O3
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2
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| 1 |
IC50 = 25 nM
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| 2 |
IC50 = 106 nM
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CP0053449
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(R)-2-(7-(1-(4-fluorophenyl)-N-methylmethylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C22H23FN2O4S
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1
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| 1 |
IC50 = 25 nM
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CP0391760
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2-[4-[2-[[2-chloro-4-(trifluoromethoxy)phenyl]sulfonylamino]-4-(cyclobutylcarbamoyl)phenoxy]-2,5-difluorophenyl]acetic acid
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C26H20ClF5N2O7S
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2
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| 1 |
IC50 = 25 nM
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| 2 |
IC50 = 53 nM
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CP0384321
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(+/-)-N-(2-methyl-1-(4-(trifluoromethoxy)benzoyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
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C26H23F3N2O3
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2
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| 1 |
IC50 = 26 nM
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| 2 |
IC50 > 10000 nM
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CP0055828
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(R)-2-(1-fluoro-7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C21H20F2N2O4S
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1
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| 1 |
IC50 = 26.5 nM
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CP0117317
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(R)-2-(7-(N,2-dimethylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
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C22H24N2O4S
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1
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| 1 |
IC50 = 27 nM
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CP0499543
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2-(2'-((N-ethylcyclopropanecarboxamido)methyl)-6-methoxy-4'-(5-methoxypyrimidin-2-yl)biphenyl-3-yl)acetic acid
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C27H29N3O5
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2
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| 1 |
IC50 = 27 nM
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| 2 |
IC50 = 107 nM
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CP0519971
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2-(2'-((N-ethylcyclopropanecarboxamido)methyl)-6-methoxy-4'-(1-methyl-1H-pyrazol-4-yl)biphenyl-3-yl)acetic acid
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C26H29N3O4
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2
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| 1 |
IC50 = 27 nM
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| 2 |
IC50 = 37 nM
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CP0440874
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2-[4-[[2-cyano-4-[(2,4-dichlorophenyl)sulfonylamino]-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
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C24H17Cl2N3O6S
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2
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| 1 |
IC50 = 27 nM
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| 2 |
IC50 = 130 nM
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CP0496653
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2-(3-chloro-5-(2-(2-chloro-4-(trifluoromethyl)phenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)acetic acid
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C24H19Cl2F3N2O6S
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1
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| 1 |
IC50 = 28 nM
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CP0447089
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2-[2-[[4-(benzenesulfonyl)-2-methylpiperazin-1-yl]methyl]-4-chlorophenoxy]acetic acid
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C20H23ClN2O5S
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1
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| 1 |
IC50 = 28 nM
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CP0473220
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(R)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)acetic acid
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C20H23ClN2O5S
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1
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| 1 |
IC50 = 28 nM
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CP0530195
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2-[4-methoxy-3-[2-[(4-methylphenyl)sulfonylamino]benzoyl]phenyl]acetic acid
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C23H21NO6S
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1
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| 1 |
IC50 = 28 nM
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CP0526340
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(+/-)-4-(aminooxy)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-4-oxo-N-phenylbutanamide
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C27H27N3O4
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1
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| 1 |
IC50 = 29 nM
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CP0127125
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2-[3-[1-[(2,4-dichlorophenyl)methyl]-2-oxo-3H-1,4-benzodiazepin-5-yl]-4-methoxyphenyl]acetic acid
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C25H20Cl2N2O4
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2
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| 1 |
IC50 = 29 nM
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| 2 |
IC50 = 240 nM
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CP0425708
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2-[2-[(2-methoxy-5-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
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C19H18N2O5S
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1
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| 1 |
IC50 = 29 nM
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CP0073641
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2-[4-methoxy-3-[2-oxo-1-[[4-(trifluoromethyl)phenyl]methyl]-3H-1,4-benzodiazepin-5-yl]phenyl]acetic acid
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C26H21F3N2O4
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1
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| 1 |
IC50 = 30 nM
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CP0392772
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2-[4-[4-(butylcarbamoyl)-2-[(2,3-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
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C26H26Cl2N2O7S
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2
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| 1 |
IC50 = 32 nM
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| 2 |
IC50 = 300 nM
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CP0419061
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2-[4-[[2-tert-butyl-4-[(2,4-dichlorophenyl)sulfonylamino]-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
Show/Hide
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C27H26Cl2N2O6S
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1
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| 1 |
IC50 = 32 nM
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CP0440872
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2-[4-[[4-[(2,4-dichlorophenyl)sulfonylamino]-2-(2-methylpropyl)-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
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C27H26Cl2N2O6S
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2
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| 1 |
IC50 = 32 nM
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| 2 |
IC50 = 48 nM
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CP0239695
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(R)-2-(7-(3-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C21H21FN2O4S
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1
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| 1 |
IC50 = 33 nM
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CP0508741
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2-[5-acetyl-2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
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C21H20N2O5S
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2
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| 1 |
IC50 = 33 nM
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| 2 |
IC50 = 63 nM
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CP0395522
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5-[7-(5,5-diphenyl-4H-1,2-oxazol-3-yl)-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
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C34H28FN3O4
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1
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| 1 |
IC50 = 33.7 nM
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CP0459106
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(+/-)-N-(1-(4-tert-butylbenzoyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
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C29H32N2O2
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1
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| 1 |
IC50 = 34 nM
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CP0261505
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2-(2-benzoyl-6,8-difluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C20H16F2N2O3
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1
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| 1 |
IC50 = 35 nM
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CP0162671
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(R)-2-(7-(4-fluorophenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C20H19FN2O4S
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1
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| 1 |
IC50 = 35.5 nM
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CP0371874
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2-[4-(4-chlorophenyl)-2-(1-phenylpyrazole-4-carbonyl)phenoxy]acetic acid
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C24H17ClN2O4
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2
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| 1 |
IC50 = 37 nM
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| 2 |
IC50 = 448 nM
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CP0239678
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(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-3-(methylsulfonyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C22H23FN2O6S2
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1
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| 1 |
IC50 = 38 nM
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CP0461325
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5-[7-(5-ethyl-5-phenyl-4H-1,2-oxazol-3-yl)-3-(4-fluorophenyl)-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
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C30H28FN3O4
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1
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| 1 |
IC50 = 38.7 nM
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CP0506324
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4-(((2R,4S)-1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-4-oxobutanoic acid
Show/Hide
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C27H26N2O4
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2
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| 1 |
IC50 = 39 nM
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| 2 |
IC50 = 400 nM
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CP0529082
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(+/-)-N-(2-methyl-1-(4-methylbenzoyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
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C26H26N2O2
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1
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| 1 |
IC50 = 41 nM
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CP0462639
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2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-5-methylsulfonylbenzimidazol-1-yl]acetic acid
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C20H20N2O6S2
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2
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| 1 |
IC50 = 41 nM
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| 2 |
IC50 = 50 nM
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CP0541450
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4-[(4-benzoyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl)-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C26H28N2O4
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2
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| 1 |
IC50 = 41 nM
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| 2 |
Ki = 10 nM
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CP0532321
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3-(1-phenyl-1H-pyrazole-4-carbonyl)biphenyl-4-yloxyacetic acid
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C24H18N2O4
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2
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| 1 |
IC50 = 42 nM
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| 2 |
IC50 = 485 nM
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CP0401616
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2-[3-[3-(5-benzhydryl-2-oxopyridin-1-yl)propyl]phenoxy]acetic acid
Show/Hide
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C29H27NO4
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1
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| 1 |
IC50 = 42 nM
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CP0199029
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2-(2-benzoyl-8-propan-2-yl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
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C23H24N2O3
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1
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| 1 |
IC50 = 42 nM
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CP0489267
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2-[2-[(5-acetyl-2-methoxyphenyl)methylsulfanyl]-6-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
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C19H17FN2O4S
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2
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| 1 |
IC50 = 45 nM
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| 2 |
IC50 = 89 nM
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CP0548523
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2-[2-[(2-bromo-5-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
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C18H15BrN2O4S
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1
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| 1 |
IC50 = 45 nM
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CP0408403
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4-nitro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
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C18H13N3O6
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2
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| 1 |
IC50 = 47 nM
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| 2 |
IC50 = 236 nM
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CP0544209
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2-(3-(4-carbamoyl-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
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C21H18N2O6S
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1
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| 1 |
IC50 = 47 nM
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CP0409146
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4-methyl-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
Show/Hide
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C19H16N2O4
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2
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| 1 |
IC50 = 48 nM
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| 2 |
IC50 = 587 nM
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CP0381784
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2-(3-(7-chloroquinolin-4-yl)-5-methoxy-2-methyl-1H-indol-1-yl)acetic acid
Show/Hide
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C21H17ClN2O3
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1
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| 1 |
IC50 = 50 nM
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CP0469170
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2-(5-methyl-6-(4-(methylsulfonyl)benzyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C17H17NO4S2
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2
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| 1 |
IC50 = 50 nM
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| 2 |
IC50 = 31000 nM
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CP0511435
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2-(2-{[(3S)-4-(benzylsulfonyl)-3-methylpiperazin-1-yl]methyl}-4-chlorophenyl)-N-(methylsulfonyl)acetamide
Show/Hide
|
C22H28ClN3O5S2
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1
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| 1 |
IC50 = 50 nM
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CP0425385
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2-(2-benzoyl-4-bromophenoxy)acetic acid
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C15H11BrO4
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2
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| 1 |
IC50 = 53 nM
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| 2 |
IC50 = 437 nM
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CP0949926
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{4-bromo-2-[(quinolin-8-ylhydrazono)methyl]phenoxy}acetic acid
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C18H14BrN3O3
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2
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| 1 |
IC50 = 54 nM
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| 2 |
IC50 = 643 nM
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CP0506594
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2-[4-[[4-[(2,4-dichlorophenyl)sulfonylamino]-2-propyl-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
Show/Hide
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C26H24Cl2N2O6S
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2
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| 1 |
IC50 = 57 nM
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| 2 |
IC50 = 110 nM
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CP0461374
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5-[3-(4-fluorophenyl)-7-[5-(hydroxymethyl)-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C29H26FN3O5
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1
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| 1 |
IC50 = 58.5 nM
|
|
|
|
CP0494077
|
2-[2-[[5-(benzylcarbamoyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C25H22FN3O4S
|
2
|
| 1 |
IC50 = 59 nM
|
|
|
| 2 |
IC50 = 94 nM
|
|
|
|
CP0453602
|
2-(4-bromo-2-tert-butylphenoxy)acetic acid
Show/Hide
|
C12H15BrO3
|
2
|
| 1 |
IC50 = 61 nM
|
|
|
| 2 |
IC50 = 423 nM
|
|
|
|
CP0199053
|
2-(2-benzoyl-8-methoxy-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C21H20N2O4
|
1
|
| 1 |
IC50 = 62 nM
|
|
|
|
CP0055133
|
(R)-2-(7-(N,1-dimethyl-1H-pyrazole-4-sulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C19H22N4O4S
|
1
|
| 1 |
IC50 = 63 nM
|
|
|
|
CP0539414
|
(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylpentanamide
Show/Hide
|
C28H30N2O2
|
1
|
| 1 |
IC50 = 64 nM
|
|
|
|
CP0467286
|
2-(2,5-dimethyl-3-(6-(trifluoromethyl)quinolin-4-yl)-1H-indol-1-yl)acetic acid
Show/Hide
|
C22H17F3N2O2
|
1
|
| 1 |
IC50 = 68 nM
|
|
|
|
CP0506029
|
2-(5-methyl-6-(4-(morpholinosulfonyl)benzyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C20H22N2O5S2
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0110764
|
2-[4-methoxy-3-[2-oxo-1-[[4-(trifluoromethoxy)phenyl]methyl]-3H-1,4-benzodiazepin-5-yl]phenyl]acetic acid
Show/Hide
|
C26H21F3N2O5
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
|
CP0156867
|
2-[2-(cyclohexanecarbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H24N2O3
|
2
|
| 1 |
IC50 = 70 nM
|
|
|
| 2 |
IC50 = 200 nM
|
|
|
|
CP0156868
|
2-[6-chloro-8-fluoro-2-(naphthalene-1-carbonyl)-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C24H18ClFN2O3
|
3
|
| 1 |
IC50 = 70 nM
|
|
|
| 2 |
IC50 = 530 nM
|
|
|
| 3 |
IC50 = 660 nM
|
|
|
|
CP0405110
|
2-[2-[(4-benzoyl-3-methylpiperazin-1-yl)methyl]-4-chlorophenoxy]acetic acid
Show/Hide
|
C21H23ClN2O4
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0503271
|
2-(4-chloro-2-(((3S,5R)-3,5-dimethyl-4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C23H27ClN2O4
|
1
|
| 1 |
IC50 = 71 nM
|
|
|
|
CP0487212
|
2-[2-[(3-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O3S
|
1
|
| 1 |
IC50 = 72 nM
|
|
|
|
CP0506429
|
2-[2-[[5-(diethylcarbamoyl)-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C22H24FN3O4S
|
2
|
| 1 |
IC50 = 72 nM
|
|
|
| 2 |
IC50 = 130 nM
|
|
|
|
CP0489432
|
5-[3-(4-fluorophenyl)-4-oxo-7-(5-phenyl-5-propyl-4H-1,2-oxazol-3-yl)quinazolin-2-yl]pentanoic acid
Show/Hide
|
C31H30FN3O4
|
1
|
| 1 |
IC50 = 73.4 nM
|
|
|
|
CP0410059
|
2-((R)-8-((S)-2-(4-fluorophenyl)-N-methylpropanamido)-6,7,8,9-tetrahydropyrido[3,2-b]indolizin-5-yl)acetic acid
Show/Hide
|
C23H24FN3O3
|
2
|
| 1 |
IC50 = 73.8 nM
|
|
|
| 2 |
Ki = 21.1 nM
|
|
|
|
CP0417942
|
(+/-)-N-((2-methyl-1-(3-methylbenzoyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0452150
|
2-[4-[4-(butylcarbamoyl)-2-[(4-chlorophenyl)sulfamoyl]phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C26H27ClN2O7S
|
1
|
| 1 |
IC50 = 76 nM
|
|
|
|
CP0048953
|
(R)-3-(3-(4-fluorophenylsulfonamido)-1,2,3,4-tetrahydrocarbazol-9-yl)propanoic acid
Show/Hide
|
C21H21FN2O4S
|
2
|
| 1 |
IC50 = 77 nM
|
|
|
| 2 |
Ki = 290 nM
|
|
|
|
CP0473222
|
3-(4-Chloro-2-{[(3S)-3-methyl-4-(phenylacetyl)piperazin-1-yl]methyl}phenyl)propanoic acid
Show/Hide
|
C23H27ClN2O3
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0503269
|
2-(2-((4-(benzylsulfonyl)-1,4-diazepan-1-yl)methyl)-4-chlorophenoxy)acetic acid
Show/Hide
|
C21H25ClN2O5S
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0473199
|
5-[3-(4-fluorophenyl)-7-[5-(methoxymethyl)-5-phenyl-4H-1,2-oxazol-3-yl]-4-oxoquinazolin-2-yl]pentanoic acid
Show/Hide
|
C30H28FN3O5
|
1
|
| 1 |
IC50 = 79.7 nM
|
|
|
|
CP0846863
|
(4-bromo-2-{[(5-phenyl-1,2,4-triazin-3-yl)hydrazono]methyl}phenoxy)acetic acid
Show/Hide
|
C18H14BrN5O3
|
2
|
| 1 |
IC50 = 89 nM
|
|
|
| 2 |
IC50 = 3210 nM
|
|
|
|
CP0469168
|
2-(5-methyl-6-(4-(methylsulfonyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C16H15NO6S3
|
2
|
| 1 |
IC50 = 90 nM
|
|
|
| 2 |
IC50 > 100000 nM
|
|
|
|
CP0522575
|
2-[5-fluoro-2-[[2-methoxy-5-(morpholine-4-carbonyl)phenyl]methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C22H22FN3O5S
|
2
|
| 1 |
IC50 = 91 nM
|
|
|
| 2 |
IC50 = 107 nM
|
|
|
|
CP0459105
|
(+/-)-N-(1-(3,4-dimethylbenzoyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C27H28N2O2
|
1
|
| 1 |
IC50 = 92 nM
|
|
|
|
CP0539416
|
(+/-)-N-(1-(4-chlorobenzoyl)-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C25H23ClN2O2
|
1
|
| 1 |
IC50 = 93 nM
|
|
|
|
CP0459723
|
2-[3-[2-(5-benzhydryl-2-oxopyridin-1-yl)ethoxy]phenoxy]acetic acid
Show/Hide
|
C28H25NO5
|
1
|
| 1 |
IC50 = 99 nM
|
|
|
|
CP0405109
|
2-(4-chloro-2-((4-(2-phenylacetyl)piperazin-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C21H23ClN2O4
|
1
|
| 1 |
IC50 = 100 nM
|
|
|
|
CP0417940
|
(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylbenzamide
Show/Hide
|
C30H26N2O2
|
1
|
| 1 |
IC50 = 105 nM
|
|
|
|
CP0480119
|
2-[2-[(3-methylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 105 nM
|
|
|
|
CP0398263
|
2-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)phenyl)propanoic acid
Show/Hide
|
C24H22Cl2N2O6S
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0343442
|
2-(2-benzoyl-6-methyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C21H20N2O3
|
1
|
| 1 |
IC50 = 107 nM
|
|
|
|
CP0445960
|
4-fluoro-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
Show/Hide
|
C18H13FN2O4
|
2
|
| 1 |
IC50 = 108 nM
|
|
|
| 2 |
IC50 = 1320 nM
|
|
|
|
CP0392975
|
2-[4-[4-(butylcarbamoyl)-2-(2-phenylethylamino)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C28H32N2O5
|
1
|
| 1 |
IC50 = 110 nM
|
|
|
|
CP0466069
|
4-[[(3aS,9R,9aR)-6-chloro-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
|
C27H26ClF3N2O5
|
2
|
| 1 |
IC50 = 110 nM
|
|
|
| 2 |
Ki = 2.3 nM
|
|
|
|
CP0563966
|
4-[cyclopropyl-(4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl)amino]-4-oxobutanoic acid
Show/Hide
|
C27H30N2O5
|
2
|
| 1 |
IC50 = 120 nM
|
|
|
| 2 |
Ki = 3 nM
|
|
|
|
CP0376330
|
2-(4-bromo-2-formylphenoxy)acetic acid
Show/Hide
|
C9H7BrO4
|
2
|
| 1 |
IC50 = 124 nM
|
|
|
| 2 |
IC50 = 481 nM
|
|
|
|
CP0433532
|
2-(3-(7-chloroquinolin-4-yl)-2,6-dimethyl-1H-indol-1-yl)acetic acid
Show/Hide
|
C21H17ClN2O2
|
1
|
| 1 |
IC50 = 125 nM
|
|
|
|
CP0502787
|
2-(3-(4-amino-2-(4-chlorophenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C20H17ClN2O5S
|
1
|
| 1 |
IC50 = 130 nM
|
|
|
|
CP0482038
|
2-[3-[2-[(2,4-dichlorophenyl)sulfonylamino]benzoyl]-4-methoxyphenyl]acetic acid
Show/Hide
|
C22H17Cl2NO6S
|
1
|
| 1 |
IC50 = 140 nM
|
|
|
|
CP0432250
|
2-[2-[(2-methoxy-5-propan-2-yloxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C21H22N2O5S
|
1
|
| 1 |
IC50 = 150 nM
|
|
|
|
CP0441809
|
4-methoxy-2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
Show/Hide
|
C19H16N2O5
|
2
|
| 1 |
IC50 = 151 nM
|
|
|
| 2 |
IC50 = 4200 nM
|
|
|
|
CP0227496
|
2-(5-bromobiphenyl-2-yloxy)acetic acid
Show/Hide
|
C14H11BrO3
|
1
|
| 1 |
IC50 = 158 nM
|
|
|
|
CP0566097
|
2-[2-[(4-chlorophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 160 nM
|
|
|
|
CP0453605
|
ethyl 2-[4-bromo-2-(1-phenylpyrazole-4-carbonyl)phenoxy]acetate
Show/Hide
|
C20H17BrN2O4
|
2
|
| 1 |
IC50 = 165 nM
|
|
|
| 2 |
IC50 = 3000 nM
|
|
|
|
CP0542936
|
4-[cyclopropyl-(10-phenylmethoxycarbonyl-2,3,4,4a,9,9a-hexahydro-1H-acridin-9-yl)amino]-4-oxobutanoic acid
Show/Hide
|
C28H32N2O5
|
2
|
| 1 |
IC50 = 175 nM
|
|
|
| 2 |
Ki = 32 nM
|
|
|
|
CP0337477
|
2-(5-nitrobiphenyl-2-yloxy)acetic acid
Show/Hide
|
C14H11NO5
|
1
|
| 1 |
IC50 = 178 nM
|
|
|
|
CP0288553
|
2-(1-(7-chloroquinolin-4-yl)-5-methoxy-2-methyl-1H-indol-3-yl)acetic acid
Show/Hide
|
C21H17ClN2O3
|
1
|
| 1 |
IC50 = 180 nM
|
|
|
|
CP0384320
|
N-[(2R,4S)-1-(3-methoxybenzoyl)-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N-phenylacetamide
Show/Hide
|
C26H26N2O3
|
2
|
| 1 |
IC50 = 180 nM
|
|
|
| 2 |
IC50 = 400 nM
|
|
|
|
CP0055418
|
2-[6-chloro-2-(3-chlorobenzoyl)-8-fluoro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl]acetic acid
Show/Hide
|
C20H15Cl2FN2O3
|
3
|
| 1 |
IC50 = 180 nM
|
|
|
| 2 |
IC50 = 190 nM
|
|
|
| 3 |
IC50 = 1280 nM
|
|
|
|
CP0526296
|
2-[2-[(3-chlorophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 186 nM
|
|
|
|
CP0506028
|
2-(6-(4-(N,N-dimethylsulfamoyl)benzyl)-5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C18H20N2O4S2
|
1
|
| 1 |
IC50 = 190 nM
|
|
|
|
CP0539415
|
(+/-)-N-(1-benzyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C25H26N2O
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0403513
|
2-[4-[2-[(4-chlorophenyl)methylcarbamoylamino]-4-(ethylcarbamoyl)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C26H26ClN3O6
|
1
|
| 1 |
IC50 = 200 nM
|
|
|
|
CP0428974
|
(+/-)-N-(1-cinnamoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C27H26N2O2
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0410998
|
2-[2-[(4-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O3S
|
1
|
| 1 |
IC50 = 210 nM
|
|
|
|
CP0515980
|
4-[cyclopropyl-(3-phenylmethoxycarbonyl-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl)amino]-4-oxobutanoic acid
Show/Hide
|
C26H28N2O5
|
2
|
| 1 |
IC50 = 210 nM
|
|
|
| 2 |
Ki = 25 nM
|
|
|
|
CP0257990
|
(R)-2-(7-(N-methyl-4-(trifluoromethyl)phenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C22H21F3N2O4S
|
1
|
| 1 |
IC50 = 214 nM
|
|
|
|
CP0452548
|
N-[(2R,4S)-2-methyl-1-[3-(trifluoromethoxy)benzoyl]-3,4-dihydro-2H-quinolin-4-yl]-N-phenylacetamide
Show/Hide
|
C26H23F3N2O3
|
2
|
| 1 |
IC50 = 217 nM
|
|
|
| 2 |
IC50 > 10000 nM
|
|
|
|
CP0423511
|
2-[2-[(4-bromophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13BrN2O2S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0526295
|
2-[2-[(4-methylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0499513
|
2-[4-[[3-chloro-4-[(2,4-dichlorophenyl)sulfonylamino]-2-methyl-1H-indol-5-yl]oxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C24H19Cl3N2O6S
|
1
|
| 1 |
IC50 = 220 nM
|
|
|
|
CP0516568
|
2-(5-methyl-6-(4-(morpholinosulfonyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C19H20N2O7S3
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0439323
|
2-[4-[4-(butylcarbamoyl)-2-[(4-chlorophenyl)methylamino]phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C27H29ClN2O5
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0423505
|
2-[2-[(3-acetylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H16N2O3S
|
1
|
| 1 |
IC50 = 230 nM
|
|
|
|
CP0496149
|
(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-ethylacetamide
Show/Hide
|
C21H24N2O2
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0055134
|
(R)-2-(7-(N,3,5-trimethylisoxazole-4-sulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C20H23N3O5S
|
1
|
| 1 |
IC50 = 250 nM
|
|
|
|
CP0290306
|
2-(5-cyanobiphenyl-2-yloxy)acetic acid
Show/Hide
|
C15H11NO3
|
1
|
| 1 |
IC50 = 251 nM
|
|
|
|
CP0916787
|
{4-bromo-2-[(pyridin-2-ylhydrazono)methyl]phenoxy}acetic acid
Show/Hide
|
C14H12BrN3O3
|
2
|
| 1 |
IC50 = 255 nM
|
|
|
| 2 |
IC50 = 3490 nM
|
|
|
|
CP0081602
|
(R)-2-(7-(N-methylpyridine-2-sulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C20H21N3O4S
|
1
|
| 1 |
IC50 = 308 nM
|
|
|
|
CP0400762
|
2-[6-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]pyridin-3-yl]acetic acid
Show/Hide
|
C24H23Cl2N3O6S
|
1
|
| 1 |
IC50 = 310 nM
|
|
|
|
CP0524811
|
2-(2-((4-benzoylpiperazin-1-yl)methyl)-4-(trifluoromethyl)phenoxy)acetic acid
Show/Hide
|
C21H21F3N2O4
|
1
|
| 1 |
IC50 = 316 nM
|
|
|
|
CP0506031
|
2-(6-(2-chloro-4-(methylsulfonyl)benzyl)-2,5-dimethyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C18H18ClNO4S2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0403516
|
N-butyl-3-[(2,4-dichlorophenyl)sulfonylamino]-4-[4-[2-(methanesulfonamido)-2-oxoethyl]-2-methoxyphenoxy]benzamide
Show/Hide
|
C27H29Cl2N3O8S2
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0432251
|
2-[2-[(3-bromo-5-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H15BrN2O4S
|
1
|
| 1 |
IC50 = 330 nM
|
|
|
|
CP0399060
|
N-butyl-3-[(2,4-dichlorophenyl)sulfonylamino]-4-[2-methoxy-4-(2H-tetrazol-5-ylmethyl)phenoxy]benzamide
Show/Hide
|
C26H26Cl2N6O5S
|
1
|
| 1 |
IC50 = 350 nM
|
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CP0499090
|
(R)-2-(8-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[4,3-b]indolizin-5-yl)acetic acid
Show/Hide
|
C20H20FN3O4S
|
2
|
| 1 |
IC50 = 351 nM
|
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|
| 2 |
Ki = 139 nM
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CP0423509
|
2-[2-[(3-bromophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13BrN2O2S
|
1
|
| 1 |
IC50 = 370 nM
|
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CP0423514
|
2-[2-[(2-chlorophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13ClN2O2S
|
1
|
| 1 |
IC50 = 370 nM
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CP0475055
|
2-(3-(4-acetyl-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C22H19NO6S
|
1
|
| 1 |
IC50 = 380 nM
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CP0524965
|
2-[2-[(3,4-dichlorophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H12Cl2N2O2S
|
1
|
| 1 |
IC50 = 380 nM
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CP0066637
|
2-(2-benzylsulfanylbenzimidazol-1-yl)acetic acid
Show/Hide
|
C16H14N2O2S
|
1
|
| 1 |
IC50 = 388 nM
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CP0522568
|
2-(5-methyl-6-(4-(pyrrolidin-1-ylsulfonyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C19H20N2O6S3
|
1
|
| 1 |
IC50 = 390 nM
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|
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CP0441807
|
2-(4-bromo-2-(isoxazole-5-carbonyl)phenoxy)acetic acid
Show/Hide
|
C12H8BrNO5
|
2
|
| 1 |
IC50 = 391 nM
|
|
|
| 2 |
IC50 = 2650 nM
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CP0397179
|
2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]sulfonylphenyl]acetic acid
Show/Hide
|
C25H24Cl2N2O7S2
|
1
|
| 1 |
IC50 = 400 nM
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CP0382773
|
N-[(2R,4S)-1-benzoyl-2-methyl-3,4-dihydro-2H-quinolin-4-yl]-N-phenylacetamide
Show/Hide
|
C25H24N2O2
|
2
|
| 1 |
IC50 = 420 nM
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|
|
| 2 |
IC50 > 10000 nM
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CP0392974
|
2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]-2,2-difluoroacetic acid
Show/Hide
|
C26H24Cl2F2N2O7S
|
1
|
| 1 |
IC50 = 420 nM
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CP0506325
|
(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-benzylacetamide
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
IC50 = 430 nM
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|
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CP0423507
|
2-[2-[(3-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H16N2O4S
|
1
|
| 1 |
IC50 = 450 nM
|
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CP0432253
|
2-[2-[(2,5-dichlorophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H12Cl2N2O2S
|
1
|
| 1 |
IC50 = 470 nM
|
|
|
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CP0417212
|
2-[2-(3-phenylpropylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H18N2O2S
|
1
|
| 1 |
IC50 = 475 nM
|
|
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CP0462637
|
2-[2-[[5-[benzyl(ethyl)carbamoyl]-2-methoxyphenyl]methylsulfanyl]-5-fluorobenzimidazol-1-yl]acetic acid
Show/Hide
|
C27H26FN3O4S
|
2
|
| 1 |
IC50 = 495 nM
|
|
|
| 2 |
IC50 = 725 nM
|
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CP0287604
|
2-(5-(thiazol-2-yl)biphenyl-2-yloxy)acetic acid
Show/Hide
|
C17H13NO3S
|
1
|
| 1 |
IC50 = 501 nM
|
|
|
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CP0401619
|
2-[3-[3-(5-benzhydryl-2-oxopyridin-1-yl)propyl]phenoxy]butanoic acid
Show/Hide
|
C31H31NO4
|
1
|
| 1 |
IC50 = 502 nM
|
|
|
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CP0376329
|
2-(2-acetyl-4-bromophenoxy)acetic acid
Show/Hide
|
C10H9BrO4
|
2
|
| 1 |
IC50 = 510 nM
|
|
|
| 2 |
IC50 = 4520 nM
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|
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CP0512038
|
2-(1-phenyl-1H-pyrazole-4-carbonyl)phenoxyacetic acid
Show/Hide
|
C18H14N2O4
|
2
|
| 1 |
IC50 = 510 nM
|
|
|
| 2 |
IC50 = 5350 nM
|
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|
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CP0432254
|
2-[2-[(2-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H16N2O4S
|
1
|
| 1 |
IC50 = 520 nM
|
|
|
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CP0384318
|
(+/-)-3-((1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-3-oxopropanoic acid
Show/Hide
|
C26H24N2O4
|
1
|
| 1 |
IC50 = 540 nM
|
|
|
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CP0889465
|
[2-({[(2,4-dichlorophenoxy)acetyl]hydrazono}methyl)phenoxy]acetic acid
Show/Hide
|
C17H14Cl2N2O5
|
2
|
| 1 |
IC50 = 555 nM
|
|
|
| 2 |
IC50 = 6320 nM
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CP0476526
|
2-[6-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-2,3-dihydro-1-benzofuran-3-yl]acetic acid
Show/Hide
|
C27H26Cl2N2O7S
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
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CP0480118
|
2-[2-[(2-bromophenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C16H13BrN2O2S
|
1
|
| 1 |
IC50 = 580 nM
|
|
|
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CP0549416
|
2-[2-(2-phenoxyethylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O3S
|
1
|
| 1 |
IC50 = 590 nM
|
|
|
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CP0473223
|
2-(4-chloro-2-((4-(phenylsulfonyl)-1,4-diazepan-1-yl)methyl)phenoxy)acetic acid
Show/Hide
|
C20H23ClN2O5S
|
1
|
| 1 |
IC50 = 631 nM
|
|
|
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CP0400763
|
2-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenyl]sulfinylphenyl]acetic acid
Show/Hide
|
C25H24Cl2N2O6S2
|
1
|
| 1 |
IC50 = 660 nM
|
|
|
|
CP0414999
|
2-(3-(4-chloro-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C20H16ClNO5S
|
1
|
| 1 |
IC50 = 680 nM
|
|
|
|
CP0439419
|
2-[4-[4-(butylcarbamoyl)-2-[(3,5-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C26H26Cl2N2O7S
|
2
|
| 1 |
IC50 = 680 nM
|
|
|
| 2 |
IC50 = 4380 nM
|
|
|
|
CP0503270
|
(S)-2-(4-chloro-2-((3-methyl-4-(phenylsulfonyl)piperazin-1-yl)methyl)phenoxy)-2-methylpropanoic acid
Show/Hide
|
C22H27ClN2O5S
|
1
|
| 1 |
IC50 = 708 nM
|
|
|
|
CP0534082
|
2-(5-methylbiphenyl-2-yloxy)acetic acid
Show/Hide
|
C15H14O3
|
1
|
| 1 |
IC50 = 708 nM
|
|
|
|
CP0475056
|
3-(4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3-methoxyphenyl)propanoic acid
Show/Hide
|
C25H24Cl2N2O7S
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0475829
|
2-[2-[(5-chloro-2-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H15ClN2O3S
|
1
|
| 1 |
IC50 = 740 nM
|
|
|
|
CP0399189
|
2-[4-[2-[(2,4-dichlorophenyl)sulfonylamino]-4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenoxy]-3-methoxyphenyl]acetic acid
Show/Hide
|
C25H21Cl2N3O7S
|
1
|
| 1 |
IC50 = 770 nM
|
|
|
|
CP0417482
|
2-[2-(3-phenoxypropylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H18N2O3S
|
1
|
| 1 |
IC50 = 786 nM
|
|
|
|
CP0417225
|
2-[2-[(2-methylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 810 nM
|
|
|
|
CP0240868
|
2-(2-benzoyl-6-chloro-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C20H17ClN2O3
|
1
|
| 1 |
IC50 = 820 nM
|
|
|
|
CP0433261
|
2-[3-[2-(benzenesulfonamido)phenoxy]phenyl]acetic acid
Show/Hide
|
C20H17NO5S
|
1
|
| 1 |
IC50 = 860 nM
|
|
|
|
CP0049438
|
(S)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
|
C21H21FN2O4S
|
1
|
| 1 |
IC50 = 864 nM
|
|
|
|
CP0303839
|
2-[2-(2-phenylethylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O2S
|
1
|
| 1 |
IC50 = 881 nM
|
|
|
|
CP0453603
|
2-(4-bromo-2-(hydroxymethyl)phenoxy)acetic acid
Show/Hide
|
C9H9BrO4
|
2
|
| 1 |
IC50 = 886 nM
|
|
|
| 2 |
IC50 = 6870 nM
|
|
|
|
CP0504724
|
(+/-)-benzyl 2-methyl-4-(N-phenylacetamido)-3,4-dihydroquinoline-1(2H)-carboxylate
Show/Hide
|
C26H26N2O3
|
1
|
| 1 |
IC50 = 910 nM
|
|
|
|
CP0432252
|
2-[2-[(4-bromo-3-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H15BrN2O4S
|
1
|
| 1 |
IC50 = 980 nM
|
|
|
|
CP0423515
|
2-[2-(6-ethoxy-6-oxohexyl)sulfanylbenzimidazol-1-yl]acetic acid
Show/Hide
|
C17H22N2O4S
|
1
|
| 1 |
IC50 = 1010 nM
|
|
|
|
CP0475054
|
2-(3-(4-(diethylcarbamoyl)-2-(4-methylphenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C26H28N2O6S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0425710
|
2-[2-[(2-methoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H16N2O3S
|
1
|
| 1 |
IC50 = 1100 nM
|
|
|
|
CP0502560
|
2-(5-methyl-6-(4-(trifluoromethyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C16H12F3NO4S2
|
1
|
| 1 |
IC50 = 1130 nM
|
|
|
|
CP0410695
|
2-[2-[(2-methoxy-5-methylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H18N2O3S
|
1
|
| 1 |
IC50 = 1200 nM
|
|
|
|
CP0489274
|
2-(2-pentylsulfanylbenzimidazol-1-yl)acetic acid
Show/Hide
|
C14H18N2O2S
|
1
|
| 1 |
IC50 = 1240 nM
|
|
|
|
CP0503534
|
2-(3,5-dimethyl-6-(4-(methylsulfonyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C17H17NO6S3
|
1
|
| 1 |
IC50 = 1300 nM
|
|
|
|
CP0494062
|
2-(2-hexylsulfanylbenzimidazol-1-yl)acetic acid
Show/Hide
|
C15H20N2O2S
|
1
|
| 1 |
IC50 = 1360 nM
|
|
|
|
CP0496654
|
2-(3-(4-methoxy-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
Show/Hide
|
C21H19NO6S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0566104
|
2-[2-(4-phenoxybutylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C19H20N2O3S
|
1
|
| 1 |
IC50 = 1400 nM
|
|
|
|
CP0520363
|
(+/-)-N-(2-methyl-1-(2-methylbenzoyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
IC50 = 1420 nM
|
|
|
|
CP0428975
|
(+/-)-N-(2-methyl-1-pentanoyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C23H28N2O2
|
1
|
| 1 |
IC50 = 1460 nM
|
|
|
|
CP0502237
|
2-(3,5-dimethyl-6-(4-(methylsulfonyl)benzyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C18H19NO4S2
|
1
|
| 1 |
IC50 = 1500 nM
|
|
|
|
CP0480045
|
2-[2-[2-(4-chlorophenoxy)ethylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C17H15ClN2O3S
|
2
|
| 1 |
IC50 = 1500 nM
|
|
|
| 2 |
IC50 = 6600 nM
|
|
|
|
CP0871310
|
[2-(({[5-(4-methoxyphenyl)-1,2,4-triazin-3-yl]hydrazono}methyl)phenoxy]acetic acid
Show/Hide
|
C19H17N5O4
|
2
|
| 1 |
IC50 = 1580 nM
|
|
|
| 2 |
IC50 > 100000 nM
|
|
|
|
CP0283177
|
2-(2-benzoyl-7-methyl-3,4-dihydro-1H-pyrido[4,3-b]indol-5-yl)acetic acid
Show/Hide
|
C21H20N2O3
|
1
|
| 1 |
IC50 = 1590 nM
|
|
|
|
CP0425709
|
2-[2-[(2,5-dimethoxyphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H18N2O4S
|
1
|
| 1 |
IC50 = 1600 nM
|
|
|
|
CP0502236
|
2-(6-(4-fluorophenylsulfonyl)-5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C15H12FNO4S2
|
1
|
| 1 |
IC50 = 1630 nM
|
|
|
|
CP0452549
|
(+/-)-N-(2-methyl-1-(2-phenylacetyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
|
C26H26N2O2
|
1
|
| 1 |
IC50 = 1750 nM
|
|
|
|
CP0506030
|
2-(2,5-dimethyl-6-(4-(methylsulfonyl)benzyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C18H19NO4S2
|
1
|
| 1 |
IC50 = 1800 nM
|
|
|
|
CP0547147
|
N-[(3aS,9R,9aR)-4-benzoyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-N-ethylacetamide
Show/Hide
|
C23H26N2O2
|
2
|
| 1 |
IC50 = 1840 nM
|
|
|
| 2 |
Ki = 26 nM
|
|
|
|
CP0510301
|
2-(2-formylphenoxy)acetic acid
Show/Hide
|
C9H8O4
|
2
|
| 1 |
IC50 = 1970 nM
|
|
|
| 2 |
IC50 = 50000 nM
|
|
|
|
CP0549143
|
2-[2-(2-naphthalen-1-yloxyethylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C21H18N2O3S
|
1
|
| 1 |
IC50 = 2000 nM
|
|
|
|
CP0462641
|
2-[2-[[5-(1-hydroxyethyl)-2-methoxyphenyl]methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C19H20N2O4S
|
1
|
| 1 |
IC50 = 2200 nM
|
|
|
|
CP0529080
|
(+/-)-4-((1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)amino)-4-oxobut-2-enoic acid
Show/Hide
|
C27H24N2O4
|
1
|
| 1 |
IC50 = 2280 nM
|
|
|
|
CP0432294
|
2-[2-(5-ethoxy-5-oxopentyl)sulfanylbenzimidazol-1-yl]acetic acid
Show/Hide
|
C16H20N2O4S
|
1
|
| 1 |
IC50 = 2360 nM
|
|
|
|
CP0404710
|
4-(4-((1H-tetrazol-5-yl)methyl)phenoxy)-3-(2,4-dichlorophenylsulfonamido)-N-ethylbenzamide
Show/Hide
|
C23H20Cl2N6O4S
|
1
|
| 1 |
IC50 = 2370 nM
|
|
|
|
CP0423516
|
2-(2-butylsulfanylbenzimidazol-1-yl)acetic acid
Show/Hide
|
C13H16N2O2S
|
1
|
| 1 |
IC50 = 2370 nM
|
|
|
|
CP0432933
|
2-[2-(2-naphthalen-2-yloxyethylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C21H18N2O3S
|
1
|
| 1 |
IC50 = 2500 nM
|
|
|
|
CP0412498
|
2-[3-[2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]phenyl]acetic acid
Show/Hide
|
C20H15Cl2NO5S
|
1
|
| 1 |
IC50 = 2510 nM
|
|
|
|
CP0417480
|
2-[2-(3-anilinopropylsulfanyl)benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H19N3O2S
|
1
|
| 1 |
IC50 = 2690 nM
|
|
|
|
CP0437110
|
2-(5-methyl-6-(phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C15H13NO4S2
|
1
|
| 1 |
IC50 = 2750 nM
|
|
|
|
CP0410694
|
2-[2-[(2-bromo-3-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
Show/Hide
|
C18H15BrN2O4S
|
1
|
| 1 |
IC50 = 2900 nM
|
|
|
|
CP0469167
|
2-(6-(4-cyanophenylsulfonyl)-5-methyl-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
|
C16H12N2O4S2
|
1
|
| 1 |
IC50 = 3000 nM
|
|
|
|
CP0471527
|
(+/-)-(4-(ethyl(phenyl)amino)-2-methyl-3,4-dihydroquinolin-1(2H)-yl)(phenyl)methanone
Show/Hide
|
C25H26N2O
|
1
|
| 1 |
IC50 = 3170 nM
|
|
|
|
CP0384323
|
(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)acetamide
Show/Hide
|
C19H20N2O2
|
1
|
| 1 |
IC50 = 3620 nM
|
|
|
|
CP0916786
|
{2-[({[(4-methylphenyl)amino]acetyl}hydrazono)methyl]phenoxy}acetic acid
Show/Hide
|
C18H19N3O4
|
2
|
| 1 |
IC50 = 3660 nM
|
|
|
| 2 |
IC50 = 60200 nM
|
|
|
|
CP0502561
|
2-(6-(4-(methylsulfonyl)phenylsulfonyl)-6H-thieno[2,3-b]pyrrol-4-yl)acetic acid
Show/Hide
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C15H13NO6S3
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1
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| 1 |
IC50 = 4000 nM
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CP0462647
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2-[2-(4-ethoxy-4-oxobutyl)sulfanylbenzimidazol-1-yl]acetic acid
Show/Hide
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C15H18N2O4S
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1
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| 1 |
IC50 = 4410 nM
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CP0513055
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2-(4-(4-(methylsulfonyl)phenylsulfonyl)-4H-thieno[3,2-b]pyrrol-6-yl)acetic acid
Show/Hide
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C15H13NO6S3
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1
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| 1 |
IC50 = 5000 nM
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CP0433490
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2-(2-methyl-1-(pyrimidin-4-yl)-1H-indol-3-yl)acetic acid
Show/Hide
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C15H13N3O2
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1
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| 1 |
IC50 = 5200 nM
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CP0384319
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(+/-)-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylbenzenesulfonamide
Show/Hide
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C29H26N2O3S
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1
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| 1 |
IC50 = 5500 nM
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CP0498372
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2-[2-(2-anilinoethylsulfanyl)benzimidazol-1-yl]acetic acid
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C17H17N3O2S
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1
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| 1 |
IC50 = 7690 nM
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CP0384324
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(+/-)-trans-N-(1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
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C25H24N2O2
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1
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| 1 |
IC50 > 10000 nM
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CP0502786
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2-(3-(4-((ethylamino)methyl)-2-(phenylsulfonamido)phenoxy)phenyl)acetic acid
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C23H24N2O5S
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1
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| 1 |
IC50 > 10000 nM
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CP0032219
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(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-2-(methylsulfonyl)-6,7,8,9-tetrahydropyrido[1,2-a]indol-10-yl)acetic acid
Show/Hide
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C22H23FN2O6S2
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1
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| 1 |
IC50 > 10000 nM
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CP0399061
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1-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]cyclopentane-1-carboxylic acid
Show/Hide
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C30H32Cl2N2O7S
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1
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| 1 |
IC50 > 10000 nM
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CP0403515
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1-[4-[4-(butylcarbamoyl)-2-[(2,4-dichlorophenyl)sulfonylamino]phenoxy]-3-methoxyphenyl]cyclopropane-1-carboxylic acid
Show/Hide
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C28H28Cl2N2O7S
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1
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| 1 |
IC50 > 10000 nM
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CP0498371
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2-[2-[5-(ethylamino)-5-oxopentyl]sulfanylbenzimidazol-1-yl]acetic acid
Show/Hide
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C16H21N3O3S
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1
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| 1 |
IC50 > 10000 nM
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CP0400266
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2-[2-[(4-methoxycarbonylphenyl)methylsulfanyl]benzimidazol-1-yl]acetic acid
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C18H16N2O4S
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1
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| 1 |
IC50 = 10600 nM
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CP0408759
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2-[3-(1-benzyl-2-oxoquinazolin-4-yl)-4-methoxyphenyl]acetic acid
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C24H20N2O4
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1
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| 1 |
IC50 = 11000 nM
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CP0883494
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[2-(({[(3-methyl-1H-pyrazol-5-yl)carbonyl]hydrazono}methyl)phenoxy]acetic acid
Show/Hide
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C14H14N4O4
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2
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| 1 |
IC50 = 11200 nM
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| 2 |
IC50 > 100000 nM
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CP0461933
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2-[2-(3-ethoxy-3-oxopropyl)sulfanylbenzimidazol-1-yl]acetic acid
Show/Hide
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C14H16N2O4S
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1
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| 1 |
IC50 = 11400 nM
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CP0881027
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(2-{[(1H-benzimidazol-1-ylacetyl)hydrazono]methyl}phenoxy)acetic acid
Show/Hide
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C18H16N4O4
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2
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| 1 |
IC50 = 12800 nM
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| 2 |
IC50 = 81700 nM
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CP0502666
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(+/-)-3-((1-benzoyl-2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)(phenyl)carbamoyl)benzoic acid
Show/Hide
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C31H26N2O4
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1
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| 1 |
IC50 = 40300 nM
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CP0459076
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(+/-)-N-(2-methyl-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
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C18H20N2O
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1
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| 1 |
IC50 > 50000 nM
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CP0868052
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(+/-)-(2-methyl-4-(phenylamino)-3,4-dihydroquinolin-1(2H)-yl)(phenyl)methanone
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C23H22N2O
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1
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| 1 |
IC50 > 50000 nM
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CP0491156
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4-(2-(2,4-dichlorophenylsulfonamido)-4-(ethylcarbamoyl)phenoxy)-3-methoxybenzoic acid
Show/Hide
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C23H20Cl2N2O7S
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1
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| 1 |
IC50 > 50000 nM
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CP0529081
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(+/-)-N-(2-methyl-1-(phenylsulfonyl)-1,2,3,4-tetrahydroquinolin-4-yl)-N-phenylacetamide
Show/Hide
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C24H24N2O3S
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1
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| 1 |
IC50 = 62000 nM
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CP0443722
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5-[3-(4-fluorophenyl)-4-oxo-7-(5-phenyl-1,2-oxazol-3-yl)quinazolin-2-yl]pentanoic acid
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C28H22FN3O4
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1
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| 1 |
Ki = 2.6 nM
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CP0515999
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4-[[(2aS,8R,8aR)-3-[3-(trifluoromethoxy)benzoyl]-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C26H25F3N2O5
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1
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| 1 |
Ki = 5 nM
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CP0571158
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US9290454, 3.1
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C31H29FN2O4
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1
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| 1 |
Ki = 5.8 nM
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CP0548231
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US9290454, 4.4
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C29H26F2N2O4
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1
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| 1 |
Ki = 5.9 nM
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CP0444398
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4-[[(3aS,9R,9aR)-4-[(1S)-1-(4-fluorophenyl)ethoxy]carbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C28H31FN2O5
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1
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| 1 |
Ki = 6 nM
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CP0561731
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US9290454, 3.2
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C31H28F2N2O4
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1
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| 1 |
Ki = 6.5 nM
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CP0566728
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C27H27F3N2O5
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1
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| 1 |
Ki = 7 nM
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CP0561732
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5-[2-(4-fluorophenyl)-6-[[5-[(4-fluorophenyl)methyl]-1,2,4-oxadiazol-3-yl]carbamoyl]-1-oxoisoquinolin-3-yl]pentanoic acid
Show/Hide
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C30H24F2N4O5
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1
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| 1 |
Ki = 7.8 nM
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CP0383896
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4-[[(2aS,8R,8aR)-3-(3-fluorobenzoyl)-2,2a,8,8a-tetrahydro-1H-cyclobuta[b]quinolin-8-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C25H25FN2O4
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1
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| 1 |
Ki = 8.1 nM
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CP0568400
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US9290454, 3.3
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C30H29FN2O5
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1
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| 1 |
Ki = 8.5 nM
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CP0566729
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclobutylamino]-4-oxobutanoic acid
Show/Hide
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C28H29F3N2O5
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1
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| 1 |
Ki = 8.6 nM
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CP0566730
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-(cyclobutylmethyl)amino]-4-oxobutanoic acid
Show/Hide
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C29H31F3N2O5
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1
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| 1 |
Ki = 9 nM
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CP0408532
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US9290454, 3.4
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C30H26FN3O4
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1
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| 1 |
Ki = 9.2 nM
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CP0566734
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2-[(4-benzoyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl)-cyclopropylcarbamoyl]oxyacetic acid
Show/Hide
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C25H26N2O5
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1
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| 1 |
Ki = 9.4 nM
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CP0930607
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5-(6-(5-(4-fluorobenzyl)isoxazol-3-ylcarbamoyl)-2-(4-fluorophenyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
Show/Hide
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C31H25F2N3O5
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1
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| 1 |
Ki = 11 nM
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CP0563952
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-ethylamino]-4-oxobutanoic acid
Show/Hide
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C26H27F3N2O5
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1
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| 1 |
Ki = 12 nM
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CP0563953
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4-[[(3aS,9R,9aR)-4-[(4-fluorophenyl)methoxycarbonyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C27H29FN2O5
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1
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| 1 |
Ki = 12 nM
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CP0408584
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US9290454, 3.5
Show/Hide
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C30H29FN2O5
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1
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| 1 |
Ki = 13 nM
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CP0911253
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5-(2-(4-fluorophenyl)-6-(5-(1-(4-fluorophenyl)ethyl)-1,2,4-oxadiazol-3-ylcarbamoyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
Show/Hide
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C31H26F2N4O5
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1
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| 1 |
Ki = 13 nM
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CP0411535
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US9290454, 4.2
Show/Hide
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C32H32FN3O4
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1
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| 1 |
Ki = 14 nM
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CP0516004
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4-[[(3aS,9R,9aR)-7-(difluoromethyl)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C28H27F5N2O5
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1
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| 1 |
Ki = 14 nM
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CP0567226
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4-[[(3aS,9R,9aR)-4-[(1R)-1-(4-fluorophenyl)ethoxy]carbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C28H31FN2O5
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1
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| 1 |
Ki = 14 nM
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CP0568403
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US9290454, 8.2
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C32H31F2N3O5S
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1
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| 1 |
Ki = 15 nM
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CP0566727
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-methylamino]-4-oxobutanoic acid
Show/Hide
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C25H25F3N2O5
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1
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| 1 |
Ki = 16 nM
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CP0572465
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US9290454, 3.6
Show/Hide
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C30H29FN2O5
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1
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| 1 |
Ki = 19 nM
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CP0568402
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US9290454, 4.3
Show/Hide
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C30H26FN3O5
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1
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| 1 |
Ki = 21 nM
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CP0948986
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5-(6-(5-(2,3-dihydro-1H-inden-2-yl)-1,2,4-oxadiazol-3-ylcarbamoyl)-2-(4-fluorophenyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
Show/Hide
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C32H27FN4O5
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1
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| 1 |
Ki = 22 nM
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CP0568401
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US9290454, 4.1
Show/Hide
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C32H31F2N3O4
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1
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| 1 |
Ki = 24 nM
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CP0957547
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5-(6-(5-(6-fluorobenzo[d]oxazol-2-yl)-5-methyl-4,5-dihydroisoxazol-3-ylcarbamoyl)-2-(4-fluorophenyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
Show/Hide
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C32H26F2N4O6
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1
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| 1 |
Ki = 26 nM
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CP0574980
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4-[[(3aS,9R,9aR)-4-(5-phenyl-1,3,4-oxadiazol-2-yl)-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C27H28N4O4
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1
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| 1 |
Ki = 28 nM
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CP0372689
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2-[6-[(4-fluorophenyl)sulfonylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]acetic acid
Show/Hide
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C20H19FN2O4S
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2
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| 1 |
Ki = 30 nM
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| 2 |
Ki ~ 21000 nM
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CP0566732
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4-[[(3aS,9R,9aR)-7-ethyl-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C29H31F3N2O5
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1
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| 1 |
Ki = 31 nM
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CP0555541
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-(3,3,3-trifluoropropyl)amino]-4-oxobutanoic acid
Show/Hide
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C27H26F6N2O5
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1
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| 1 |
Ki = 35 nM
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CP0541449
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4-[[(3aS,9R,9aR)-7-(hydroxymethyl)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C28H29F3N2O6
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1
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| 1 |
Ki = 38 nM
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CP0444402
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4-[[(3aS,9R,9aR)-7-cyclopropyl-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C30H31F3N2O5
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1
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| 1 |
Ki = 43 nM
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CP0429722
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US9290454, 1.2
Show/Hide
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C30H28F2N2O4
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1
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| 1 |
Ki = 49 nM
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CP0574977
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-propan-2-ylamino]-4-oxobutanoic acid
Show/Hide
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C27H29F3N2O5
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1
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| 1 |
Ki = 50 nM
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CP0574979
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4-[[(3aS,9R,9aR)-4-(phenylcarbamoyl)-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C26H29N3O4
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1
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| 1 |
Ki = 56 nM
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CP0574978
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4-[[(3aS,9R,9aS)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-(1-methylcyclopropyl)amino]-4-oxobutanoic acid
Show/Hide
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C28H29F3N2O5
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1
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| 1 |
Ki = 64 nM
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CP0566731
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(2R)-4-[[(3aS,9R,9aR)-4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-2-methyl-4-oxobutanoic acid
Show/Hide
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C28H32N2O5
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1
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| 1 |
Ki = 82 nM
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CP0444400
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N-[(3aS,9R,9aR)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-N-cyclopropyl-3-(2H-tetrazol-5-yl)propanamide
Show/Hide
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C27H27F3N6O3
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1
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| 1 |
Ki = 98 nM
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CP0465980
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4-[[(3aS,9R,9aR)-7-(4-fluorophenyl)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C33H30F4N2O5
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1
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| 1 |
Ki = 110 nM
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CP0485660
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3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
Show/Hide
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C21H21FN2O4S
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1
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| 1 |
Ki = 250 nM
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CP0566733
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4-[[(3aS,9R,9aR)-7-pyrimidin-5-yl-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C31H29F3N4O5
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1
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| 1 |
Ki = 300 nM
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CP0511773
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4-[[(3aS,9R,9aR)-4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-2-methyl-4-oxobutanoic acid
Show/Hide
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C28H32N2O5
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1
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| 1 |
Ki = 510 nM
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CP0516000
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4-[[(3aS,9R,9aR)-4-[2-(4-fluoroanilino)-2-oxoethyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-4-oxobutanoic acid
Show/Hide
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C27H30FN3O4
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1
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| 1 |
Ki = 660 nM
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CP0857301
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(R)-5-(6-(1-(4-fluorophenyl)ethylcarbamoyl)-1-oxo-1,2-dihydroisoquinolin-3-yl)pentanoic acid
Show/Hide
|
C23H23FN2O4
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1
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| 1 |
Ki = 703 nM
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CP0444399
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2-[[(3aS,9R,9aR)-4-[4-(trifluoromethoxy)benzoyl]-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylcarbamoyl]benzoic acid
Show/Hide
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C31H27F3N2O5
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1
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| 1 |
Ki = 840 nM
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CP0432582
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3-[6-(2-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
Show/Hide
|
C21H21FN2O4S
|
1
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| 1 |
Ki = 970 nM
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CP0439385
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3-(6-Benzenesulfonylamino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid
Show/Hide
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C21H22N2O4S
|
1
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| 1 |
Ki = 1200 nM
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CP0432581
|
3-[6-(3-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
Show/Hide
|
C21H21FN2O4S
|
1
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| 1 |
Ki = 1300 nM
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CP0516005
|
5-[cyclopropyl-(4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl)amino]-5-oxopentanoic acid
Show/Hide
|
C28H32N2O5
|
1
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| 1 |
Ki = 1490 nM
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CP0485086
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3-[6-(3-Chloro-4-fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H20ClFN2O4S
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1
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| 1 |
Ki = 1700 nM
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CP0504929
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3-[6-(4-Methoxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C22H24N2O5S
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1
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| 1 |
Ki = 2100 nM
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CP0442320
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2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-ethanesulfonic acid
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C20H21FN2O5S2
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1
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| 1 |
Ki = 2400 nM
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CP0499224
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3-[6-(4-Chloro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H21ClN2O4S
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1
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| 1 |
Ki = 3000 nM
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CP0420031
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3-[6-(Toluene-4-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C22H24N2O4S
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1
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| 1 |
Ki = 3200 nM
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CP0445762
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3-[6-(Biphenyl-4-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C27H26N2O4S
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1
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| 1 |
Ki = 3300 nM
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CP0501591
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3-[6-(2,4-Difluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H20F2N2O4S
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1
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| 1 |
Ki = 3600 nM
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CP0420032
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3-[6-(Toluene-3-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C22H24N2O4S
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1
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| 1 |
Ki = 4200 nM
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CP0496861
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3-[6-(3,4-Difluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H20F2N2O4S
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1
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| 1 |
Ki = 4200 nM
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CP0435410
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2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H21FN2O4S
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1
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| 1 |
Ki = 4400 nM
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CP0497843
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5-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-pentanoic acid
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C23H25FN2O4S
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1
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| 1 |
Ki = 4600 nM
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CP0559094
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US9290454, 2.1
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C26H20F2N2O4
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1
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| 1 |
Ki = 4920 nM
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CP0497313
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4-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid
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C25H21FN2O4S
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1
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| 1 |
Ki = 6400 nM
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CP0378830
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(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[3,4-b]indolizin-10-yl)acetic acid
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C20H20FN3O4S
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1
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| 1 |
Ki = 6725 nM
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CP0073515
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(R)-2-(7-(4-fluoro-N-methylphenylsulfonamido)-6,7,8,9-tetrahydropyrido[2,3-b]indolizin-10-yl)acetic acid
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C20H20FN3O4S
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1
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| 1 |
Ki = 7189 nM
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CP0499223
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3-[6-(4-Hydroxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C21H22N2O5S
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1
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| 1 |
Ki = 7400 nM
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CP0511254
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3-[6-(Naphthalene-2-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C25H24N2O4S
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1
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| 1 |
Ki = 7400 nM
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CP0392612
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3-[6-(4-Phenoxy-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C27H26N2O5S
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1
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| 1 |
Ki = 7500 nM
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CP0420033
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3-[6-(Thiophene-2-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C19H20N2O4S2
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1
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| 1 |
Ki = 7600 nM
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CP0547148
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4-[[(3aS,9R,9aR)-4-phenylmethoxycarbonyl-1,2,3,3a,9,9a-hexahydrocyclopenta[b]quinolin-9-yl]-cyclopropylamino]-2,2-dimethyl-4-oxobutanoic acid
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C29H34N2O5
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1
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| 1 |
Ki = 7800 nM
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CP0497842
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4-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-butyric acid
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C22H23FN2O4S
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1
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| 1 |
Ki = 8300 nM
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CP0404848
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3-(6-Benzylamino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid
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C22H24N2O2
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1
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| 1 |
Ki = 17000 nM
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CP0509498
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2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-butyric acid
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C22H23FN2O4S
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1
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| 1 |
Ki = 18000 nM
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CP0445494
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(Z)-3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-acrylic acid
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C21H19FN2O4S
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1
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| 1 |
Ki = 19000 nM
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CP0497847
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3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid
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C25H21FN2O4S
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1
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| 1 |
Ki = 27000 nM
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CP0511275
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2-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-benzoic acid
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C25H21FN2O4S
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1
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| 1 |
Ki = 33000 nM
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CP0372688
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2-[6-[(4-fluorophenyl)sulfonylamino]-1,2,3,4-tetrahydrocarbazol-9-yl]ethylphosphonic acid
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C20H22FN2O5PS
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1
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| 1 |
Ki > 50000 nM
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CP0420114
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3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-butyric acid
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C22H23FN2O4S
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1
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| 1 |
Ki > 50000 nM
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CP0445761
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3-[6-(Toluene-2-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C22H24N2O4S
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1
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| 1 |
Ki > 50000 nM
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CP0445885
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3-[6-(3-Phenyl-ureido)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C22H23N3O3
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1
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| 1 |
Ki > 50000 nM
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CP0485087
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3-[6-(Propane-1-sulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-propionic acid
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C18H24N2O4S
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1
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| 1 |
Ki > 50000 nM
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CP0497816
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3-(6-Benzoylamino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid
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C22H22N2O3
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1
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| 1 |
Ki > 50000 nM
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CP0497841
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3-(6-Amino-1,2,3,4-tetrahydro-carbazol-9-yl)-propionic acid
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C15H18N2O2
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1
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| 1 |
Ki > 50000 nM
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CP0511249
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3-[6-(4-Fluoro-benzenesulfonylamino)-1,2,3,4-tetrahydro-carbazol-9-yl]-2-methyl-propionic acid
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C22H23FN2O4S
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1
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| 1 |
Ki > 50000 nM
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